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Identification
NameCetirizine
Accession NumberDB00341  (APRD00630)
TypeSmall Molecule
GroupsApproved
Description

A potent second-generation histamine H1 antagonist that is effective in the treatment of allergic rhinitis, chronic urticaria, and pollen-induced asthma. Unlike many traditional antihistamines, it does not cause drowsiness or anticholinergic side effects. [PubChem]

Structure
Thumb
Synonyms
Cetirizin
Cetirizina
Cetirizinum
External Identifiers Not Available
Approved Prescription Products
NameDosageStrengthRouteLabellerMarketing StartMarketing End
Cetirizinetablet20 mgoralPro Doc LimiteeNot applicableNot applicableCanada
Dom-cetirizinetablet20 mgoralDominion PharmacalNot applicableNot applicableCanada
Ipg-cetirizinetablet20 mgoralMarcan Pharmaceuticals IncNot applicableNot applicableCanada
Mar-cetirizinetablet20 mgoralMarcan Pharmaceuticals Inc2015-10-13Not applicableCanada
Novo-cetirizinetablet20 mgoralNovopharm LimitedNot applicableNot applicableCanada
PMS-cetirizinetablet20 mgoralPharmascience Inc2008-10-14Not applicableCanada
Priva-cetirizinetablet20 mgoralPharmapar Inc2015-10-19Not applicableCanada
Reactine 20mg Tablettablet20 mgoralMcneil Consumer Healthcare Division Of Johnson & Johnson Inc2002-01-14Not applicableCanada
Rhinaris Relieftablet20 mgoralPendopharm Division Of De Pharmascience IncNot applicableNot applicableCanada
Zyrtectablet, film coated10 mg/1oralbryant ranch prepack2008-10-01Not applicableUs
Approved Generic Prescription Products
NameDosageStrengthRouteLabellerMarketing StartMarketing End
Apo-cetirizinetablet20 mgoralApotex Inc2016-04-22Not applicableCanada
Cetirizine Hydrochloridetablet5 mg/1oralbryant ranch prepack2009-10-01Not applicableUs
Cetirizine Hydrochloridesyrup1 mg/mLoralQualitest Pharmaceuticals2009-09-25Not applicableUs
Cetirizine Hydrochloridesolution5 mg/5mLoralAmneal Pharmaceuticals2009-10-07Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralBreckenridge Pharmaceutical, Inc.2013-12-03Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralProficient Rx LP2013-12-03Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralTaro Pharmaceuticals U.S.A., Inc.2014-05-01Not applicableUs
Cetirizine Hydrochloridesyrup1 mg/mLoralTeva Pharmaceuticals USA Inc2008-05-302015-11-30Us
Cetirizine Hydrochloridesyrup1 mg/mLoralCaraco Pharmaceutical Laboratories, Ltd.2009-11-16Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralREMEDYREPACK INC.2010-12-01Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralPreferred Pharmaceuticals, Inc.2015-04-20Not applicableUs
Cetirizine Hydrochloridesyrup1 mg/mLoralDr. Reddy's Laboratories Limited2009-08-202016-03-03Us
Cetirizine Hydrochloridetablet5 mg/1oralREMEDYREPACK INC.2010-11-23Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralPreferred Pharmaceuticals, Inc.2014-04-02Not applicableUs
Cetirizine Hydrochloridesyrup5 mg/5mLoralSilarx Pharmaceuitcals, Inc2012-05-11Not applicableUs
Cetirizine Hydrochloridesyrup1 mg/mLoralPerrigo New York Inc2008-07-24Not applicableUs
Cetirizine Hydrochloridesyrup1 mg/mLoralPreferred Pharmaceuticals, Inc2010-12-20Not applicableUs
Cetirizine Hydrochloridesyrup5 mg/5mLoralSilarx Pharmaceuitcals, Inc2012-05-11Not applicableUs
Cetirizine Hydrochloridesyrup1 mg/mLoralWockhardt Llc.2009-08-28Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralHeritage Pharmaceuticals Inc.2009-04-07Not applicableUs
Cetirizine Hydrochloridesyrup1 mg/mLoralCarilion Materials Management2008-07-24Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralREMEDYREPACK INC.2013-06-03Not applicableUs
Approved Over the Counter Products
NameDosageStrengthRouteLabellerMarketing StartMarketing End
24 Hour Allergyliquid5 mg/5mLoralMeijer Distribution Inc2008-04-16Not applicableUs
24 Hour Allergytablet10 mg/1oralMeijer Distribution Inc1997-07-07Not applicableUs
24 Hour Allergycapsule10 mg/1oralWalgreens2013-03-01Not applicableUs
24 Hour Allergy Lil Drug Store Productstablet10 mg/1oralLil' Drug Store Products, Inc2014-11-01Not applicableUs
24-hour All Day Allergytablet10 mg/1oralMc Kesson2012-04-27Not applicableUs
7 Select All Day Allergytablet10 mg/1oral7 Eleven2014-04-29Not applicableUs
7 Select Childrens Allergy Reliefsolution5 mg/5mLoral7 Eleven2014-08-05Not applicableUs
All Day Allergytablet10 mg/1oralHy Vee Inc1997-08-28Not applicableUs
All Day Allergycapsule10 mg/1oralThe Kroger Co.2013-12-30Not applicableUs
All Day Allergycapsule10 mg/1oralFreds Inc2013-08-01Not applicableUs
All Day Allergycapsule10 mg/1oralHy Vee2013-09-30Not applicableUs
All Day Allergycapsule10 mg/1oralP and L Development of New York Corporation2013-02-14Not applicableUs
All Day Allergyliquid5 mg/5mLoralKroger Company2008-05-08Not applicableUs
All Day Allergycapsule10 mg/1oralCardinal Health (Leader) 372052013-03-03Not applicableUs
All Day Allergytablet10 mg/1oralMedicine Shoppe International Inc2008-01-16Not applicableUs
All Day Allergycapsule10 mg/1oralH E B2013-10-09Not applicableUs
All Day Allergytablet10 mg/1oralHannaford Brothers Company2008-01-16Not applicableUs
All Day Allergysolution5 mg/5mLoralAmerisource Bergen2011-05-20Not applicableUs
All Day Allergytablet10 mg/1oralLIVE BETTER (The Great Atlantic & Pacific Tea Company)2013-06-07Not applicableUs
All Day Allergyliquid5 mg/5mLoralKroger Company2011-08-05Not applicableUs
All Day Allergytablet10 mg/1oralMc Kesson (Health Mart)2012-02-08Not applicableUs
All Day Allergycapsule10 mg/1oralTOP CARE (Topco Associates LLC)2013-04-30Not applicableUs
All Day Allergytablet10 mg/1oralLIVE BETTER (The Great Atlantic & Pacific Tea Company)2011-11-23Not applicableUs
All Day Allergytablet10 mg/1oralKroger Company2008-01-08Not applicableUs
All Day Allergycapsule10 mg/1oralCare One (American Sales Company)2013-12-30Not applicableUs
All Day Allergy 24 Hourtablet10 mg/1oralMc Kesson (Health Mart)2012-01-01Not applicableUs
All Day Allergy Antihistaminetablet10 mg/1oralP and L Development of New York Corporation2012-12-05Not applicableUs
All Day Allergy Antihistaminetablet10 mg/1oralCare One (American Sales Company)2010-09-07Not applicableUs
All Day Allergy Antihistaminecapsule10 mg/1oralChain Drug Consortium, LLC2013-06-01Not applicableUs
All Day Allergy Relieftablet10 mg/1oralASSURED / DOLLAR TREE (Greenbrier International, Inc.)2010-07-06Not applicableUs
All Day Allergy Reliefcapsule10 mg/1oralQUALITY CHOICE (Chain Drug Marketing Association)2013-03-03Not applicableUs
All Day Allergy Relieftablet10 mg/1oralAssured (Greenbrier International, Inc.)2012-10-19Not applicableUs
All Day Allergy Relieftablet10 mg/1oralH E B2014-02-08Not applicableUs
All Day Allergy Relieftablet10 mg/1oralP And L Development Of New York Corporation (Ready In Case)2010-09-01Not applicableUs
All Day Allergy Relieftablet10 mg/1oralP And L Development Of New York Corporation (Ready In Case)2014-07-31Not applicableUs
All Day Allergy Relief 24 Hourtablet10 mg/1oralOUR FAMILY (Nash Finch Company)2013-03-15Not applicableUs
All Day Allergy Relief 24 Hourtablet10 mg/1oralMc Kesson (Sunmark)2013-03-15Not applicableUs
All Day Allergy Relief 24 Hourtablet10 mg/1oralDolgencorp, Inc. (DOLLAR GENERAL & REXALL)2012-10-19Not applicableUs
Aller-relieftablet10 mgoralApotex Inc1999-08-17Not applicableCanada
Aller-relief 10mgtablet10 mgoralPharmascience Inc2011-04-07Not applicableCanada
Allergy Childrens 24 Hourliquid5 mg/5mLoralMeijer Distribution Inc2011-01-14Not applicableUs
Allergy Relieftablet10 mg/1oralAllegiant Health2014-12-16Not applicableUs
Allergy Reliefcapsule, liquid filled10 mg/1oralTarget Corporation2014-09-30Not applicableUs
Allergy Relieftablet10 mg/1oralShopko Stores Operating Co., LLC2013-07-08Not applicableUs
Allergy Reliefcapsule, liquid filled10 mg/1oralPublix Supermarkets, Inc.2015-01-31Not applicableUs
Allergy Reliefsolution5 mg/5mLoralCVS Pharmacy2015-12-03Not applicableUs
Allergy Reliefcapsule10 mg/1oralHarmon Stores2015-02-28Not applicableUs
Allergy Relieftablet10 mgoralApotex Inc1999-08-17Not applicableCanada
Allergy Relieftablet5 mgoralPharmascience IncNot applicableNot applicableCanada
Allergy Relieftablet10 mg/1oralWestern Family Foods Inc2008-01-25Not applicableUs
Allergy Reliefcapsule10 mg/1oralWestern Family Foods, Inc.2013-12-30Not applicableUs
Allergy Relieftablet, film coated5 mg/1oralWal Mart Stores Inc2011-02-08Not applicableUs
Allergy Reliefsolution1 mg/mLoralH E B2011-05-20Not applicableUs
Allergy Relieftablet10 mg/1oralRite Aid Corporation2008-01-16Not applicableUs
Allergy Relieftablet10 mg/1oralPublix Super Markets Inc2009-01-21Not applicableUs
Allergy Relief 24 Hourtablet10 mg/1oralSafeway2008-02-15Not applicableUs
Allergy Relief All Daytablet10 mg/1oralDolgencorp, Inc. (DOLLAR GENERAL & REXALL)2013-05-17Not applicableUs
Allergy Relief All Daytablet10 mg/1oralDolgencorp, Inc. (DOLLAR GENERAL & REXALL)2013-05-17Not applicableUs
Allergy Relief Childrenssolution5 mg/5mLoralCVS Pharmacy2015-09-11Not applicableUs
Allergy Relief Childrensliquid5 mg/5mLoralWestern Family Foods Inc2010-10-25Not applicableUs
Allergy Relief Childrensliquid5 mg/5mLoralCVS Pharmacy2010-08-18Not applicableUs
Allergy Relief Childrens Indoor/outdoortablet, chewable10 mg/1oralWOONSOCKET PRESCRIPTION CENTER,INCORPORATED2008-10-31Not applicableUs
Allergy Relief Indoor and Outdoor Allergiestablet, film coated10 mg/1oralCVS Pharmacy2009-01-14Not applicableUs
Allergy Relief Liquid Gelscapsule10 mgoralApotex IncNot applicableNot applicableCanada
Allerofftablet10 mg/1oralCorporacion Infarmasa2010-01-01Not applicableUs
Allerofftablet10 mg/1oralCorporacion Infarmasa2010-01-01Not applicableUs
Alleroffsyrup1 mg/1oralCorporacion Infarmasa2010-01-15Not applicableUs
Apo-cetirizinetablet5 mgoralApotex Inc2000-03-22Not applicableCanada
Apo-cetirizinetablet10 mgoralApotex Inc1998-10-21Not applicableCanada
Aptrizine 24-hour All Day Allergytablet10 mg/1oralA P J Laboratories Limited2013-02-21Not applicableUs
Being Well Allergytablet10 mg/1oralSave A Lot Food Stores Ltd2008-05-19Not applicableUs
Berkley and Jensen Allergy Relieftablet10 mg/1oralBJWC2013-11-26Not applicableUs
Berkley and Jensen Cetirizine Hydrochloridetablet10 mg/1oralBJWC2009-04-27Not applicableUs
Berkley and Jensen Childrens Cetirizine Hydrochlorideliquid5 mg/5mLoralBJWC2011-05-13Not applicableUs
Best Choice Childrens Cetirizinesolution5 mg/5mLoralValu Merchandisers Company2011-09-08Not applicableUs
Best Choice Childrens Cetirizinesolution5 mg/5mLoralValu Merchandisers Company2008-04-22Not applicableUs
Careone All Day Allergysolution5 mg/5mLoralAmerican Sales Company2015-12-21Not applicableUs
Careone All Day Allergytablet10 mg/1oralAmerican Sales Company2008-01-23Not applicableUs
Careone All Day Allergy Childrensliquid5 mg/5mLoralAmerican Sales Company2008-04-18Not applicableUs
Careone Childrens All Day Allergyliquid5 mg/5mLoralAmerican Sales Company2013-12-27Not applicableUs
Careone Childrens Allergy Reliefsolution5 mg/5mLoralAmerican Sales Company2016-04-06Not applicableUs
Cetirizinetablet10 mg/1oralbryant ranch prepack2008-01-16Not applicableUs
Cetirizineliquid5 mg/5mLoralRebel Distributors Corp2008-06-17Not applicableUs
Cetirizinetablet10 mg/1oralLife Line Home Care Services, Inc.2012-02-03Not applicableUs
Cetirizinetablet10 mg/1oralNcs Health Care Of Ky, Inc Dba Vangard Labs2007-12-27Not applicableUs
Cetirizinetablet10 mgoralApotex IncNot applicableNot applicableCanada
Cetirizinetablet5 mgoralApotex IncNot applicableNot applicableCanada
Cetirizine HClcapsule10 mg/1oralSMART SENSE (Kmart)2013-05-01Not applicableUs
Cetirizine HCl 10 Mg All Day Allergy Relieftablet10 mg/1oralFreds Inc2013-03-01Not applicableUs
Cetirizine Hydrochloridetablet, chewable5 mg/1oralJubilant Cadista Pharmaceuticals Inc.2015-02-19Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralKinray2011-12-07Not applicableUs
Cetirizine Hydrochloridesolution5 mg/5mLoralAmneal Pharmaceuticals of New York, LLC2009-10-07Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralTorrent Pharmaceuticals Limited2010-04-15Not applicableUs
Cetirizine Hydrochloridetablet, chewable5 mg/1oralSandoz Inc2008-02-14Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralCardinal Health2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet, film coated5 mg/1oralCaraco Pharmaceutical Laboratories, Ltd.2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet5 mg/1oralUnichem Pharmaceuticals (USA), Inc.2010-11-30Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralLake Erie Medical DBA Quality Care Products LLC2009-10-01Not applicableUs
Cetirizine Hydrochlorideliquid5 mg/5mLoralPerrigo New York Inc2008-04-15Not applicableUs
Cetirizine Hydrochloridesolution5 mg/5mLoralBlacksmith Brands Inc.2008-04-22Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralArmy & Air Force Exchange Service2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralClinical Solutions Wholesale2009-10-01Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralAmneal Pharmaceuticals2010-01-21Not applicableUs
Cetirizine Hydrochloridetablet, chewable10 mg/1oralChain Drug Consortium, LLC2013-09-10Not applicableUs
Cetirizine Hydrochloridetablet5 mg/1oralPack Pharmaceuticals LLC2009-10-01Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralDispensing Solutions, Inc.2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet, film coated5 mg/1oralMylan Pharmaceuticals Inc.2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet, chewable5 mg/1oralSun Pharma Global FZE2011-09-09Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralMc Kesson2011-08-01Not applicableUs
Cetirizine Hydrochloridesolution5 mg/5mLoralSilarx Pharmaceuticals, Inc2011-05-06Not applicableUs
Cetirizine Hydrochloridetablet5 mg/1oralTorrent Pharmaceuticals Limited2010-04-15Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralSandoz Inc2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralTaro Pharmaceuticals U.S.A., Inc.2009-07-22Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralCardinal Health2012-03-30Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralAmerican Health Packaging2015-07-20Not applicableUs
Cetirizine Hydrochloridesolution5 mg/5mLoralAmneal Pharmaceuticals of New York, LLC2009-10-07Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralPreferred Pharmaceuticals, Inc.2012-10-22Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralMed Vantx, Inc.2009-10-19Not applicableUs
Cetirizine Hydrochloridetablet5 mg/1oralKAISER FOUNDATION HOSPITALS2013-12-13Not applicableUs
Cetirizine Hydrochloridesolution5 mg/5mLoralSilarx Pharmaceuticals, Inc2011-05-02Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralApotheca Inc.2010-01-01Not applicableUs
Cetirizine Hydrochloridetablet5 mg/1oralSandoz Inc2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralAidarex Pharmaceuticals LLC2009-10-01Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralTaro Pharmaceuticals U.S.A., Inc.2008-04-22Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralDr.Reddy's Laboratories Limited2008-01-15Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralFamily Dollar Services, Inc.2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralApotex Corp.2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralProficient Rx LP2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralPreferred Pharmaceuticals, Inc.2009-10-01Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralKAISER FOUNDATION HOSPITALS2013-12-13Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralMedline Industries, Inc.2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralRebel Distributors Corp2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralOhm Laboratories Inc.2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralDr.Reddy's Laboratories Limited2008-01-15Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralIpca Laboratories Limited2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralUnique Pharmaceutical Laboratories2009-10-01Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralTri Marc Labs2010-06-25Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralRebel Distributors Corp2007-12-27Not applicableUs
Cetirizine Hydrochloridesyrup5 mg/5mLoralPharmaceutical Associates, Inc.2009-09-15Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralMajor Pharmaceuticals2010-06-25Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralUnichem Pharmaceuticals (USA), Inc.2010-11-30Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralTopco Associates LLC2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralREMEDYREPACK INC.2015-03-26Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralMylan Institutional Inc.2012-03-30Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralPhysicians Total Care, Inc.2008-05-01Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralValu Merchandisers Company2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet5 mg/1oralUnique Pharmaceutical Laboratories2009-10-01Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralRugby Laboratories, Inc.2012-03-23Not applicableUs
Cetirizine Hydrochloridetablet5 mg/1oralUnichem Pharmaceuticals (USA), Inc.2010-11-30Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralSunmark2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralDIRECT RX2014-01-01Not applicableUs
Cetirizine Hydrochloridetablet, chewable10 mg/1oralMajor Pharmaceuticals2008-02-14Not applicableUs
Cetirizine Hydrochloridetablet, film coated5 mg/1oralPhysicians Total Care, Inc.2008-01-29Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralPublix Super Markets Inc2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralCVS Pharmacy2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralWin Co Foods, Llc2012-01-20Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralBlenheim Pharmacal, Inc.2009-10-01Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralRugby Laboratories2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet, chewable10 mg/1oralJubilant Cadista Pharmaceuticals Inc.2015-02-19Not applicableUs
Cetirizine Hydrochloridetablet5 mg/1oralAmneal Pharmaceuticals2010-01-21Not applicableUs
Cetirizine Hydrochloridetablet, film coated5 mg/1oralAvera Mc Kennan Hospital2015-05-29Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralRising Pharmaceuticals, Inc.2009-10-01Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralSelect Brand2007-12-27Not applicableUs
Cetirizine Hydrochlorideliquid5 mg/5mLoralTris Pharma Inc2012-11-21Not applicableUs
Cetirizine Hydrochloridetablet, chewable10 mg/1oralSandoz Inc2008-02-14Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralLake Erie Medical & Surgical Supply DBA Quality Care Products LLC2012-02-23Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralPerrigo New York Inc2007-12-27Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralTaro Pharmaceuticals U.S.A., Inc.2011-05-20Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralCaraco Pharmaceutical Laboratories, Ltd.2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralUnichem Pharmaceuticals (USA), Inc.2010-11-30Not applicableUs
Cetirizine Hydrochloridesolution1 mg/mLoralTaro Pharmaceutical Industries, Ltd.2011-05-20Not applicableUs
Cetirizine Hydrochloridetablet5 mg/1oralREMEDYREPACK INC.2015-03-30Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralChain Drug Consortium, LLC2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralMajor Pharmaceuticals2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralNorthstar Rx LLC2009-10-19Not applicableUs
Cetirizine Hydrochloridetablet, film coated10 mg/1oralMylan Pharmaceuticals Inc.2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralShopko Stores Operating Co., LLC2007-12-27Not applicableUs
Cetirizine Hydrochloridetablet, chewable10 mg/1oralSun Pharma Global FZE2011-09-09Not applicableUs
Cetirizine Hydrochloridetablet10 mg/1oralPhysicians Total Care, Inc.2008-01-02Not applicableUs
Cetirizine Hydrochloride (allergy)tablet10 mg/1oralAurohealth LLC2015-08-05Not applicableUs
Cetirizine Hydrochloride (allergy)tablet5 mg/1oralAurohealth LLC2015-08-05Not applicableUs
Cetirizine Hydrochloride (hives Relief)tablet10 mg/1oralAurohealth LLC2015-08-05Not applicableUs
Cetirizine Hydrochloride (hives Relief)tablet5 mg/1oralAurohealth LLC2015-08-05Not applicableUs
Cetirizine Hydrochloride Hivessolution1 mg/mLoralCaraco Pharmaceutical Laboratories, Ltd2011-12-01Not applicableUs
Cetirizine Hydrochloride Hives Relieftablet10 mg/1oralAmneal Pharmaceuticals2010-01-21Not applicableUs
Cetirizine Hydrochloride Hives Relieftablet5 mg/1oralAmneal Pharmaceuticals2010-01-21Not applicableUs
Cetirizine Hydroloride Allergysolution1 mg/mLoralCaraco Pharmaceutical Laboratories, Ltd2011-12-01Not applicableUs
Cetrizine Hydrochloridesolution1 mg/mLoralMajor Pharmaceuticals2014-02-24Not applicableUs
Childrens 24 Hour Allergysolution5 mg/5mLoralMeijer Distribution Inc2011-05-20Not applicableUs
Childrens 24 Hour Allergysolution5 mg/5mLoralMeijer Distribution Inc2015-12-02Not applicableUs
Childrens 24 Hour Allergysolution5 mg/5mLoralMeijer Distribution Inc2011-09-08Not applicableUs
Childrens All Day Allergysolution5 mg/5mLoralMc Kesson2011-05-20Not applicableUs
Childrens All Day Allergyliquid5 mg/5mLoralMajor Pharmaceuticals2010-07-26Not applicableUs
Childrens All Day Allergysolution5 mg/5mLoralKroger Company2011-05-20Not applicableUs
Childrens All Day Allergysolution5 mg/5mLoralHy Vee Inc2014-02-17Not applicableUs
Childrens All Day Allergysolution5 mg/5mLoralHy Vee Inc2016-03-20Not applicableUs
Childrens All Day Allergysolution5 mg/5mLoralKroger Company2011-09-08Not applicableUs
Childrens All Day Allergysolution5 mg/5mLoralKroger Company2016-03-10Not applicableUs
Childrens All Day Allergysolution5 mg/5mLoralKroger Company2015-10-23Not applicableUs
Childrens All Day Allergysolution5 mg/5mLoralMc Kesson2008-04-22Not applicableUs
Childrens All Day Allergy (leader)liquid5 mg/5mLoralCardinal Health2009-09-29Not applicableUs
Childrens All Day Allergy Reliefsolution1 mg/mLoralTarget Corporation2008-04-22Not applicableUs
Childrens Allergyliquid5 mg/5mLoralWalgreen Company2008-04-25Not applicableUs
Childrens Allergyliquid5 mg/5mLoralH E B2010-11-01Not applicableUs
Childrens Allergysolution1 mg/mLoralPublix Super Markets Inc2011-05-20Not applicableUs
Childrens Allergyliquid5 mg/5mLoralQUALITY CHOICE (Chain Drug Marketing Association)2014-12-31Not applicableUs
Childrens Allergysolution5 mg/5mLoralPublix Super Markets Inc2015-12-21Not applicableUs
Childrens Allergyliquid5 mg/5mLoralPublix Super Markets Inc2009-01-15Not applicableUs
Childrens Allergy Reliefsolution5 mg/5mLoralPreferred Plus (Kinray)2011-09-08Not applicableUs
Childrens Allergy Reliefsolution5 mg/5mLoralShopko Stores Operating Co., LLC2016-03-22Not applicableUs
Childrens Allergy Reliefliquid5 mg/5mLoralTarget Corporation2015-01-31Not applicableUs
Childrens Allergy Reliefsolution1 mg/mLoralAurohealth LLC2010-02-02Not applicableUs
Childrens Allergy Reliefsolution5 mg/5mLoralCVS Pharmacy2015-09-22Not applicableUs
Childrens Allergy Reliefsolution1 mg/mLoralC.D.M.A., Inc.2014-11-20Not applicableUs
Childrens Allergy Reliefsolution5 mg/5mLoralRite Aid Corporation2016-03-23Not applicableUs
Childrens Allergy Reliefsolution5 mg/5mLoralWal Mart Stores Inc2011-05-20Not applicableUs
Childrens Allergy Reliefsolution5 mg/5mLoralWal Mart Stores Inc2008-04-22Not applicableUs
Childrens Allergy Reliefliquid5 mg/5mLoralCVS Pharmacy2009-07-15Not applicableUs
Childrens Allergy Reliefliquid5 mg/5mLoralSafeway2014-05-15Not applicableUs
Childrens Allergy Relieftablet, chewable10 mg/1oralL.N.K. International, Inc.2008-10-31Not applicableUs
Childrens Allergy Reliefliquid5 mg/5mLoralShopko Stores Operating Co., LLC2013-07-08Not applicableUs
Childrens Allergy Reliefliquid5 mg/5mLoralRite Aid Corporation2008-04-17Not applicableUs
Childrens Allergy Relieftablet, chewable10 mg/1oralRite Aid2008-10-31Not applicableUs
Childrens Allergy Relieftablet, chewable10 mg/1oralWal Mart Stores Inc2008-10-31Not applicableUs
Childrens Allergy Reliefsolution1 mg/mLoralFRED'S, INC.2015-01-31Not applicableUs
Childrens Cetirizine Hydrochloridesolution1 mg/mLoralHealth Mart2011-05-20Not applicableUs
Childrens Cetirizine Hydrochloridesolution5 mg/5mLoralChain Drug Consortium, LLC (Premier Value)2008-04-22Not applicableUs
Childrens Cetirizine Hydrochloridesolution5 mg/5mLoralPrecision Dose Inc.2009-03-17Not applicableUs
Childrens Cetirizine Hydrochloride Allergysolution1 mg/mLoralAurobindo Pharma Limited2010-02-02Not applicableUs
Childrens Cetirizine Hydrochloride Allergysolution1 mg/mLoralAurohealth LLC2015-06-24Not applicableUs
Childrens Cetirizine Hydrochloride Hives Reliefsolution1 mg/mLoralAurobindo Pharma Limited2010-02-02Not applicableUs
Childrens Cetirizine Hydrochloride Hives Reliefsolution1 mg/mLoralAurohealth LLC2015-06-24Not applicableUs
Childrens Cetirizine Hydrochloride Sugar Free Grapesolution1 mg/mLoralTaro Pharmaceuticals U.S.A., Inc.2011-09-08Not applicableUs
Childrens Cetirizine Hydrochloride Sugar Free Grapesolution1 mg/mLoralPreferred Pharmaceuticals Inc.2016-02-15Not applicableUs
Childrens Cetirzinesolution5 mg/5mLoralChain Drug Consortium2011-05-20Not applicableUs
Childrens Wal Zyrsolution5 mg/5mLoralWalgreen Company2015-09-22Not applicableUs
Childrens Wal Zyr 24 Hour Allergyliquid5 mg/5mLoralWalgreen Company2010-10-15Not applicableUs
Childrens Wal-zyrtablet, chewable10 mg/1oralWALGREEN CO.2008-10-31Not applicableUs
Childrens Zyrtecsyrup5 mg/5mLoralJohnson & Johnson Consumer Inc., Mc Neil Consumer Healthcare Division2009-06-01Not applicableUs
Childrens Zyrtec Allergysyrup5 mg/5mLoralJohnson & Johnson Consumer Inc., Mc Neil Consumer Healthcare Division2009-01-20Not applicableUs
Childrens Zyrtec Allergytablet, orally disintegrating10 mg/1oralJohnson & Johnson Consumer Inc., Mc Neil Consumer Healthcare Division2014-01-20Not applicableUs
Cvs Childrens Allergy Reliefsolution5 mg/5mLoralCVS Pharmacy2011-05-20Not applicableUs
Cvs Pharmacy Childrens Allergy Reliefsolution5 mg/5mLoralCVS Pharmacy2011-09-08Not applicableUs
Dg Health All Day Allergytablet10 mg/1oralDolgencorp Inc2010-01-08Not applicableUs
Equaline All Day Allergysolution5 mg/5mLoralSupervalu Inc2011-07-26Not applicableUs
Equaline All Day Allergytablet10 mg/1oralSupervalu Inc2008-01-23Not applicableUs
Equaline Childrens All Day Allergysolution5 mg/5mLoralSupervalu Inc2015-11-17Not applicableUs
Equaline Childrens All Day Allergysolution5 mg/5mLoralSupervalu Inc2008-05-20Not applicableUs
Equate Allergy Relieftablet10 mg/1oralWal Mart Stores Inc2008-01-09Not applicableUs
Equate Allergy Relieftablet, film coated10 mg/1oralWal Mart Stores, Inc.2013-07-25Not applicableUs
Equate Childrens Allergy Reliefsolution5 mg/5mLoralWal Mart Stores Inc2011-09-08Not applicableUs
Exchange Select Allergy Relieftablet10 mg/1oralArmy & Air Force Exchange Service2014-02-06Not applicableUs
Extra Strength Allergy Relieftablet10 mgoralPharmascience Inc2009-08-20Not applicableCanada
Extra Strength Allergy Relieftablet10 mgoralPharmel IncNot applicableNot applicableCanada
Extra Strength Allergy Relieftablet10 mgoralVita Health Products IncNot applicableNot applicableCanada
Family Wellness Childrens All Day Allergyliquid5 mg/5mLoralFamily Dollar Services Inc2012-08-02Not applicableUs
Family Wellness Childrens All Day Allergysolution5 mg/5mLoralFamily Dollar Services Inc2015-10-31Not applicableUs
Fulton Street Market Cetirizine Hydrochloridetablet10 mg/1oralAccess Business Group LLC2009-07-01Not applicableUs
Good Neighbor Pharmacy All Day Allergytablet10 mg/1oralAmerisource Bergen2008-01-15Not applicableUs
Good Neighbor Pharmacy All Day Allergyliquid5 mg/5mLoralAmerisource Bergen2008-04-22Not applicableUs
Good Neighbor Pharmacy Allergy Childrens All Dayliquid5 mg/5mLoralAmerisource Bergen2010-10-29Not applicableUs
Good Neighbor Pharmacy Childrens All Day Allergysolution5 mg/5mLoralAmerisource Bergen2015-11-10Not applicableUs
Good Sense All Day Allergytablet10 mg/1oralL Perrigo Company2008-01-16Not applicableUs
Good Sense Childrens All Day Allergyliquid5 mg/5mLoralL Perrigo Company1992-06-15Not applicableUs
Good Sense Childrens All Day Allergysolution5 mg/5mLoralL. Perrigo Company2014-01-03Not applicableUs
Good Sense Childrens All Day Allergysolution5 mg/5mLoralL. Perrigo Company2016-01-11Not applicableUs
Good Sense Childrens All Day Allergyliquid5 mg/5mLoralL Perrigo Company2008-04-18Not applicableUs
H-E-B Allergy Reliefsolution5 mg/5mLoralH E B2008-04-22Not applicableUs
Harmon Face Values Allergy Relieftablet10 mg/1oralHarmon Stores Inc.2011-12-18Not applicableUs
Harris Teeter All Day Allergytablet, film coated10 mg/1oralHarris Teeter, LLC2015-06-24Not applicableUs
Harris Teeter All Day Allergy Childrensliquid5 mg/5mLoralHarris Teeter, LLC2015-06-24Not applicableUs
Harris Teeter Childrens All Day Allergysolution5 mg/5mLoralHarris Teeter, LLC2016-01-08Not applicableUs
Health Mart Allergy Complete Childrensliquid5 mg/5mLoralMc Kesson2012-01-11Not applicableUs
Health Mart Childrens All Day Allergysolution5 mg/5mLoralMcKesson2016-02-26Not applicableUs
Health Mart Pharmacy Childrens Cetirizine Hydrochloridesolution1 mg/mLoralHealth Mart2008-04-22Not applicableUs
Healthmart Childrens Cetirizinesolution5 mg/5mLoralMc Kesson2011-09-08Not applicableUs
Healthy Accents Cetirizine Hydrochloridetablet10 mg/1oralDZA Brands LLC2008-01-15Not applicableUs
Healthy Accents Childrens Allergysolution5 mg/5mLoralDZA Brands LLC2015-12-09Not applicableUs
Healthy Accents Childrens Allergyliquid5 mg/5mLoralDZA Brands LLC2008-04-28Not applicableUs
Heb Allergy Reliefsolution5 mg/5mLoralH E B2011-09-08Not applicableUs
Indoor/outdoor Allergy Relief Softgelscapsule10 mg/1oralCVS Pharmacy2013-03-01Not applicableUs
Ipg-cetirizinetablet10 mgoralMarcan Pharmaceuticals IncNot applicableNot applicableCanada
Ipg-cetirizinetablet5 mgoralMarcan Pharmaceuticals IncNot applicableNot applicableCanada
Jamp-cetirizinetablet10 mgoralJamp Pharma Corporation2016-04-05Not applicableCanada
Jamp-cetirizinetablet5 mgoralJamp Pharma CorporationNot applicableNot applicableCanada
Kirkland Signature Aller Tec Allergytablet10 mg/1oralCostco Wholesale Company2008-03-25Not applicableUs
Kirklands Childrens Aller Tecliquid5 mg/5mLoralCostco Wholesale Company2009-08-14Not applicableUs
Leader All Day Allergytablet10 mg/1oralCardinal Health2008-01-16Not applicableUs
Leader All Day Allergytablet10 mg/1oralCardinal Health2007-12-27Not applicableUs
Leader All Day Allergytablet10 mg/1oralCardinal Health2014-06-04Not applicableUs
Leader Childrens All Day Allergysolution5 mg/5mLoralCardinal Health2016-02-03Not applicableUs
Leader Childrens All Day Allergyliquid5 mg/5mLoralCardinal Health2010-11-09Not applicableUs
Leader Childrens Allergy Reliefsolution1 mg/mLoralCardinal Health2011-05-20Not applicableUs
Mar-cetirizinetablet10 mgoralMarcan Pharmaceuticals Inc2015-10-13Not applicableCanada
Mar-cetirizinetablet5 mgoralMarcan Pharmaceuticals IncNot applicableNot applicableCanada
Members Mark Cetirizinetablet, film coated10 mg/1oralSam's West Inc2008-03-24Not applicableUs
Our Family Childrens Cetirizinesolution5 mg/5mLoralNash Finch Company2011-05-20Not applicableUs
Pedia Care Childrens 24 Hour Allergysolution5 mg/5mLoralMedtech Products Inc.2011-09-08Not applicableUs
Preferred Plus All Day Allergytablet10 mg/1oralKinray2014-09-22Not applicableUs
Premier Value Childrens Cetirizinesolution5 mg/5mLoralChain Drug Constortium2011-09-08Not applicableUs
Quality Choice Cetirizine Hydrochloridetablet10 mg/1oralChain Drug Marketing Association Inc.2007-12-27Not applicableUs
Quality Choice Childrens Allergy Reliefsolution1 mg/mLoralChain Drug Marketing Association Inc.2011-09-08Not applicableUs
Quality Choice Childrens Allergy Reliefsolution5 mg/5mLoralChain Drug Marketing Association2008-04-22Not applicableUs
Quality Choice Childrens Allergy Reliefsolution5 mg/5mLoralChain Drug Marketing Association2011-05-20Not applicableUs
Reactinetablet5 mgoralMcneil Consumer Healthcare Division Of Johnson & Johnson Inc1997-03-06Not applicableCanada
Reactinesyrup5 mgoralMcneil Consumer Healthcare Division Of Johnson & Johnson Inc1999-12-21Not applicableCanada
Reactinetablet10 mgoralMcneil Consumer Healthcare Division Of Johnson & Johnson Inc1997-03-06Not applicableCanada
Reactine Allergy Liquid Gelscapsule (immediate release)10 mgoralMcneil Consumer Healthcare Division Of Johnson & Johnson Inc2012-04-01Not applicableCanada
Reactine Chewable Tablets 10 mgtablet (chewable)10 mgoralMcneil Consumer Healthcare Division Of Johnson & Johnson IncNot applicableNot applicableCanada
Reactine Chewable Tablets 5 mgtablet (chewable)5 mgoralMcneil Consumer Healthcare Division Of Johnson & Johnson IncNot applicableNot applicableCanada
Reactine Fast Melt Juniortablet (orally disintegrating)10 mgoralMcneil Consumer Healthcare Division Of Johnson & Johnson Inc2014-03-21Not applicableCanada
Reactine Tab 10mgtablet10 mgoralPfizer Canada Inc1991-12-311997-08-04Canada
Rexall All Day Allergy Relieftablet10 mg/1oralDolgencorp, LLC2012-09-06Not applicableUs
Rexall All Day Allergy Relief Childrenssolution5 mg/5mLoralDolgencorp, LLC2015-11-07Not applicableUs
Rexall Allergy Reliefliquid5 mg/5mLoralDolgencorp, LLC2010-08-07Not applicableUs
Rhinaris Relieftablet10 mgoralPendopharm Division Of De Pharmascience IncNot applicableNot applicableCanada
Rhinaris Relieftablet5 mgoralPendopharm Division Of De Pharmascience IncNot applicableNot applicableCanada
Rite Aid Childrens Allergy Reliefsolution5 mg/5mLoralRite Aid Corporation2008-04-22Not applicableUs
Rite Aid Childrens Allergy Reliefsolution1 mg/mLoralRite Aid Corporation2011-05-20Not applicableUs
Rite Aid Childrens Allergy Reliefsolution5 mg/5mLoralRite Aid Corporation2011-09-08Not applicableUs
Rx Act All Day Allergy Relieftablet10 mg/1oralH E B2008-01-31Not applicableUs
Safeway Children Allergy Reliefsolution5 mg/5mLoralSafeway Inc.2011-05-20Not applicableUs
Shoprite Allergytablet10 mg/1oralWakefern Food Corporation2013-08-14Not applicableUs
Shoprite Childrens Allergysolution5 mg/5mLoralWakefern Food Corporation2016-02-15Not applicableUs
Shoprite Childrens Allergyliquid5 mg/5mLoralWakefern Food Corporation2013-07-02Not applicableUs
Signature Care Allergy Relieftablet10 mg/1oralSafeway2015-09-17Not applicableUs
Signature Care Childrens Allergy Reliefsolution5 mg/5mLoralSafeway2015-09-28Not applicableUs
Simply Right Cetirizine Hydrochloridetablet10 mg/1oralSam's West Inc2013-04-10Not applicableUs
Simply Right Childrens Cetirizineliquid5 mg/5mLoralSam's West Inc2012-01-26Not applicableUs
Simply Right Childrens Cetirizinesolution5 mg/5mLoralSam's West Inc2011-09-08Not applicableUs
Smart Sense All Day Allergytablet10 mg/1oralKmart Corporation2011-01-18Not applicableUs
Smart Sense Allergy Relieftablet10 mg/1oralKmart Corporation2014-04-18Not applicableUs
Smart Sense Allergy Reliefsolution5 mg/5mLoralKmart Corporation2016-04-04Not applicableUs
Smart Sense Allergy Relief Childrenssolution5 mg/5mLoralKmart Corporation2015-10-21Not applicableUs
Smart Sense Childrens Allergysolution5 mg/5mLoralKmart Corporation2014-01-02Not applicableUs
Smart Sense Childrens Cetirizine Hydrochlorideliquid5 mg/5mLoralKmart Corporation2013-02-07Not applicableUs
Sound Body All Day Allergytablet, film coated10 mg/1oralBig Lots Stores, Inc.2015-04-28Not applicableUs
Sunmark All Day Allergytablet10 mg/1oralMc Kesson2008-01-21Not applicableUs
Sunmark All Day Allergy Childrensliquid5 mg/5mLoralMc Kesson2008-04-23Not applicableUs
Sunmark Childrens All Day Allergyliquid5 mg/5mLoralMc Kesson2010-09-09Not applicableUs
Sunmark Childrens Cetirizinesolution5 mg/5mLoralMc Kesson2011-09-08Not applicableUs
Target Childrens All Day Allergy Relief Sugar Free Grapesolution1 mg/mLoralTarget Corporation2011-09-08Not applicableUs
Topcare All Day Allergytablet10 mg/1oralTopco Associates LLC2008-01-10Not applicableUs
Topcare Childrens All Day Allergyliquid5 mg/5mLoralTopco Associates LLC2008-04-17Not applicableUs
Topcare Childrens All Day Allergysolution5 mg/5mLoralTopco Associates LLC2016-02-02Not applicableUs
Topcare Childrens All Day Allergyliquid5 mg/5mLoralTopco Associates LLC2013-12-23Not applicableUs
Up and Up All Day Allergy Relieftablet10 mg/1oralTarget Corporation2009-05-27Not applicableUs
Up and Up Allergy Reliefsolution5 mg/5mLoralTarget Corporation2015-01-23Not applicableUs
Up and Up Allergy Reliefsolution5 mg/5mLoralTarget Corporation2014-12-23Not applicableUs
Up and Up Allergy Relieftablet, film coated10 mg/1oralTarget Corporation2014-12-17Not applicableUs
Up and Up Childrens All Day Allergy Reliefliquid5 mg/5mLoralTarget Corporation2009-06-12Not applicableUs
Up and Up Childrens All Day Allergy Reliefliquid5 mg/5mLoralTarget Corporation2011-01-18Not applicableUs
Up and Up Childrens All Day Allergy Reliefsolution1 mg/mLoralTarget Corporation2011-05-20Not applicableUs
Up and Up Childrens Allergy Reliefsolution5 mg/5mLoralTarget Corporation2015-10-15Not applicableUs
Wal Zyrtablet10 mg/1oralWalgreen Company2008-01-09Not applicableUs
Wal Zyrsolution5 mg/5mLoralWalgreen Company2015-12-12Not applicableUs
Wal Zyr All Day Allergytablet10 mg/1oralWalgreen Company2008-01-09Not applicableUs
Wal Zyr Childrenssolution5 mg/5mLoralWalgreen Company2015-08-11Not applicableUs
Wal Zyr Childrensliquid5 mg/5mLoralWalgreen Company1989-08-15Not applicableUs
Wal-zyrtablet10 mg/1oralWalgreen Company2014-09-02Not applicableUs
Wal-zyr 24 Hour Allergytablet10 mg/1oralWalgreens2013-12-30Not applicableUs
Wal-zyr All Day Allergysolution5 mg/5mLoralWalgreen Company2011-05-20Not applicableUs
Wal-zyr Cetirizine Hydrochloridesolution5 mg/5mLoralWalgreen Company2011-09-08Not applicableUs
Wal-zyr Cetirizine Hydrochloridesolution5 mg/5mLoralWalgreen Company2008-04-22Not applicableUs
Western Family Childrens Allergy Reliefsolution5 mg/5mLoralWestern Family Foods Inc2011-05-20Not applicableUs
Zero Allergytablet10 mg/1oralEfficient Laboratories Inc2013-04-01Not applicableUs
Zyrteccapsule, liquid filled10 mg/1oralJohnson & Johnson Consumer Inc., Mc Neil Consumer Healthcare Division2010-02-08Not applicableUs
Zyrtec - Tab 10mgtablet10 mgoralUcb Inc1996-12-062001-07-05Canada
Zyrtec Allergytablet, orally disintegrating10 mg/1oralJohnson & Johnson Consumer Inc., Mc Neil Consumer Healthcare Division2014-01-20Not applicableUs
Zyrtec Allergytablet, film coated10 mg/1oralJohnson & Johnson Consumer Inc., Mc Neil Consumer Healthcare Division2008-10-01Not applicableUs
Unapproved/Other Products Not Available
International Brands
NameCompany
AlerlisinNot Available
CetrynNot Available
FormistinNot Available
HitrizinNot Available
VirlixNot Available
ZirtekNot Available
ZyrlexNot Available
Brand mixtures
NameLabellerIngredients
12 Hour Allergy DMeijer Distribution Inc
All Day Allergy DMajor Pharmaceuticals
All Day Allergy Relief DH E B
All Day Allergy-DL. Perrigo Company
Allergy and Congestion Relief D Original Prescription StrengthRite Aid Corporation
Allergy Relief DShopko Stores Operating Co., LLC
Careone All Day Allergy DAmerican Sales Company
Cetiri DRite Aid Corporation
Cetirizine HCl and Pseudoephedrine HCl ERPhysicians Total Care, Inc.
Cetirizine Hydrochloride and Pseudoephedrine HydrochloridePerrigo New York Inc
Equaline All Day Allergy DSupervalu Inc
Equate Allergy Relief DWal Mart Stores Inc
Good Neighbor Pharmacy All Day Allergy DAmerisource Bergen
Good Sense All Day Allergy DL Perrigo Company
Harris Teeter All Day Allergy DHarris Teeter, LLC
Health Mart Allergy Complete DMc Kesson
Healthy Accents Cetirizine-DDZA Brands LLC
Kirkland Signature Aller Tec DCostco Wholesale Company
Leader Allergy D 12Cardinal Health
Reactine CompleteMcneil Consumer Healthcare Division Of Johnson & Johnson Inc
Shoprite Allergy D 12Wakefern Food Corporation
Signature Care Allergy Relief DSafeway
Smart Sense All Day Allergy DKmart Corporation
Smart Sense Allergy Relief DKmart Corporation
Sunmark All Day Allergy DMc Kesson
Topcare All Day Allergy DTopco Associates LLC
Up and Up All Day Allergy Relief DTarget Corporation
Up and Up Allergy Plus Congestion Relief DTarget Corporation
Wal Zyr DWalgreen Company
Wal Zyr D Allergy and CongestionWalgreen Company
Zyrtec D Allergy and CongestionPhysicians Total Care, Inc.
Zyrtec-D Allergy and CongestionJohnson & Johnson Consumer Inc., Mc Neil Consumer Healthcare Division
Salts
Name/CASStructureProperties
Cetirizine hydrochloride
ThumbNot applicableDBSALT001214
Categories
UNIIYO7261ME24
CAS number83881-51-0
WeightAverage: 388.888
Monoisotopic: 388.155370383
Chemical FormulaC21H25ClN2O3
InChI KeyInChIKey=ZKLPARSLTMPFCP-UHFFFAOYSA-N
InChI
InChI=1S/C21H25ClN2O3/c22-19-8-6-18(7-9-19)21(17-4-2-1-3-5-17)24-12-10-23(11-13-24)14-15-27-16-20(25)26/h1-9,21H,10-16H2,(H,25,26)
IUPAC Name
2-(2-{4-[(4-chlorophenyl)(phenyl)methyl]piperazin-1-yl}ethoxy)acetic acid
SMILES
OC(=O)COCCN1CCN(CC1)C(C1=CC=CC=C1)C1=CC=C(Cl)C=C1
Taxonomy
DescriptionThis compound belongs to the class of organic compounds known as diphenylmethanes. These are compounds containing a diphenylmethane moiety, which consists of a methane wherein two hydrogen atoms are replaced by two phenyl groups.
KingdomOrganic compounds
Super ClassBenzenoids
ClassBenzene and substituted derivatives
Sub ClassDiphenylmethanes
Direct ParentDiphenylmethanes
Alternative Parents
Substituents
  • Diphenylmethane
  • Aralkylamine
  • N-alkylpiperazine
  • Halobenzene
  • Chlorobenzene
  • Piperazine
  • 1,4-diazinane
  • Aryl halide
  • Aryl chloride
  • Tertiary aliphatic amine
  • Tertiary amine
  • Azacycle
  • Organoheterocyclic compound
  • Monocarboxylic acid or derivatives
  • Ether
  • Dialkyl ether
  • Carboxylic acid
  • Carboxylic acid derivative
  • Hydrocarbon derivative
  • Organooxygen compound
  • Organonitrogen compound
  • Organochloride
  • Organohalogen compound
  • Carbonyl group
  • Amine
  • Aromatic heteromonocyclic compound
Molecular FrameworkAromatic heteromonocyclic compounds
External DescriptorsNot Available
Pharmacology
IndicationFor the relief of symptoms associated with seasonal allergic rhinitis, perennial allergic rhinitis and the treatment of the uncomplicated skin manifestations of chronic idiopathic urticaria
PharmacodynamicsCetirizine, the active metabolite of the piperazine H1-receptor antagonist hydroxyzine, is used to treat chronic idiopathic urticaria, perennial allergic rhinitis, seasonal allergic rhinitis, allergic asthma, physical urticaria, and atopic dermatitis.
Mechanism of actionCetirizine competes with histamine for binding at H1-receptor sites on the effector cell surface, resulting in suppression of histaminic edema, flare, and pruritus. The low incidence of sedation can be attributed to reduced penetration of cetirizine into the CNS as a result of the less lipophilic carboxyl group on the ethylamine side chain.
Related Articles
Absorptionmean peak plasma concentration (Cmax) of 114 ng/mL at a time (Tmax) of 2.2 hours postdose was observed for cetirizine
Volume of distributionNot Available
Protein bindingVery high (93%) plasma protein binding
MetabolismNot Available
Route of eliminationNot Available
Half life8.3 hours
Clearance
  • 53 mL/min [healthy]
ToxicitySomnolence (sleepiness or unusual drowsiness), restlessness, irritability
Affected organisms
  • Humans and other mammals
PathwaysNot Available
SNP Mediated EffectsNot Available
SNP Mediated Adverse Drug ReactionsNot Available
ADMET
Predicted ADMET features
PropertyValueProbability
Human Intestinal Absorption+0.6863
Blood Brain Barrier+0.7576
Caco-2 permeable-0.5879
P-glycoprotein substrateSubstrate0.7862
P-glycoprotein inhibitor IInhibitor0.7364
P-glycoprotein inhibitor IINon-inhibitor0.7624
Renal organic cation transporterNon-inhibitor0.5232
CYP450 2C9 substrateNon-substrate0.8408
CYP450 2D6 substrateNon-substrate0.9116
CYP450 3A4 substrateNon-substrate0.7
CYP450 1A2 substrateNon-inhibitor0.9045
CYP450 2C9 inhibitorNon-inhibitor0.907
CYP450 2D6 inhibitorNon-inhibitor0.8885
CYP450 2C19 inhibitorNon-inhibitor0.9025
CYP450 3A4 inhibitorNon-inhibitor0.9465
CYP450 inhibitory promiscuityLow CYP Inhibitory Promiscuity0.6917
Ames testNon AMES toxic0.7815
CarcinogenicityNon-carcinogens0.9426
BiodegradationNot ready biodegradable0.9974
Rat acute toxicity2.6841 LD50, mol/kg Not applicable
hERG inhibition (predictor I)Weak inhibitor0.866
hERG inhibition (predictor II)Inhibitor0.6517
ADMET data is predicted using admetSAR, a free tool for evaluating chemical ADMET properties. (23092397 )
Pharmacoeconomics
Manufacturers
  • Banner pharmacaps inc
  • Actavis mid atlantic llc
  • Amneal pharmaceuticals
  • Apotex inc
  • Aurobindo pharma ltd
  • Cypress pharmaceutical inc
  • Dr reddys laboratories ltd
  • Perrigo israel pharmaceuticals ltd
  • Ranbaxy laboratories ltd
  • Sun pharmaceutical industries inc
  • Taro pharmaceutical industries ltd
  • Teva pharmaceuticals usa
  • Vintage pharmaceuticals llc
  • Wockhardt ltd
  • Perrigo r and d co
  • Mcneil consumer healthcare div mcneil ppc inc
  • Caraco pharmaceutical laboratories ltd
  • Sandoz inc
  • Pfizer inc
  • Actavis elizabeth llc
  • Amneal pharmaceuticals ny llc
  • Cadista pharmaceuticals inc
  • Contract pharmacal corp
  • Mylan pharmaceuticals inc
  • Orchid healthcare
  • Torrent pharmaceuticals llc
  • Unichem laboratories ltd
  • Unique pharmaceutical laboratories
Packagers
Dosage forms
FormRouteStrength
Capsuleoral10 mg/1
Capsule, liquid filledoral10 mg/1
Capsuleoral10 mg
Syruporal1 mg/1
Tablet, film coated, extended releaseoral
Syruporal1 mg/mL
Syruporal5 mg/5mL
Tabletoral5 mg/1
Tablet, chewableoral5 mg/1
Tablet, film coatedoral10 mg/1
Tablet, film coatedoral5 mg/1
Solutionoral1 mg/mL
Tablet, chewableoral10 mg/1
Tabletoral10 mg/1
Tablet, extended releaseoral
Liquidoral5 mg/5mL
Syruporal5 mg
Tabletoral10 mg
Tabletoral5 mg
Tabletoral20 mg
Capsule (immediate release)oral10 mg
Tablet (chewable)oral10 mg
Tablet (chewable)oral5 mg
Tablet (extended-release)oral
Tablet (orally disintegrating)oral10 mg
Solutionoral5 mg/5mL
Tablet, orally disintegratingoral10 mg/1
Prices
Unit descriptionCostUnit
Cetirizine HCl 100 10 mg tablet Bottle259.71USD bottle
Cetirizine HCl 100 5 mg tablet Bottle259.71USD bottle
Zyrtec 10 mg tablet2.66USD tablet
Zyrtec 5 mg tablet2.66USD tablet
Zyrtec itchy eye 0.025% drops2.62USD ml
Cetirizine hcl 5 mg chew tablet2.5USD tablet
Cetirizine hcl 10 mg tablet2.49USD tablet
Cetirizine hcl 5 mg tablet2.49USD tablet
Zyrtec-d tablet1.33USD tablet
Child's zyrtec chew tablet0.9USD tablet
CVS Pharmacy allergy relief 10 mg tablet0.74USD each
DrugBank does not sell nor buy drugs. Pricing information is supplied for informational purposes only.
Patents
Patent NumberPediatric ExtensionApprovedExpires (estimated)
US6455533 No1998-07-022018-07-02Us
US6469009 No1999-07-132019-07-13Us
US6489329 No1996-04-082016-04-08Us
US7014867 No2002-06-102022-06-10Us
US7226614 No2002-06-102022-06-10Us
Properties
StateSolid
Experimental Properties
PropertyValueSource
melting point112.5 °CPhysProp
water solubility101 mg/LNot Available
logP2.8Not Available
Predicted Properties
PropertyValueSource
Water Solubility0.0658 mg/mLALOGPS
logP2.98ALOGPS
logP0.86ChemAxon
logS-3.8ALOGPS
pKa (Strongest Acidic)3.6ChemAxon
pKa (Strongest Basic)7.79ChemAxon
Physiological Charge0ChemAxon
Hydrogen Acceptor Count5ChemAxon
Hydrogen Donor Count1ChemAxon
Polar Surface Area53.01 Å2ChemAxon
Rotatable Bond Count8ChemAxon
Refractivity106.87 m3·mol-1ChemAxon
Polarizability41.88 Å3ChemAxon
Number of Rings3ChemAxon
Bioavailability1ChemAxon
Rule of FiveYesChemAxon
Ghose FilterYesChemAxon
Veber's RuleYesChemAxon
MDDR-like RuleYesChemAxon
Spectra
Mass Spec (NIST)Not Available
SpectraNot Available
References
Synthesis Reference

Manne Reddy, “Polymorphic forms of dihydrochloride salts of cetirizine and processes for preparation thereof.” U.S. Patent US20040186112, issued September 23, 2004.

US20040186112
General ReferencesNot Available
External Links
ATC CodesR06AE07
AHFS Codes
  • 04:08.00
PDB EntriesNot Available
FDA labelDownload (54.2 KB)
MSDSNot Available
Interactions
Drug Interactions
Drug
AclidiniumAclidinium may increase the anticholinergic activities of Cetirizine.
AmphetamineAmphetamine may decrease the sedative activities of Cetirizine.
AzelastineCetirizine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
BaclofenThe risk or severity of adverse effects can be increased when Baclofen is combined with Cetirizine.
Benzylpenicilloyl PolylysineCetirizine may decrease effectiveness of Benzylpenicilloyl Polylysine as a diagnostic agent.
BetahistineThe therapeutic efficacy of Betahistine can be decreased when used in combination with Cetirizine.
Botulinum Toxin Type ACetirizine may increase the anticholinergic activities of Botulinum Toxin Type A.
Botulinum Toxin Type BCetirizine may increase the anticholinergic activities of Botulinum Toxin Type B.
BrimonidineBrimonidine may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
BuprenorphineCetirizine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
CathinoneCathinone may decrease the sedative activities of Cetirizine.
Cimetropium BromideCetirizine may increase the anticholinergic activities of Cimetropium Bromide.
DoxylamineDoxylamine may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
DronabinolDronabinol may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
DroperidolDroperidol may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
EluxadolineCetirizine may increase the activities of Eluxadoline.
EthanolCetirizine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Glucagon recombinantThe risk or severity of adverse effects can be increased when Cetirizine is combined with Glucagon recombinant.
HyaluronidaseThe therapeutic efficacy of Hyaluronidase can be decreased when used in combination with Cetirizine.
HydrocodoneCetirizine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
HydroxyzineHydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
Ipratropium bromideIpratropium bromide may increase the anticholinergic activities of Cetirizine.
ItoprideThe therapeutic efficacy of Itopride can be decreased when used in combination with Cetirizine.
LorazepamThe risk or severity of adverse effects can be increased when Lorazepam is combined with Cetirizine.
LumacaftorThe serum concentration of Cetirizine can be decreased when it is combined with Lumacaftor.
Magnesium SulfateMagnesium Sulfate may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
MethotrimeprazineCetirizine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
MetyrosineCetirizine may increase the sedative activities of Metyrosine.
MianserinMianserin may increase the anticholinergic activities of Cetirizine.
MinocyclineMinocycline may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
MirabegronThe risk or severity of adverse effects can be increased when Cetirizine is combined with Mirabegron.
MirtazapineCetirizine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
MorphineThe risk or severity of adverse effects can be increased when Cetirizine is combined with Morphine.
NabiloneNabilone may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
OrphenadrineCetirizine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
ParaldehydeCetirizine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
ParoxetineThe risk or severity of adverse effects can be increased when Cetirizine is combined with Paroxetine.
PerampanelPerampanel may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
Potassium ChlorideCetirizine may increase the ulcerogenic activities of Potassium Chloride.
PramipexoleCetirizine may increase the sedative activities of Pramipexole.
PramlintidePramlintide may increase the anticholinergic activities of Cetirizine.
ProcyclidineThe risk or severity of adverse effects can be increased when Procyclidine is combined with Cetirizine.
RamosetronCetirizine may increase the activities of Ramosetron.
RanolazineThe serum concentration of Cetirizine can be increased when it is combined with Ranolazine.
RopiniroleCetirizine may increase the sedative activities of Ropinirole.
RotigotineCetirizine may increase the sedative activities of Rotigotine.
RufinamideThe risk or severity of adverse effects can be increased when Rufinamide is combined with Cetirizine.
SaquinavirThe serum concentration of Cetirizine can be increased when it is combined with Saquinavir.
SecretinThe therapeutic efficacy of Secretin can be decreased when used in combination with Cetirizine.
Sodium oxybateSodium oxybate may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
SulpirideThe therapeutic efficacy of Sulpiride can be decreased when used in combination with Cetirizine.
SuvorexantCetirizine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
TacrineThe therapeutic efficacy of Cetirizine can be decreased when used in combination with Tacrine.
TapentadolTapentadol may increase the central nervous system depressant (CNS depressant) activities of Cetirizine.
TesmilifeneThe serum concentration of Cetirizine can be decreased when it is combined with Tesmilifene.
ThalidomideCetirizine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
TiotropiumCetirizine may increase the anticholinergic activities of Tiotropium.
TopiramateThe risk or severity of adverse effects can be increased when Cetirizine is combined with Topiramate.
TrichlormethiazideThe serum concentration of Trichlormethiazide can be increased when it is combined with Cetirizine.
UmeclidiniumUmeclidinium may increase the anticholinergic activities of Cetirizine.
VerapamilThe serum concentration of Cetirizine can be increased when it is combined with Verapamil.
ZolpidemCetirizine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Food Interactions
  • Avoid alcohol.
  • Take without regard to meals.

Targets

Kind
Protein
Organism
Human
Pharmacological action
yes
Actions
antagonist
General Function:
Histamine receptor activity
Specific Function:
In peripheral tissues, the H1 subclass of histamine receptors mediates the contraction of smooth muscles, increase in capillary permeability due to contraction of terminal venules, and catecholamine release from adrenal medulla, as well as mediating neurotransmission in the central nervous system.
Gene Name:
HRH1
Uniprot ID:
P35367
Molecular Weight:
55783.61 Da
References
  1. Chen X, Ji ZL, Chen YZ: TTD: Therapeutic Target Database. Nucleic Acids Res. 2002 Jan 1;30(1):412-5. [PubMed:11752352 ]
  2. Christophe B, Carlier B, Gillard M, Chatelain P, Peck M, Massingham R: Histamine H1 receptor antagonism by cetirizine in isolated guinea pig tissues: influence of receptor reserve and dissociation kinetics. Eur J Pharmacol. 2003 May 30;470(1-2):87-94. [PubMed:12787835 ]
  3. Tashiro M, Sakurada Y, Iwabuchi K, Mochizuki H, Kato M, Aoki M, Funaki Y, Itoh M, Iwata R, Wong DF, Yanai K: Central effects of fexofenadine and cetirizine: measurement of psychomotor performance, subjective sleepiness, and brain histamine H1-receptor occupancy using 11C-doxepin positron emission tomography. J Clin Pharmacol. 2004 Aug;44(8):890-900. [PubMed:15286093 ]
  4. Tillement JP, Testa B, Bree F: Compared pharmacological characteristics in humans of racemic cetirizine and levocetirizine, two histamine H1-receptor antagonists. Biochem Pharmacol. 2003 Oct 1;66(7):1123-6. [PubMed:14505791 ]
  5. Cavero I, Mestre M, Guillon JM, Heuillet E, Roach AG: Preclinical in vitro cardiac electrophysiology: a method of predicting arrhythmogenic potential of antihistamines in humans? Drug Saf. 1999;21 Suppl 1:19-31; discussion 81-7. [PubMed:10597865 ]
  6. Tamura T, Masaki S, Ohmori K, Karasawa A: Effect of olopatadine and other histamine H1 receptor antagonists on the skin inflammation induced by repeated topical application of oxazolone in mice. Pharmacology. 2005 Dec;75(1):45-52. Epub 2005 Jun 7. [PubMed:15942272 ]
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Drug created on June 13, 2005 07:24 / Updated on July 29, 2016 01:52