Mechanism of action of cariprazine.

Article Details

Citation

Stahl SM

Mechanism of action of cariprazine.

CNS Spectr. 2016 Apr;21(2):123-7. doi: 10.1017/S1092852916000043. Epub 2016 Mar 9.

PubMed ID
26956157 [ View in PubMed
]
Abstract

Cariprazine is a new therapeutic agent recently approved for the treatment of both schizophrenia and manic or mixed episodes associated with bipolar disorder, and is under investigation for the treatment of both bipolar depression and major depressive disorder.

DrugBank Data that Cites this Article

Drugs
Drug Targets
DrugTargetKindOrganismPharmacological ActionActions
Cariprazine5-hydroxytryptamine receptor 1AProteinHumans
Unknown
Partial agonist
Details
Cariprazine5-hydroxytryptamine receptor 2AProteinHumans
Unknown
Antagonist
Details
Cariprazine5-hydroxytryptamine receptor 2BProteinHumans
Unknown
Antagonist
Details
CariprazineDopamine D2 receptorProteinHumans
Unknown
Partial agonist
Details
CariprazineDopamine D3 receptorProteinHumans
Unknown
Partial agonist
Details
CariprazineHistamine H1 receptorProteinHumans
Unknown
Antagonist
Details