| Reteplase | target | Urokinase plasminogen activator surface receptor | Details |
| Reteplase | target | Fibrinogen alpha chain | Details |
| Reteplase | target | Plasminogen | Details |
| Erythropoietin | target | Erythropoietin receptor | Details |
| Salmon Calcitonin | target | Calcitonin receptor | Details |
| Interferon alfa-n3 | enzyme | Cytochrome P450 1A2 | Details |
| Interferon alfa-n3 | target | Interferon alpha/beta receptor 1 | Details |
| Interferon alfa-n3 | target | Interferon alpha/beta receptor 2 | Details |
| Pegfilgrastim | target | Granulocyte colony-stimulating factor receptor | Details |
| Pegfilgrastim | enzyme | Neutrophil elastase | Details |
| Sargramostim | target | Bone marrow proteoglycan | Details |
| Sargramostim | target | Interleukin-3 receptor subunit alpha | Details |
| Sargramostim | target | Syndecan-2 | Details |
| Sargramostim | target | Granulocyte-macrophage colony-stimulating factor receptor subunit alpha | Details |
| Sargramostim | target | Cytokine receptor common subunit beta | Details |
| Peginterferon alfa-2b | target | Interferon alpha/beta receptor 1 | Details |
| Peginterferon alfa-2b | enzyme | Cytochrome P450 1A2 | Details |
| Peginterferon alfa-2b | target | Interferon alpha/beta receptor 2 | Details |
| Peginterferon alfa-2b | enzyme | Cytochrome P450 2D6 | Details |
| Peginterferon alfa-2b | enzyme | Cytochrome P450 2C9 | Details |
| Asparaginase Escherichia coli | carrier | Thyroxine-binding globulin | Details |
| Asparaginase Escherichia coli | target | L-asparagine | Details |
| Thyrotropin alfa | target | Thyrotropin receptor | Details |
| Antihemophilic factor, human recombinant | target | Phytanoyl-CoA dioxygenase, peroxisomal | Details |
| Antihemophilic factor, human recombinant | target | 78 kDa glucose-regulated protein | Details |
| Antihemophilic factor, human recombinant | target | Calreticulin | Details |
| Antihemophilic factor, human recombinant | target | Protein ERGIC-53 | Details |
| Antihemophilic factor, human recombinant | target | Prolow-density lipoprotein receptor-related protein 1 | Details |
| Antihemophilic factor, human recombinant | enzyme | Prothrombin | Details |
| Antihemophilic factor, human recombinant | target | Coagulation factor IX | Details |