Uterine Leiomyomas

Also known as: Uterine Fibroids (UF) / Leiomyoma / Leiomyomas / Fibroids / Fibroid / Uterine Fibroids (Leiomyomas) / Leiomyoma, Uterine / Uterine Leiomyoma / Uterine Myoma / Uterine Myomas / Fibroids, Uterine / Uterine Fibroids / Uterine Fibroid / Leiomyoma (morphologic abnormality) / Leiomyomatous neoplasm (morphologic abnormality) / Leiomyoma NOS / Leiomyoma of uterus, unspecified / Uterine fibroma / Fibroid Uterus / Uterine leiomyoma (disorder) / Uterine fibromyoma / Leiomyoma of uterus / Leiomyoma (disorder)

DrugDrug NameDrug Description
DB11979ElagolixA gonadotropin releasing hormone receptor antagonist used to treat moderate to severe pain in endometriosis.
DB00783EstradiolAn estrogenic steroid used to treat vasomotor symptoms of vulvar and vaginal atrophy in menopause, hypoestrogenism, prevention of postmenopausal osteoporosis, treatment of breast cancer, and advanced androgen-dependent carcinoma of the prostate.
DB00007LeuprolideA peptide-based GnRH receptor superagonist used for the palliative treatment of prostate cancer, uterine leiomyomata, endometriosis, and central precocious puberty.
DB00717NorethisteroneA synthetic second-generation progestin used for contraception, prevention of endometrial hyperplasia in hormone replacement therapy, and in the treatment of other hormone-mediated illnesses such as endometriosis.
DB11853RelugolixAn oral GnRH receptor antagonist for androgen deprivation therapy in the treatment of advanced prostate cancer.
DrugDrug NameTargetType
DB11979ElagolixGonadotropin-releasing hormone receptortarget
DB11979ElagolixCytochrome P450 3A Subfamilyenzyme
DB11979ElagolixCytochrome P450 2D6enzyme
DB11979ElagolixCytochrome P450 2C8enzyme
DB11979ElagolixP-glycoprotein 1transporter
DB11979ElagolixSolute carrier organic anion transporter family member 1B1transporter
DB00783EstradiolEstrogen receptor alphatarget
DB00783EstradiolNuclear receptor subfamily 1 group I member 2target
DB00783EstradiolSex hormone-binding globulincarrier
DB00783EstradiolEstrogen receptor betatarget
DB00783EstradiolCytochrome P450 1A2enzyme
DB00783EstradiolUDP-glucuronosyltransferase 1-1enzyme
DB00783EstradiolSerum albumincarrier
DB00783EstradiolFatty acid-binding protein, intestinalcarrier
DB00783EstradiolCytochrome P450 3A4enzyme
DB00783EstradiolCytochrome P450 3A5enzyme
DB00783EstradiolCytochrome P450 3A7enzyme
DB00783EstradiolSolute carrier family 22 member 2transporter
DB00783EstradiolSolute carrier family 22 member 3transporter
DB00783EstradiolMultidrug resistance-associated protein 7transporter
DB00783EstradiolSolute carrier family 22 member 11transporter
DB00783EstradiolATP-binding cassette sub-family G member 2transporter
DB00783EstradiolSolute carrier organic anion transporter family member 1B1transporter
DB00783EstradiolP-glycoprotein 1transporter
DB00783EstradiolCytochrome P450 1A1enzyme
DB00783EstradiolCytochrome P450 1B1enzyme
DB00783EstradiolCytochrome P450 2C19enzyme
DB00783EstradiolCytochrome P450 2C8enzyme
DB00783EstradiolCytochrome P450 2C9enzyme
DB00783EstradiolSolute carrier family 22 member 8transporter
DB00783EstradiolSolute carrier organic anion transporter family member 1B3transporter
DB00783EstradiolSolute carrier organic anion transporter family member 1C1transporter
DB00783EstradiolNeuronal acetylcholine receptor subunit alpha-4target
DB00783EstradiolG-protein coupled estrogen receptor 1target
DB00783EstradiolATP synthase subunit atarget
DB00783EstradiolBeclin-1target
DB00783EstradiolUDP-glucuronosyltransferase 2B15enzyme
DB00783EstradiolCatechol O-methyltransferaseenzyme
DB00783EstradiolUDP-glucuronosyltransferases (UGTs)enzyme
DB00783EstradiolCytochrome P450 19A1enzyme
DB00007LeuprolideGonadotropin-releasing hormone receptortarget
DB00717NorethisteroneProgesterone receptortarget
DB00717NorethisteroneP-glycoprotein 1transporter
DB00717NorethisteroneCytochrome P450 2C19enzyme
DB00717NorethisteroneSerum albumincarrier
DB00717NorethisteroneSex hormone-binding globulincarrier
DB00717NorethisteroneAldo-keto reductase family 1 member C4enzyme
DB00717Norethisterone3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2enzyme
DB00717Norethisterone3-oxo-5-alpha-steroid 4-dehydrogenaseenzyme
DB00717Norethisterone3-oxo-5-beta-steroid 4-dehydrogenaseenzyme
DB00717NorethisteroneCytochrome P450 3A4enzyme
DB00717NorethisteroneCytochrome P450 1A2enzyme
DB00717NorethisteroneCytochrome P450 2A6enzyme
DB00717NorethisteroneGlucocorticoid receptortarget
DB00717NorethisteroneAndrogen receptortarget
DB11853RelugolixSerum albumincarrier
DB11853RelugolixAlpha-1-acid glycoprotein 1carrier
DB11853RelugolixP-glycoprotein 1transporter
DB11853RelugolixATP-binding cassette sub-family G member 2transporter
DB11853RelugolixCytochrome P450 3A Subfamilyenzyme
DB11853RelugolixCytochrome P450 2C8enzyme
DB11853RelugolixCytochrome P450 2B6enzyme
DB11853RelugolixGonadotropin-releasing hormone receptortarget
DrugDrug NamePhaseStatusCount
DB00297Bupivacaine0Recruiting1
DB00429Carboprost tromethamine0Recruiting1
DB16024Indocyanine green0Completed1
DB00620Triamcinolone0Recruiting1
DB01282Carbetocin1Completed1
DB00882Clomifene1Completed1
DB00048Collagenase clostridium histolyticum1Completed1
DB00668Epinephrine1Completed1
DB01006Letrozole1Completed1
DB00834Mifepristone1Completed1
DB00302Tranexamic acid1Completed1
DB08867Ulipristal1Terminated1
DB11971Vilaprisan1Completed3
DB11971Vilaprisan1Terminated1
DB00050Cetrorelix1 / 2Completed1
DB00097Choriogonadotropin alfa1 / 2Completed1
DB09126Chorionic Gonadotropin (Human)1 / 2Completed1
DB00644Gonadorelin1 / 2Completed1
DB00032Menotropins1 / 2Completed1
DB06825Triptorelin1 / 2Completed1
DB06680Asoprisnil2Completed3
DB11979Elagolix2Completed2
DB00783Estradiol2Completed2
DB00007Leuprolide2Completed1
DB00007Leuprolide2Terminated1
DB00281Lidocaine2Completed1
DB00834Mifepristone2Completed1
DB00834Mifepristone2Terminated1
DB00717Norethisterone2Completed2
DB04951Pirfenidone2Completed1
DB00396Progesterone2Completed1
DB11853Relugolix2Completed1
DB00296Ropivacaine2Completed1
DB00641Simvastatin2Recruiting1
DB11599Starch, corn2Recruiting1
DB05253Telapristone acetate2Completed7
DB05253Telapristone acetate2Terminated3
DB08867Ulipristal2Completed3
DB11971Vilaprisan2Completed2
DB00151Cysteine2 / 3Recruiting1
DB09123Dienogest2 / 3Recruiting1
DB00834Mifepristone2 / 3Completed2
DB00834Mifepristone2 / 3Terminated1
DB00929Misoprostol2 / 3Unknown Status1
DB00126Ascorbic acid3Completed1
DB06680Asoprisnil3Completed6
DB00297Bupivacaine3Recruiting1
DB01234Dexamethasone3Active Not Recruiting1
DB15230Dithiopyr3Withdrawn1
DB11979Elagolix3Active Not Recruiting1
DB11979Elagolix3Completed3
DB12116Epigallocatechin gallate3Recruiting1
DB00668Epinephrine3Completed1
DB00783Estradiol3Active Not Recruiting1
DB00783Estradiol3Completed7
DB00783Estradiol3Recruiting1
DB00644Gonadorelin3Completed1
DB00014Goserelin3Completed1
DB14307Green tea leaf3Recruiting1
DB01592Iron3Completed1
DB01592Iron3Withdrawn1
DB00007Leuprolide3Completed2
DB00007Leuprolide3Withdrawn1
DB17083Linzagolix3Completed2
DB00834Mifepristone3Completed1
DB00929Misoprostol3Completed2
DB00717Norethisterone3Active Not Recruiting1
DB00717Norethisterone3Completed7
DB00717Norethisterone3Recruiting1
DB11853Relugolix3Completed6
DB11853Relugolix3Recruiting1
DB05253Telapristone acetate3Terminated6
DB05253Telapristone acetate3Withdrawn1
DB00302Tranexamic acid3Unknown Status1
DB08867Ulipristal3Completed8
DB08867Ulipristal3Terminated1
DB08867Ulipristal3Withdrawn1
DB00067Vasopressin3Completed1
DB11971Vilaprisan3Active Not Recruiting1
DB11971Vilaprisan3Terminated3
DB11971Vilaprisan3Withdrawn1
DB00482Celecoxib4Terminated1
DB00050Cetrorelix4Completed1
DB00304Desogestrel4Terminated1
DB09123Dienogest4Terminated1
DB09123Dienogest4Unknown Status1
DB00378Dydrogesterone4Completed1
DB11979Elagolix4Completed1
DB00783Estradiol4Recruiting1
DB13257Ferrous sulfate anhydrous4Terminated1
DB00644Gonadorelin4Completed1
DB00014Goserelin4Completed1
DB00014Goserelin4Terminated1
DB01006Letrozole4Completed1
DB01006Letrozole4Not Yet Recruiting1
DB00007Leuprolide4Unknown Status3
DB00367Levonorgestrel4Completed1
DB00281Lidocaine4Completed2
DB00834Mifepristone4Terminated1
DB00929Misoprostol4Completed1
DB00929Misoprostol4Terminated1
DB00788Naproxen4Recruiting1
DB00717Norethisterone4Recruiting1
DB00107Oxytocin4Unknown Status1
DB00230Pregabalin4Terminated1
DB00165Pyridoxine4Terminated1
DB11853Relugolix4Recruiting1
DB00728Rocuronium4Completed1
DB00877Sirolimus4Recruiting1
DB00302Tranexamic acid4Completed1
DB00302Tranexamic acid4Terminated1
DB08867Ulipristal4Completed1
DB08867Ulipristal4Terminated2
DB08867Ulipristal4Unknown Status5
DB03128AcetylcholineNot AvailableCompleted1
DB00297BupivacaineNot AvailableUnknown Status2
DB00169CholecalciferolNot AvailableUnknown Status1
DB01189DesfluraneNot AvailableCompleted1
DB01234DexamethasoneNot AvailableCompleted1
DB00644GonadorelinNot AvailableCompleted2
DB00007LeuprolideNot AvailableUnknown Status1
DB00325NitroprussideNot AvailableCompleted1
DB00368NorepinephrineNot AvailableCompleted1
DB00107OxytocinNot AvailableCompleted1
DB00388PhenylephrineNot AvailableCompleted1
DB00899RemifentanilNot AvailableCompleted1
DB09070TiboloneNot AvailableNot Yet Recruiting1
DB00302Tranexamic acidNot AvailableRecruiting1
DB00302Tranexamic acidNot AvailableUnknown Status1
DB06825TriptorelinNot AvailableCompleted1
DB08867UlipristalNot AvailableUnknown Status1
DB00067VasopressinNot AvailableCompleted1