Antarelix (EP 24332) a novel water soluble LHRH antagonist.
Article Details
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Deghenghi R, Boutignon F, Wuthrich P, Lenaerts V
Antarelix (EP 24332) a novel water soluble LHRH antagonist.
Biomed Pharmacother. 1993;47(2-3):107-10.
- PubMed ID
- 7693007 [ View in PubMed]
- Abstract
A novel water soluble LHRH antagonist (EP 24332-Antarelix) is described. Its activity in vitro and in vivo in several animal models is given. Antarelix (Ac-D-Nal, D-Cpa, D-Pal, Ser, Tyr, D-Hci, Leu, Lys-(iPr), Pro, D-Ala-NH2) in view of its potency, modest histamine-liberating activity and high water solubility has been selected for further development.
DrugBank Data that Cites this Article
- Drug Targets
Drug Target Kind Organism Pharmacological Action Actions Teverelix Gonadotropin-releasing hormone receptor Protein Humans YesAntagonistDetails