Benzazepines

Name
Benzazepines
Accession Number
DBCAT000451
Description

Compounds with BENZENE fused to AZEPINES.

Drugs
DrugDrug Description
LorazepamA long-acting benzodiazepine commonly used to treat panic disorders, severe anxiety, and seizures.
TemazepamA short-acting benzodiazepine commonly used to treat panic disorders, severe anxiety, and insomnia.
OlanzapineAn antipsychotic drug used in the management of schizophrenia, bipolar 1 disorder, and agitation associated with these disorders.
DiltiazemA calcium channel blocker used to treat hypertension and to manage chronic stable angina.
ClobazamA benzodiazepine used as adjunct treatment in seizures associated with Lennox-Gastaut syndrome.
AlprazolamA long-acting benzodiazepine with intermediate onset commonly used to treat panic disorders and generalized anxiety in addition to anxiety associated with depression.
ChlordiazepoxideA benzodiazepine used to treat the withdrawal symptoms of acute alcoholism, to treat preoperative anxiety, and to treat anxiety over a short term period.
AdinazolamFor the treatment of anxiety and status epilepticus.
Clorazepic acidA benzodiazepine used to treat anxiety, partial seizures, and alcohol withdrawal.
PirenzepineAn antimuscarinic agent used to treat peptic ulcers, gastric ulcers, and duodenal ulcers.
GalantamineA benzazepine derivative used to treat mild to moderate dementia associated with Alzheimer's Disease.
FlurazepamA long-acting benzodiazepine with a rapid onset of action that is commonly used to treat insomnia.
FenoldopamA dopamine D1 receptor agonist used for the short term management of hypertension.
HalazepamUsed to relieve anxiety, nervousness, and tension associated with anxiety disorders.
DiazepamA long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.
OxazepamAn intermediate-acting benzodiazepine with slow onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawals, and insomnia.
TriazolamA benzodiazepine used for short term treatment of insomnia.
ClonazepamA long-acting benzodiazepine with intermediate onset commonly used to treat panic disorders, severe anxiety, and seizures.
FlumazenilA benzodiazepine antagonist that is used for the complete or partial reversal of the sedative effects caused by benzodiazepines in various clinical settings, such as induced general anesthesia for diagnostic and therapeutic procedures.
EstazolamA benzodiazepine used for the short-term management of insomnia.
VareniclineA partial agonist at nicotinic acetylcholine receptors used as an aid in smoking cessation.
HaloxazolamNot Available
CamazepamCamazepam has been used in placebo controlled studies for the treatment of patients suffering from anxiety and depression.
DelorazepamMainly used as an anti-anxiety agent. Studies have found delorazepam to be more effective in the first 4 weeks of use than antidepressants; however, after 4 weeks, antidepressants showed superior...
FlunitrazepamFor short-term treatment of severe insomnias, that are not responsive to other hypnotics.
Ethyl loflazepateNot Available
CloxazolamUsed primarily as an anti-anxiety agent. Typically used short term, and may be given as a single dose of up to 100mcg/kg to reduce anxiety and tension experienced prior to...
BromazepamA short-acting benzodiazepine with intermediate onset commonly used to treat panic disorders and severe anxiety.
FludiazepamUsed for the short-term treatment of anxiety disorders.
KetazolamA long-acting benzodiazepine used to manage anxiety and insomnia.
PrazepamFor the treatment of anxiety disorders.
QuazepamA long -acting benzodiazepine used to manage insomnia.
CinolazepamFor the management of anxiety disorders or for the short-term relief of the symptoms of anxiety or anxiety associated with depressive symptoms.
NitrazepamA long-acting benzodiazepine with intermediate onset commonly used to treat panic disorders, severe anxiety, insomnia, and seizures.
Omacetaxine mepesuccinateA cephalotaxine used in the treatment of Chronic Myeloid Leukemia (CML) that is intolerant to or resistant to two or more tyrosine kinase inhibitors.
TalampanelFor the treatment of epilepsy.
EVT 201Investigated for use/treatment in insomnia.
TarazepideInvestigated for use/treatment in gastrointestinal diseases and disorders (miscellaneous).
S-8510Investigated for use/treatment in alzheimer's disease and dementia.
DextofisopamInvestigated for use/treatment in irritable bowel syndrome (IBS).
TofisopamFor the treatment of anxiety and alcohol withdrawal.
EtizolamIndicated for the treatment of generalized anxiety disorder with depression, panic disorder and insomnia.
AptazapineInvestigated for the treatment of depression.
EvacetrapibEvacetrapib has been used in trials studying the basic science and treatment of Dyslipidemia, Hyperlipidemia, Hypercholesterolemia, Hepatic Insufficiency, and Cardiovascular Disease.
SJG-136SJG-136 has been used in trials studying the treatment of Recurrent Fallopian Tube Cancer, Secondary Acute Myeloid Leukemia, de Novo Myelodysplastic Syndromes, Recurrent Ovarian Epithelial Cancer, and Secondary Myelodysplastic Syndromes,...
BMS-906024BMS-906024 has been used in trials studying the treatment of Cancer, Lymphoblastic Leukemia, Acute T-cell, and Precursor T-Cell Lymphoblastic Lymphoma.
GI-181771XGski181771 X is under investigation in clinical trial NCT00600743 (Effect of a CCK-1R Agonist on Food Intake in Humans).
NetazepideNetazepide has been used in trials studying the prevention and treatment of Dyspepsia, Hypergastrinaemia, Barrett's Esophagus, ECL-cell Hyperplasia, and Rebound Hyperacidity, among others.
RemimazolamRemimazolam has been used in trials studying the supportive care and treatment of Anesthesia, Colonoscopy, Bronchoscopy, and General Anesthesia.
BenzodiazepineBenzodiazepine is under investigation for the prevention of Delirium and C.Surgical Procedure; Cardiac. Benzodiazepine has been investigated for the treatment of Obesity, Sleep Apnea, Obstructive, and Disorders of Gallbladder, Biliary...
IndiplonIndiplon has been used in trials studying the treatment of Insomnia and Depression.
PF-477736PF-00477736 has been used in trials studying the treatment of Neoplasms.
CE-326597CE-326,597 has been used in trials studying the treatment of Obesity.
TetrazepamNot Annotated
PinazepamNot Annotated
MedazepamNot Annotated
LoprazolamLoprazolam is an imidazobenzodiazepine with anxiolytic, anticonvulsant, hypnotic, sedative and skeletal muscle relaxant properties. It is indicated for the short-term treatment of insomnia including difficulty in falling asleep and/or frequent...
DoxefazepamNot Annotated
LormetazepamFor the treatment of short-term insomnia
NordazepamAn intermediate in the metabolism of DIAZEPAM to OXAZEPAM. It may have actions similar to those of diazepam.
Oxazepam acetateNot Annotated
CinazepamNot Annotated
BMS-214662BMS-214662 has been used in trials studying the treatment of Childhood Myelodysplastic Syndromes, Refractory Anemia With Excess Blasts, Recurrent Adult Acute Myeloid Leukemia, Relapsing Chronic Myelogenous Leukemia, and Adult Acute...
IomazenilIomazenil is under investigation in clinical trial NCT01590277 (Ability of Partial Inverse Agonist, Iomazenil, to Block Ethanol Effects in Humans).
RSV-604RSV-604 is under investigation in clinical trial NCT00416442 (Safety, Tolerability and Pharmacokinetic Study of Single and Multiple Intravenous Doses of RSV604 in Healthy Subjects.).
TolvaptanA selective vasopressin V2-receptor antagonist to slow kidney function decline in patients at risk for rapidly progressing autosomal dominant polycystic kidney disease (ADPKD). Also used to treat hypervolemic and euvolemic hyponatremia.
IvabradineA HCN channel blocker used to reduce the risk of hospitalization for worsening heart failure in adult patients and for treatment of stable symptomatic heart failure as a result of dilated cardiomyopathy in pediatric patients.
Vadastuximab TalirineVadastuximab Talirine has been used in trials studying the treatment of Acute myeloid leukemia, Myelodysplastic Syndrome, Acute Myelogenous Leukemia, and Acute Promyelocytic Leukemia.
Rovalpituzumab TesirineRovalpituzumab Tesirine has been used in trials studying the treatment of GLIOBLASTOMA, Malignant Melanoma, Other Solid Tumors, Small Cell Lung Cancer, and Medullary Thyroid Cancer, among others.
BMS-986115BMS-986115 has been used in trials studying the treatment of Various Advanced Cancer.
PyrazolamNot Annotated
MexazolamA benzodiazepine indicated to treat anxiety with or without psychoneurotic conditions.
OxazolamNot Annotated
R-82913Not Available
Drugs & Drug Targets
DrugTargetType
LorazepamTranslocator proteintarget
LorazepamUDP-glucuronosyltransferase 2B15enzyme
LorazepamGABA-A receptor (anion channel)target
LorazepamCytochrome P450 3A4enzyme
TemazepamTranslocator proteintarget
TemazepamGamma-aminobutyric acid receptor subunit alpha-1target
TemazepamGamma-aminobutyric acid receptor subunit alpha-2target
TemazepamGamma-aminobutyric acid receptor subunit alpha-3target
TemazepamGamma-aminobutyric acid receptor subunit alpha-4target
TemazepamGamma-aminobutyric acid receptor subunit alpha-5target
TemazepamGamma-aminobutyric acid receptor subunit alpha-6target
TemazepamGamma-aminobutyric acid receptor subunit beta-1target
TemazepamGamma-aminobutyric acid receptor subunit beta-2target
TemazepamGamma-aminobutyric acid receptor subunit beta-3target
TemazepamGamma-aminobutyric acid receptor subunit gamma-1target
TemazepamGamma-aminobutyric acid receptor subunit gamma-2target
TemazepamGamma-aminobutyric acid receptor subunit gamma-3target
TemazepamGamma-aminobutyric acid receptor subunit deltatarget
TemazepamGamma-aminobutyric acid receptor subunit epsilontarget
TemazepamGamma-aminobutyric acid receptor subunit pitarget
TemazepamGamma-aminobutyric acid receptor subunit rho-1target
TemazepamGamma-aminobutyric acid receptor subunit rho-2target
TemazepamGamma-aminobutyric acid receptor subunit thetatarget
TemazepamGamma-aminobutyric acid receptor subunit rho-3target
TemazepamCytochrome P450 3A4enzyme
TemazepamCytochrome P450 2B6enzyme
TemazepamCytochrome P450 2C9enzyme
TemazepamGABA-A receptor (anion channel)target
OlanzapineDopamine D1 receptortarget
OlanzapineMuscarinic acetylcholine receptor M1target
OlanzapineMuscarinic acetylcholine receptor M3target
Olanzapine5-hydroxytryptamine receptor 2Atarget
OlanzapineDopamine D4 receptortarget
OlanzapineHistamine H1 receptortarget
OlanzapineMuscarinic acetylcholine receptor M4target
OlanzapineMuscarinic acetylcholine receptor M2target
OlanzapineDopamine D2 receptortarget
Olanzapine5-hydroxytryptamine receptor 2Ctarget
OlanzapineDopamine D3 receptortarget
OlanzapineAlpha-1B adrenergic receptortarget
OlanzapineCytochrome P450 1A2enzyme
Olanzapine5-hydroxytryptamine receptor 3Atarget
Olanzapine5-hydroxytryptamine receptor 6target
OlanzapineAlpha-1A adrenergic receptortarget
OlanzapineDopamine D5 receptortarget
OlanzapineSerum albumincarrier
OlanzapineAlpha-1-acid glycoprotein 1carrier
OlanzapineDimethylaniline monooxygenase [N-oxide-forming] 3enzyme
OlanzapineCytochrome P450 2D6enzyme
OlanzapineP-glycoprotein 1transporter
OlanzapineCytochrome P450 2C19enzyme
OlanzapineD(1) dopamine receptortarget
OlanzapineBeta adrenergic receptortarget
Olanzapine5-hydroxytryptamine receptor 1target
OlanzapineGABA-A receptor (benzodiazepine site)target
OlanzapineCytochrome P450 2C9enzyme
OlanzapineUDP-glucuronosyltransferase 1-4enzyme
OlanzapineCytochrome P450 3A4enzyme
OlanzapineCytochrome P450 3A Subfamilyenzyme
DiltiazemVoltage-dependent calcium channel gamma-1 subunittarget
DiltiazemCytochrome P450 3A4enzyme
DiltiazemCytochrome P450 2C19enzyme
DiltiazemCytochrome P450 2D6enzyme
DiltiazemCytochrome P450 3A5enzyme
DiltiazemCytochrome P450 3A7enzyme
DiltiazemP-glycoprotein 1transporter
DiltiazemCytochrome P450 2C8enzyme
DiltiazemSerum albumincarrier
DiltiazemAlpha-1-acid glycoprotein 1carrier
DiltiazemVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
ClobazamCytochrome P450 2C19enzyme
ClobazamCytochrome P450 3A4enzyme
ClobazamCytochrome P450 2B6enzyme
ClobazamCytochrome P450 2C18enzyme
ClobazamSodium- and chloride-dependent GABA transporter 1transporter
ClobazamSodium- and chloride-dependent GABA transporter 3transporter
ClobazamP-glycoprotein 1transporter
ClobazamGABA-A receptor (anion channel)target
ClobazamCytochrome P450 2D6enzyme
AlprazolamGamma-aminobutyric acid receptor subunit alpha-1target
AlprazolamGamma-aminobutyric acid receptor subunit alpha-6target
AlprazolamTranslocator proteintarget
AlprazolamGamma-aminobutyric acid receptor subunit alpha-3target
AlprazolamGamma-aminobutyric acid receptor subunit alpha-4target
AlprazolamGamma-aminobutyric acid receptor subunit alpha-5target
AlprazolamGamma-aminobutyric acid receptor subunit alpha-2target
AlprazolamCytochrome P450 3A4enzyme
AlprazolamCytochrome P450 2C9enzyme
AlprazolamCytochrome P450 3A5enzyme
AlprazolamCytochrome P450 3A7enzyme
AlprazolamGABA-A receptor (anion channel)target
AlprazolamSerum albumincarrier
Alprazolamalpha1-acid glycoproteincarrier
ChlordiazepoxideGABA-A receptor (anion channel)target
AdinazolamCytochrome P450 2C19enzyme
AdinazolamCytochrome P450 3A4enzyme
AdinazolamGamma-aminobutyric acid receptor subunit alpha-1target
AdinazolamGamma-aminobutyric acid receptor subunit alpha-2target
AdinazolamGamma-aminobutyric acid receptor subunit alpha-3target
AdinazolamGamma-aminobutyric acid receptor subunit alpha-5target
AdinazolamGamma-aminobutyric acid receptor subunit gamma-1target
AdinazolamGamma-aminobutyric acid receptor subunit gamma-2target
AdinazolamGamma-aminobutyric acid receptor subunit gamma-3target
AdinazolamGamma-aminobutyric acid receptor subunit beta-1target
AdinazolamGamma-aminobutyric acid receptor subunit beta-2target
AdinazolamGamma-aminobutyric acid receptor subunit beta-3target
AdinazolamGamma-aminobutyric acid receptor subunit deltatarget
AdinazolamGamma-aminobutyric acid receptor subunit epsilontarget
AdinazolamGamma-aminobutyric acid receptor subunit pitarget
AdinazolamGamma-aminobutyric acid receptor subunit rho-1target
AdinazolamGamma-aminobutyric acid receptor subunit rho-2target
AdinazolamGamma-aminobutyric acid receptor subunit rho-3target
Clorazepic acidTranslocator proteintarget
Clorazepic acidCytochrome P450 3A4enzyme
Clorazepic acidGABA-A receptor (anion channel)target
PirenzepineMuscarinic acetylcholine receptor M1target
GalantamineAcetylcholinesterasetarget
GalantamineCytochrome P450 3A4enzyme
GalantamineCytochrome P450 2D6enzyme
GalantamineAcetylcholine receptor subunit alphatarget
GalantamineAcetylcholine receptor subunit betatarget
GalantamineAcetylcholine receptor subunit deltatarget
GalantamineAcetylcholine receptor subunit gammatarget
GalantamineAcetylcholine receptor subunit epsilontarget
GalantamineNeuronal acetylcholine receptor subunit alpha-2target
GalantamineNeuronal acetylcholine receptor subunit alpha-3target
GalantamineNeuronal acetylcholine receptor subunit alpha-4target
GalantamineNeuronal acetylcholine receptor subunit alpha-5target
GalantamineNeuronal acetylcholine receptor subunit alpha-6target
GalantamineNeuronal acetylcholine receptor subunit alpha-7target
GalantamineNeuronal acetylcholine receptor subunit alpha-9target
GalantamineNeuronal acetylcholine receptor subunit alpha-10target
GalantamineNeuronal acetylcholine receptor subunit beta-2target
GalantamineNeuronal acetylcholine receptor subunit beta-3target
GalantamineNeuronal acetylcholine receptor subunit beta-4target
GalantamineCholinesterasetarget
FlurazepamGamma-aminobutyric acid receptor subunit alpha-1target
FlurazepamGamma-aminobutyric acid receptor subunit beta-1target
FlurazepamGamma-aminobutyric acid receptor subunit beta-3target
FlurazepamGamma-aminobutyric acid receptor subunit alpha-5target
FlurazepamGamma-aminobutyric acid receptor subunit alpha-3target
FlurazepamGamma-aminobutyric acid receptor subunit alpha-2target
FlurazepamGamma-aminobutyric acid receptor subunit beta-2target
FlurazepamGamma-aminobutyric acid receptor subunit alpha-4target
FlurazepamGamma-aminobutyric acid receptor subunit alpha-6target
FlurazepamGamma-aminobutyric acid receptor subunit gamma-1target
FlurazepamGamma-aminobutyric acid receptor subunit gamma-2target
FlurazepamGamma-aminobutyric acid receptor subunit gamma-3target
FlurazepamGamma-aminobutyric acid receptor subunit deltatarget
FlurazepamGamma-aminobutyric acid receptor subunit epsilontarget
FlurazepamGamma-aminobutyric acid receptor subunit pitarget
FlurazepamGamma-aminobutyric acid receptor subunit rho-2target
FlurazepamGamma-aminobutyric acid receptor subunit thetatarget
FlurazepamGamma-aminobutyric acid receptor subunit rho-1target
FlurazepamCytochrome P450 3A4enzyme
FlurazepamGamma-aminobutyric acid receptor subunit rho-3target
FlurazepamP-glycoprotein 1transporter
FlurazepamCytochrome P450 2E1enzyme
FlurazepamCytochrome P450 2A6enzyme
FlurazepamSolute carrier family 22 member 2transporter
FenoldopamDopamine D5 receptortarget
FenoldopamDopamine D1 receptortarget
FenoldopamAlpha-2B adrenergic receptortarget
FenoldopamAlpha-2C adrenergic receptortarget
FenoldopamAlpha-2A adrenergic receptortarget
FenoldopamAlpha-1B adrenergic receptortarget
FenoldopamAlpha-1D adrenergic receptortarget
FenoldopamAlpha-1A adrenergic receptortarget
HalazepamGamma-aminobutyric acid receptor subunit alpha-1target
HalazepamGamma-aminobutyric acid receptor subunit alpha-2target
HalazepamGamma-aminobutyric acid receptor subunit alpha-3target
HalazepamGamma-aminobutyric acid receptor subunit alpha-5target
HalazepamGamma-aminobutyric acid receptor subunit gamma-1target
HalazepamGamma-aminobutyric acid receptor subunit gamma-2target
HalazepamGamma-aminobutyric acid receptor subunit gamma-3target
HalazepamGamma-aminobutyric acid receptor subunit beta-1target
HalazepamGamma-aminobutyric acid receptor subunit beta-2target
HalazepamGamma-aminobutyric acid receptor subunit beta-3target
HalazepamGamma-aminobutyric acid receptor subunit deltatarget
HalazepamGamma-aminobutyric acid receptor subunit epsilontarget
HalazepamGamma-aminobutyric acid receptor subunit pitarget
HalazepamGamma-aminobutyric acid receptor subunit rho-1target
HalazepamGamma-aminobutyric acid receptor subunit rho-2target
HalazepamGamma-aminobutyric acid receptor subunit rho-3target
HalazepamGABA-A receptor (anion channel)target
DiazepamTranslocator proteintarget
DiazepamGamma-aminobutyric acid receptor subunit alpha-1target
DiazepamGamma-aminobutyric acid receptor subunit alpha-2target
DiazepamGamma-aminobutyric acid receptor subunit alpha-3target
DiazepamCytochrome P450 3A4enzyme
DiazepamSerum albumincarrier
DiazepamCytochrome P450 2C9enzyme
DiazepamCytochrome P450 2C19enzyme
DiazepamCytochrome P450 3A5enzyme
DiazepamCytochrome P450 3A7enzyme
DiazepamGamma-aminobutyric acid receptor subunit alpha-5target
DiazepamGamma-aminobutyric acid receptor subunit beta-1target
DiazepamGamma-aminobutyric acid receptor subunit beta-2target
DiazepamGamma-aminobutyric acid receptor subunit beta-3target
DiazepamGamma-aminobutyric acid receptor subunit gamma-1target
DiazepamGamma-aminobutyric acid receptor subunit gamma-2target
DiazepamGamma-aminobutyric acid receptor subunit gamma-3target
DiazepamGamma-aminobutyric acid receptor subunit deltatarget
DiazepamGamma-aminobutyric acid receptor subunit epsilontarget
DiazepamGamma-aminobutyric acid receptor subunit pitarget
DiazepamGamma-aminobutyric acid receptor subunit rho-1target
DiazepamGamma-aminobutyric acid receptor subunit rho-2target
DiazepamGamma-aminobutyric acid receptor subunit rho-3target
DiazepamGamma-aminobutyric acid receptor subunit thetatarget
DiazepamP-glycoprotein 1transporter
DiazepamCytochrome P450 2B6enzyme
DiazepamProstaglandin G/H synthase 1enzyme
DiazepamCytochrome P450 2C18enzyme
DiazepamCytochrome P450 2C8enzyme
DiazepamCytochrome P450 2E1enzyme
DiazepamGABA-A receptor (anion channel)target
OxazepamGamma-aminobutyric acid receptor subunit alpha-1target
OxazepamGamma-aminobutyric acid receptor subunit alpha-2target
OxazepamGamma-aminobutyric acid receptor subunit alpha-3target
OxazepamGamma-aminobutyric acid receptor subunit alpha-4target
OxazepamGamma-aminobutyric acid receptor subunit alpha-5target
OxazepamGamma-aminobutyric acid receptor subunit alpha-6target
OxazepamGamma-aminobutyric acid receptor subunit beta-1target
OxazepamGamma-aminobutyric acid receptor subunit beta-2target
OxazepamGamma-aminobutyric acid receptor subunit beta-3target
OxazepamGamma-aminobutyric acid receptor subunit gamma-1target
OxazepamGamma-aminobutyric acid receptor subunit gamma-2target
OxazepamGamma-aminobutyric acid receptor subunit gamma-3target
OxazepamGamma-aminobutyric acid receptor subunit deltatarget
OxazepamGamma-aminobutyric acid receptor subunit epsilontarget
OxazepamGamma-aminobutyric acid receptor subunit pitarget
OxazepamGamma-aminobutyric acid receptor subunit rho-1target
OxazepamGamma-aminobutyric acid receptor subunit rho-2target
OxazepamGamma-aminobutyric acid receptor subunit thetatarget
OxazepamGamma-aminobutyric acid receptor subunit rho-3target
OxazepamUDP-glucuronosyltransferase 2B15enzyme
OxazepamUDP-glucuronosyltransferase 2B7enzyme
OxazepamUDP-glucuronosyltransferase 1-9enzyme
OxazepamGABA-A receptor (anion channel)target
TriazolamTranslocator proteintarget
TriazolamCytochrome P450 3A4enzyme
TriazolamCytochrome P450 3A5enzyme
TriazolamCytochrome P450 3A7enzyme
TriazolamGamma-aminobutyric acid receptor subunit alpha-1target
TriazolamGamma-aminobutyric acid receptor subunit alpha-2target
TriazolamGamma-aminobutyric acid receptor subunit alpha-3target
TriazolamGamma-aminobutyric acid receptor subunit alpha-4target
TriazolamGamma-aminobutyric acid receptor subunit alpha-5target
TriazolamGamma-aminobutyric acid receptor subunit alpha-6target
TriazolamGamma-aminobutyric acid receptor subunit beta-1target
TriazolamGamma-aminobutyric acid receptor subunit beta-2target
TriazolamGamma-aminobutyric acid receptor subunit beta-3target
TriazolamGamma-aminobutyric acid receptor subunit gamma-1target
TriazolamGamma-aminobutyric acid receptor subunit gamma-2target
TriazolamGamma-aminobutyric acid receptor subunit gamma-3target
TriazolamGamma-aminobutyric acid receptor subunit deltatarget
TriazolamGamma-aminobutyric acid receptor subunit epsilontarget
TriazolamGamma-aminobutyric acid receptor subunit pitarget
TriazolamGamma-aminobutyric acid receptor subunit rho-1target
TriazolamGamma-aminobutyric acid receptor subunit rho-2target
TriazolamGamma-aminobutyric acid receptor subunit rho-3target
TriazolamGamma-aminobutyric acid receptor subunit thetatarget
TriazolamCytochrome P450 2C8enzyme
TriazolamGABA-A receptor (anion channel)target
ClonazepamTranslocator proteintarget
ClonazepamCytochrome P450 3A4enzyme
ClonazepamSerum albumincarrier
ClonazepamCytochrome P450 2E1enzyme
ClonazepamArylamine N-acetyltransferase 2enzyme
ClonazepamGABA-A receptor (anion channel)target
ClonazepamNuclear receptor subfamily 1 group I member 2target
FlumazenilGamma-aminobutyric acid receptor subunit alpha-1target
FlumazenilGamma-aminobutyric acid receptor subunit gamma-2target
FlumazenilGamma-aminobutyric acid receptor subunit alpha-5target
FlumazenilGABA-A receptor (anion channel)target
EstazolamCytochrome P450 3A4enzyme
EstazolamGamma-aminobutyric acid receptor subunit alpha-1target
EstazolamGamma-aminobutyric acid receptor subunit alpha-2target
EstazolamGamma-aminobutyric acid receptor subunit alpha-3target
EstazolamGamma-aminobutyric acid receptor subunit alpha-5target
EstazolamGamma-aminobutyric acid receptor subunit gamma-1target
EstazolamGamma-aminobutyric acid receptor subunit gamma-2target
EstazolamGamma-aminobutyric acid receptor subunit gamma-3target
EstazolamGamma-aminobutyric acid receptor subunit beta-1target
EstazolamGamma-aminobutyric acid receptor subunit beta-2target
EstazolamGamma-aminobutyric acid receptor subunit beta-3target
EstazolamGamma-aminobutyric acid receptor subunit deltatarget
EstazolamGamma-aminobutyric acid receptor subunit epsilontarget
EstazolamGamma-aminobutyric acid receptor subunit pitarget
EstazolamGamma-aminobutyric acid receptor subunit rho-1target
EstazolamGamma-aminobutyric acid receptor subunit rho-2target
EstazolamGamma-aminobutyric acid receptor subunit rho-3target
EstazolamGABA-A receptor (anion channel)target
VareniclineNeuronal acetylcholine receptor subunit alpha-4target
VareniclineNeuronal acetylcholine receptor subunit alpha-7target
VareniclineNeuronal acetylcholine receptor subunit alpha-3target
VareniclineNeuronal acetylcholine receptor subunit alpha-6target
VareniclineNeuronal acetylcholine receptor subunit beta-2target
VareniclineSolute carrier family 22 member 2transporter
FlunitrazepamGamma-aminobutyric acid receptor subunit alpha-2target
FlunitrazepamGamma-aminobutyric acid receptor subunit alpha-4target
FlunitrazepamGamma-aminobutyric acid receptor subunit alpha-5target
FlunitrazepamGamma-aminobutyric acid receptor subunit alpha-6target
FlunitrazepamGamma-aminobutyric acid receptor subunit alpha-3target
FlunitrazepamTranslocator proteintarget
FlunitrazepamCytochrome P450 2C19enzyme
FlunitrazepamUDP-glucuronosyltransferase 2B7enzyme
FlunitrazepamCytochrome P450 2A6enzyme
FlunitrazepamCytochrome P450 2B6enzyme
FlunitrazepamCytochrome P450 2C9enzyme
FlunitrazepamCytochrome P450 3A4enzyme
FlunitrazepamCytochrome P450 2E1enzyme
FlunitrazepamUDP-glucuronosyltransferase 1-1enzyme
FlunitrazepamUDP-glucuronosyltransferase 1-3enzyme
FlunitrazepamGamma-aminobutyric acid receptor subunit alpha-1target
FlunitrazepamGamma-aminobutyric acid receptor subunit beta-3target
FlunitrazepamGamma-aminobutyric acid receptor subunit gamma-2target
BromazepamGamma-aminobutyric acid receptor subunit alpha-2target
BromazepamGamma-aminobutyric acid receptor subunit alpha-1target
BromazepamGamma-aminobutyric acid receptor subunit alpha-3target
BromazepamGamma-aminobutyric acid receptor subunit alpha-4target
BromazepamGamma-aminobutyric acid receptor subunit alpha-5target
BromazepamGamma-aminobutyric acid receptor subunit alpha-6target
BromazepamGamma-aminobutyric acid receptor subunit beta-1target
BromazepamGamma-aminobutyric acid receptor subunit beta-2target
BromazepamGamma-aminobutyric acid receptor subunit beta-3target
BromazepamGamma-aminobutyric acid receptor subunit gamma-1target
BromazepamGamma-aminobutyric acid receptor subunit gamma-2target
BromazepamGamma-aminobutyric acid receptor subunit gamma-3target
BromazepamGamma-aminobutyric acid receptor subunit deltatarget
BromazepamGamma-aminobutyric acid receptor subunit epsilontarget
BromazepamGamma-aminobutyric acid receptor subunit pitarget
BromazepamGamma-aminobutyric acid receptor subunit rho-1target
BromazepamGamma-aminobutyric acid receptor subunit rho-2target
BromazepamGamma-aminobutyric acid receptor subunit thetatarget
BromazepamGamma-aminobutyric acid receptor subunit rho-3target
BromazepamCytochrome P450 1A2enzyme
BromazepamCytochrome P450 2C19enzyme
BromazepamCytochrome P450 2E1enzyme
FludiazepamGamma-aminobutyric acid receptor subunit alpha-2target
FludiazepamGamma-aminobutyric acid receptor subunit alpha-1target
FludiazepamGamma-aminobutyric acid receptor subunit alpha-3target
FludiazepamGamma-aminobutyric acid receptor subunit alpha-5target
FludiazepamGamma-aminobutyric acid receptor subunit gamma-1target
FludiazepamGamma-aminobutyric acid receptor subunit gamma-2target
FludiazepamGamma-aminobutyric acid receptor subunit gamma-3target
FludiazepamGamma-aminobutyric acid receptor subunit beta-1target
FludiazepamGamma-aminobutyric acid receptor subunit beta-2target
FludiazepamGamma-aminobutyric acid receptor subunit beta-3target
FludiazepamGamma-aminobutyric acid receptor subunit deltatarget
FludiazepamGamma-aminobutyric acid receptor subunit epsilontarget
FludiazepamGamma-aminobutyric acid receptor subunit pitarget
FludiazepamGamma-aminobutyric acid receptor subunit rho-1target
FludiazepamGamma-aminobutyric acid receptor subunit rho-2target
FludiazepamGamma-aminobutyric acid receptor subunit rho-3target
KetazolamTranslocator proteintarget
KetazolamGamma-aminobutyric acid receptor subunit alpha-1target
KetazolamGamma-aminobutyric acid receptor subunit beta-1target
KetazolamGamma-aminobutyric acid receptor subunit gamma-1target
KetazolamGamma-aminobutyric acid receptor subunit deltatarget
KetazolamGamma-aminobutyric acid receptor subunit epsilontarget
KetazolamCytochrome P450 3A4enzyme
KetazolamP-glycoprotein 1transporter
KetazolamSerum albumincarrier
PrazepamGamma-aminobutyric acid receptor subunit alpha-1target
PrazepamGamma-aminobutyric acid receptor subunit alpha-2target
PrazepamGamma-aminobutyric acid receptor subunit alpha-3target
PrazepamGamma-aminobutyric acid receptor subunit alpha-5target
PrazepamGamma-aminobutyric acid receptor subunit gamma-1target
PrazepamGamma-aminobutyric acid receptor subunit gamma-2target
PrazepamGamma-aminobutyric acid receptor subunit gamma-3target
PrazepamGamma-aminobutyric acid receptor subunit beta-1target
PrazepamGamma-aminobutyric acid receptor subunit beta-2target
PrazepamGamma-aminobutyric acid receptor subunit beta-3target
PrazepamGamma-aminobutyric acid receptor subunit deltatarget
PrazepamGamma-aminobutyric acid receptor subunit epsilontarget
PrazepamGamma-aminobutyric acid receptor subunit pitarget
PrazepamGamma-aminobutyric acid receptor subunit rho-1target
PrazepamGamma-aminobutyric acid receptor subunit rho-2target
PrazepamGamma-aminobutyric acid receptor subunit rho-3target
PrazepamCytochrome P450 3A4enzyme
PrazepamGABA-A receptor (anion channel)target
QuazepamGamma-aminobutyric acid receptor subunit alpha-1target
QuazepamGamma-aminobutyric acid receptor subunit alpha-2target
QuazepamGamma-aminobutyric acid receptor subunit alpha-3target
QuazepamGamma-aminobutyric acid receptor subunit alpha-5target
QuazepamGamma-aminobutyric acid receptor subunit gamma-1target
QuazepamGamma-aminobutyric acid receptor subunit gamma-2target
QuazepamGamma-aminobutyric acid receptor subunit gamma-3target
QuazepamGamma-aminobutyric acid receptor subunit beta-1target
QuazepamGamma-aminobutyric acid receptor subunit beta-3target
QuazepamGamma-aminobutyric acid receptor subunit deltatarget
QuazepamGamma-aminobutyric acid receptor subunit epsilontarget
QuazepamGamma-aminobutyric acid receptor subunit pitarget
QuazepamGamma-aminobutyric acid receptor subunit rho-1target
QuazepamGamma-aminobutyric acid receptor subunit rho-2target
QuazepamGamma-aminobutyric acid receptor subunit rho-3target
QuazepamCytochrome P450 2C19enzyme
QuazepamCytochrome P450 2C9enzyme
QuazepamCytochrome P450 3A4enzyme
QuazepamGABA-A receptor (anion channel)target
QuazepamCytochrome P450 2B6enzyme
CinolazepamGamma-aminobutyric acid receptor subunit alpha-1target
CinolazepamGamma-aminobutyric acid receptor subunit alpha-2target
CinolazepamGamma-aminobutyric acid receptor subunit alpha-3target
CinolazepamGamma-aminobutyric acid receptor subunit alpha-5target
CinolazepamGamma-aminobutyric acid receptor subunit gamma-1target
CinolazepamGamma-aminobutyric acid receptor subunit gamma-2target
CinolazepamGamma-aminobutyric acid receptor subunit gamma-3target
CinolazepamGamma-aminobutyric acid receptor subunit beta-1target
CinolazepamGamma-aminobutyric acid receptor subunit beta-2target
CinolazepamGamma-aminobutyric acid receptor subunit beta-3target
CinolazepamGamma-aminobutyric acid receptor subunit deltatarget
CinolazepamGamma-aminobutyric acid receptor subunit epsilontarget
CinolazepamGamma-aminobutyric acid receptor subunit pitarget
CinolazepamGamma-aminobutyric acid receptor subunit rho-1target
CinolazepamGamma-aminobutyric acid receptor subunit rho-2target
CinolazepamGamma-aminobutyric acid receptor subunit rho-3target
NitrazepamGamma-aminobutyric acid receptor subunit alpha-1target
NitrazepamSodium channel protein type 1 subunit alphatarget
NitrazepamGamma-aminobutyric acid receptor subunit alpha-2target
NitrazepamGamma-aminobutyric acid receptor subunit alpha-3target
NitrazepamGamma-aminobutyric acid receptor subunit alpha-4target
NitrazepamGamma-aminobutyric acid receptor subunit alpha-5target
NitrazepamGamma-aminobutyric acid receptor subunit alpha-6target
NitrazepamGamma-aminobutyric acid receptor subunit beta-1target
NitrazepamGamma-aminobutyric acid receptor subunit beta-2target
NitrazepamGamma-aminobutyric acid receptor subunit beta-3target
NitrazepamGamma-aminobutyric acid receptor subunit gamma-1target
NitrazepamGamma-aminobutyric acid receptor subunit gamma-2target
NitrazepamGamma-aminobutyric acid receptor subunit gamma-3target
NitrazepamGamma-aminobutyric acid receptor subunit deltatarget
NitrazepamGamma-aminobutyric acid receptor subunit epsilontarget
NitrazepamGamma-aminobutyric acid receptor subunit pitarget
NitrazepamGamma-aminobutyric acid receptor subunit rho-1target
NitrazepamGamma-aminobutyric acid receptor subunit rho-2target
NitrazepamGamma-aminobutyric acid receptor subunit rho-3target
NitrazepamGamma-aminobutyric acid receptor subunit thetatarget
NitrazepamCytochrome P450 3A4enzyme
NitrazepamCytochrome P450 2E1enzyme
Omacetaxine mepesuccinate50S ribosomal protein L2target
Omacetaxine mepesuccinate60S ribosomal protein L3target
TalampanelGlutamate receptor 1target
TalampanelGlutamate receptor 2target
TalampanelGlutamate receptor 3target
TalampanelGlutamate receptor 4target
TofisopamcAMP-specific 3',5'-cyclic phosphodiesterase 4Atarget
TofisopamcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10Atarget
TofisopamcGMP-inhibited 3',5'-cyclic phosphodiesterase Atarget
TofisopamcGMP-dependent 3',5'-cyclic phosphodiesterasetarget
TofisopamCytochrome P450 3A4enzyme
EtizolamCytochrome P450 3A4enzyme
EtizolamCytochrome P450 2C18enzyme
EtizolamCytochrome P450 2C19enzyme
EtizolamPlatelet-activating factor receptortarget
EtizolamGamma-aminobutyric acid receptor subunit alpha-1target
EtizolamGamma-aminobutyric acid receptor subunit alpha-2target
EtizolamGamma-aminobutyric acid receptor subunit alpha-3target
EtizolamGamma-aminobutyric acid receptor subunit gamma-2target
BenzodiazepineCytochrome P450 3A4enzyme
LormetazepamGamma-aminobutyric acid receptor subunit alpha-2target
LormetazepamGamma-aminobutyric acid receptor subunit gamma-2target
LormetazepamGamma-aminobutyric acid receptor subunit alpha-3target
LormetazepamGamma-aminobutyric acid receptor subunit alpha-5target
LormetazepamGamma-aminobutyric acid receptor subunit alpha-1target
TolvaptanVasopressin V2 receptortarget
TolvaptanCytochrome P450 3A4enzyme
TolvaptanP-glycoprotein 1transporter
TolvaptanVasopressin V1a receptortarget
IvabradineCytochrome P450 3A4enzyme
IvabradinePotassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2target
MexazolamGABA-A receptor (benzodiazepine site)target
MexazolamCytochrome P450 3A4enzyme
R-82913Gag-Pol polyproteintarget
R-82913Gag-Pol polyproteintarget