| DB00187 | Esmolol | A cardioselective beta-adrenergic blocker used for the short-term control of ventricular rate and heart rate in various types of tachycardia, including perioperative tachycardia and hypertension. |
| DB00195 | Betaxolol | A cardioselective beta blocking agent commonly used to treat hypertension and elevated intraocular pressure (when administered ophthalmically). |
| DB00264 | Metoprolol | A beta-blocker used in the treatment of hypertension and angina, and used to reduce mortality due to myocardial infarction. |
| DB00298 | Dapiprazole | Used in the treatment of iatrogenically induced mydriasis produced by adrenergic (phenylephrine) or parasympatholytic (tropicamide) agents used in certain eye examinations. |
| DB00335 | Atenolol | A synthetic beta-1 selective blocker used in the management of hypertension and chronic angina, and to reduce mortality in known or suspected myocardial infarction in hemodynamically stable patients. |
| DB00346 | Alfuzosin | An alpha-1 adrenergic antagonist used in the management of benign prostatic hypertrophy (BPH). |
| DB00370 | Mirtazapine | A tetracyclic antidepressant used in the treatment of major depression and is used off-label as a drug for insomnia and to increase appetite. |
| DB00373 | Timolol | A non-selective beta adrenergic blocker used in the treatment of elevated intraocular pressure in ocular hypertension or open angle glaucoma. |
| DB00392 | Profenamine | An antidyskinetic phenothiazine used to treat the symptoms of Parkinson's disease. |
| DB00457 | Prazosin | An alpha-blocker that causes a decrease in total peripheral resistance and is used to treat hypertension. |
| DB00489 | Sotalol | A methane sulfonanilide beta adrenergic antagonist used to treat life-threatening ventricular arrhythmias and to maintain sinus rhythm in atrial fibrillation or flutter. |
| DB00521 | Carteolol | A beta adrenergic antagonist used to treat arrhythmia, angina, hypertension, and glaucoma. |
| DB00571 | Propranolol | A non-selective beta adrenergic antagonist used to treat hypertension, angina, atrial fibrillation, myocardial infarction, migraine, essential tremor, hypertrophic subaortic stenosis, and pheochromocytoma. |
| DB00590 | Doxazosin | An alpha-1 adrenergic receptor used to treat mild to moderate hypertension and urinary obstruction due to benign prostatic hyperplasia. |
| DB00598 | Labetalol | An alpha and beta adrenergic antagonist used to treat hypertension, angina, and sympathetic overactivity syndrome. |
| DB00612 | Bisoprolol | A beta-1 adrenergic blocking agent used to prevent myocardial infarction and heart failure and to treat mild to moderate hypertension. |
| DB00692 | Phentolamine | An alpha adrenergic antagonist used to reverse soft tissue anesthesia. |
| DB00699 | Nicergoline | For the treatment of senile dementia, migraines of vascular origin, transient ischemia, platelet hyper-aggregability, and macular degeneration. |
| DB00706 | Tamsulosin | An alpha-1A and alpha-1B adrenergic receptor antagonist used to treat benign prostatic hyperplasia, ureteral stones, prostatitis, and female voiding dysfunction. |
| DB00797 | Tolazoline | A vasodilator used to treat pulmonary artery anomalies. |
| DB00866 | Alprenolol | For the treatment of hypertension, angina, and arrhythmia |
| DB00908 | Quinidine | A medication used to restore normal sinus rhythm, treat atrial fibrillation and flutter, and treat ventricular arrhythmias. |
| DB00925 | Phenoxybenzamine | An alpha adrenergic agonist used to treat pheochromocytoma and episodes of hypertension and sweating. |
| DB00960 | Pindolol | A beta adrenoceptor antagonist used to treat hypertension, edema, ventricular tachycardias, and atrial fibrillation. |
| DB01049 | Ergoloid mesylate | A nootropic with an unknown mechanism of action indicated in individuals over sixty who manifest signs and symptoms of an idiopathic decline in mental capacity. |
| DB01136 | Carvedilol | A non selective beta-adrenergic antagonist used to treat mild to severe chronic heart failure, hypertension, and left ventricular dysfunction following myocardial infarction in clinically stable patients. |
| DB01158 | Bretylium | A norepinephrine release inhibitor used for the prophylaxis and therapy of ventricular fibrillation, as well as the treatment of life-threatening ventricular arrhythmias. |
| DB01162 | Terazosin | An alpha-1 adrenergic antagonist used in the treatment of symptomatic benign prostatic hyperplasia and management of hypertension. |
| DB01193 | Acebutolol | A selective β1-receptor antagonist used for the management of hypertension and ventricular premature beats in adults. |
| DB01203 | Nadolol | A non-selective beta-adrenergic antagonist used for the management of arrhythmias, angina pectoris, and hypertension. |
| DB01210 | Levobunolol | A beta-adrenergic antagonist used for the reduction of elevated intraocular pressure in patients with ocular hypertension or open-angle glaucoma. |
| DB01214 | Metipranolol | A beta-adrenergic antagonist used for the reduction of elevated intraocular pressure in patients with ocular hypertension or open-angle glaucoma. |
| DB01295 | Bevantolol | For the treatment of angina pectoris and hypertension. |
| DB01297 | Practolol | Used in the emergency treatment of cardiac arrhythmias. |
| DB01359 | Penbutolol | A beta-adrenergic antagonist used for the management of mild to moderate arterial hypertension, alone or in combination with other antihypertensive agents. |
| DB01392 | Yohimbine | An alpha-2-adrenergic blocker and sympatholytic found in supplements used to. |
| DB01580 | Oxprenolol | A non-selective beta-adrenergic antagonist used to treat hypertension, angina pectoris, arrhythmias, and anxiety. |
| DB04581 | 1-benzylimidazole | 1-benzylimidazole, an N-imidazole derivative, has been shown to have strong cardiotonic activity. |
| DB04846 | Celiprolol | Celiprolol is indicated for the management of mild to moderate hypertension and effort-induced angina pectoris. |
| DB06207 | Silodosin | An alpha-1 adrenergic receptor antagonist used to treat symptoms associated with benign prostatic hyperplasia (BPH). |
| DB06678 | Esmirtazapine | Investigated for use/treatment in insomnia and sleep disorders. |
| DB06726 | Bufuralol | Bufuralol is a new, non-selective -adrenoceptor blocking agent. |
| DB08807 | Bopindolol | For the management of hypertension, edema, ventricular tachycardias, and atrial fibrillation. |
| DB08808 | Bupranolol | Used to manage hypertension and tachycardia. Also used to treat glaucoma. |
| DB08815 | Lurasidone | An atypical antipsychotic used to treat schizophrenia and depressive episodes associated with bipolar I disorder. |
| DB08950 | Indoramin | Indoramin is a discontinued piperidine antiadrenergic drug with the trade names Baratol and Doralese. It is a selective alpha-1 adrenergic antagonist with no reflex tachycardia and direct myocardial depression action. |
| DB08952 | Indenolol | Indenolol is a drug of the beta-adrenergic blocker class. |
| DB08954 | Ifenprodil | Ifenprodil is a selective NMDA receptor (glutamate) antagonist. |
| DB09013 | Befunolol | Used in the management of open angle glaucoma. PMID: 12480285. |
| DB09204 | Arotinolol | Artinolol was introduced to be used as an antihypertensive agent since 1986. It has been studied for other functions like tremor control for patients with Parkinson disease and it is... |
| DB09205 | Moxisylyte | By the WHO, moxisylyte is indicated for the symptomatic management of sequelae of cerebral infarction or hemorrhage. The cerebral infarction is characterized by the blockage of the artery either by... |
| DB09206 | Trimazosin | Trimazosin is a sympatholytic alpha blocker. |
| DB11481 | Atipamezole | For the reversal of the sedative and analgesic effects of dexmedetomidine and medetomidine in dogs. |
| DB11770 | Talinolol | Talinolol has been investigated for the basic science of Gastrointestinal Motility Disorder. |
| DB12092 | Naftopidil | Naftopidil has been investigated for the treatment of Disorder of Urinary Stent. |
| DB12212 | Landiolol | Landiolol has been used in trials studying the treatment of Pharmacokinetics/Dynamics Study. |
| DB12230 | Bunazosin | Bunazosin has been used in trials studying the treatment of High Blood Pressure. |
| DB12551 | Idazoxan | Idazoxan has been used in trials studying the basic science of Molecular Imaging, Alzheimer Disease, and Major Depressive Disorder. |
| DB12661 | Urapidil | Urapidil has been investigated for the treatment of Hypertension During Pre-Eclampsia. |
| DB12752 | Bucindolol | Bucindolol has been investigated in Heart Failure. |
| DB13345 | Dihydroergocristine | An ergot alkaloid used to delay progressive mental decline in conditions like Alzheimer's. |
| DB13508 | Cloranolol | Not Annotated |
| DB13530 | Mepindolol | Mepindolol is a 2-methyl derivative of pindolol. It is a beta blocker. |
| DB13757 | Epanolol | Epanolol is an beta blocker. |
| DB13775 | Tertatolol | Tertatolol is a beta blocker. |
| DB04861 | Nebivolol | A beta blocking agent used to treat hypertension and aid in the management of heart failure. |
| DB13443 | Esatenolol | Esatenolol is a beta blocker. |
| DB06216 | Asenapine | An atypical antipsychotic used to treat patients with bipolar I disorder and patients with schizophrenia. |
| DB01182 | Propafenone | A Class 1C antiarrhythmic agent used in the management of paroxysmal atrial fibrillation/flutter and ventricular arrhythmias. |
| DB09351 | Levobetaxolol | Used in the treatment of open-angle glaucoma and ocular hypertension [FDA Label]. |
| DB13510 | Buflomedil | Not Annotated |
| DB01126 | Dutasteride | An antiandrogenic compound that is used for the treatment of symptomatic benign prostatic hyperplasia (BPH) in adult males by inhibiting 5-alpha reductase. |
| DB01216 | Finasteride | An antiandrogenic compound that is used for the treatment of symptomatic benign prostatic hyperplasia (BPH) and male pattern hair loss in adult males by inhibiting Type II 5-alpha reductase. |
| DB00246 | Ziprasidone | An atypical antipsychotic used to manage schizophrenia, bipolar mania, and agitation in patients with schizophrenia. |
| DB00679 | Thioridazine | A phenothiazine antipsychotic used to treat schizophrenia and generalized anxiety disorder. |
| DB00875 | Flupentixol | A thioxanthene neuroleptic used to treat schizophrenia and depression. |
| DB00420 | Promazine | A phenothiazine used to manage schizophrenia. |
| DB00656 | Trazodone | A serotonin uptake inhibitor used to treat major depressive disorder. |
| DB00734 | Risperidone | A second-generation antipsychotic medication used to treat a number of mental health disorders including schizophrenia, bipolar mania, psychosis, or as an adjunct in severe depression. |
| DB00777 | Propiomazine | Propiomazine is largely used for its antihistamininc sleep inducing effects in treating insomnia. |
| DB00831 | Trifluoperazine | A phenothiazine used to treat depression, anxiety, and agitation. |
| DB01149 | Nefazodone | An antidepressant used in the treatment of depression. |
| DB01403 | Methotrimeprazine | A phenothiazine used in the management of psychosis, particular those of schizophrenia, and manic phases of bipolar disorder. |
| DB04855 | Dronedarone | An antiarrhythmic agent used in the reduce the risk of hospitalization in patients with paroxysmal or persistent atrial fibrillation. |
| DB00622 | Nicardipine | A calcium channel blocker used for the short-term treatment of hypertension and chronic stable angina. |
| DB01267 | Paliperidone | An atypical antipsychotic used in the treatment of schizophrenia and other schizoaffective or delusional disorders. |
| DB01224 | Quetiapine | A psychotropic agent used for the management of bipolar disorder, schizophrenia, and major depressive disorder. |
| DB00363 | Clozapine | An antipsychotic drug used in treatment resistant schizophrenia and to decrease suicide risk in schizophrenic patients. |
| DB01238 | Aripiprazole | An atypical antipsychotic used in the treatment of a wide variety of mood and psychotic disorders, such as schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's syndrome. |
| DB00334 | Olanzapine | An antipsychotic drug used in the management of schizophrenia, bipolar 1 disorder, and agitation associated with these disorders. |
| DB00450 | Droperidol | A butyrophenone derivative and dopamine antagonist used to prevent and treat postoperative nausea and vomiting. |
| DB01624 | Zuclopenthixol | An antipsychotic indicated for the management of schizophrenia. The acuphase formulation is indicated for initial treatment of acute psychosis or exacerbation of psychosis, while the depot formulation is best for maintenance. |
| DB00321 | Amitriptyline | A tricyclic antidepressant indicated in the treatment of depressive illness, either endogenous or psychotic, and to relieve depression associated anxiety. |
| DB01142 | Doxepin | A psychotropic agent used for the treatment of depression, anxiety, manic-depressive disorder, and insomnia. |
| DB00458 | Imipramine | A tricyclic antidepressant indicated for the treatment of depression and to reduce childhood enuresis. |
| DB00540 | Nortriptyline | A tricyclic antidepressant used in the treatment of depression. |
| DB00543 | Amoxapine | A tricyclic antidepressant used in the treatment of neurotic or reactive depressive disorders and endogenous or psychotic depression. |
| DB00726 | Trimipramine | A tricyclic antidepressant used to treat depression. |
| DB00477 | Chlorpromazine | A phenothiazine antipsychotic used to treat nausea, vomiting, preoperative anxiety, schizophrenia, bipolar disorder, and severe behavioral problems in children. |
| DB01614 | Acepromazine | Acepromazine was first used in humans in the 1950s as an antipsychotic agent. It is now rarely used in humans. Acepromazine is frequently used in animals as a sedative and... |
| DB01622 | Thioproperazine | An antipsychotic indicated for the management of acute and chronic schizophrenia, including cases that are refractory to more common neuroleptics. May also be used to treat manic syndromes. |
| DB04946 | Iloperidone | An atypical antipsychotic agent used for the acute treatment of schizophrenia in adults. |
| DB09239 | Niguldipine | Niguldipine is a calcium channel blocker drug (CCB) with a1-adrenergic antagonist properties. |
| DB00661 | Verapamil | A calcium channel blocker used for the short-term treatment of angina, arrhythmia, and hypertension. |
| DB06153 | Pizotifen | A serotonin and tryptamine antagonist indicated for migraine prophylaxis. |
| DB12278 | Propiverine | An antimuscarinic agent used to treat urinary incontinence or increased urinary frequency or urgency. |
| DB01608 | Periciazine | A phenothiazine used with other medications to treat aggressiveness, impulsiveness, and hostility associated with psychiatric conditions such as schizophrenia. |
| DB09128 | Brexpiprazole | A serotonin–dopamine activity modulator used in the treatment of major depressive disorder as an adjunct and schizophrenia. |
| DB01200 | Bromocriptine | A dopamine D2 receptor agonist used for the treatment of galactorrhea due to hyperprolactinemia and other prolactin-related conditions, as well as in early Parkinsonian Syndrome. |
| DB11785 | Anisodamine | Anisodamine has been investigated for the treatment of Intestinal Diseases. |
| DB00696 | Ergotamine | A alpha-1 selective adrenergic agonist vasoconstrictor used to treat migraines with or without aura and cluster headaches. |
| DB00320 | Dihydroergotamine | An ergot alkaloid used in the acute treatment of migraine headache and cluster headache. |
| DB14185 | Aripiprazole lauroxil | An antipsychotic used to treat schizophrenia in adults. |
| DB03322 | Dexpropranolol | Not Available |
| DB00226 | Guanadrel | Used to treat and control hypertension. |
| DB01170 | Guanethidine | An antihypertensive agent used in the management of moderate and severe hypertension, either alone or as an adjunct, and for the management of renal hypertension. |
| DB12057 | ORM-12741 | ORM-12741 has been used in trials studying the basic science and treatment of Alzheimer's Disease. |