Hypertension,Essential

Also known as: Primary Hypertension / Essential Hypertension / Hypertension, Essential Hypertension / Essential,Hypertension / Hypertension, Essential / Essential hypertension, unspecified / Essential hypertension (disorder) / Essential (primary) hypertension / Unspecified essential hypertension

DrugDrug NameDrug Description
DB00381AmlodipineA calcium channel blocker used to treat hypertension and angina.
DB01076AtorvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
DB12221CanrenoneAn antimineralocorticoid and active metabolite of spironolactone used in the treatment of primary hyperaldosteronism and edematous states caused by secondary hyperaldosteronism (e.g. heart failure).
DB09279FimasartanAn angiotensin II receptor antagonist (ARB) used to treat hypertension and heart failure.
DB01275HydralazineAn antihypertensive agent used for the management of essential hypertension or severe hypertension associated with conditions requiring immediate action, heart failure, and pre-eclampsia or eclampsia .
DB00999HydrochlorothiazideA thiazide diuretic used to treat edema associated with a number of conditions, and hypertension.
DB11783ImidaprilAn ACE inhibitor used in the treatment of essential hypertension.
DB00790PerindoprilAn ACE inhibitor prodrug used to treat hypertension, mild to moderate congestive heart failure, and to reduce cardiovascular risk in patients with hypertension or post-myocardial infarction.
DB01098RosuvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
DB00421SpironolactoneAn aldosterone receptor antagonist used to treat edema, hypertension, heart failure, and aldosteronism.
DB15959TripamideNot Annotated
DrugDrug NameTargetType
DB00381AmlodipineCarbonic anhydrase 1target
DB00381AmlodipineCytochrome P450 3A4enzyme
DB00381AmlodipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
DB00381AmlodipineCytochrome P450 1A1enzyme
DB00381AmlodipineCytochrome P450 2B6enzyme
DB00381AmlodipineVoltage-dependent N-type calcium channel subunit alpha-1Btarget
DB00381AmlodipineVoltage-dependent L-type calcium channel subunit beta-1target
DB00381AmlodipineVoltage-dependent calcium channel subunit alpha-2/delta-3target
DB00381AmlodipineCytochrome P450 3A5enzyme
DB00381AmlodipineP-glycoprotein 1transporter
DB00381AmlodipineCytochrome P450 2C8enzyme
DB00381AmlodipineCytochrome P450 2D6enzyme
DB00381AmlodipineSphingomyelin phosphodiesterasetarget
DB00381AmlodipineVoltage-dependent T-type calcium channel subunit alpha-1Itarget
DB00381AmlodipineVoltage-dependent N-type calcium channeltarget
DB00381AmlodipineCytochrome P450 2C19enzyme
DB00381AmlodipineCytochrome P450 2C9enzyme
DB01076Atorvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
DB01076AtorvastatinCytochrome P450 3A4enzyme
DB01076AtorvastatinDipeptidyl peptidase 4target
DB01076AtorvastatinCytochrome P450 2D6enzyme
DB01076AtorvastatinCytochrome P450 2C9enzyme
DB01076AtorvastatinCytochrome P450 2C19enzyme
DB01076AtorvastatinCytochrome P450 3A5enzyme
DB01076AtorvastatinCytochrome P450 3A7enzyme
DB01076AtorvastatinP-glycoprotein 1transporter
DB01076AtorvastatinSolute carrier organic anion transporter family member 1A2transporter
DB01076AtorvastatinSolute carrier organic anion transporter family member 1B1transporter
DB01076AtorvastatinMultidrug resistance-associated protein 4transporter
DB01076AtorvastatinMultidrug resistance-associated protein 5transporter
DB01076AtorvastatinMultidrug resistance-associated protein 1transporter
DB01076AtorvastatinCytochrome P450 2B6enzyme
DB01076AtorvastatinCytochrome P450 2C8enzyme
DB01076AtorvastatinAryl hydrocarbon receptortarget
DB01076AtorvastatinSolute carrier organic anion transporter family member 2B1transporter
DB01076AtorvastatinSolute carrier organic anion transporter family member 1B3transporter
DB01076AtorvastatinUDP-glucuronosyltransferase 1-1enzyme
DB01076AtorvastatinUDP-glucuronosyltransferase 1-3enzyme
DB01076AtorvastatinCanalicular multispecific organic anion transporter 1transporter
DB01076AtorvastatinBile salt export pumptransporter
DB01076AtorvastatinSerum albumincarrier
DB01076AtorvastatinHistone deacetylase 2target
DB01076AtorvastatinNuclear receptor subfamily 1 group I member 3target
DB09279FimasartanType-1 angiotensin II receptortarget
DB09279FimasartanSolute carrier organic anion transporter family member 1B1transporter
DB09279FimasartanATP-binding cassette sub-family G member 2transporter
DB01275HydralazineMembrane primary amine oxidasetarget
DB01275HydralazineProlyl 4-hydroxylase subunit alpha-1target
DB01275HydralazineCytochrome P450 3A4enzyme
DB01275HydralazineSerum albumincarrier
DB01275HydralazineHypoxia-inducible factor 1-alphatarget
DB00999HydrochlorothiazideSolute carrier family 12 member 3target
DB00999HydrochlorothiazideSolute carrier family 22 member 6transporter
DB00999HydrochlorothiazideCalcium-activated potassium channel subunit alpha-1target
DB00999HydrochlorothiazideSerum albumincarrier
DB00999HydrochlorothiazideSolute carrier family 22 member 11transporter
DB00999HydrochlorothiazideMultidrug resistance-associated protein 4transporter
DB00999HydrochlorothiazideSolute carrier family 22 member 8transporter
DB00790PerindoprilAngiotensin-converting enzymetarget
DB00790PerindoprilSolute carrier family 15 member 1transporter
DB00790PerindoprilSolute carrier family 15 member 2transporter
DB00790PerindoprilCholinesteraseenzyme
DB00790PerindoprilSecreted frizzled-related protein 4target
DB01098Rosuvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
DB01098RosuvastatinCytochrome P450 2C9enzyme
DB01098RosuvastatinMultidrug resistance-associated protein 4transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1A2transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1B3transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 2B1transporter
DB01098RosuvastatinCystine/glutamate transportertransporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1B1transporter
DB01098RosuvastatinBile salt export pumptransporter
DB01098RosuvastatinATP-binding cassette sub-family G member 2transporter
DB01098RosuvastatinSerum albumincarrier
DB01098RosuvastatinCanalicular multispecific organic anion transporter 1transporter
DB01098RosuvastatinSolute carrier family 22 member 8transporter
DB01098RosuvastatinSodium/bile acid cotransportertransporter
DB01098RosuvastatinIntegrin alpha-Ltarget
DB00421SpironolactoneMineralocorticoid receptortarget
DB00421SpironolactoneCytochrome P450 2C8enzyme
DB00421SpironolactoneCanalicular multispecific organic anion transporter 1transporter
DB00421SpironolactoneP-glycoprotein 1transporter
DB00421SpironolactoneSolute carrier organic anion transporter family member 1A2transporter
DB00421SpironolactoneCytochrome P450 11B1, mitochondrialenzyme
DB00421SpironolactoneAndrogen receptortarget
DB00421SpironolactoneProgesterone receptortarget
DB00421SpironolactoneGlucocorticoid receptortarget
DB00421SpironolactoneNuclear receptor subfamily 1 group I member 2target
DB00421SpironolactoneBile salt export pumptransporter
DB00421SpironolactoneSerum albumincarrier
DB00421Spironolactonealpha1-acid glycoproteincarrier
DB00421SpironolactoneEstrogen receptortarget
DB00421SpironolactoneCytochrome P450 11B2, mitochondrialenzyme
DB00421SpironolactoneVoltage-dependent L-type calcium channeltarget
DrugDrug NamePhaseStatusCount
DB05229Beraprost0Recruiting1
DB00310Chlorthalidone0Not Yet Recruiting1
DB00381Amlodipine1Completed2
DB11720Angiotensin 1-71Terminated1
DB11842Angiotensin II1Not Yet Recruiting1
DB11842Angiotensin II1Terminated1
DB01076Atorvastatin1Completed4
DB13919Candesartan1Completed2
DB00796Candesartan cilexetil1Completed2
DB01136Carvedilol1Unknown Status1
DB00390Digoxin1Completed1
DB09279Fimasartan1Completed10
DB00999Hydrochlorothiazide1Completed2
DB01026Ketoconazole1Completed1
DB09237Levamlodipine1Completed2
DB00678Losartan1Completed1
DB01115Nifedipine1Completed2
DB00388Phenylephrine1Terminated1
DB13107QGC-0011Completed2
DB01045Rifampicin1Completed1
DB09153Sodium chloride1Completed1
DB00966Telmisartan1Completed3
DB01116Trimethaphan1Terminated1
DB16498Vasomera1Completed2
DB00682Warfarin1Completed1
DB05739CYT006-AngQb1 / 2Completed1
DB01197Captopril1 / 2Terminated1
DB00584Enalapril1 / 2Terminated1
DB11242Gelatin1 / 2Completed1
DB00999Hydrochlorothiazide1 / 2Terminated1
DB11110Magnesium citrate1 / 2Completed1
DB00437Allopurinol2Completed1
DB00381Amlodipine2Completed6
DB00381Amlodipine2Unknown Status2
DB15059Aprocitentan2Completed1
DB08822Azilsartan medoxomil2Completed1
DB13919Candesartan2Completed1
DB13919Candesartan2Unknown Status1
DB00796Candesartan cilexetil2Completed3
DB00796Candesartan cilexetil2Unknown Status1
DB00584Enalapril2Completed1
DB00700Eplerenone2Completed2
DB15207Esaxerenone2Completed1
DB00898Ethanol2Active Not Recruiting1
DB09279Fimasartan2Completed3
DB00999Hydrochlorothiazide2Completed1
DB01029Irbesartan2Completed1
DB15367LY-26230912Completed1
DB00528Lercanidipine2Completed2
DB00722Lisinopril2Completed1
DB00678Losartan2Completed1
DB00678Losartan2Unknown Status1
DB01065Melatonin2Active Not Recruiting1
DB04861Nebivolol2Completed1
DB01115Nifedipine2Completed1
DB00275Olmesartan2Recruiting1
DB11837Osilodrostat2Completed1
DB13107QGC-0012Completed1
DB12350Rostafuroxin2Completed1
DB12350Rostafuroxin2Unknown Status1
DB09292Sacubitril2Completed1
DB09292Sacubitril2Recruiting1
DB00421Spironolactone2Completed1
DB00820Tadalafil2Completed1
DB00966Telmisartan2Completed1
DB00177Valsartan2Completed3
DB00177Valsartan2Recruiting1
DB00381Amlodipine2 / 3Completed1
DB00381Amlodipine2 / 3Unknown Status2
DB00125Arginine2 / 3Completed1
DB12236Bexagliflozin2 / 3Completed1
DB00177Valsartan2 / 3Completed1
DB09026Aliskiren3Completed4
DB00381Amlodipine3Completed20
DB00381Amlodipine3Unknown Status1
DB00335Atenolol3Completed1
DB01076Atorvastatin3Completed1
DB01076Atorvastatin3Recruiting1
DB05358Azilsartan medoxomil3Completed4
DB08822Azilsartan medoxomil3Completed6
DB08822Azilsartan medoxomil3Unknown Status1
DB00612Bisoprolol3Completed1
DB13919Candesartan3Unknown Status1
DB00796Candesartan cilexetil3Completed2
DB01197Captopril3Not Yet Recruiting1
DB01136Carvedilol3Unknown Status1
DB00310Chlorthalidone3Completed5
DB00700Eplerenone3Completed2
DB00876Eprosartan3Completed1
DB15207Esaxerenone3Completed2
DB00973Ezetimibe3Recruiting1
DB09279Fimasartan3Completed5
DB09279Fimasartan3Recruiting2
DB00695Furosemide3Completed1
DB00999Hydrochlorothiazide3Completed18
DB11783Imidapril3Unknown Status1
DB00808Indapamide3Not Yet Recruiting1
DB00808Indapamide3Recruiting1
DB01029Irbesartan3Completed2
DB00678Losartan3Completed5
DB00678Losartan3Unknown Status1
DB00275Olmesartan3Completed20
DB00275Olmesartan3Not Yet Recruiting1
DB00275Olmesartan3Unknown Status1
DB00790Perindopril3Completed3
DB01098Rosuvastatin3Completed1
DB09292Sacubitril3Completed4
DB00641Simvastatin3Completed1
DB00421Spironolactone3Completed1
DB00966Telmisartan3Completed1
DB00177Valsartan3Completed4
DB00177Valsartan3Recruiting1
DB00945Acetylsalicylic acid4Completed1
DB09026Aliskiren4Completed2
DB00594Amiloride4Unknown Status1
DB00381Amlodipine4Completed9
DB00381Amlodipine4Not Yet Recruiting2
DB00381Amlodipine4Recruiting1
DB00381Amlodipine4Unknown Status2
DB09204Arotinolol4Completed1
DB00335Atenolol4Completed1
DB00335Atenolol4Terminated1
DB01076Atorvastatin4Unknown Status1
DB08822Azilsartan medoxomil4Completed1
DB00612Bisoprolol4Not Yet Recruiting1
DB13919Candesartan4Completed1
DB13919Candesartan4Unknown Status1
DB12221Canrenone4Completed1
DB01136Carvedilol4Completed1
DB00310Chlorthalidone4Not Yet Recruiting1
DB00310Chlorthalidone4Unknown Status1
DB00590Doxazosin4Completed2
DB00584Enalapril4Completed2
DB00584Enalapril4Unknown Status1
DB00700Eplerenone4Completed1
DB00876Eprosartan4Completed1
DB09279Fimasartan4Completed1
DB00158Folic acid4Completed1
DB00999Hydrochlorothiazide4Completed5
DB00999Hydrochlorothiazide4Not Yet Recruiting2
DB00999Hydrochlorothiazide4Unknown Status2
DB00808Indapamide4Recruiting1
DB01029Irbesartan4Completed1
DB09236Lacidipine4Completed1
DB00528Lercanidipine4Completed2
DB09237Levamlodipine4Unknown Status1
DB00722Lisinopril4Completed2
DB00678Losartan4Completed2
DB00678Losartan4Not Yet Recruiting1
DB00678Losartan4Unknown Status2
DB09238Manidipine4Completed1
DB00264Metoprolol4Completed2
DB01115Nifedipine4Completed1
DB01115Nifedipine4Unknown Status1
DB00275Olmesartan4Completed4
DB00275Olmesartan4Not Yet Recruiting1
DB00275Olmesartan4Terminated1
DB00790Perindopril4Recruiting1
DB00790Perindopril4Unknown Status1
DB00881Quinapril4Completed1
DB00178Ramipril4Completed3
DB00178Ramipril4Unknown Status1
DB00641Simvastatin4Unknown Status1
DB00966Telmisartan4Completed2
DB00966Telmisartan4Not Yet Recruiting2
DB00966Telmisartan4Unknown Status2
DB00177Valsartan4Completed6
DB00177Valsartan4Unknown Status1
DB00594AmilorideNot AvailableCompleted1
DB00381AmlodipineNot AvailableCompleted5
DB00381AmlodipineNot AvailableRecruiting1
DB00381AmlodipineNot AvailableUnknown Status1
DB11842Angiotensin IINot AvailableCompleted1
DB00125ArginineNot AvailableRecruiting1
DB08822Azilsartan medoxomilNot AvailableCompleted1
DB08822Azilsartan medoxomilNot AvailableNot Yet Recruiting1
DB00612BisoprololNot AvailableRecruiting1
DB01373CalciumNot AvailableActive Not Recruiting1
DB01373CalciumNot AvailableCompleted1
DB13919CandesartanNot AvailableCompleted1
DB00310ChlorthalidoneNot AvailableCompleted2
DB00310ChlorthalidoneNot AvailableRecruiting1
DB01394ColchicineNot AvailableCompleted1
DB00700EplerenoneNot AvailableRecruiting1
DB15207EsaxerenoneNot AvailableCompleted1
DB00492FosinoprilNot AvailableCompleted1
DB00999HydrochlorothiazideNot AvailableCompleted3
DB01088IloprostNot AvailableCompleted1
DB01029IrbesartanNot AvailableRecruiting1
DB09237LevamlodipineNot AvailableNot Yet Recruiting1
DB09237LevamlodipineNot AvailableUnknown Status1
DB00722LisinoprilNot AvailableCompleted1
DB00678LosartanNot AvailableCompleted1
DB00331MetforminNot AvailableCompleted1
DB01115NifedipineNot AvailableNot Yet Recruiting1
DB00727NitroglycerinNot AvailableRecruiting1
DB00275OlmesartanNot AvailableCompleted2
DB00107OxytocinNot AvailableTerminated1
DB00790PerindoprilNot AvailableCompleted3
DB01001SalbutamolNot AvailableRecruiting1
DB00421SpironolactoneNot AvailableCompleted1
DB00966TelmisartanNot AvailableCompleted1
DB00966TelmisartanNot AvailableRecruiting1
DB11815TilarginineNot AvailableUnknown Status1
DB00177ValsartanNot AvailableCompleted1