The Cost of Knowledge: Evaluating Open vs. Paid Data for Pharma
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Substrate
Enzyme
Products
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Acalabrutinib M27 Metabolite (ACP-5862)
DBMET02878
Not Available
Acalabrutinib M2 Metabolite
Details
Acalabrutinib M5 Metabolite (ACP-5530)
DBMET02885
Not Available
Acalabrutinib M7 Metabolite (ACP-5531)
Details
Acalabrutinib M7 Metabolite (ACP-5531)
DBMET02886
Not Available
Acalabrutinib M10 Metabolite (ACP-5461)
Details
Aceclofenac
DB06736
Not Available
Diclofenac
Details
Aceclofenac
DB06736
Cytochrome P450 2C9
5-OH-aceclofenac
Details
Aceclofenac
DB06736
Cytochrome P450 2C9
4'-Hydroxyaceclofenac
Details
Aceclofenac
DB06736
Prostaglandin G/H synthase 1
5-Hydroxyaceclofenac
Details
Aceclofenac
DB06736
Cytochrome P450 2C9
4'-OH-aceclofenac
Details
Acemetacin
DB13783
Not Available
Indomethacin
Details
Acemetacin
DB13783
Not Available
des-4-chlorobenzoyl-indomethacin
Details
Acemetacin
DB13783
Not Available
O-desmethyl-des-4-chlorobenzoyl
Details
Acemetacin
DB13783
Not Available
O-demethylated acemetacin
Details
Acenocoumarol
DB01418
Cytochrome P450 2C9
/
Cytochrome P450 1A2
/
Cytochrome P450 2C19
6-Hydroxy-R-acenocoumarol
Details
Acenocoumarol
DB01418
Cytochrome P450 2C9
/
Cytochrome P450 2C19
8-Hydroxy-R-acenocoumarol
Details
Acenocoumarol
DB01418
Cytochrome P450 2C9
/
Cytochrome P450 2C19
7-Hydroxy-R-acenocoumarol
Details
acetaldehyde
DBMET00328
Aldehyde dehydrogenase, mitochondrial
Acetate
Details
Acetaminophen
DB00316
UDP-glucuronosyltransferase 1-9
/
UDP-glucuronosyltransferase 1-6
/
UDP-glucuronosyltransferase 1-1
/
UDP-glucuronosyltransferase 2B15
/
UDP-glucuronosyltransferase 1-10
Acetaminophen glucuronide
Details
Acetaminophen
DB00316
Cytochrome P450 2E1
/
Cytochrome P450 3A4
/
Cytochrome P450 1A2
/
Cytochrome P450 2D6
/
Cytochrome P450 2A6
NAPQI
Details
Acetaminophen
DB00316
Sulfotransferase 1A1
/
Sulfotransferase 1A3/1A4
/
Bile salt sulfotransferase
Acetaminophen sulfate
Details
Acetate
DBMET01513
Not Available
Carbon dioxide
Details
Acetate
DBMET01513
Not Available
Water
Details
Acetohexamide
DB00414
Not Available
Hydroxyhexamide
Details
Acetyl Coenzyme A
DBMET03175
Not Available
Propionyl Coenzyme A
Details
Acetylbenzocaine
DBMET03291
Not Available
4-Acetaminobenzoic acid
Details
Acetylcysteine
DB06151
Aminoacylase-1
Cysteine
Details
Acetylsalicylic acid
DB00945
Carboxylesterase
Salicylic acid
Details
Acetylsalicylic acid
DB00945
UDP-glucuronosyltransferase 1-6
Phenolic glucuronide
/
Salicylic acid acyl glucuronide
Details
Acetylsalicylic acid
DB00945
Cytochrome P450 2C9
Gentisic acid
Details
Acetylsalicylic acid
DB00945
Medium-chain fatty-acid--CoA ligase
Salicyluric acid
Details
Acrolein
DBMET01126
Aldehyde dehydrogenase, dimeric NADP-preferring
/
Retinal dehydrogenase 1
Acrylic Acid
Details
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