Hypercholesterolaemia

Also known as: High Blood Cholesterol Level / Hypercholesterolemia / High Blood Cholesterol / High Cholesterol / Elevated levels of cholesterol / Hypercholesteremia / Hypercholesterolemia (disorder) / Hypercholesteraemia / Elevated cholesterol / Cholesterol total increased / Cholesterol levels raised / Cholesterol high / Cholesterol blood excessive / Cholesterol blood increased / Blood cholesterol increased

DrugDrug NameDrug Description
DB01076AtorvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
DB00627NiacinA B vitamin used to treat hypertriglyceridemia and pellagra.
DB00175PravastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and to reduce the risk of cardiovascular events, including myocardial infarction and stroke.
DB01098RosuvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
DB00641SimvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular events including myocardial infarction and stroke.
DB15921Tocopheryl nicotinateA vitamin E supplement indicated in the treatment of high cholesterol and narrowing of peripheral arteries.
DrugDrug NameTargetType
DB01076Atorvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
DB01076AtorvastatinCytochrome P450 3A4enzyme
DB01076AtorvastatinDipeptidyl peptidase 4target
DB01076AtorvastatinCytochrome P450 2D6enzyme
DB01076AtorvastatinCytochrome P450 2C9enzyme
DB01076AtorvastatinCytochrome P450 2C19enzyme
DB01076AtorvastatinCytochrome P450 3A5enzyme
DB01076AtorvastatinCytochrome P450 3A7enzyme
DB01076AtorvastatinP-glycoprotein 1transporter
DB01076AtorvastatinSolute carrier organic anion transporter family member 1A2transporter
DB01076AtorvastatinSolute carrier organic anion transporter family member 1B1transporter
DB01076AtorvastatinMultidrug resistance-associated protein 4transporter
DB01076AtorvastatinMultidrug resistance-associated protein 5transporter
DB01076AtorvastatinMultidrug resistance-associated protein 1transporter
DB01076AtorvastatinCytochrome P450 2B6enzyme
DB01076AtorvastatinCytochrome P450 2C8enzyme
DB01076AtorvastatinAryl hydrocarbon receptortarget
DB01076AtorvastatinSolute carrier organic anion transporter family member 2B1transporter
DB01076AtorvastatinSolute carrier organic anion transporter family member 1B3transporter
DB01076AtorvastatinUDP-glucuronosyltransferase 1-1enzyme
DB01076AtorvastatinUDP-glucuronosyltransferase 1-3enzyme
DB01076AtorvastatinCanalicular multispecific organic anion transporter 1transporter
DB01076AtorvastatinBile salt export pumptransporter
DB01076AtorvastatinSerum albumincarrier
DB01076AtorvastatinHistone deacetylase 2target
DB01076AtorvastatinNuclear receptor subfamily 1 group I member 3target
DB00627NiacinHydroxycarboxylic acid receptor 2target
DB00627NiacinNicotinamide N-methyltransferasetarget
DB00627NiacinNicotinate-nucleotide pyrophosphorylase [carboxylating]target
DB00627NiacinHydroxycarboxylic acid receptor 3target
DB00627NiacinSolute carrier family 22 member 5transporter
DB00627NiacinSolute carrier organic anion transporter family member 2B1transporter
DB00627NiacinMonocarboxylate transporter 1transporter
DB00627NiacinCytochrome P450 2D6enzyme
DB00627NiacinSodium-coupled monocarboxylate transporter 1transporter
DB00627NiacinMonocarboxylate transporter 4transporter
DB00627NiacinThyroxine-binding globulincarrier
DB00627NiacinCytochrome P450 3A4enzyme
DB00627NiacinCytochrome P450 2E1enzyme
DB00175Pravastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
DB00175PravastatinSolute carrier organic anion transporter family member 2B1transporter
DB00175PravastatinP-glycoprotein 1transporter
DB00175PravastatinSolute carrier organic anion transporter family member 1A2transporter
DB00175PravastatinSolute carrier family 22 member 6transporter
DB00175PravastatinSolute carrier family 22 member 8transporter
DB00175PravastatinCanalicular multispecific organic anion transporter 1transporter
DB00175PravastatinSolute carrier family 22 member 11transporter
DB00175PravastatinATP-binding cassette sub-family G member 2transporter
DB00175PravastatinSolute carrier family 22 member 7transporter
DB00175PravastatinSolute carrier organic anion transporter family member 1B1transporter
DB00175PravastatinMonocarboxylate transporter 1transporter
DB00175PravastatinBile salt export pumptransporter
DB00175PravastatinSolute carrier organic anion transporter family member 1B3transporter
DB00175PravastatinHistone deacetylase 2target
DB01098Rosuvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
DB01098RosuvastatinCytochrome P450 2C9enzyme
DB01098RosuvastatinMultidrug resistance-associated protein 4transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1A2transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1B3transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 2B1transporter
DB01098RosuvastatinCystine/glutamate transportertransporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1B1transporter
DB01098RosuvastatinBile salt export pumptransporter
DB01098RosuvastatinATP-binding cassette sub-family G member 2transporter
DB01098RosuvastatinSerum albumincarrier
DB01098RosuvastatinCanalicular multispecific organic anion transporter 1transporter
DB01098RosuvastatinSolute carrier family 22 member 8transporter
DB01098RosuvastatinSodium/bile acid cotransportertransporter
DB01098RosuvastatinIntegrin alpha-Ltarget
DB00641Simvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
DB00641SimvastatinCytochrome P450 3A4enzyme
DB00641SimvastatinCytochrome P450 2C8enzyme
DB00641SimvastatinCytochrome P450 2C9enzyme
DB00641SimvastatinCytochrome P450 3A5enzyme
DB00641SimvastatinP-glycoprotein 1transporter
DB00641SimvastatinSolute carrier organic anion transporter family member 1A2transporter
DB00641SimvastatinSolute carrier organic anion transporter family member 1B1transporter
DB00641SimvastatinCytochrome P450 2B6enzyme
DB00641SimvastatinCytochrome P450 2D6enzyme
DB00641SimvastatinUDP-glucuronosyltransferase 1-1enzyme
DB00641SimvastatinUDP-glucuronosyltransferase 1-3enzyme
DB00641SimvastatinUDP-glucuronosyltransferase 2B7enzyme
DB00641SimvastatinCanalicular multispecific organic anion transporter 1transporter
DB00641SimvastatinIntegrin alpha-Ltarget
DB00641SimvastatinBile salt export pumptransporter
DB00641SimvastatinCytochrome P450 2C19enzyme
DB00641SimvastatinSolute carrier organic anion transporter family member 2B1transporter
DB00641SimvastatinSolute carrier organic anion transporter family member 1B3transporter
DB00641SimvastatinHistone deacetylase 2target
DB00641SimvastatinCocaine esteraseenzyme
DB00641SimvastatinLiver carboxylesterase 1enzyme
DrugDrug NamePhaseStatusCount
DB00973Ezetimibe0Completed1
DB11755Tetrahydrocannabivarin0Completed1
DB09302Alirocumab1Completed10
DB06630Anacetrapib1Completed1
DB01076Atorvastatin1Completed6
DB12456Bococizumab1Completed5
DB12456Bococizumab1Terminated1
DB00973Ezetimibe1Completed7
DB01039Fenofibrate1Completed1
DB15089Frovocimab1Completed1
DB05123Gemcabene1Completed3
DB06205Hyaluronidase (human recombinant)1Terminated1
DB11789Hyodeoxycholic Acid1Unknown Status1
DB14901Inclisiran1Completed1
DB11629Laropiprant1Completed1
DB00627Niacin1Completed2
DB14862PF-068153451Terminated1
DB08860Pitavastatin1Completed1
DB06817Raltegravir1Completed1
DB01098Rosuvastatin1Completed2
DB00641Simvastatin1Completed3
DB00877Sirolimus1Completed1
DB09153Sodium chloride1Terminated1
DB00864Tacrolimus1Completed1
DB16336Tafolecimab1Completed1
DB126293,5-diiodothyropropionic acid1 / 2Terminated1
DB17642AEM-281 / 2Completed1
DB09302Alirocumab2Completed8
DB11780Allicin2Withdrawn1
DB06630Anacetrapib2Terminated1
DB00125Arginine2Completed1
DB01076Atorvastatin2Completed17
DB01076Atorvastatin2Terminated1
DB11936Bempedoic acid2Completed8
DB11936Bempedoic acid2Recruiting1
DB11105Benzalkonium2Completed1
DB06698Betahistine2Terminated1
DB12456Bococizumab2Completed4
DB01432Cholestyramine2Completed1
DB00930Colesevelam2Completed1
DB05035Eprotirome2Completed1
DB00783Estradiol2Completed1
DB15354Evinacumab2Completed1
DB09303Evolocumab2Completed2
DB00973Ezetimibe2Active Not Recruiting1
DB00973Ezetimibe2Completed12
DB05449FM-VP42Completed1
DB12469Fasudil2Completed1
DB01039Fenofibrate2Completed1
DB01095Fluvastatin2Completed1
DB15089Frovocimab2Completed1
DB05123Gemcabene2Completed5
DB14901Inclisiran2Completed1
DB16215Lapaquistat2Completed1
DB16215Lapaquistat2Terminated1
DB11629Laropiprant2Completed1
DB00166Lipoic acid2Completed1
DB08827Lomitapide2Completed3
DB00227Lovastatin2Completed2
DB05192MB078112Withdrawn1
DB00331Metformin2Completed2
DB00959Methylprednisolone2Completed1
DB05528Mipomersen2Completed4
DB00627Niacin2Completed2
DB14890Obicetrapib2Completed4
DB11133Omega-3 fatty acids2Completed1
DB08860Pitavastatin2Completed1
DB00175Pravastatin2Completed4
DB01098Rosuvastatin2Completed3
DB00658Sevelamer2Completed1
DB00641Simvastatin2Completed1
DB05317TAK-4752Completed1
DB05317TAK-4752Terminated1
DB16336Tafolecimab2Completed1
DB12435Tipelukast2Completed1
DB00284Acarbose3Completed1
DB09302Alirocumab3Completed22
DB09302Alirocumab3Unknown Status1
DB00381Amlodipine3Completed4
DB06630Anacetrapib3Completed2
DB01076Atorvastatin3Completed51
DB01076Atorvastatin3Terminated7
DB11936Bempedoic acid3Completed5
DB00542Benazepril3Completed1
DB00796Candesartan cilexetil3Completed1
DB01136Carvedilol3Completed1
DB00310Chlorthalidone3Completed2
DB04540Cholesterol3Completed1
DB01432Cholestyramine3Completed2
DB00930Colesevelam3Completed1
DB00286Conjugated estrogens3Completed1
DB00343Diltiazem3Completed1
DB00590Doxazosin3Completed1
DB00783Estradiol3Completed1
DB11655Evacetrapib3Terminated2
DB09303Evolocumab3Completed8
DB00973Ezetimibe3Active Not Recruiting1
DB00973Ezetimibe3Completed73
DB00973Ezetimibe3Recruiting1
DB00973Ezetimibe3Terminated4
DB00973Ezetimibe3Unknown Status1
DB01023Felodipine3Completed1
DB01039Fenofibrate3Completed5
DB13873Fenofibric acid3Completed1
DB01095Fluvastatin3Completed4
DB01095Fluvastatin3Terminated1
DB00695Furosemide3Completed1
DB00222Glimepiride3Completed1
DB01275Hydralazine3Completed1
DB00999Hydrochlorothiazide3Completed1
DB14901Inclisiran3Active Not Recruiting3
DB01306Insulin aspart3Completed1
DB01307Insulin detemir3Completed1
DB00047Insulin glargine3Completed1
DB00030Insulin human3Completed1
DB01029Irbesartan3Completed1
DB16215Lapaquistat3Completed6
DB16215Lapaquistat3Terminated4
DB11629Laropiprant3Completed2
DB11629Laropiprant3Unknown Status1
DB12448Lifibrol3Completed1
DB00722Lisinopril3Completed2
DB00227Lovastatin3Completed4
DB00227Lovastatin3Terminated1
DB00603Medroxyprogesterone acetate3Completed1
DB00331Metformin3Completed2
DB00264Metoprolol3Completed1
DB05528Mipomersen3Completed5
DB00627Niacin3Completed8
DB00627Niacin3Unknown Status1
DB14890Obicetrapib3Active Not Recruiting2
DB14890Obicetrapib3Recruiting1
DB11133Omega-3 fatty acids3Completed2
DB14377Palm oil3Terminated1
DB15212Pemafibrate3Recruiting1
DB01132Pioglitazone3Completed1
DB08860Pitavastatin3Completed7
DB00175Pravastatin3Completed6
DB00175Pravastatin3Terminated1
DB00396Progesterone3Completed1
DB00178Ramipril3Completed1
DB00912Repaglinide3Completed1
DB00206Reserpine3Completed1
DB00412Rosiglitazone3Completed1
DB01098Rosuvastatin3Completed43
DB01098Rosuvastatin3Terminated3
DB01098Rosuvastatin3Unknown Status1
DB00641Simvastatin3Completed44
DB00641Simvastatin3Terminated5
DB11325Soy sterol3Completed1
DB05317TAK-4753Completed6
DB05317TAK-4753Terminated4
DB16336Tafolecimab3Completed1
DB16336Tafolecimab3Recruiting1
DB00966Telmisartan3Completed2
DB01162Terazosin3Completed1
DB12647Tocotrienol3Terminated1
DB06281Torcetrapib3Completed1
DB06281Torcetrapib3Terminated1
DB00384Triamterene3Completed1
DB00177Valsartan3Completed4
DB09302Alirocumab4Completed3
DB00381Amlodipine4Completed3
DB00381Amlodipine4Unknown Status1
DB01076Atorvastatin4Completed30
DB01076Atorvastatin4Terminated3
DB01076Atorvastatin4Unknown Status3
DB01393Bezafibrate4Completed1
DB00930Colesevelam4Completed6
DB00375Colestipol4Completed1
DB11874Crocin4Completed1
DB06292Dapagliflozin4Completed1
DB09303Evolocumab4Unknown Status2
DB09303Evolocumab4Withdrawn1
DB00973Ezetimibe4Completed29
DB00973Ezetimibe4Terminated3
DB00973Ezetimibe4Unknown Status5
DB01039Fenofibrate4Completed2
DB01095Fluvastatin4Completed2
DB01095Fluvastatin4Unknown Status1
DB14901Inclisiran4Active Not Recruiting1
DB11629Laropiprant4Completed2
DB00238Nevirapine4Completed1
DB00627Niacin4Completed3
DB11133Omega-3 fatty acids4Completed1
DB11133Omega-3 fatty acids4Unknown Status1
DB09539Omega-3-acid ethyl esters4Completed1
DB09539Omega-3-acid ethyl esters4Unknown Status1
DB00790Perindopril4Unknown Status1
DB08860Pitavastatin4Completed6
DB11097Plantago seed4Completed1
DB00175Pravastatin4Completed5
DB00175Pravastatin4Unknown Status1
DB00503Ritonavir4Completed1
DB01098Rosuvastatin4Active Not Recruiting1
DB01098Rosuvastatin4Completed11
DB01098Rosuvastatin4Terminated2
DB01098Rosuvastatin4Unknown Status2
DB00641Simvastatin4Completed21
DB00641Simvastatin4Terminated1
DB00641Simvastatin4Unknown Status2
DB00177Valsartan4Completed1
DB00945Acetylsalicylic acidNot AvailableCompleted2
DB09302AlirocumabNot AvailableRecruiting1
DB09302AlirocumabNot AvailableTerminated1
DB00381AmlodipineNot AvailableCompleted1
DB01060AmoxicillinNot AvailableCompleted1
DB01076AtorvastatinNot AvailableCompleted8
DB01076AtorvastatinNot AvailableUnknown Status1
DB11936Bempedoic acidNot AvailableCompleted1
DB11936Bempedoic acidNot AvailableRecruiting1
DB13015CardarineNot AvailableCompleted1
DB04540CholesterolNot AvailableRecruiting1
DB04540CholesterolNot AvailableTerminated1
DB01432CholestyramineNot AvailableCompleted1
DB00758ClopidogrelNot AvailableUnknown Status1
DB01394ColchicineNot AvailableRecruiting1
DB09303EvolocumabNot AvailableRecruiting1
DB00973EzetimibeNot AvailableCompleted12
DB00973EzetimibeNot AvailableRecruiting1
DB00973EzetimibeNot AvailableTerminated1
DB01095FluvastatinNot AvailableCompleted1
DB07215GW-590735Not AvailableCompleted1
DB14901InclisiranNot AvailableRecruiting2
DB11629LaropiprantNot AvailableTerminated1
DB00227LovastatinNot AvailableCompleted1
DB00331MetforminNot AvailableWithdrawn1
DB00627NiacinNot AvailableCompleted1
DB00627NiacinNot AvailableTerminated1
DB11220OctacosanolNot AvailableCompleted1
DB08860PitavastatinNot AvailableCompleted1
DB08860PitavastatinNot AvailableRecruiting1
DB08860PitavastatinNot AvailableTerminated1
DB00175PravastatinNot AvailableCompleted4
DB00175PravastatinNot AvailableTerminated1
DB01098RosuvastatinNot AvailableCompleted7
DB01098RosuvastatinNot AvailableTerminated1
DB01098RosuvastatinNot AvailableUnknown Status1
DB00641SimvastatinNot AvailableCompleted11
DB00641SimvastatinNot AvailableUnknown Status1
DB00300Tenofovir disoproxilNot AvailableCompleted1
DB00177ValsartanNot AvailableRecruiting1
DB14038beta-SitosterolNot AvailableCompleted1