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Identification
NameBenzocaine
Accession NumberDB01086  (APRD00539)
TypeSmall Molecule
GroupsApproved
Description

A surface anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings. [PubChem]

Structure
Thumb
Synonyms
SynonymLanguageCode
4-aminobenzoic acid ethyl esterNot AvailableNot Available
Amben ethyl esterNot AvailableNot Available
BenzocainaNot AvailableNot Available
BenzocaineNot AvailableNot Available
BenzocainumNot AvailableNot Available
Ethyl AminobenzoateNot AvailableNot Available
Ethyl p-AminobenzoateNot AvailableNot Available
Ethyl p-AminophenylcarboxylateNot AvailableNot Available
p-(Ethoxycarbonyl)anilineNot AvailableNot Available
p-CarbethoxyanilineNot AvailableNot Available
p-Ethoxycarboxylic AnilineNot AvailableNot Available
Prescription ProductsNot Available
Generic Prescription ProductsNot Available
Over the Counter Products
NameDosageStrengthRouteLabellerMarketing StartMarketing End
Colgate Orabasepaste, dentifrice.02 g/gtopicalColgate Oral Pharmaceuticals, Inc.2010-08-31Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Hurricaine Topical Anesthetic Gelgel200 mg/gdental; oral; periodontalBeutlich LP, Pharmaceuticals1993-02-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Hurricaine Topical Anesthetic Liquidliquid200 mg/gdental; oral; periodontalBeutlich LP, Pharmaceuticals1969-05-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Hurricaine Topical Anestheticspray200 mg/gdental; oral; periodontalBeutlich Pharmaceuticals, LLC1979-06-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Hurricaine Topical Anestheticgel200 mg/gdental; oral; periodontalBeutlich LP, Pharmaceuticals1971-08-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Hurricaine Topical Anestheticgel200 mg/gdental; oral; periodontalBeutlich LP, Pharmaceuticals1971-08-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Hurricaine Topical Anesthetic Gelgel200 mg/gdental; oral; periodontalBeutlich LP, Pharmaceuticals1986-08-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Hurricaine Topical Anestheticgel200 mg/gdental; oral; periodontalBeutlich Pharmaceuticals LLC1998-09-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Hurricaine Topical Anesthetic Liquidliquid200 mg/gdental; oral; periodontalBeutlich LP, Pharmaceuticals1986-08-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Walgreens Intense Toothachepaste, dentifrice20 g/100gtopicalWalgreens2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Severe Oral Pain Relieverliquid20 g/100goralWalgreens2012-01-10Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Walgreens Severe Oral Pain Relieverliquid20 g/100goralWalgreens2012-01-10Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Walgreens Severe Toothache Reliefpaste, dentifrice20 g/100gtopicalWalgreens2013-08-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Walgreens Maximum Strengthpaste, dentifrice20 g/100gtopicalWalgreens2013-08-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Walgreens Baby Teethinggel, dentifrice7.5 g/100goralWalgreens2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Walgreens Baby Teethinggel, dentifrice7.5 g/100goralWalgreens2013-09-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Walgreens Pain Relieving For Boilsointment20 g/100gtopicalWalgreen Company2014-05-28Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Walgreens Maximum Strengthpaste, dentifrice20 g/100gtopicalWalgreens2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Anbesol Regular Strengthsolution100 mg/mLtopicalPfizer Consumer Healthcare2004-05-11Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Anbesol Maximum Strengthsolution200 mg/mLtopicalPfizer Consumer Healthcare2005-05-11Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Baby Anbesolgel75 mg/gtopicalWyeth Consumer Healthcare2004-04-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Anbesol Regular Strengthgel100 mg/gtopicalPfizer Consumer Healthcare2005-05-11Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Anbesol Jrgel100 mg/gtopicalPfizer Consumer Healthcare2005-05-11Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Anbesol Maximum Strengthgel200 mg/gtopicalPfizer Consumer Healthcare2005-05-11Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Oral Pain Relief Anesthetic Anestheticgel200 mg/goralMajor Pharmaceuticals2009-08-19Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Kank-a Mouth Painliquid200 mg/mLbuccalBlistex Inc.2011-12-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Carmex Cold Sore Treatment External Analgesiccream10 g/100gtopicalCarma Laboratories, Inc.2014-05-28Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel Maximum Strengthliquid.2 mL/mLtopicalChurch & Dwight Co., Inc.2010-04-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel Instant Pain Relief Regular Strengthgel100 mg/gtopicalChurch & Dwight Co., Inc.2010-06-10Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel For Toothache Maximum Strengthswab.2 mL/mLtopicalChurch & Dwight Co., Inc.2010-08-11Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel Instant Pain Relief Maximum Strengthgel.4; 200; 1 mg/g; mg/g; mg/gtopicalChurch & Dwight Co., Inc.2010-06-11Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel For All Mouth Sores Maximum Strengthswab.2 mL/mLtopicalChurch & Dwight Co., Inc.2010-08-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel Instant Relief For Teething Pain Cooling Cucumbergel75 mg/gtopicalChurch & Dwight Co., Inc.2010-06-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel Severe Toothache Maximum Strength Fast-Acting Formulaliquid.2 mL/mLtopicalChurch & Dwight Co., Inc.2011-03-21Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel Instant Relief For Teething Pain Longer Lastinggel75 mg/gtopicalChurch & Dwight Co., Inc.2011-03-22Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel Instant Relief For Teething Painswab.075 mL/mLtopicalChurch & Dwight Co., Inc.2010-08-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel Nighttime Instant Relief For Teething Pain Longer Lasting Extra Strengthgel100 mg/gtopicalChurch & Dwight Co., Inc.2010-06-18Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel Instant Relief For Teething Pain Daytime Nighttime Twin PackkitChurch & Dwight Co., Inc.2011-03-22Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Orajel For Cold Sorescream200; 744.4 mg/g; mg/gtopicalChurch & Dwight Co., Inc.2010-07-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mandelay Male Genital Desensitizergel2.13 g/28.35gtopicalMajestic Drug Co., INC.1995-10-31Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Red Cross Oral Pain Reliefliquid200 mg/mLtopicalThe Mentholatum Company2013-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cepacol Fizzlerstablet, orally disintegrating6 mgoralCombe Incorporated2009-09-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Sheffield Baby Teething Gelgel75 mg/goralFaria LLC dba Sheffield Pharmaceuticals2003-06-17Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Sheffield Pain Reliefgel200 mg/goralFaria LLC dba Sheffield Pharmaceuticals2006-01-30Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Alcohol Prep Padsswab.06; .7 mL/1; mLtopicalTarget Corporation2010-02-19Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Rite Aid Maximum Strengthgel, dentifrice20 g/100goralRite Aid2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Rite Aid Maximum Strengthgel, dentifrice.04; 20; .1 g/100g; g/100g; g/100goralRite Aid2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Rite Aid Maximum Strengthliquid20 g/100gdentalRite Aid2015-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Rite Aid Baby Caregel, dentifrice7.5 g/100goralRite Aid2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Rite Aid Liquid Anesthetic Oral Pain Reliefgel200 mg/mLoralRite Aid Corporation2010-07-08Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Rite Aid Oral Pain Relieverliquid20 g/100goralRite Aid2013-08-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Rite Aid Professional Strengthliquid20 g/100goralRite Aid2014-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Rite Aid Maximum Strengthpaste, dentifrice20 g/100gtopicalRite Aid2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
My Fair Baby Instant Pain Reliefgel7.5 g/100gtopicalDelta Brands Inc2014-06-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Bactimicina For Sore Throatlozenge15 mgoralDLC Laboratories, Inc.2011-05-24Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Pain Relief Alcohol Swabsswab.06; .7 mL/1; mLtopicalAmerisource Bergen2007-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Boy Butter Extreme H2O Desensitizing Lubricantcream4.25 g/85.05gtopicalBoy Butter Lubes2011-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Boy Butter Extreme H2O Desensitizing Lubricantcream34.05 g/454gtopicalBoy Butter Lubes2011-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Boy Butter Extreme Desensitizing Lubricantcream34.05 g/454gtopicalBoy Butter Lubes2011-05-23Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Boy Butter Desensitizing Lubricantcream6.39 g/85.2gtopicalBoy Butter Lubes2011-05-23Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Boy Butter Extreme H2O Desensitizing Lubricantcream7.1 g/142gtopicalBoy Butter Lubes2011-05-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Boy Butter Desensitizing Lubricantcream10.65 g/142gtopicalBoy Butter Lubes2011-05-23Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Boy Butter Desensitizing Lubricantcream73.9395789 mg/mLtopicalBoy Butter Lubes2012-09-25Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Boy Butter Desensitizing Lubricantcream71.9395789 mg/mLtopicalBoy Butter Lubes2012-09-25Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gumnumb Topical Anestheticgel200 mg/gdentalCrosstex International Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gumnumb Topical Anestheticgel200 mg/gdentalCrosstex International Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gumnumb Topical Anestheticgel200 mg/gdentalCrosstex International Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gumnumb Topical Anestheticgel200 mg/gdentalCrosstex International Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gumnumb Topical Anestheticgel200 mg/gdentalCrosstex International Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gumnumb Topical Anestheticgel200 mg/gdentalCrosstex International Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Terrasil Boil Pain Reliefointment3.5 g/100gtopicalAidance Skincare & Topical Solutions, LLC2014-06-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Oral Gel Maximum Strengthgel20 g/100gtopicalBudpak Inc.2010-02-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Baby Teething Oral Pain Relievergel7.5 g/100gtopicalBudpak Inc.2010-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Budpak Baby Teething Oral Pain Relievergel7.5 g/100gtopicalBudpak Inc.2013-12-26Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Budpak Oral Maximum Strengthgel.2 g/gtopicalBudpak Inc.2013-06-10Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Kroger Toothache Pain Reliefpaste, dentifrice20 g/100gtopicalKroger2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Sting Relief Padsswab.06 mL/mLtopicalJiangsu Province Jian Er Kang Medical Dressing Co. ,Ltd.2010-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mouth Sore Medicationliquid200 mg/gtopicalZEE MEDICAL2010-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topcare Maximum Strengthliquid20 g/100goralTopco2014-10-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Leader Oral Analgesicgel20 g/100goralCardinal Health2012-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Heb Severe Toothachepaste, dentifrice20 g/100gtopicalHEB2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Benzodentcream.2 g/gtopicalChattem, Inc.1994-05-12Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Oral Analgesic Maximum Strengthliquid.2 mL/mLtopicalMeijer Distribution Inc.2010-05-13Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Good Neighbor Pain Reliefliquid200 mg/mLoralAmerisource Bergen Drug Corporation (Good Neighbor Pharmacy)2008-08-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Benzocaineswab60 mg/mLtopicalUnifirst First Aid Corporation2014-08-26Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Oral B Instant Pain Reliefgel.2 mL/mLoralHealth Tech, Inc.Not AvailableNot AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Kmart Smart Sensepaste, dentifrice20 g/100gtopicalK Mart2013-12-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Pina Coladagel220 mg/gdentalPatterson Dental Supply Inc1963-02-19Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Strawberrygel220 mg/gdentalPatterson Dental Supply Inc1963-02-19Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Mintgel220 mg/gdentalPatterson Dental Supply Inc1963-02-19Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Raspberrygel220 mg/gdentalPatterson Dental Supply Inc1963-02-19Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Bubble Gumgel220 mg/gdentalPatterson Dental Supply Inc1963-02-19Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Cherrygel220 mg/gdentalPatterson Dental Supply Inc1963-02-19Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Zilactin-bgel.1 g/gtopicalBlairex Laboratories, Inc.2005-06-29Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Herbasoul Male Genital Desensitizer Creamcream4.5 g/100gtopicalBodon Med Laboratories Ltd.2010-02-23Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Jianze Sting Relief Padsliquid6 g/100gtopicalChangzhou Jianze Sanitary Material Co., Ltd.2012-06-14Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Goodsense Oral Pain Reliefgel20 g/100gtopicalGeiss, Destin and Dunn, Inc.2014-05-09Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Atopalm Oral Pain Reliefgel10 g/100goralNeo Pharm, Usa2012-02-06Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ultracare Anesthetic Bubble Gumgel6.96 g/30mLdentalUltradent Products, Inc.1986-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ultracare Anesthetic Walterberrygel6.96 g/30mLdentalUltradent Products, Inc.1993-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ultracare Anesthetic Butter Rumgel6.96 g/30mLdentalUltradent Products, Inc.1986-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ultracare Anesthetic Pina Coladagel6.96 g/30mLdentalUltradent Products, Inc.1986-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ultracare Anesthetic Creme de Menthegel6.96 g/30mLdentalUltradent Products, Inc.1986-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Oral Analgesic Maximum Strengthgel200 mg/gtopicalLif Elabs, A Division Of Atico International Usa, Inc.2010-11-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Opahlgel6.4 g/32gdental; oralDharma Research, Inc.2013-11-02Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Opahlgel6.4 g/32gdental; oralDharma Research, Inc.2013-11-02Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Opahlgel6.4 g/32gdental; oralDharma Research, Inc.2013-11-02Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Opahlgel6.4 g/32gdental; oralDharma Research, Inc.2013-11-02Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Opahlgel6.4 g/32gdental; oralDharma Research, Inc.2013-11-02Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Opahlgel6.4 g/32gdental; oralDharma Research, Inc.2013-11-02Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Opahlgel6.4 g/32gdental; oralDharma Research, Inc.2013-11-02Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Opahlgel6.4 g/32gdental; oralDharma Research, Inc.2013-11-02Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Opahl Dye Freegel6.4 g/32gdental; oralDharma Research, Inc.2013-11-02Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Anestenkaliquid.2 mg/2mLtopicalMenper Distributors, Inc2014-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Nene Denteliquid2.1 mg/30mLtopicalMenper Distributors, Inc2014-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Baby Anestenkaliquid2.1 mg/30mLtopicalMenper Distributors2014-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Benz O Stheticspray20 mL/100mLtopicalGeritrex Corp.2012-02-13Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Benz O Stheticgel20 g/100gtopicalGeritrex Corp.2012-01-26Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Comfortcaine Topical Anestheticgel200 mg/gdentalDental Technologies, Inc.1997-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Comfortcaine Topical Anestheticgel200 mg/gdentalDental Technologies, Inc.1997-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Comfortcaine Topical Anestheticgel200 mg/gdentalDental Technologies, Inc.1997-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Comfortcaine Topical Anestheticgel200 mg/gdentalDental Technologies, Inc.1997-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Comfortcaine Topical Anestheticgel200 mg/gdentalDental Technologies, Inc.1997-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Comfortcaine Topical Anestheticgel200 mg/gdentalDental Technologies, Inc.1997-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Alpha-caine Topical Anestheticgel200 mg/gtopicalDental Technologies, Inc.1999-12-31Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Alpha-caine Topical Anestheticgel200 mg/gtopicalDental Technologies, Inc.1999-12-31Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Alpha-caine Topical Anestheticgel200 mg/gtopicalDental Technologies, Inc.1999-12-31Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Alpha-caine Topical Anestheticgel200 mg/gtopicalDental Technologies, Inc.1999-12-31Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Anestheticgel200 mg/gtopicalMoore Medical LLC2012-07-12Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Dollar General Toothache Reliefpaste, dentifrice20 g/100gtopicalDollar General2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Rexall Maximum Strengthliquid20 g/100gdentalRexall2015-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Oral Pain Relieverliquid20 g/100goralDolgencorp LLC2012-01-10Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Sting Relief Medicated Padswab.06 mgtopicalTongzhou Ruihong Medical Products Factory2013-05-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Finafta Babyliquid7.5 mg/100mgoralEfficient Laboratories Inc.2000-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Finafta MultiOralliquid7.5 mL/100mLoralEfficient Laboratories Inc.2004-09-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Maximum Strengthpaste, dentifrice20 g/100gtopicalCVS Pharmacy2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Oral Anestheticliquid200 mg/mLoralCVS Pharmacy2010-07-08Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Intense Cvs Intense Toothachepaste, dentifrice20 g/100gtopicalCVS Pharmacy2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Maximum Strength Boil Reliefointment20 g/100gtopicalCVS Pharmacy, Inc.2014-10-13Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Pharmacy Maximum Strengthgel, dentifrice20 g/100goralCVS Pharmacy2011-01-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Pharmacy Maximum Strengthgel, dentifrice20 g/100goralCVS Pharmacy2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Pharmacy Maximum Strengthliquid20 g/100gdentalCVS Pharmacy2015-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Severe Oral Pain Relieverliquid20 g/100goralCVS Pharmacy2011-12-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Fast Acting Baby Teethinggel75 mg/goralCVS Pharmacy2010-07-08Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Fast Acting Baby Teethinggel75 mg/goralCVS Pharmacy2010-07-08Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mouth Sore Relief Professional Strengthliquid200 mg/goralCVS Pharmacy2009-10-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Instant Toothache Pain Reliefliquid20 g/100goralCVS Pharmacy2009-10-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Pharmacy Nighttime Oral Pain Reliefgel, dentifrice10 g/100gdentalCVS Pharmacy2013-08-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Pharmacy Mouth Sore Gelgel, dentifrice.02; 20; .1 g/100g; g/100g; g/100goralCVS Pharmacy2012-10-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cvs Pharmacy Instant Toothachegel, dentifrice20 g/100gdentalCVS Pharmacy2012-10-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Brace Reliefgel9 mg/mLoralInfa Lab,Inc2005-01-03Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Dentek Instant Pain Relief Maximum Strengthliquid200 mg/mLtopicalDen Tek Oral Care. Inc.2014-02-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Pain Reliefliquid200 mg/gtopicalSafetec of America, Inc.2010-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mark 3gel6.4 g/32gdental; oralCargus International, Inc.2014-02-28Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mark 3gel6.4 g/32gdental; oralCargus International, Inc.2014-02-28Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mark 3gel6.4 g/32gdental; oralCargus International, Inc.2014-02-28Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mark 3gel6.4 g/32gdental; oralCargus International, Inc.2014-03-03Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mark 3gel6.4 g/32gdental; oralCargus International, Inc.2014-03-03Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mark 3gel6.4 g/32gdental; oralCargus International, Inc.2014-03-03Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mark 3gel6.4 g/32gdental; oralCargus International, Inc.2012-03-03Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mark 3gel6.4 g/32gdental; oralCargus International, Inc.2014-03-03Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Preboostliquid4 g/100mLtopical944 Corp2014-02-18Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Little Colds Sore Throat Relief Melt Awaysgranule6 mgoralMedtech Products Inc.2009-12-31Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Outgroliquid.009 mg/mLtopicalMedtech Products Inc.2013-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Shunga Male Genital Desensitizeraerosol, spray1.125 g/15gtopicalEau Zone Oils & Fragrances LTD2010-08-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Oralabs Cold Sore Treatmentointment5 mg/gtopicalOra Labs2014-08-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Tanacliquid1.3 mg/13mLoralInsight Pharmaceuticals LLC2011-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Boil Easecream5 g/28gtopicalInsight Pharmaceuticals2010-06-21Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Americaineointment5.6 g/28gtopicalInsight Pharmaceuticals2009-07-10Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Americaineaerosol, spray11.4 g/57gtopicalInsight Pharmaceuticals2009-07-14Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cepacol Sensations Warminglozenge4 mgoralReckitt Benckiser LLC2012-06-10Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cepacol Sensations Hydralozenge3 mgoralReckitt Benckiser LLC2012-05-28Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Cepacol Sensations Sore Throat Hydra citrus splashlozenge3 mgoralReckitt Benckiser LLC2013-07-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Quality Choice Maximum Strength Oral Pain Relievinggel20 g/100gtopicalChain Drug Marketing Association Inc2013-05-31Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Baby Sensigelgel7.5 g/100gtopicalDr. Fresh, Inc2011-10-12Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Baby Sensigel Night Time Formulagel10 g/100gtopicalDr. Fresh, Inc2011-10-07Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Sensigelgel20 g/100gtopicalDr. Fresh, Inc.2011-09-26Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Dukal Sting Relief Padswab60; .6 mg/mL; mL/mLtopicalDukal Corporation2010-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Physicians Care Sting Relief Padswab.06; .6 mL/mL; mL/mLtopicalDukal Corporation2010-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Insect Bite Reliefliquid15 mg/mLtopicalSwabplus Inc.2003-03-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Insect Bite Reliefsolution150 mg/mLtopicalSwabplus Inc.2003-03-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Mouth Sore Relief Applicatorliquid200 mg/mLoralSwabplus Inc.2005-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Iodent Maximum Strength Oral Analgesicgel20 g/100gtopicalUnited Exchange Corp2013-05-31Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Sally Hansen Ouch-relief Wax KitkittopicalCoty US LLC2012-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Sally Hansen Ouch-relief Wax Strip KitkittopicalCoty US LLC2012-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Sally Hansen Ouch-relief Numbing Wipescloth.0543 gtopicalCoty US LLC2015-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Bencocaine Topical Anestheticgel200 mg/gdentalBenco Dental2014-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Bencocaine Topical Anestheticgel200 mg/gdentalBenco Dental2014-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Bencocaine Topical Anestheticgel200 mg/gdentalBenco Dental2014-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Bencocaine Topical Anestheticgel200 mg/gdentalBenco Dental2014-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Bencocaine Topical Anestheticgel200 mg/gdentalBenco Dental2014-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Bencocaine Topical Anestheticgel200 mg/gdentalBenco Dental2014-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Bencocaine Topical Anestheticgel200 mg/gdentalBenco Dental2014-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Bencocaine Topical Anestheticgel200 mg/gdentalBenco Dental2014-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Bencocaine Topical Anestheticgel200 mg/gdentalBenco Dental2014-06-27Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Winco Foods Maximum Strength Oral Analgesicgel200 mg/gtopicalWin Co Foods, Llc2014-12-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Chloraseptic Warming Sore Throatlozenge15 mgoralPrestige Brands Holdings, Inc.2012-01-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Chloraseptic Warming Sore Throatlozenge15 mgoralPrestige Brands Holdings, Inc.2012-09-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Cherrygel200 mg/gdentalSafco Dental Supply Co.2012-08-06Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Mintgel200 mg/gdentalSafco Dental Supply Co.2012-08-06Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Bananagel200 mg/gdentalSafco Dental Supply Co.2012-08-06Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Pina Coladagel200 mg/gdentalSafco Dental Supply Co.2012-08-06Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Bubble Gumgel200 mg/gdentalSafco Dental Supply Co.2012-08-06Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Strawberrygel200 mg/gdentalSafco Dental Supply Co.2012-08-06Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Topical Anesthetic Raspberrygel200 mg/gdentalSafco Dental Supply Co.2012-08-06Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Benzocaineswab.12 mLtopicalDynarex Corporation2011-01-24Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Benzocaineswab60 mg/mLtopicalDynarex Corporation2011-07-20Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gelato Topical Anestheticspray, metered11.4 g/57gdentalMycone Dental Supply Co., Inc DBA Keystone Industries and Deepak Products Inc2013-07-29Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gelato Topical Anestheticgel200 mg/gdentalMycone Dental Supply Co., Inc DBA Keystone Industries and Deepak Products Inc2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gelato Topical Anestheticgel200 mg/gdentalMycone Dental Supply Co., Inc DBA Keystone Industries and Deepak Products Inc2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gelato Topical Anestheticgel200 mg/gdentalMycone Dental Supply Co., Inc DBA Keystone Industries and Deepak Products Inc2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gelato Topical Anestheticgel200 mg/gdentalMycone Dental Supply Co., Inc DBA Keystone Industries and Deepak Products Inc2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gelato Topical Anestheticgel200 mg/gdentalMycone Dental Supply Co., Inc DBA Keystone Industries and Deepak Products Inc2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gelato Topical Anestheticgel200 mg/gdentalMycone Dental Supply Co., Inc DBA Keystone Industries and Deepak Products Inc2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gelato Topical Anestheticgel200 mg/gdentalMycone Dental Supply Co., Inc DBA Keystone Industries and Deepak Products Inc2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gelato Topical Anestheticgel200 mg/gdentalMycone Dental Supply Co., Inc DBA Keystone Industries and Deepak Products Inc2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gelato Topical Anestheticgel200 mg/gdentalMycone Dental Supply Co., Inc DBA Keystone Industries and Deepak Products Inc2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Dental Reliefliquid200 mg/gtopicalCintas First Aid & Safety2012-06-13Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Pac-dent Top Gelgel200 mg/gdentalPac Dent International, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Pac-dent Top Gelgel200 mg/gdentalPac Dent International, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Pac-dent Top Gelgel200 mg/gdentalPac Dent International, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Pac-dent Top Gelgel200 mg/gdentalPac Dent International, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Pac-dent Top Gelgel200 mg/gdentalPac Dent International, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Purelife Topical Anestheticgel200 mg/gdentalPure Life Dental2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Purelife Topical Anestheticgel200 mg/gdentalPure Life Dental2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Purelife Topical Anestheticgel200 mg/gdentalPure Life Dental2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Purelife Topical Anestheticgel200 mg/gdentalPure Life Dental2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Purelife Topical Anestheticgel200 mg/gdentalPure Life Dental2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Purelife Topical Anestheticgel200 mg/gdentalPure Life Dental2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Purelife Topical Anestheticgel200 mg/gdentalPure Life Dental2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Purelife Topical Anestheticgel200 mg/gdentalPure Life Dental2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gps Topical Anestheticgel200 mg/gdentalGroup Practice Solutions, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gps Topical Anestheticgel200 mg/gdentalGroup Practice Solutions, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gps Topical Anestheticgel200 mg/gdentalGroup Practice Solutions, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gps Topical Anestheticgel200 mg/gdentalGroup Practice Solutions, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gps Topical Anestheticgel200 mg/gdentalGroup Practice Solutions, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Gps Topical Anestheticgel200 mg/gdentalGroup Practice Solutions, Inc.2013-07-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Makesense Junior Pain Reliefgel7.5 g/100gtopicalCherry Hill Sales Co2014-07-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Makesense Pain Reliefgel20 g/100gtopicalCherry Hill Sales Co2014-07-15Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Top Quality Mfg. Topical Anestheticgel200 mg/gdentalTop Quality Manufacturing, Inc.2014-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Top Quality Mfg. Topical Anestheticgel200 mg/gdentalTop Quality Manufacturing, Inc.2014-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Top Quality Mfg. Topical Anestheticgel200 mg/gdentalTop Quality Manufacturing, Inc.2014-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Top Quality Mfg. Topical Anestheticgel200 mg/gdentalTop Quality Manufacturing, Inc.2014-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Top Quality Mfg. Topical Anestheticgel200 mg/gdentalTop Quality Manufacturing, Inc.2014-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Top Quality Mfg. Topical Anestheticgel200 mg/gdentalTop Quality Manufacturing, Inc.2014-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Top Quality Mfg. Topical Anestheticgel200 mg/gdentalTop Quality Manufacturing, Inc.2014-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Tiger Supply Inc Topical Anestheticgel200 mg/gdentalTiger Supply Inc.2013-05-08Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Tiger Supply Inc Topical Anestheticgel200 mg/gdentalTiger Supply Inc.2013-05-08Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Tiger Supply Inc Topical Anestheticgel200 mg/gdentalTiger Supply Inc.2013-05-08Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Tiger Supply Inc Topical Anestheticgel200 mg/gdentalTiger Supply Inc.2013-05-08Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Tiger Supply Inc Topical Anestheticgel200 mg/gdentalTiger Supply Inc.2013-05-08Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Tiger Supply Inc Topical Anestheticgel200 mg/gdentalTiger Supply Inc.2013-05-08Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ismile Topical Anestheticgel200 mg/gdentalI Smile Dental Products, Inc.2014-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ismile Topical Anestheticgel200 mg/gdentalI Smile Dental Products, Inc.2014-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ismile Topical Anestheticgel200 mg/gdentalI Smile Dental Products, Inc.2014-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ismile Topical Anestheticgel200 mg/gdentalI Smile Dental Products, Inc.2014-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ismile Topical Anestheticgel200 mg/gdentalI Smile Dental Products, Inc.2014-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Ismile Topical Anestheticgel200 mg/gdentalI Smile Dental Products, Inc.2014-06-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Allegenal-mcream7.5 g/100gtopicalHalal Nutritional Center2015-01-28Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Male Desensitizer Pleasure Balmgel3 g/100mLtopicalKama Sutra2011-02-14Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Pleasure Balm Kama Sutragel5 g/100mLtopicalKama Sutra2013-09-12Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
Certus Sting Relief Prep Padswab.06 mL/mLtopicalCertus Medical, Inc.2011-05-01Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
20/20 Topical Anestheticstrip10 mgdentalAdvanced Dental Anesthetics2012-02-28Not AvailableUs 0a2ef1ad1c84951dc1392a8bbe1f3cb241c91ed59e44ad8268635315440d978c
International Brands
NameCompany
AnacaineNot Available
AnaesthesinNot Available
Anbesol BabyNot Available
DermoplastNot Available
Brand mixtures
Brand NameIngredients
Anbesol GelBenzocaine + Phenol
Anbesol LiquidBenzocaine + Camphor + Menthol + Phenol
AnivyBenzocaine + Chlorphenesin + Titanium Dioxide + Zinc Oxide
AppedrineBenzocaine + Iron (Ferrous Fumarate) + Nicotinamide + Thiamine Hydrochloride + Vitamin a (Vitamin a Acetate) + Vitamin B2 + Vitamin C (Sodium Ascorbate) + Vitamin D
ArkodyneBenzalkonium Chloride + Benzocaine + Oxyquinoline Sulfate
AuralganAntipyrine + Benzocaine
Burn O Sol SprayBenzocaine + Chlorhexidine Acetate
CepacolBenzocaine + Cetylpyridinium Chloride
CetacaineBenzocaine + Butamben + Tetracaine Hydrochloride
ChlorasepticBenzocaine + Menthol
EndosprayBenzocaine + Tetracaine Hydrochloride
Extra Strength LanacaneBenzocaine + Resorcinol
Extra Strength VagisilBenzocaine + Resorcinol
Lanacane Anti-Bacterial First Aid SprayBenzethonium Chloride + Benzocaine
Lanacane CreamBenzocaine + Resorcinol
OnrectalBenzocaine + Bismuth Subcarbonate (Oxycarbonate) + Bismuth Subgallate + Hamamelis Virginiana + Naphazoline Hydrochloride + Zinc Oxide
Orajel Denture PlusBenzocaine + Menthol
Orajel Mouth Sore MedicineBenzocaine + Zinc Chloride
Orajel Mouth-AidBenzalkonium Chloride + Benzocaine + Zinc Chloride
Orajel Multi-Action Cold Sore MedicineAllantoin + Benzocaine + Camphor + Dimethicone + Menthol + White Petrolatum
Orajel Ultra Canker Sore MedicineBenzocaine + Menthol
RectogelBenzocaine + Zinc Sulfate
SolarcaineBenzocaine + Triclosan
Sting EzeBenzocaine + Phenol
SaltsNot Available
Categories
CAS number94-09-7
WeightAverage: 165.1891
Monoisotopic: 165.078978601
Chemical FormulaC9H11NO2
InChI KeyBLFLLBZGZJTVJG-UHFFFAOYSA-N
InChI
InChI=1S/C9H11NO2/c1-2-12-9(11)7-3-5-8(10)6-4-7/h3-6H,2,10H2,1H3
IUPAC Name
ethyl 4-aminobenzoate
SMILES
CCOC(=O)C1=CC=C(N)C=C1
Taxonomy
DescriptionThis compound belongs to the class of organic compounds known as benzoic acid esters. These are ester derivatives of benzoic acid.
KingdomOrganic compounds
Super ClassBenzenoids
ClassBenzene and substituted derivatives
Sub ClassBenzoic acids and derivatives
Direct ParentBenzoic acid esters
Alternative Parents
Substituents
  • Benzoate ester
  • Aminobenzoic acid or derivatives
  • Benzylether
  • Substituted aniline
  • Benzoyl
  • Aniline
  • Primary aromatic amine
  • Carboxylic acid ester
  • Monocarboxylic acid or derivatives
  • Carboxylic acid derivative
  • Hydrocarbon derivative
  • Primary amine
  • Organooxygen compound
  • Organonitrogen compound
  • Carbonyl group
  • Amine
  • Aromatic homomonocyclic compound
Molecular FrameworkAromatic homomonocyclic compounds
External Descriptors
Pharmacology
IndicationFor general use as a lubricant and topical anesthetic on esophagus, larynx, mouth, nasal cavity, rectum, respiratory tract or trachea, urinary tract, vagina. It is also used to suppress gag reflex.
PharmacodynamicsBenzocaine is a local anesthetic commonly used as a topical pain reliever. It is the active ingredient in many over-the-counter analgesic ointments. It is also indicated for general use as a lubricant and topical anesthetic on intratracheal catheters and pharyngeal and nasal airways to obtund the pharyngeal and tracheal reflexes; on nasogastric and endoscopic tubes; urinary catheters; laryngoscopes; proctoscopes; sigmoidoscopes and vaginal specula.
Mechanism of actionBenzocaine binds to sodium channels and reversibly stabilizes the neuronal membrane which decreases its permeability to sodium ions. Depolarization of the neuronal membrane is inhibited thereby blocking the initiation and conduction of nerve impulses.
AbsorptionNot Available
Volume of distributionNot Available
Protein bindingNot Available
MetabolismNot Available
Route of eliminationNot Available
Half lifeNot Available
ClearanceNot Available
ToxicityLD50=3040 mg/kg (rat, oral)
Affected organisms
  • Humans and other mammals
PathwaysNot Available
SNP Mediated EffectsNot Available
SNP Mediated Adverse Drug ReactionsNot Available
ADMET
Predicted ADMET features
PropertyValueProbability
Human Intestinal Absorption+0.9963
Blood Brain Barrier+0.9609
Caco-2 permeable+0.7814
P-glycoprotein substrateNon-substrate0.8329
P-glycoprotein inhibitor INon-inhibitor0.9589
P-glycoprotein inhibitor IINon-inhibitor0.9612
Renal organic cation transporterNon-inhibitor0.8818
CYP450 2C9 substrateNon-substrate0.8426
CYP450 2D6 substrateNon-substrate0.7934
CYP450 3A4 substrateNon-substrate0.7513
CYP450 1A2 substrateInhibitor0.9107
CYP450 2C9 substrateNon-inhibitor0.9071
CYP450 2D6 substrateNon-inhibitor0.9231
CYP450 2C19 substrateNon-inhibitor0.9025
CYP450 3A4 substrateNon-inhibitor0.937
CYP450 inhibitory promiscuityLow CYP Inhibitory Promiscuity0.7883
Ames testNon AMES toxic0.8825
CarcinogenicityCarcinogens 0.513
BiodegradationReady biodegradable0.7718
Rat acute toxicity1.7665 LD50, mol/kg Not applicable
hERG inhibition (predictor I)Weak inhibitor0.9721
hERG inhibition (predictor II)Non-inhibitor0.9668
Pharmacoeconomics
ManufacturersNot Available
Packagers
Dosage forms
FormRouteStrength
Aerosol, spraytopical1.125 g/15g
Aerosol, spraytopical11.4 g/57g
Clothtopical.0543 g
Creamtopical.2 g/g
Creamtopical10 g/100g
Creamtopical10.65 g/142g
Creamtopical200; 744.4 mg/g; mg/g
Creamtopical34.05 g/454g
Creamtopical4.25 g/85.05g
Creamtopical4.5 g/100g
Creamtopical5 g/28g
Creamtopical6.39 g/85.2g
Creamtopical7.1 g/142g
Creamtopical7.5 g/100g
Creamtopical71.9395789 mg/mL
Creamtopical73.9395789 mg/mL
Geldental200 mg/g
Geldental220 mg/g
Geldental6.96 g/30mL
Geldental; oral6.4 g/32g
Geldental; oral; periodontal200 mg/g
Geloral.2 mL/mL
Geloral10 g/100g
Geloral20 g/100g
Geloral200 mg/g
Geloral200 mg/mL
Geloral75 mg/g
Geloral9 mg/mL
Geltopical.1 g/g
Geltopical.2 g/g
Geltopical.4; 200; 1 mg/g; mg/g; mg/g
Geltopical10 g/100g
Geltopical100 mg/g
Geltopical2.13 g/28.35g
Geltopical20 g/100g
Geltopical200 mg/g
Geltopical3 g/100mL
Geltopical5 g/100mL
Geltopical7.5 g/100g
Geltopical75 mg/g
Gel, dentifricedental10 g/100g
Gel, dentifricedental20 g/100g
Gel, dentifriceoral.02; 20; .1 g/100g; g/100g; g/100g
Gel, dentifriceoral.04; 20; .1 g/100g; g/100g; g/100g
Gel, dentifriceoral20 g/100g
Gel, dentifriceoral7.5 g/100g
Granuleoral6 mg
Kit
Kittopical
Liquidbuccal200 mg/mL
Liquiddental20 g/100g
Liquiddental; oral; periodontal200 mg/g
Liquidoral1.3 mg/13mL
Liquidoral20 g/100g
Liquidoral200 mg/g
Liquidoral200 mg/mL
Liquidoral7.5 mg/100mg
Liquidoral7.5 mL/100mL
Liquidtopical.009 mg/mL
Liquidtopical.2 mg/2mL
Liquidtopical.2 mL/mL
Liquidtopical15 mg/mL
Liquidtopical2.1 mg/30mL
Liquidtopical200 mg/g
Liquidtopical200 mg/mL
Liquidtopical4 g/100mL
Liquidtopical6 g/100g
Lozengeoral15 mg
Lozengeoral3 mg
Lozengeoral4 mg
Ointmenttopical20 g/100g
Ointmenttopical3.5 g/100g
Ointmenttopical5 mg/g
Ointmenttopical5.6 g/28g
Paste, dentifricetopical.02 g/g
Paste, dentifricetopical20 g/100g
Solutiontopical100 mg/mL
Solutiontopical150 mg/mL
Solutiontopical200 mg/mL
Spraydental; oral; periodontal200 mg/g
Spraytopical20 mL/100mL
Spray, metereddental11.4 g/57g
Stripdental10 mg
Swabtopical.06 mg
Swabtopical.06 mL/mL
Swabtopical.06; .6 mL/mL; mL/mL
Swabtopical.06; .7 mL/1; mL
Swabtopical.075 mL/mL
Swabtopical.12 mL
Swabtopical.2 mL/mL
Swabtopical60 mg/mL
Swabtopical60; .6 mg/mL; mL/mL
Tablet, orally disintegratingoral6 mg
Prices
Unit descriptionCostUnit
Americaine Anesthetic 20% Gel 28 gm Tube22.99USD tube
Americaine 20% ear drops1.26USD ml
Oticaine 20% ear drops0.83USD ml
Americaine lubricant0.71USD g
Hurricaine 20% liquid swab0.6USD swab
Hurricaine 20% spray0.52USD ml
Anbesol baby 7.5% gel0.41USD g
Cepacol 6 mg fizzlers tablet0.39USD tablet
Benzocaine powder0.09USD g
Dermoplast pain relieving spry0.07USD ml
Dermoplast spray0.07USD ml
DrugBank does not sell nor buy drugs. Pricing information is supplied for informational purposes only.
PatentsNot Available
Properties
StateSolid
Experimental Properties
PropertyValueSource
melting point92 °CPhysProp
boiling point310 °CPhysProp
water solubility1310 mg/L (at 30 °C)YALKOWSKY,SH & HE,Y (2003)
logP1.86HANSCH,C ET AL. (1995)
pKa2.51 (at 25 °C)PERRIN,DD (1965)
Predicted Properties
PropertyValueSource
Water Solubility2.85 mg/mLALOGPS
logP2.2ALOGPS
logP1.5ChemAxon
logS-1.8ALOGPS
pKa (Strongest Basic)2.78ChemAxon
Physiological Charge0ChemAxon
Hydrogen Acceptor Count2ChemAxon
Hydrogen Donor Count1ChemAxon
Polar Surface Area52.32 Å2ChemAxon
Rotatable Bond Count3ChemAxon
Refractivity47.53 m3·mol-1ChemAxon
Polarizability17.46 Å3ChemAxon
Number of Rings1ChemAxon
Bioavailability1ChemAxon
Rule of FiveYesChemAxon
Ghose FilterYesChemAxon
Veber's RuleYesChemAxon
MDDR-like RuleYesChemAxon
Spectra
Mass Spec (NIST)Download (7.74 KB)
SpectraGC-MSMS/MSLC-MSMS1D NMR2D NMR
References
Synthesis ReferenceNot Available
General ReferenceNot Available
External Links
ATC CodesC05AD03D04AB04N01BA05R02AD01
AHFS Codes
  • 52:16.00
  • 84:08.00
PDB EntriesNot Available
FDA labelNot Available
MSDSDownload (73.3 KB)
Interactions
Drug Interactions
Drug
Nitric OxideMay enhance the adverse/toxic effect of Methemoglobinemia Associated Agents. Combinations of these agents may increase the likelihood of significant methemoglobinemia.
PrilocaineMethemoglobinemia Associated Agents may enhance the adverse/toxic effect of Prilocaine. Combinations of these agents may increase the likelihood of significant methemoglobinemia.
Food InteractionsNot Available

Targets

1. Sodium channel protein type 10 subunit alpha

Kind: protein

Organism: Human

Pharmacological action: yes

Actions: inhibitor

Components

Name UniProt ID Details
Sodium channel protein type 10 subunit alpha Q9Y5Y9 Details

References:

  1. Overington JP, Al-Lazikani B, Hopkins AL: How many drug targets are there? Nat Rev Drug Discov. 2006 Dec;5(12):993-6. Pubmed
  2. Imming P, Sinning C, Meyer A: Drugs, their targets and the nature and number of drug targets. Nat Rev Drug Discov. 2006 Oct;5(10):821-34. Pubmed
  3. Ahern CA, Eastwood AL, Dougherty DA, Horn R: Electrostatic contributions of aromatic residues in the local anesthetic receptor of voltage-gated sodium channels. Circ Res. 2008 Jan 4;102(1):86-94. Epub 2007 Oct 25. Pubmed
  4. Hanck DA, Nikitina E, McNulty MM, Fozzard HA, Lipkind GM, Sheets MF: Using lidocaine and benzocaine to link sodium channel molecular conformations to state-dependent antiarrhythmic drug affinity. Circ Res. 2009 Aug 28;105(5):492-9. Epub 2009 Aug 6. Pubmed
  5. Lipkind GM, Fozzard HA: Molecular modeling of local anesthetic drug binding by voltage-gated sodium channels. Mol Pharmacol. 2005 Dec;68(6):1611-22. Epub 2005 Sep 20. Pubmed

Enzymes

1. Liver carboxylesterase 1

Kind: protein

Organism: Human

Pharmacological action: unknown

Actions: inhibitor

Components

Name UniProt ID Details
Liver carboxylesterase 1 P23141 Details

References:

  1. Bell FP: The effect of local anesthetics on arterial lipid metabolism. Inhibition of sterol esterification in vitro. Atherosclerosis. 1981 Jan-Feb;38(1-2):81-8. Pubmed

Transporters

1. Multidrug resistance protein 1

Kind: protein

Organism: Human

Pharmacological action: unknown

Actions: inhibitor

Components

Name UniProt ID Details
Multidrug resistance protein 1 P08183 Details

References:

  1. Nagy H, Goda K, Fenyvesi F, Bacso Z, Szilasi M, Kappelmayer J, Lustyik G, Cianfriglia M, Szabo G Jr: Distinct groups of multidrug resistance modulating agents are distinguished by competition of P-glycoprotein-specific antibodies. Biochem Biophys Res Commun. 2004 Mar 19;315(4):942-9. Pubmed

Comments
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Drug created on June 13, 2005 07:24 / Updated on September 16, 2013 17:13