Moderately to Severely Active Ulcerative Colitis

DrugDrug NameDrug Description
DB00051AdalimumabA monoclonal anti-tumor necrosis factor alpha antibody used in the treatment of a wide variety of inflammatory conditions such as rheumatoid arthritis, Crohn's disease, and ankylosing spondylitis.
DB14766EtrasimodAn S1P receptors modulator used to treat moderate to severely active ulcerative colitis in adults
DB14845FilgotinibA Janus kinase (JAK) 1 selective inhibitor used to treat cases of rheumatoid arthritis that are unresponsive to conventional treatments.
DB00065InfliximabA monoclonal anti tumor necrosis factor alpha antibody used in the treatment of a wide variety of inflammatory conditions such as rheumatoid arthritis, Crohn's disease, and ankylosing spondylitis.
DB14910MirikizumabAn anti-IL-23 monoclonal antibody used as a second-line therapy for moderate-to-severe active ulcerative colitis.
DB12612OzanimodA sphingosine 1-phosphate receptor modulator being studied to treat Multiple Sclerosis (MS) and inflammatory bowel disease (IBD).
DB15091UpadacitinibAn oral Janus kinase (JAK)1-selective inhibitor used in the treatment of moderate to severe rheumatoid arthritis, active psoriatic arthritis, ankylosing spondylitis, and severe atopic dermatitis, including in patients who did not respond well to other therapies.
DB09033VedolizumabAn integrin blocker and anti-inflammatory agent used to manage ulcerative colitis and Crohn's disease in adults.
DrugDrug NameTargetType
DB00051AdalimumabTumor necrosis factortarget
DB14766EtrasimodCytochrome P450 2C8enzyme
DB14766EtrasimodCytochrome P450 2C9enzyme
DB14766EtrasimodCytochrome P450 2C19enzyme
DB14766EtrasimodCytochrome P450 2J2enzyme
DB14766EtrasimodCytochrome P450 3A4enzyme
DB14766EtrasimodSphingosine 1-phosphate receptor 1target
DB14766EtrasimodSphingosine 1-phosphate receptor 4target
DB14766EtrasimodSphingosine 1-phosphate receptor 5target
DB14845FilgotinibTyrosine-protein kinase JAK1target
DB14845FilgotinibCocaine esteraseenzyme
DB14845FilgotinibLiver carboxylesterase 1enzyme
DB14845FilgotinibP-glycoprotein 1transporter
DB00065InfliximabTumor necrosis factortarget
DB14910MirikizumabInterleukin-23 subunit alphatarget
DB12612OzanimodSphingosine 1-phosphate receptor 1target
DB12612OzanimodSphingosine 1-phosphate receptor 5target
DB12612OzanimodAmine oxidase [flavin-containing] Btransporter
DB12612OzanimodATP-binding cassette sub-family G member 2transporter
DB12612OzanimodP-glycoprotein 1transporter
DB12612OzanimodFatty aldehyde dehydrogenaseenzyme
DB12612OzanimodAlcohol dehydrogenase class-3enzyme
DB12612OzanimodArylamine N-acetyltransferase 2enzyme
DB12612OzanimodCytochrome P450 2C8enzyme
DB12612OzanimodAmine oxidase [flavin-containing] Benzyme
DB12612OzanimodAldo-keto reductase family 1 member C1enzyme
DB12612OzanimodAldo-keto reductase family 1 member C2enzyme
DB12612OzanimodCytochrome P450 3A4enzyme
DB15091UpadacitinibTyrosine-protein kinase JAK1target
DB15091UpadacitinibCytochrome P450 3A4enzyme
DB15091UpadacitinibCytochrome P450 2D6enzyme
DB15091UpadacitinibP-glycoprotein 1transporter
DB15091UpadacitinibATP-binding cassette sub-family G member 2transporter
DB15091UpadacitinibSolute carrier organic anion transporter family member 1B1transporter
DB09033VedolizumabIntegrin alpha-4target
DB09033VedolizumabIntegrin beta-7target
DrugDrug NamePhaseStatusCount
DB14766Etrasimod3Active Not Recruiting1
DB09033Vedolizumab3Recruiting1