Dopamine Agents

Name
Dopamine Agents
Accession Number
DBCAT000436  (DBCAT002741)
Description

Any drugs that are used for their effects on dopamine receptors, on the life cycle of dopamine, or on the survival of dopaminergic neurons.

ATC Classification
Drugs
DrugDrug Description
RopiniroleA non-ergoline dopamine agonist used to treat the symptoms of Parkinson's disease and Restless Legs Syndrome.
PramipexoleA non-ergot dopamine agonist used to treat the signs and symptoms of idiopathic Parkinson's disease and Restless Legs Syndrome (RLS).
ApomorphineA morphine derivative D2 dopamine agonist used to treat hypomobile "off" episodes of advanced Parkinson's disease.
AmantadineA medication used to treat dyskinesia in Parkinson's patients receiving levodopa, as well as extrapyramidal side effects of medications.
PergolideA long-acting dopamine agonist that is uncommonly used for the management of Parkinson's disease, due to the risk for cardiac valvulopathy.
BromocriptineA dopamine D2 receptor agonist used for the treatment of galactorrhea due to hyperprolactinemia and other prolactin-related conditions, as well as in early Parkinsonian Syndrome.
LevodopaA dopamine precursor used in the management of Parkinson's disease, often in combination with carbidopa, as well as other conditions associated with parkinsonism.
RotigotineA non-selective dopamine agonist used for the treatment of Parkinson's Disease and Restless Leg Syndrome.
PiribedilA dopamine agonist used with or without levodopa in the treatment of Parkinson's disease.
DihydroergocryptineA dopamine agonist indicated in the treatment of cerebrovascular diseases and atherosclerosis.
AmphetamineA CNS stimulant and sympathomimetic agent indicated for the treatment of Attention Deficit Hyperactivity Disorder (ADHD).
BenzatropineAn anticholinergic drug used to treat Parkinson's disease (PD) and extrapyramidal symptoms, except tardive dyskinesia.
ZiprasidoneAn atypical antipsychotic used to manage schizophrenia, bipolar mania, and agitation in patients with schizophrenia.
CabergolineA dopamine receptor agonist used for the treatment of hyperprolactinemic conditions due to various causes.
DihydroergotamineAn ergot alkaloid used in the acute treatment of migraine headache and cluster headache.
ThiethylperazineA drug used for the treatment of nausea and vomiting.
SulpirideA selective D2 dopamine receptor antagonist indicated to treat chronic and acute schizophrenia.
LoxapineA antipsychotic used for the treatment of schizophrenia.
RemoxiprideAn discontinued atypical antipsychotic selective for dopamine D2 receptors.
PromazineA phenothiazine used to manage schizophrenia.
MethylphenidateA stimulant used in the management of Attention Deficit Hyperactivity Disorder (ADHD).
ProchlorperazineA phenothiazine derivative used in the treatment of schizophrenia and anxiety and to relieve severe nausea and vomiting.
DroperidolA butyrophenone derivative and dopamine antagonist used to prevent and treat postoperative nausea and vomiting.
ChlorpromazineA phenothiazine antipsychotic used to treat nausea, vomiting, preoperative anxiety, schizophrenia, bipolar disorder, and severe behavioral problems in children.
HaloperidolAn antipsychotic agent used to treat schizophrenia and other psychoses, as well as symptoms of agitation, irritability, and delirium.
TriflupromazineUsed mainly in the management of psychoses. Also used to control nausea and vomiting.
AmoxapineA tricyclic antidepressant used in the treatment of neurotic or reactive depressive disorders and endogenous or psychotic depression.
MazindolA sympathomimetic used to treat obesity in combination with lifestyle modifications.
LisurideFor the management of Parkinson's Disease
FluphenazineA phenothiazine used to treat patients requiring long-term neuroleptic therapy.
ThioridazineA phenothiazine antipsychotic used to treat schizophrenia and generalized anxiety disorder.
RisperidoneA second-generation antipsychotic medication used to treat a number of mental health disorders including schizophrenia, bipolar mania, psychosis, or as an adjunct in severe depression.
FenoldopamA dopamine D1 receptor agonist used for the short term management of hypertension.
TrifluoperazineA phenothiazine used to treat depression, anxiety, and agitation.
PerphenazineA phenothiazine used to treat schizophrenia as well as nausea and vomiting.
BenzphetamineA sympathomimetic used to manage exogenous obesity short term.
FlupentixolA thioxanthene neuroleptic used to treat schizophrenia and depression.
CocaineAn ester local anesthetic used during diagnostic procedures and surgeries in or through the nasal cavities.
MesoridazineA phenothiazine antipsychotic used to treat schizophrenia, organic brain disorders, alcoholism, and psychoneuroses.
DopamineA catecholamine neurotransmitter used to treat hemodynamic imbalances, poor perfusion of vital organs, low cardiac output, and hypotension.
MemantineAn NMDA receptor antagonist used to treat moderate to severe dementia in Alzheimer's.
Ergoloid mesylateA nootropic with an unknown mechanism of action indicated in individuals over sixty who manifest signs and symptoms of an idiopathic decline in mental capacity.
PimozideAn antipsychotic used to manage debilitating motor and phonic tics in patients with Tourette's Disorder.
BupropionA norepinephrine and dopamine reuptake inhibitor used in the treatment of major depressive disorder (MDD), seasonal affective disorder (SAD), and as an aid to smoking cessation.
DomperidoneA dopamine receptor antagonist used as a peristaltic stimulant and anti-emetic agent for dyspepsia, indigestion, epigastric pain, nausea, and vomiting.
MetoclopramideAn antiemetic agent and dopamine D2 antagonist used in the treatment of gastroesophageal reflux disease, prevention of nausea and vomiting, and to stimulate gastric emptying.
ChlorprothixeneA thioxanthene antipsychotic.
LisdexamfetamineA central nervous system (CNS) stimulant used to treat attention deficit hyperactivity disorder (ADHD) and moderate to severe eating disorders.
PaliperidoneAn atypical antipsychotic used in the treatment of schizophrenia and other schizoaffective or delusional disorders.
MethotrimeprazineA phenothiazine used in the management of psychosis, particular those of schizophrenia, and manic phases of bipolar disorder.
DextroamphetamineA sympathomimetic agent used in the treatment of attention deficit hyperactivity disorder (ADHD) and narcolepsy.
MetamfetamineA sympathomimetic agent used in the treatment of attention deficit hyperactivity disorder (ADHD) and exogenous obesity.
ThiothixeneAn antipsychotic indicated for the management of schizophrenia.
ZuclopenthixolAn antipsychotic indicated for the management of schizophrenia. The acuphase formulation is indicated for initial treatment of acute psychosis or exacerbation of psychosis, while the depot formulation is best for maintenance.
NomifensineNomifensine, formerly marketed as Merital capsules, was associated with an increased incidence of hemolytic anemia. The approved application holder removed Merital capsules from the market on January 23, 1986. FDA...
FluspirileneAn antipsychotic agent used in the treatment of schizophrenia.
AmisulprideA dopamine D2 receptor antagonist used in the treatment of acute and chronic schizophrenia, and in the prevention and treatment of postoperative nausea and vomiting in adults.
DexmethylphenidateA norepinephrine-dopamine reuptake inhibitor used in the treatment of ADHD in conjunction with other therapies.
LurasidoneAn atypical antipsychotic used to treat schizophrenia and depressive episodes associated with bipolar I disorder.
QuinagolideA dopamine D2 receptor agonist used for the treatment of hyperprolactinemia.
BrexpiprazoleA serotonin–dopamine activity modulator used in the treatment of major depressive disorder as an adjunct, schizophrenia, and agitation associated with dementia due to Alzheimer’s disease.
DopexamineDopexamine has been used in trials studying the diagnostic and treatment of Free Flap, Oral Cancer, Hypotension, Septic Shock, and Head and Neck Cancer.
PerazineA phenothiazine antipsychotic used in the acute and chronic treatment of psychotic disorders.
BenserazideA medication used to treat Parkinson's disease, parkinsonism, and restless leg syndrome.
BenperidolA neuroleptic butyrophenone derivative indicated in the treatment of psychoses, manic episodes, and psychomotor agitation.
MetergolineAn ergot-derivative that acts as an antagonist at certain 5-HT receptor subtypes and as an agonist at dopamine receptors. It is often used in situations where inhibition of prolactin is desirable.
TolcaponeA catechol-O-methyltransferase (COMT) inhibitor used as adjunct therapy in the symptomatic management of idiopathic Parkinson's disease.
EntacaponeA selective reversible catechol-O-methyltransferase inhibitor for the treatment of Parkinson's disease.
SelegilineA monoamine oxidase inhibitor used to treat major depressive disorder and Parkinson's.
RasagilineAn irreversible inhibitor of monoamine oxidase used for the symptomatic management of idiopathic Parkinson's disease as initial monotherapy and as adjunct therapy to levodopa.
EtilevodopaInvestigated for use/treatment in parkinson's disease.
MelevodopaA methyl ester of levodopa indicated in combination with carbidopa for the treatment of Parkinson's disease.
BudipineNot Annotated
SafinamideA MAO-B inhibitor used as an add-on treatment to levodopa/carbidopa for Parkinson's disease during "off" episodes.
OpicaponeA catechol-O-methyltransferase inhibitor used as an adjunct treatment for Parkinson's Disease in adults currently receiving levodopa and a dopa decarboxylase inhibitor.
SolriamfetolSolriamfetol is indicated for treatment of daytime sleepiness associated with obstructive sleep apnea and narcolepsy, but is not a treatment for the underlying airway obstruction in apnea patients[FDA Label][A176534,A176744].
AripiprazoleAn atypical antipsychotic used in the treatment of a wide variety of mood and psychotic disorders, such as schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's syndrome.
EticloprideNot Annotated
SerdexmethylphenidateA prodrug of the CNS stimulant dexmethylphenidate used as a first-line treatment for Attention Deficit Hyperactivity Disorder (ADHD).
AcepromazineAcepromazine was first used in humans in the 1950s as an antipsychotic agent. It is now rarely used in humans. Acepromazine is frequently used in animals as a sedative and...
AceprometazineAceprometazine is often used in combination with meprobamate for the treatment of sleep disorders.
VanoxerineAn investigational dopamine transporter antagonist suggested to be beneficial in the treatment of cocaine addiction.
YKP-1358Investigated for use/treatment in schizophrenia and schizoaffective disorders.
BromoprideA substituted benzamide, closely related to metoclopramide, used as an antiemetic.
AS-8112AS-8112 is a synthetic compound that acts as a selective antagonist at the dopamine receptor subtypes D2 and D3, and the serotonin receptor 5-HT3. It has been shown to exert...
DihydroergocornineA nootropic with an unknown mechanism of action indicated in individuals over sixty who manifest signs and symptoms of an idiopathic decline in mental capacity.
AzaperoneAzaperone is a pyridinylpiperazine and butyrophenone agent that is capable of eliciting neuroleptic sedative and antiemetic effects. It is subsequently employed predominantly as a veterinary tranquilizer and mainly for pigs...
TetrahydropalmatineTetrahydropalmatine is under investigation in clinical trial NCT02118610 (Treatment of Schizophrenia With L-tetrahydropalmatine (l-THP): a Novel Dopamine Antagonist With Anti-inflammatory and Antiprotozoal Activity).
EcopipamEcopipam has been used in trials studying the treatment of Tourette's Syndrome, Lesch-Nyhan Disease, Pathological Gambling, and Self-injurious Behavior.
RacloprideRaclopride has been used in trials studying Parkinson Disease.
JNJ-37822681JNJ-37822681 has been used in trials studying the treatment of Schizophrenia.
DihydrexidineDihydrexidine has been used in trials studying the treatment of SPD, Cocaine-Related Disorders, and Schizotypal Personality Disorder.
TiaprideA dopamine D2 and D3 receptor antagonist indicated in the treatment of chorea in Huntington's disease, as well as agitation and anxiety in the elderly or with acute or chronic alcoholism.
SultoprideSultopride is used in Japan, Hong Kong, and Europe to treat schizophrenia. It is of the drug class atypical antipsychotics .
IbopamineA sympathomimetic, indicated in the induction of mydriasis and treatment of pos-surgical ocular hypotonia.
TergurideNot Annotated
TrifluperidolNot Annotated
PenfluridolNot Annotated
ClopenthixolClopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
DexpramipexoleDexpramipexole is under investigation in clinical trial NCT01511029 (Study to Evaluate the QTC Interval in Healthy Volunteers Dosed With Dexpramipexole (QTC = Electrocardiogram (ECG) Interval Measured From the Onset of...
FallyprideFallypride is under investigation in clinical trial NCT02310360 (Striatal and Extra-striatal Dopamine Release in Response to Food in Healthy Humans).
DAR-0100ADAR-0100A is under investigation in clinical trial NCT01466205 (Clinical Testing of a D1 Agonist for Cognitive Enhancement in Schizotypal Personality Disorder).
DihydroergotoxineNot Annotated
GBR-12783A selective inhibitor of dopamine uptake.
SpiperoneSpiperone is a dopamine antagonist that binds dopamine and serotonin receptors.
MesdopetamMesdopetam is under investigation in clinical trial NCT04435431 (A Clinical Study of Mesdopetam in Patients With Parkinson's Disease Experiencing Levodopa Induced Dyskinesia).
FoslevodopaFoslevodopa is under investigation in clinical trial NCT04750226 (Study to Assess Adverse Events and Change in Disease Activity of 24-hour Continuous Subcutaneous Infusion of ABBV-951 in Adult Participants With Advanced...
DocarpamineNot Available
Drugs & Drug Targets
DrugTargetType
RopiniroleDopamine D2 receptortarget
RopiniroleDopamine D3 receptortarget
RopiniroleDopamine D4 receptortarget
RopiniroleCytochrome P450 1A2enzyme
RopiniroleAlpha adrenergic receptortarget
PramipexoleDopamine D3 receptortarget
PramipexoleDopamine D4 receptortarget
PramipexoleDopamine D2 receptortarget
Pramipexole5-hydroxytryptamine receptor 1Atarget
PramipexoleAlpha-2A adrenergic receptortarget
PramipexoleSolute carrier family 22 member 2transporter
PramipexoleSolute carrier family 22 member 1transporter
PramipexoleSolute carrier family 22 member 3transporter
ApomorphineDopamine D2 receptortarget
ApomorphineDopamine D1 receptortarget
ApomorphineDopamine D4 receptortarget
ApomorphineDopamine D3 receptortarget
ApomorphineDopamine D5 receptortarget
ApomorphineAlpha-2C adrenergic receptortarget
ApomorphineAlpha-2B adrenergic receptortarget
Apomorphine5-hydroxytryptamine receptor 2Ctarget
Apomorphine5-hydroxytryptamine receptor 1Atarget
Apomorphine5-hydroxytryptamine receptor 2Atarget
Apomorphine5-hydroxytryptamine receptor 2Btarget
ApomorphineAlpha-2A adrenergic receptortarget
Apomorphine5-hydroxytryptamine receptor 1Dtarget
Apomorphine5-hydroxytryptamine receptor 1Btarget
ApomorphineCatechol O-methyltransferaseenzyme
ApomorphineSulfotransferase 1A1enzyme
ApomorphineSulfotransferase 1A2enzyme
ApomorphineSulfotransferase 1A3/1A4enzyme
ApomorphineEstrogen sulfotransferaseenzyme
ApomorphineSulfotransferase family cytosolic 1B member 1enzyme
ApomorphineCytochrome P450 2B6enzyme
ApomorphineCytochrome P450 2C8enzyme
ApomorphineCytochrome P450 3A4enzyme
ApomorphineCytochrome P450 3A5enzyme
ApomorphineUDP-glucuronosyltransferases (UGTs)enzyme
ApomorphineSerum albumincarrier
ApomorphineSynaptic vesicular amine transportertransporter
AmantadineDopamine D2 receptortarget
AmantadineMatrix protein 2target
AmantadineAromatic-L-amino-acid decarboxylaseenzyme
AmantadineAmine oxidase [flavin-containing] Benzyme
AmantadineSolute carrier family 22 member 2transporter
AmantadineSolute carrier family 22 member 1transporter
AmantadineGlutamate receptor ionotropic, NMDA 3Atarget
AmantadineNeuronal acetylcholine receptor subunit alpha-7target
AmantadineNeuronal acetylcholine receptor subunit alpha-4target
AmantadineNeuronal acetylcholine receptor subunit alpha-3target
PergolideDopamine D2 receptortarget
PergolideDopamine D1 receptortarget
PergolideDopamine D3 receptortarget
Pergolide5-hydroxytryptamine receptor 1Atarget
PergolideAlpha-1A adrenergic receptortarget
PergolideAlpha-2 adrenergic receptorstarget
PergolideAlpha-1B adrenergic receptortarget
PergolideAlpha-1D adrenergic receptortarget
PergolideDopamine D4 receptortarget
PergolideDopamine D5 receptortarget
Pergolide5-hydroxytryptamine receptor 1Btarget
Pergolide5-hydroxytryptamine receptor 1Dtarget
Pergolide5-hydroxytryptamine receptor 2Atarget
Pergolide5-hydroxytryptamine receptor 2Btarget
Pergolide5-hydroxytryptamine receptor 2Ctarget
PergolideCytochrome P450 3A4enzyme
BromocriptineDopamine D2 receptortarget
BromocriptineCytochrome P450 3A4enzyme
Bromocriptine5-hydroxytryptamine receptor 1Dtarget
BromocriptineAlpha-2A adrenergic receptortarget
BromocriptineDopamine D3 receptortarget
Bromocriptine5-hydroxytryptamine receptor 1Atarget
BromocriptineAlpha-2C adrenergic receptortarget
BromocriptineAlpha-2B adrenergic receptortarget
Bromocriptine5-hydroxytryptamine receptor 2Btarget
BromocriptineDopamine D4 receptortarget
Bromocriptine5-hydroxytryptamine receptor 2Atarget
Bromocriptine5-hydroxytryptamine receptor 1Btarget
Bromocriptine5-hydroxytryptamine receptor 2Ctarget
BromocriptineDopamine D5 receptortarget
BromocriptineDopamine D1 receptortarget
BromocriptineAlpha-1A adrenergic receptortarget
BromocriptineAlpha-1B adrenergic receptortarget
BromocriptineAlpha-1D adrenergic receptortarget
Bromocriptine5-hydroxytryptamine receptor 7target
BromocriptineP-glycoprotein 1transporter
LevodopaDopamine D1 receptortarget
LevodopaDopamine D2 receptortarget
LevodopaAromatic-L-amino-acid decarboxylaseenzyme
LevodopaSolute carrier family 15 member 1transporter
LevodopaMonocarboxylate transporter 10transporter
LevodopaDopamine D3 receptortarget
LevodopaDopamine D4 receptortarget
LevodopaDopamine D5 receptortarget
LevodopaLarge neutral amino acids transporter small subunit 1transporter
LevodopaLarge neutral amino acids transporter small subunit 2transporter
LevodopaSerum albumincarrier
RotigotineDopamine D3 receptortarget
RotigotineDopamine D5 receptortarget
RotigotineDopamine D4 receptortarget
RotigotineDopamine D2 receptortarget
Rotigotine5-hydroxytryptamine receptor 1Atarget
RotigotineDopamine D1 receptortarget
RotigotineCytochrome P450 2D6enzyme
RotigotineCytochrome P450 3A4enzyme
RotigotineAlpha-2B adrenergic receptortarget
RotigotineCytochrome P450 2C19enzyme
PiribedilDopamine D2 receptortarget
PiribedilDopamine D3 receptortarget
DihydroergocryptineCytochrome P450 3A4enzyme
AmphetamineSodium-dependent dopamine transportertarget
AmphetamineCocaine- and amphetamine-regulated transcript proteintarget
AmphetamineTrace amine-associated receptor 1target
AmphetamineCytochrome P450 2D6enzyme
AmphetamineSolute carrier family 22 member 3transporter
AmphetamineSolute carrier family 22 member 5transporter
AmphetamineSynaptic vesicular amine transportertarget
AmphetamineCytochrome P450 2A6enzyme
AmphetamineSodium-dependent noradrenaline transportertarget
AmphetamineAlpha adrenergic receptortarget
AmphetamineBeta adrenergic receptortarget
AmphetamineDopamine D2 receptortarget
AmphetamineAmine oxidase [flavin-containing] Btarget
AmphetamineSodium-dependent serotonin transportertarget
AmphetamineMonoamine oxidasetarget
BenzatropineMuscarinic acetylcholine receptor M1target
BenzatropineSodium-dependent dopamine transportertarget
BenzatropineHistamine H1 receptortarget
BenzatropineSerum albumincarrier
BenzatropineSodium-dependent serotonin transportertarget
BenzatropineSodium-dependent noradrenaline transportertarget
ZiprasidoneAlpha-1A adrenergic receptortarget
ZiprasidoneDopamine D2 receptortarget
Ziprasidone5-hydroxytryptamine receptor 2Ctarget
ZiprasidoneDopamine D3 receptortarget
Ziprasidone5-hydroxytryptamine receptor 1Atarget
Ziprasidone5-hydroxytryptamine receptor 1Dtarget
ZiprasidoneHistamine H1 receptortarget
Ziprasidone5-hydroxytryptamine receptor 2Atarget
ZiprasidoneDopamine D4 receptortarget
Ziprasidone5-hydroxytryptamine receptor 7target
ZiprasidoneCytochrome P450 3A4enzyme
ZiprasidoneAlpha-2A adrenergic receptortarget
ZiprasidoneAlpha-1B adrenergic receptortarget
ZiprasidoneAlpha-2B adrenergic receptortarget
ZiprasidoneAlpha-2C adrenergic receptortarget
ZiprasidoneDopamine D1 receptortarget
ZiprasidoneDopamine D5 receptortarget
ZiprasidoneMuscarinic acetylcholine receptor M1target
ZiprasidoneMuscarinic acetylcholine receptor M2target
ZiprasidoneMuscarinic acetylcholine receptor M3target
ZiprasidoneMuscarinic acetylcholine receptor M4target
ZiprasidoneMuscarinic acetylcholine receptor M5target
Ziprasidone5-hydroxytryptamine receptor 1Btarget
Ziprasidone5-hydroxytryptamine receptor 1Etarget
Ziprasidone5-hydroxytryptamine receptor 6target
ZiprasidoneAldehyde oxidaseenzyme
ZiprasidoneSerum albumincarrier
ZiprasidoneP-glycoprotein 1transporter
ZiprasidoneAlpha-1-acid glycoprotein 1carrier
Ziprasidone5-hydroxytryptamine 3 receptortarget
Ziprasidone5-hydroxytryptamine receptor 5Atarget
CabergolineDopamine D2 receptortarget
Cabergoline5-hydroxytryptamine receptor 2Btarget
CabergolineDopamine D3 receptortarget
Cabergoline5-hydroxytryptamine receptor 2Atarget
CabergolineAlpha-2B adrenergic receptortarget
Cabergoline5-hydroxytryptamine receptor 1Dtarget
CabergolineDopamine D4 receptortarget
CabergolineAlpha-2A adrenergic receptortarget
Cabergoline5-hydroxytryptamine receptor 1Atarget
CabergolineAlpha-2C adrenergic receptortarget
CabergolineDopamine D5 receptortarget
CabergolineDopamine D1 receptortarget
Cabergoline5-hydroxytryptamine receptor 1Btarget
Cabergoline5-hydroxytryptamine receptor 2Ctarget
CabergolineCytochrome P450 3A4enzyme
Cabergoline5-hydroxytryptamine receptor 7target
CabergolineAlpha-1A adrenergic receptortarget
CabergolineAlpha-1B adrenergic receptortarget
CabergolineAlpha-1D adrenergic receptortarget
CabergolineBeta-1 adrenergic receptortarget
CabergolineBeta-2 adrenergic receptortarget
CabergolineD(1) dopamine receptortarget
CabergolineP-glycoprotein 1transporter
Dihydroergotamine5-hydroxytryptamine receptor 1Dtarget
Dihydroergotamine5-hydroxytryptamine receptor 1Btarget
DihydroergotamineCytochrome P450 3A4enzyme
DihydroergotamineAlpha-2A adrenergic receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 2Btarget
DihydroergotamineP-glycoprotein 1transporter
Dihydroergotamine5-hydroxytryptamine receptor 1Atarget
Dihydroergotamine5-hydroxytryptamine receptor 1Etarget
Dihydroergotamine5-hydroxytryptamine receptor 2Atarget
Dihydroergotamine5-hydroxytryptamine receptor 2Ctarget
DihydroergotamineAlpha-1 adrenergic receptorstarget
DihydroergotamineAlpha-2 adrenergic receptorstarget
DihydroergotamineDopamine D2 receptortarget
DihydroergotamineDopamine D3 receptortarget
DihydroergotamineDopamine D4 receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 1Ftarget
Dihydroergotamine5-hydroxytryptamine receptor 4target
DihydroergotamineBeta-3 adrenergic receptortarget
ThiethylperazineDopamine D2 receptortarget
SulpirideDopamine D2 receptortarget
SulpirideDopamine D3 receptortarget
SulpirideCholinesteraseenzyme
SulpirideCarbonic anhydrase 2target
SulpirideCarbonic anhydrase 3target
SulpirideSerum albumincarrier
SulpirideSolute carrier family 22 member 1transporter
SulpirideSolute carrier family 22 member 2transporter
SulpirideMultidrug and toxin extrusion protein 1transporter
SulpirideMultidrug and toxin extrusion protein 2transporter
SulpirideDopamine D4 receptortarget
SulpirideSolute carrier family 22 member 3transporter
SulpirideP-glycoprotein 1transporter
SulpirideATP-binding cassette sub-family G member 2transporter
LoxapineDopamine D1 receptortarget
LoxapineDopamine D2 receptortarget
Loxapine5-hydroxytryptamine receptor 2Atarget
Loxapine5-hydroxytryptamine receptor 2Ctarget
Loxapine5-hydroxytryptamine receptor 1Atarget
Loxapine5-hydroxytryptamine receptor 1Btarget
Loxapine5-hydroxytryptamine receptor 1Dtarget
Loxapine5-hydroxytryptamine receptor 1Etarget
Loxapine5-hydroxytryptamine receptor 3Atarget
Loxapine5-hydroxytryptamine receptor 5Atarget
Loxapine5-hydroxytryptamine receptor 6target
Loxapine5-hydroxytryptamine receptor 7target
LoxapineAlpha-1A adrenergic receptortarget
LoxapineAlpha-1B adrenergic receptortarget
LoxapineAlpha-2A adrenergic receptortarget
LoxapineAlpha-2B adrenergic receptortarget
LoxapineAlpha-2C adrenergic receptortarget
LoxapineBeta-1 adrenergic receptortarget
LoxapineMuscarinic acetylcholine receptor M1target
LoxapineMuscarinic acetylcholine receptor M2target
LoxapineMuscarinic acetylcholine receptor M3target
LoxapineMuscarinic acetylcholine receptor M4target
LoxapineMuscarinic acetylcholine receptor M5target
LoxapineD(1) dopamine receptortarget
LoxapineDopamine D3 receptortarget
LoxapineDopamine D4 receptortarget
LoxapineDopamine D5 receptortarget
LoxapineHistamine H1 receptortarget
LoxapineHistamine H2 receptortarget
LoxapineHistamine H4 receptortarget
LoxapineSodium-dependent serotonin transportertarget
LoxapineSodium-dependent noradrenaline transportertarget
LoxapineSodium-dependent dopamine transportertarget
RemoxiprideDopamine D2 receptortarget
RemoxiprideDopamine D4 receptortarget
Remoxipride5-hydroxytryptamine receptor 2Atarget
RemoxiprideSigma non-opioid intracellular receptor 1target
RemoxiprideDopamine D3 receptortarget
RemoxiprideCytochrome P450 2D6enzyme
Remoxipridealpha1-acid glycoproteincarrier
RemoxiprideCytochrome P450 1A2enzyme
RemoxiprideCytochrome P450 2B1enzyme
RemoxiprideCytochrome P450 3A Subfamilyenzyme
PromazineDopamine D2 receptortarget
Promazine5-hydroxytryptamine receptor 2Atarget
Promazine5-hydroxytryptamine receptor 2Ctarget
PromazineAlpha-1A adrenergic receptortarget
PromazineMuscarinic acetylcholine receptor M1target
PromazineHistamine H1 receptortarget
PromazineCytochrome P450 2C19enzyme
PromazineCytochrome P450 1A2enzyme
PromazineCytochrome P450 3A4enzyme
PromazineCytochrome P450 2C9enzyme
PromazineCytochrome P450 2D6enzyme
MethylphenidateSodium-dependent dopamine transportertarget
MethylphenidateSodium-dependent noradrenaline transportertarget
MethylphenidateCarboxylesteraseenzyme
Methylphenidate5-hydroxytryptamine receptor 1Atarget
ProchlorperazineDopamine D2 receptortarget
ProchlorperazineCytochrome P450 2D6enzyme
ProchlorperazineHistamine H1 receptortarget
ProchlorperazineAlpha-1 adrenergic receptorstarget
ProchlorperazineAlpha-2 adrenergic receptorstarget
DroperidolDopamine D2 receptortarget
DroperidolAlpha-1A adrenergic receptortarget
ChlorpromazineDopamine D2 receptortarget
Chlorpromazine5-hydroxytryptamine receptor 2Atarget
ChlorpromazineCytochrome P450 2D6enzyme
ChlorpromazineCholinesteraseenzyme
ChlorpromazineCytochrome P450 1A2enzyme
ChlorpromazineSerum albumincarrier
ChlorpromazineP-glycoprotein 1transporter
ChlorpromazineDopamine D1 receptortarget
Chlorpromazine5-hydroxytryptamine receptor 1Atarget
ChlorpromazineAlpha-1A adrenergic receptortarget
ChlorpromazineAlpha-1B adrenergic receptortarget
ChlorpromazineCytochrome P450 2E1enzyme
ChlorpromazineCytochrome P450 3A4enzyme
ChlorpromazineHistamine H1 receptortarget
ChlorpromazinePotassium voltage-gated channel subfamily H member 2target
ChlorpromazineD(1) dopamine receptortarget
ChlorpromazineDopamine D3 receptortarget
ChlorpromazineDopamine D4 receptortarget
ChlorpromazineDopamine D5 receptortarget
Chlorpromazine5-hydroxytryptamine receptor 2Ctarget
Chlorpromazine5-hydroxytryptamine 2 receptortarget
ChlorpromazineAlpha-1 adrenergic receptorstarget
ChlorpromazineAlpha-2 adrenergic receptorstarget
ChlorpromazineMuscarinic acetylcholine receptor M1target
ChlorpromazineMuscarinic acetylcholine receptor M3target
ChlorpromazineSphingomyelin phosphodiesterasetarget
ChlorpromazineCalmodulintarget
Chlorpromazinealpha1-acid glycoproteintarget
Chlorpromazine5-hydroxytryptamine receptor 6target
Chlorpromazine5-hydroxytryptamine receptor 7target
ChlorpromazineHistamine H4 receptortarget
ChlorpromazineBile salt export pumptransporter
HaloperidolDopamine D2 receptortarget
HaloperidolGlutamate receptor ionotropic, NMDA 2Btarget
HaloperidolDopamine D1 receptortarget
HaloperidolCytochrome P450 1A2enzyme
HaloperidolCytochrome P450 2D6enzyme
Haloperidol5-hydroxytryptamine receptor 2Atarget
HaloperidolDopamine D3 receptortarget
HaloperidolCytochrome P450 3A4enzyme
HaloperidolCytochrome P450 3A5enzyme
HaloperidolCytochrome P450 3A7enzyme
HaloperidolP-glycoprotein 1transporter
HaloperidolCarbonyl reductase [NADPH] 1enzyme
HaloperidolUDP-glucuronosyltransferase 1-9enzyme
HaloperidolCytochrome P450 2C19enzyme
HaloperidolCytochrome P450 2C9enzyme
HaloperidolMelanin-concentrating hormone receptor 1target
HaloperidolSynaptic vesicular amine transportertarget
Haloperidol5-hydroxytryptamine receptor 2Ctarget
HaloperidolSigma non-opioid intracellular receptor 1target
HaloperidolHistamine H1 receptortarget
HaloperidolMuscarinic acetylcholine receptor M3target
HaloperidolAlpha-1A adrenergic receptortarget
HaloperidolAlpha-2A adrenergic receptortarget
HaloperidolAlpha-2B adrenergic receptortarget
HaloperidolAlpha-2C adrenergic receptortarget
Haloperidol5-hydroxytryptamine receptor 1Atarget
Haloperidol5-hydroxytryptamine receptor 6target
Haloperidol5-hydroxytryptamine receptor 7target
HaloperidolCytochrome P450 1A1enzyme
TriflupromazineDopamine D1 receptortarget
TriflupromazineDopamine D2 receptortarget
TriflupromazineMuscarinic acetylcholine receptor M1target
TriflupromazineMuscarinic acetylcholine receptor M2target
Triflupromazine5-hydroxytryptamine receptor 2Btarget
TriflupromazineP-glycoprotein 1transporter
TriflupromazineCholinesteraseenzyme
AmoxapineSodium-dependent serotonin transportertarget
AmoxapineSodium-dependent noradrenaline transportertarget
AmoxapineAlpha-2A adrenergic receptortarget
AmoxapineDopamine D2 receptortarget
AmoxapineAlpha-1A adrenergic receptortarget
AmoxapineDopamine D1 receptortarget
AmoxapineMuscarinic acetylcholine receptor M1target
AmoxapineGamma-aminobutyric acid receptor subunit alpha-1target
AmoxapineAlpha-1-acid glycoprotein 1carrier
AmoxapineCytochrome P450 2D6enzyme
Amoxapine5-hydroxytryptamine receptor 2Atarget
Amoxapine5-hydroxytryptamine receptor 2Ctarget
Amoxapine5-hydroxytryptamine receptor 6target
Amoxapine5-hydroxytryptamine receptor 7target
AmoxapineDopamine D3 receptortarget
AmoxapineDopamine D4 receptortarget
AmoxapineHistamine H1 receptortarget
AmoxapineAlpha-1 adrenergic receptorstarget
AmoxapineMuscarinic acetylcholine receptortarget
Amoxapine5-hydroxytryptamine receptor 2Btarget
Amoxapine5-hydroxytryptamine receptor 3Atarget
Amoxapine5-hydroxytryptamine receptor 1Atarget
Amoxapine5-hydroxytryptamine receptor 1Btarget
AmoxapineAlpha-2 adrenergic receptorstarget
AmoxapineHistamine H4 receptortarget
AmoxapineGABA(A) Receptortarget
AmoxapineSodium-dependent dopamine transportertarget
MazindolSodium-dependent noradrenaline transportertarget
MazindolSodium-dependent dopamine transportertarget
MazindolSodium-dependent serotonin transportertarget
MazindolSynaptic vesicular amine transportertarget
LisurideDopamine D1 receptortarget
Lisuride5-hydroxytryptamine receptor 1Atarget
LisurideDopamine D2 receptortarget
LisurideAlpha-2A adrenergic receptortarget
LisurideAlpha-2B adrenergic receptortarget
LisurideAlpha-2C adrenergic receptortarget
LisurideDopamine D3 receptortarget
Lisuride5-hydroxytryptamine receptor 1Dtarget
Lisuride5-hydroxytryptamine receptor 2Btarget
Lisuride5-hydroxytryptamine receptor 2Atarget
LisurideDopamine D4 receptortarget
Lisuride5-hydroxytryptamine receptor 2Ctarget
LisurideDopamine D5 receptortarget
Lisuride5-hydroxytryptamine receptor 1Btarget
LisurideCytochrome P450 3A4enzyme
Lisuride5-hydroxytryptamine receptor 7target
FluphenazineDopamine D2 receptortarget
FluphenazineCalmodulintarget
FluphenazineDopamine D1 receptortarget
FluphenazineCytochrome P450 2D6enzyme
FluphenazineP-glycoprotein 1transporter
FluphenazineCytochrome P450 2E1enzyme
FluphenazineAndrogen receptortarget
Fluphenazine5-hydroxytryptamine receptor 2Atarget
Fluphenazine5-hydroxytryptamine receptor 2Ctarget
ThioridazineAlpha-1A adrenergic receptortarget
ThioridazineDopamine D2 receptortarget
Thioridazine5-hydroxytryptamine receptor 2Atarget
ThioridazineDopamine D1 receptortarget
ThioridazineCytochrome P450 2C19enzyme
ThioridazineCytochrome P450 2D6enzyme
ThioridazineAlpha-1B adrenergic receptortarget
ThioridazinePotassium voltage-gated channel subfamily H member 2target
ThioridazineCytochrome P450 2E1enzyme
RisperidoneCytochrome P450 2D6enzyme
RisperidoneCytochrome P450 3A4enzyme
RisperidoneP-glycoprotein 1transporter
RisperidoneSerum albumincarrier
RisperidoneAlpha-1-acid glycoprotein 1carrier
Risperidone5-hydroxytryptamine receptor 2Atarget
RisperidoneDopamine D2 receptortarget
RisperidoneAlpha-1B adrenergic receptortarget
RisperidoneAlpha-2B adrenergic receptortarget
RisperidoneAlpha-1A adrenergic receptortarget
RisperidoneAlpha-2C adrenergic receptortarget
RisperidoneHistamine H1 receptortarget
Risperidone5-hydroxytryptamine receptor 2Ctarget
Risperidone5-hydroxytryptamine receptor 1Dtarget
Risperidone5-hydroxytryptamine receptor 1Atarget
Risperidone5-hydroxytryptamine receptor 7target
RisperidoneD(2L) dopamine receptortarget
RisperidoneDopamine D1 receptortarget
FenoldopamDopamine D5 receptortarget
FenoldopamDopamine D1 receptortarget
FenoldopamAlpha-2B adrenergic receptortarget
FenoldopamAlpha-2C adrenergic receptortarget
FenoldopamAlpha-2A adrenergic receptortarget
FenoldopamAlpha-1B adrenergic receptortarget
FenoldopamAlpha-1D adrenergic receptortarget
FenoldopamAlpha-1A adrenergic receptortarget
TrifluoperazineDopamine D2 receptortarget
TrifluoperazineAlpha-1A adrenergic receptortarget
TrifluoperazineNeuron-specific vesicular protein calcyontarget
TrifluoperazineXanthine dehydrogenase/oxidaseenzyme
TrifluoperazineUDP-glucuronosyltransferase 1-4enzyme
TrifluoperazineCytochrome P450 1A2enzyme
TrifluoperazineP-glycoprotein 1transporter
TrifluoperazineCalmodulintarget
TrifluoperazineTroponin C, slow skeletal and cardiac musclestarget
TrifluoperazineProtein S100-A4target
PerphenazineDopamine D1 receptortarget
PerphenazineDopamine D2 receptortarget
PerphenazineCalmodulintarget
PerphenazineCytochrome P450 2D6enzyme
PerphenazineCytochrome P450 1A2enzyme
PerphenazineCytochrome P450 2C18enzyme
PerphenazineCytochrome P450 2C19enzyme
PerphenazineCytochrome P450 2C8enzyme
PerphenazineCytochrome P450 2C9enzyme
PerphenazineCytochrome P450 3A4enzyme
PerphenazineSerum albumincarrier
BenzphetamineAlpha-2A adrenergic receptortarget
BenzphetamineAlpha-1A adrenergic receptortarget
BenzphetamineCytochrome P450 3A4enzyme
BenzphetamineCytochrome P450 2B6enzyme
BenzphetamineNADPH--cytochrome P450 reductaseenzyme
BenzphetamineSynaptic vesicular amine transportertarget
BenzphetamineSodium-dependent dopamine transportertarget
FlupentixolAlpha-1A adrenergic receptortarget
FlupentixolDopamine D2 receptortarget
FlupentixolDopamine D1 receptortarget
FlupentixolAromatic-L-amino-acid decarboxylaseenzyme
Flupentixol5-hydroxytryptamine receptor 2Atarget
FlupentixolP-glycoprotein 1transporter
FlupentixolMuscarinic acetylcholine receptor M1target
FlupentixolLiver carboxylesterase 1enzyme
FlupentixolDopamine D3 receptortarget
FlupentixolDopamine D4 receptortarget
Flupentixol5-hydroxytryptamine receptor 2Ctarget
CocaineSodium-dependent noradrenaline transportertarget
CocaineSodium channel proteintarget
CocaineSodium-dependent serotonin transportertarget
CocaineSodium-dependent dopamine transportertarget
CocaineCytochrome P450 3A4enzyme
CocaineMuscarinic acetylcholine receptor M1target
CocaineMuscarinic acetylcholine receptor M2target
CocaineCytochrome P450 2D6enzyme
CocaineSolute carrier family 22 member 2transporter
CocaineCytochrome P450 2C8enzyme
CocaineSigma non-opioid intracellular receptor 1target
CocaineLiver carboxylesterase 1target
CocaineCholinesteraseenzyme
CocaineSodium-dependent dopamine transportertransporter
Cocainealpha1-acid glycoproteincarrier
CocaineLiver carboxylesterase 1enzyme
MesoridazineDopamine D2 receptortarget
Mesoridazine5-hydroxytryptamine receptor 2Atarget
MesoridazineCytochrome P450 2D6enzyme
DopamineDopamine D1 receptortarget
DopamineDopamine beta-hydroxylasetarget
DopamineAmine oxidase [flavin-containing] Aenzyme
DopamineAmine oxidase [flavin-containing] Benzyme
DopamineCatechol O-methyltransferaseenzyme
DopamineSolute carrier family 22 member 2transporter
DopamineSolute carrier family 22 member 1transporter
DopamineSolute carrier family 22 member 3transporter
DopamineSolute carrier family 22 member 5transporter
DopaminePOU domain, class 5, transcription factor 1transporter
DopamineDopamine D5 receptortarget
DopamineDopamine D2 receptortarget
DopamineDopamine D3 receptortarget
DopamineDopamine D4 receptortarget
DopamineSodium-dependent dopamine transportertarget
DopamineDopamine beta-hydroxylaseenzyme
Dopamine5-hydroxytryptamine receptor 1Atarget
Dopamine5-hydroxytryptamine receptor 7target
DopamineD(1) dopamine receptortarget
DopamineSodium-dependent noradrenaline transportertarget
DopamineSodium-dependent serotonin transportertarget
Dopamine5-hydroxytryptamine receptor 3Atarget
Dopamine5-hydroxytryptamine receptor 3Btarget
DopamineSuperoxide dismutase [Cu-Zn]target
DopamineSynaptic vesicular amine transportertarget
MemantineCytochrome P450 2B6enzyme
MemantineSolute carrier family 22 member 2transporter
Memantine5-hydroxytryptamine receptor 3Atarget
MemantineNeuronal acetylcholine receptor subunit alpha-7target
MemantineCytochrome P450 2A6enzyme
MemantineCytochrome P450 2C19enzyme
MemantineDopamine D2 receptortarget
MemantineGlutamate receptor ionotropic, NMDA 1target
MemantineSodium/hydrogen exchanger 1transporter
MemantineSolute carrier family 22 member 4transporter
MemantineMultidrug and toxin extrusion protein 1transporter
MemantineGlutamate (NMDA) receptortarget
MemantineGABA(A) Receptortarget
MemantineGlycine receptorstarget
Ergoloid mesylateDopamine receptortarget
Ergoloid mesylateAlpha adrenergic receptortarget
Ergoloid mesylateBeta adrenergic receptortarget
Ergoloid mesylateSerotonin Receptorstarget
Ergoloid mesylateCytochrome P450 3A4enzyme
PimozideDopamine D2 receptortarget
PimozideCalmodulintarget
PimozidePotassium voltage-gated channel subfamily H member 2target
PimozideCytochrome P450 3A4enzyme
PimozideCytochrome P450 1A2enzyme
PimozideCytochrome P450 3A5enzyme
PimozideCytochrome P450 3A7enzyme
PimozideP-glycoprotein 1transporter
PimozideDopamine D3 receptortarget
PimozideCytochrome P450 2D6enzyme
BupropionSodium-dependent dopamine transportertarget
BupropionSodium-dependent noradrenaline transportertarget
BupropionCytochrome P450 2B6enzyme
BupropionCytochrome P450 2D6enzyme
BupropionAlpha-1-acid glycoprotein 1carrier
BupropionNeuronal acetylcholine receptor subunit alpha-3target
BupropionCytochrome P450 2C9enzyme
BupropionCytochrome P450 2E1enzyme
BupropionSolute carrier family 22 member 2transporter
Bupropion5-hydroxytryptamine receptor 3Atarget
DomperidoneDopamine D2 receptortarget
DomperidoneCytochrome P450 3A4enzyme
DomperidoneCytochrome P450 3A5enzyme
DomperidoneCytochrome P450 3A7enzyme
DomperidoneP-glycoprotein 1transporter
DomperidoneCytochrome P450 1A2enzyme
DomperidoneCytochrome P450 2B6enzyme
DomperidoneCytochrome P450 2C8enzyme
DomperidoneCytochrome P450 2D6enzyme
DomperidoneDopamine D3 receptortarget
MetoclopramideMuscarinic acetylcholine receptor M1target
MetoclopramideDopamine D2 receptortarget
MetoclopramideCytochrome P450 2D6enzyme
Metoclopramide5-hydroxytryptamine receptor 4target
Metoclopramide5-hydroxytryptamine receptor 3Atarget
MetoclopramideCytochrome P450 3A4enzyme
MetoclopramideCytochrome P450 1A2enzyme
MetoclopramideP-glycoprotein 1transporter
MetoclopramideAlpha-1-acid glycoprotein 1carrier
ChlorprothixeneDopamine D1 receptortarget
ChlorprothixeneDopamine D2 receptortarget
ChlorprothixeneDopamine D3 receptortarget
Chlorprothixene5-hydroxytryptamine receptor 2Atarget
ChlorprothixeneHistamine H1 receptortarget
ChlorprothixeneMuscarinic acetylcholine receptor M1target
ChlorprothixeneMuscarinic acetylcholine receptor M2target
ChlorprothixeneMuscarinic acetylcholine receptor M3target
ChlorprothixeneMuscarinic acetylcholine receptor M4target
ChlorprothixeneMuscarinic acetylcholine receptor M5target
ChlorprothixeneP-glycoprotein 1transporter
ChlorprothixeneSerotonin Receptorstarget
LisdexamfetamineSolute carrier family 15 member 1transporter
LisdexamfetamineTrace amine-associated receptor 1target
PaliperidoneDopamine D2 receptortarget
Paliperidone5-hydroxytryptamine receptor 2Atarget
PaliperidoneHistamine H1 receptortarget
PaliperidoneAlpha-1A adrenergic receptortarget
PaliperidoneAlpha-1B adrenergic receptortarget
PaliperidoneDopamine D3 receptortarget
PaliperidoneDopamine D4 receptortarget
PaliperidoneDopamine D1 receptortarget
PaliperidoneAlpha-2A adrenergic receptortarget
PaliperidoneAlpha-2B adrenergic receptortarget
PaliperidoneAlpha-2C adrenergic receptortarget
Paliperidone5-hydroxytryptamine receptor 1Atarget
Paliperidone5-hydroxytryptamine receptor 1Dtarget
Paliperidone5-hydroxytryptamine receptor 2Ctarget
Paliperidone5-hydroxytryptamine receptor 7target
PaliperidoneCytochrome P450 3A4enzyme
PaliperidoneCytochrome P450 2D6enzyme
PaliperidoneCytochrome P450 3A5enzyme
PaliperidoneP-glycoprotein 1transporter
MethotrimeprazineDopamine D3 receptortarget
MethotrimeprazineHistamine H1 receptortarget
MethotrimeprazineMuscarinic acetylcholine receptor M1target
MethotrimeprazineMuscarinic acetylcholine receptor M2target
MethotrimeprazineMuscarinic acetylcholine receptor M3target
MethotrimeprazineMuscarinic acetylcholine receptor M4target
MethotrimeprazineMuscarinic acetylcholine receptor M5target
MethotrimeprazineAlpha-1A adrenergic receptortarget
MethotrimeprazineAlpha-1B adrenergic receptortarget
MethotrimeprazineAlpha-1D adrenergic receptortarget
MethotrimeprazineCytochrome P450 2D6enzyme
MethotrimeprazineDopamine D2 receptortarget
MethotrimeprazineDopamine D1 receptortarget
MethotrimeprazineDopamine D5 receptortarget
MethotrimeprazineDopamine D4 receptortarget
MethotrimeprazineAlpha-2A adrenergic receptortarget
MethotrimeprazineAlpha-2B adrenergic receptortarget
MethotrimeprazineAlpha-2C adrenergic receptortarget
Methotrimeprazine5-hydroxytryptamine receptor 2Atarget
Methotrimeprazine5-hydroxytryptamine receptor 2Ctarget
MethotrimeprazineCytochrome P450 2E1enzyme
DextroamphetamineAlpha-1B adrenergic receptortarget
DextroamphetamineSodium-dependent dopamine transportertarget
DextroamphetamineSodium-dependent noradrenaline transportertarget
DextroamphetamineSynaptic vesicular amine transportertarget
DextroamphetamineTrace amine-associated receptor 1target
DextroamphetamineCytochrome P450 2D6enzyme
DextroamphetaminePrimary amine oxidaseenzyme
DextroamphetamineSodium-dependent dopamine transportertransporter
DextroamphetamineAlpha adrenergic receptortarget
MetamfetamineCytochrome P450 2D6enzyme
MetamfetamineSolute carrier family 22 member 3transporter
MetamfetamineSolute carrier family 22 member 5transporter
MetamfetamineSodium-dependent dopamine transportertarget
MetamfetamineSynaptic vesicular amine transportertarget
MetamfetamineTrace amine-associated receptor 1target
MetamfetamineSodium-dependent serotonin transportertarget
MetamfetamineSodium-dependent noradrenaline transportertarget
MetamfetamineChromaffin granule amine transportertarget
MetamfetamineAmine oxidase [flavin-containing] Atarget
MetamfetamineAmine oxidase [flavin-containing] Btarget
MetamfetamineAlpha-2A adrenergic receptortarget
MetamfetamineAlpha-2B adrenergic receptortarget
MetamfetamineAlpha-2C adrenergic receptortarget
ThiothixeneCytochrome P450 1A2enzyme
ThiothixeneCytochrome P450 2D6enzyme
ThiothixeneDopamine D2 receptortarget
ThiothixeneDopamine D1 receptortarget
Thiothixene5-hydroxytryptamine receptor 2Atarget
ThiothixeneSolute carrier family 22 member 1transporter
ThiothixeneSerum albumincarrier
ZuclopenthixolDopamine D1 receptortarget
ZuclopenthixolDopamine D5 receptortarget
ZuclopenthixolDopamine D2 receptortarget
ZuclopenthixolCytochrome P450 2D6enzyme
ZuclopenthixolAlpha-1A adrenergic receptortarget
ZuclopenthixolAlpha-2A adrenergic receptortarget
Zuclopenthixol5-hydroxytryptamine receptor 2Atarget
ZuclopenthixolHistamine H1 receptortarget
ZuclopenthixolCytochrome P450 3A4enzyme
NomifensineSodium-dependent noradrenaline transportertarget
NomifensineSodium-dependent dopamine transportertarget
NomifensineAlpha-1-acid glycoprotein 1carrier
NomifensineAmine oxidase [flavin-containing] Btarget
NomifensineAmine oxidase [flavin-containing] Atarget
NomifensineMyeloperoxidasetarget
NomifensineSodium-dependent serotonin transportertarget
NomifensineSynaptic vesicular amine transportertarget
FluspirileneDopamine D2 receptortarget
Fluspirilene5-hydroxytryptamine receptor 2Atarget
FluspirileneVoltage-dependent calcium channel gamma-1 subunittarget
FluspirileneCytochrome P450 3A4enzyme
AmisulprideDopamine D2 receptortarget
AmisulprideDopamine D3 receptortarget
Amisulpride5-hydroxytryptamine receptor 7target
Amisulpride5-hydroxytryptamine receptor 2Atarget
AmisulprideErythrocytecarrier
AmisulprideMultidrug and toxin extrusion protein 1transporter
AmisulprideMultidrug and toxin extrusion protein 2transporter
AmisulprideP-glycoprotein 1transporter
AmisulprideATP-binding cassette sub-family G member 2transporter
AmisulprideSolute carrier family 22 member 1transporter
AmisulprideMu-type opioid receptortarget
AmisulprideDelta-type opioid receptortarget
AmisulprideKappa-type opioid receptortarget
DexmethylphenidateSodium-dependent dopamine transportertarget
DexmethylphenidateSodium-dependent noradrenaline transportertarget
DexmethylphenidateSodium-dependent serotonin transportertarget
DexmethylphenidateCarboxylesteraseenzyme
LurasidoneCytochrome P450 3A4enzyme
LurasidoneDopamine D2 receptortarget
Lurasidone5-hydroxytryptamine receptor 2Atarget
Lurasidone5-hydroxytryptamine receptor 7target
Lurasidone5-hydroxytryptamine receptor 1Atarget
LurasidoneAlpha-2C adrenergic receptortarget
LurasidoneAlpha-2A adrenergic receptortarget
QuinagolideDopamine D2 receptortarget
QuinagolideD(1) dopamine receptortarget
BrexpiprazoleCytochrome P450 2D6enzyme
BrexpiprazoleCytochrome P450 3A4enzyme
Brexpiprazole5-hydroxytryptamine receptor 1Atarget
BrexpiprazoleDopamine D2 receptortarget
Brexpiprazole5-hydroxytryptamine receptor 2Atarget
BrexpiprazoleAlpha-2C adrenergic receptortarget
BrexpiprazoleAlpha-1B adrenergic receptortarget
BrexpiprazoleMultidrug and toxin extrusion protein 2transporter
BrexpiprazoleSerum albumincarrier
BrexpiprazoleAlpha-1-acid glycoprotein 1carrier
BrexpiprazoleDopamine D3 receptortarget
Brexpiprazole5-hydroxytryptamine receptor 2Btarget
Brexpiprazole5-hydroxytryptamine receptor 7target
BrexpiprazoleAlpha-1A adrenergic receptortarget
BrexpiprazoleAlpha-1D adrenergic receptortarget
BrexpiprazoleHistamine H1 receptortarget
BrexpiprazoleMuscarinic acetylcholine receptor M1target
BenserazideAromatic-L-amino-acid decarboxylasetarget
MetergolineSodium channel protein type 2 subunit alphatarget
TolcaponeCatechol O-methyltransferasetarget
TolcaponeCytochrome P450 2C9enzyme
EntacaponeCatechol O-methyltransferasetarget
EntacaponeCatechol O-methyltransferaseenzyme
EntacaponeUDP-glucuronosyltransferase 1-9enzyme
EntacaponeCytochrome P450 2D6enzyme
SelegilineAmine oxidase [flavin-containing] Btarget
SelegilineCytochrome P450 2B6enzyme
SelegilineAmine oxidase [flavin-containing] Atarget
SelegilineCytochrome P450 2A6enzyme
SelegilineCytochrome P450 3A4enzyme
SelegilineP-glycoprotein 1transporter
SelegilineCytochrome P450 1A2enzyme
SelegilineCytochrome P450 2C19enzyme
SelegilineCytochrome P450 2C8enzyme
SelegilineCytochrome P450 2C9enzyme
SelegilineCytochrome P450 2D6enzyme
RasagilineApoptosis regulator Bcl-2target
RasagilineAmine oxidase [flavin-containing] Btarget
RasagilineCytochrome P450 1A2enzyme
SafinamideAmine oxidase [flavin-containing] Btarget
SafinamideAmine oxidase [flavin-containing] Aenzyme
SafinamideATP-binding cassette sub-family G member 2transporter
SafinamideSolute carrier organic anion transporter family member 3A1transporter
SafinamideCytochrome P450 3A4enzyme
SafinamideCytochrome P450 1A1enzyme
SafinamideCytochrome P450 1A2enzyme
SafinamideCytochrome P450 2D6enzyme
SafinamideCytochrome P450 2C19enzyme
SafinamideCytochrome P450 3A5enzyme
OpicaponeCytochrome P450 2C19enzyme
OpicaponeCytochrome P450 2C8enzyme
OpicaponeCatechol O-methyltransferasetarget
OpicaponeSolute carrier organic anion transporter family member 1B1transporter
OpicaponeP-glycoprotein 1transporter
OpicaponeATP-binding cassette sub-family G member 2transporter
OpicaponeSolute carrier organic anion transporter family member 1B3transporter
OpicaponeSolute carrier organic anion transporter family member 2B1transporter
OpicaponeCytochrome P450 2C9enzyme
OpicaponeCytochrome P450 1A2enzyme
OpicaponeCytochrome P450 2B6enzyme
SolriamfetolSolute carrier family 22 member 2transporter
SolriamfetolSolute carrier family 22 member 4transporter
SolriamfetolSolute carrier family 22 member 5transporter
SolriamfetolSodium-dependent dopamine transportertarget
SolriamfetolSodium-dependent noradrenaline transportertarget
AripiprazoleDopamine D2 receptortarget
Aripiprazole5-hydroxytryptamine receptor 1Atarget
Aripiprazole5-hydroxytryptamine receptor 2Atarget
AripiprazoleCytochrome P450 3A4enzyme
AripiprazoleCytochrome P450 2D6enzyme
Aripiprazole5-hydroxytryptamine receptor 1Btarget
Aripiprazole5-hydroxytryptamine receptor 1Dtarget
Aripiprazole5-hydroxytryptamine receptor 1Etarget
AripiprazoleDopamine D1 receptortarget
AripiprazoleDopamine D5 receptortarget
AripiprazoleDopamine D3 receptortarget
AripiprazoleDopamine D4 receptortarget
Aripiprazole5-hydroxytryptamine receptor 2Ctarget
Aripiprazole5-hydroxytryptamine receptor 3Atarget
Aripiprazole5-hydroxytryptamine receptor 6target
Aripiprazole5-hydroxytryptamine receptor 7target
AripiprazoleHistamine H1 receptortarget
AripiprazoleAlpha-1A adrenergic receptortarget
AripiprazoleAlpha-1B adrenergic receptortarget
AripiprazoleAlpha-2A adrenergic receptortarget
AripiprazoleAlpha-2B adrenergic receptortarget
AripiprazoleAlpha-2C adrenergic receptortarget
AripiprazoleCytochrome P450 3A5enzyme
AripiprazoleCytochrome P450 3A7enzyme
AripiprazoleSerum albumincarrier
Aripiprazole5-hydroxytryptamine receptor 2Btarget
Aripiprazole5-hydroxytryptamine receptor 5Atarget
AripiprazoleBeta-1 adrenergic receptortarget
AripiprazoleBeta-2 adrenergic receptortarget
AripiprazoleHistamine H2 receptortarget
AripiprazoleHistamine H3 receptortarget
AripiprazoleHistamine H4 receptortarget
AripiprazoleMuscarinic acetylcholine receptor M1target
AripiprazoleMuscarinic acetylcholine receptor M2target
AripiprazoleMuscarinic acetylcholine receptor M3target
AripiprazoleMuscarinic acetylcholine receptor M4target
AripiprazoleMuscarinic acetylcholine receptor M5target
AripiprazoleKappa-type opioid receptortarget
AripiprazoleMu-type opioid receptortarget
AripiprazoleDelta-type opioid receptortarget
AripiprazoleGlutamate (NMDA) receptortarget
AripiprazoleSodium-dependent dopamine transportertarget
AripiprazoleSodium-dependent serotonin transportertarget
AripiprazoleP-glycoprotein 1transporter
AripiprazoleATP-binding cassette sub-family G member 2transporter
SerdexmethylphenidateSodium-dependent dopamine transportertarget
SerdexmethylphenidateSodium-dependent noradrenaline transportertarget
Serdexmethylphenidate5-hydroxytryptamine receptor 1Atarget
SerdexmethylphenidateCarboxylesteraseenzyme
AcepromazineDopamine D2 receptortarget
AcepromazineDopamine D1 receptortarget
Acepromazine5-hydroxytryptamine receptor 2Atarget
Acepromazine5-hydroxytryptamine receptor 1Atarget
AcepromazineAlpha-1A adrenergic receptortarget
AcepromazineAlpha-1B adrenergic receptortarget
AcepromazineSerum albumincarrier
AceprometazineHistamine H1 receptortarget
VanoxerineCytochrome P450 3A4enzyme
VanoxerineSodium-dependent dopamine transportertarget
VanoxerineHERG human cardiac K+ channeltarget
YKP-13585-hydroxytryptamine receptor 2Atarget
YKP-1358Dopamine D2 receptortarget
BromoprideDopamine D2 receptortarget
AS-8112Dopamine D2 receptortarget
AS-8112Dopamine D3 receptortarget
AS-81125HT3 serotonin receptortarget
DihydroergocornineSerotonin Receptorstarget
DihydroergocornineBeta adrenergic receptortarget
DihydroergocornineAlpha adrenergic receptortarget
DihydroergocornineCytochrome P450 3A4enzyme
TetrahydropalmatineDopamine D1 receptortarget
TetrahydropalmatineDopamine D2 receptortarget
TetrahydropalmatineCytochrome P450 3A4enzyme
RacloprideDopamine D2 receptortarget
JNJ-37822681Dopamine D2 receptortarget
DihydrexidineDopamine D1 receptortarget
TiaprideDopamine D2 receptortarget
TiaprideDopamine D3 receptortarget
TiaprideSerotonin Receptorstarget
TiaprideAlpha-1 adrenergic receptorstarget
TiaprideAlpha-2 adrenergic receptorstarget
TergurideCytochrome P450 3A4enzyme
PenfluridolCytochrome P450 3A4enzyme