Monotherapy

DrugDrug NameDrug Description
DB01238AripiprazoleAn atypical antipsychotic used in the treatment of a wide variety of mood and psychotic disorders, such as schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's syndrome.
DB09038EmpagliflozinAn SGLT2 inhibitor used to manage type 2 diabetes mellitus.
DB05889Inotuzumab ozogamicinAn antibody-drug conjugate used to treat B-cell precursor acute lymphoblastic leukemia (ALL).
DB00762IrinotecanA topoisomerase inhibitor used to treat metastatic carcinoma of the colon or rectum and pancreatic adenocarcinoma.
DB00108NatalizumabA monoclonal anti-integrin antibody used to treat Crohn's disease or multiple sclerosis.
DB00776OxcarbazepineAn anti-epileptic used in the treatment of partial-onset seizures.
DB00642PemetrexedA folate analog used to treat mesothelioma and non-small cell lung cancer.
DB15626SpesolimabAn interleukin-36 receptor antagonist used to treat generalized pustular psoriasis flares in adults.
DB16732Tisotumab vedotinA tissue factor-directed antibody drug conjugate that is used to treat adults with recurrent or metastatic cervical cancer with disease progression on or after chemotherapy.
DB06273TocilizumabAn interleukin-6 (IL-6) receptor antagonist used to treat Cytokine Release Syndrome (CRS), Systemic Juvenile Idiopathic Arthritis (sJIA), Giant Cell Arteritis (GCA), and Rheumatoid Arthritis (RA).
DB00361VinorelbineA vinca alkaloid used in the treatment of metastatic non-small cell lung carcinoma (NSLC) and in conjunction with other drugs in locally advanced NSCLC.
DrugDrug NameTargetType
DB01238AripiprazoleDopamine D2 receptortarget
DB01238Aripiprazole5-hydroxytryptamine receptor 1Atarget
DB01238Aripiprazole5-hydroxytryptamine receptor 2Atarget
DB01238AripiprazoleCytochrome P450 3A4enzyme
DB01238AripiprazoleCytochrome P450 2D6enzyme
DB01238Aripiprazole5-hydroxytryptamine receptor 1Btarget
DB01238Aripiprazole5-hydroxytryptamine receptor 1Dtarget
DB01238Aripiprazole5-hydroxytryptamine receptor 1Etarget
DB01238AripiprazoleDopamine D1 receptortarget
DB01238AripiprazoleDopamine D5 receptortarget
DB01238AripiprazoleDopamine D3 receptortarget
DB01238AripiprazoleDopamine D4 receptortarget
DB01238Aripiprazole5-hydroxytryptamine receptor 2Ctarget
DB01238Aripiprazole5-hydroxytryptamine receptor 3Atarget
DB01238Aripiprazole5-hydroxytryptamine receptor 6target
DB01238Aripiprazole5-hydroxytryptamine receptor 7target
DB01238AripiprazoleHistamine H1 receptortarget
DB01238AripiprazoleAlpha-1A adrenergic receptortarget
DB01238AripiprazoleAlpha-1B adrenergic receptortarget
DB01238AripiprazoleAlpha-2A adrenergic receptortarget
DB01238AripiprazoleAlpha-2B adrenergic receptortarget
DB01238AripiprazoleAlpha-2C adrenergic receptortarget
DB01238AripiprazoleCytochrome P450 3A5enzyme
DB01238AripiprazoleCytochrome P450 3A7enzyme
DB01238AripiprazoleSerum albumincarrier
DB01238Aripiprazole5-hydroxytryptamine receptor 2Btarget
DB01238Aripiprazole5-hydroxytryptamine receptor 5Atarget
DB01238AripiprazoleBeta-1 adrenergic receptortarget
DB01238AripiprazoleBeta-2 adrenergic receptortarget
DB01238AripiprazoleHistamine H2 receptortarget
DB01238AripiprazoleHistamine H3 receptortarget
DB01238AripiprazoleHistamine H4 receptortarget
DB01238AripiprazoleMuscarinic acetylcholine receptor M1target
DB01238AripiprazoleMuscarinic acetylcholine receptor M2target
DB01238AripiprazoleMuscarinic acetylcholine receptor M3target
DB01238AripiprazoleMuscarinic acetylcholine receptor M4target
DB01238AripiprazoleMuscarinic acetylcholine receptor M5target
DB01238AripiprazoleKappa-type opioid receptortarget
DB01238AripiprazoleMu-type opioid receptortarget
DB01238AripiprazoleDelta-type opioid receptortarget
DB01238AripiprazoleGlutamate (NMDA) receptortarget
DB01238AripiprazoleSodium-dependent dopamine transportertarget
DB01238AripiprazoleSodium-dependent serotonin transportertarget
DB01238AripiprazoleP-glycoprotein 1transporter
DB01238AripiprazoleATP-binding cassette sub-family G member 2transporter
DB09038EmpagliflozinSodium/glucose cotransporter 2target
DB09038EmpagliflozinUDP-glucuronosyltransferase 2B7enzyme
DB09038EmpagliflozinUDP-glucuronosyltransferase 1-3enzyme
DB09038EmpagliflozinUDP-glucuronosyltransferase 1-8enzyme
DB09038EmpagliflozinUDP-glucuronosyltransferase 1-9enzyme
DB09038EmpagliflozinP-glycoprotein 1transporter
DB09038EmpagliflozinATP-binding cassette sub-family G member 2transporter
DB09038EmpagliflozinSolute carrier family 22 member 8transporter
DB09038EmpagliflozinSolute carrier organic anion transporter family member 1B1transporter
DB09038EmpagliflozinSolute carrier organic anion transporter family member 1B3transporter
DB05889Inotuzumab ozogamicinP-glycoprotein 1transporter
DB05889Inotuzumab ozogamicinB-cell receptor CD22target
DB00762IrinotecanDNA topoisomerase I, mitochondrialtarget
DB00762IrinotecanDNA topoisomerase 1target
DB00762IrinotecanCytochrome P450 3A4enzyme
DB00762IrinotecanCytochrome P450 3A5enzyme
DB00762IrinotecanUDP-glucuronosyltransferase 1-1enzyme
DB00762IrinotecanUDP-glucuronosyltransferase 1-9enzyme
DB00762IrinotecanCytochrome P450 3A7enzyme
DB00762IrinotecanSolute carrier family 22 member 3transporter
DB00762IrinotecanSolute carrier organic anion transporter family member 1B1transporter
DB00762IrinotecanMultidrug resistance-associated protein 1transporter
DB00762IrinotecanATP-binding cassette sub-family G member 2transporter
DB00762IrinotecanSerum albumincarrier
DB00762IrinotecanP-glycoprotein 1transporter
DB00762IrinotecanCanalicular multispecific organic anion transporter 1transporter
DB00762IrinotecanHuman Carboxylesterasesenzyme
DB00108NatalizumabIntegrin alpha-4target
DB00108NatalizumabLow affinity immunoglobulin gamma Fc region receptor III-Btarget
DB00108NatalizumabHigh affinity immunoglobulin gamma Fc receptor Itarget
DB00108NatalizumabIntercellular adhesion molecule 1target
DB00776OxcarbazepineCytochrome P450 2C19enzyme
DB00776OxcarbazepineCytochrome P450 3A4enzyme
DB00776OxcarbazepineCytochrome P450 3A5enzyme
DB00776OxcarbazepineSerum albumincarrier
DB00776OxcarbazepineP-glycoprotein 1transporter
DB00776OxcarbazepineAldo-keto reductase family 1 member C1enzyme
DB00776OxcarbazepineAldo-keto reductase family 1 member C2enzyme
DB00776OxcarbazepineAldo-keto reductase family 1 member C3enzyme
DB00776OxcarbazepineAldo-keto reductase family 1 member C4enzyme
DB00776OxcarbazepineCarbonyl reductase [NADPH] 1enzyme
DB00776OxcarbazepineCarbonyl reductase [NADPH] 3enzyme
DB00776OxcarbazepineSodium channel proteintarget
DB00642PemetrexedThymidylate synthasetarget
DB00642PemetrexedDihydrofolate reductasetarget
DB00642PemetrexedTrifunctional purine biosynthetic protein adenosine-3target
DB00642PemetrexedDeoxycytidine kinaseenzyme
DB00642PemetrexedBifunctional purine biosynthesis protein PURHtarget
DB00642PemetrexedEquilibrative nucleoside transporter 1enzyme
DB00642PemetrexedSolute carrier family 22 member 8transporter
DB00642PemetrexedFolate transporter 1transporter
DB00642PemetrexedProton-coupled folate transportertransporter
DB00642PemetrexedATP-binding cassette sub-family G member 2transporter
DB00642PemetrexedMultidrug resistance-associated protein 5transporter
DB00642PemetrexedSolute carrier family 22 member 6transporter
DB00642PemetrexedSerum albumincarrier
DB00642PemetrexedSolute carrier family 22 member 11transporter
DB15626SpesolimabInterleukin-1 receptor-like 2target
DB16732Tisotumab vedotinCytochrome P450 3A4enzyme
DB16732Tisotumab vedotinTissue factortarget
DB16732Tisotumab vedotinP-glycoprotein 1transporter
DB06273TocilizumabInterleukin-6 receptor subunit alphatarget
DB06273TocilizumabCytochrome P450 3A4enzyme
DB00361VinorelbineTubulin beta chaintarget
DB00361VinorelbineCytochrome P450 3A4enzyme
DB00361VinorelbineCytochrome P450 2D6enzyme
DrugDrug NamePhaseStatusCount
DB07101Mirdametinib1 / 2Recruiting1
DB08930Dolutegravir2Completed1
DB08930Dolutegravir2Unknown Status1
DB00564Carbamazepine3Completed2
DB06218Lacosamide3Completed2