Endometriosis

Also known as: Sigmoid endometriosis / Endometriosis, unspecified / Endometriosis (morphologic abnormality) / Endometriosis (disorder) / Endometriosis, site unspecified

DrugDrug NameDrug Description
DB06719BuserelinA LHRH agonist used for the palliative treatment of hormone-dependent advanced carcinoma of the prostate gland in males and treatment of endometriosis in females.
DB01406DanazolA synthetic steroid and pituitary gonadotropin inhibitor used in the treatment of endometriosis and symptomatic treatment of severe pain and tenderness associated with benign fibrocystic breasts.
DB09123DienogestAn oral progestin used for the treatment of endometriosis as monotherapy or contraception in combination with ethinylestradiol.
DB11979ElagolixA gonadotropin releasing hormone receptor antagonist used to treat moderate to severe pain in endometriosis.
DB00783EstradiolAn estrogenic steroid used to treat vasomotor symptoms of vulvar and vaginal atrophy in menopause, hypoestrogenism, prevention of postmenopausal osteoporosis, treatment of breast cancer, and advanced androgen-dependent carcinoma of the prostate.
DB00823Ethynodiol diacetateAn oral contraceptive used to prevent pregnancy.
DB00014GoserelinA synthetic analog of luteinizing hormone-releasing hormone used to treat breast cancer and prostate cancer by reducing secretion of gonadotropins from the pituitary.
DB00007LeuprolideA peptide-based GnRH receptor superagonist used for the palliative treatment of prostate cancer, uterine leiomyomata, endometriosis, and central precocious puberty.
DB00367LevonorgestrelA progestin found in oral and IUD contraceptives and at higher doses in emergency contraceptives.
DB12474LynestrenolA progestin used for contraception and in the treatment of menstrual disorders.
DB00603Medroxyprogesterone acetateA progestin used as a contraceptive and in the treatment of secondary amenorrhea, abnormal uterine bleeding, pain from endometriosis, endometrial and renal carcinomas, paraphilia in males, and GnRH-dependent precocious puberty.
DB01357MestranolA synthetic estradiol found in oral contraceptive pills for contraception and the treatment of other conditions in the female reproductive system, such as dysmenorrhea and dysfunctional uterine bleeding.
DB00666NafarelinA gonadotropin releasing hormone agonist used to treat central precocious puberty.
DB00717NorethisteroneA synthetic second-generation progestin used for contraception, prevention of endometrial hyperplasia in hormone replacement therapy, and in the treatment of other hormone-mediated illnesses such as endometriosis.
DB09389NorgestrelA progestin used in combination with ethinyl estradiol for oral contraception and prevention of pregnancy in women.
DB11853RelugolixAn oral GnRH receptor antagonist for androgen deprivation therapy in the treatment of advanced prostate cancer.
DrugDrug NameTargetType
DB06719BuserelinLutropin-choriogonadotropic hormone receptortarget
DB06719BuserelinGonadotropin-releasing hormone receptortarget
DB06719BuserelinCytochrome P450 19A1enzyme
DB01406DanazolEstrogen receptor alphatarget
DB01406DanazolGonadotropin-releasing hormone receptortarget
DB01406DanazolPutative gonadotropin-releasing hormone II receptortarget
DB01406DanazolSex hormone-binding globulincarrier
DB01406DanazolC-C motif chemokine 2target
DB01406DanazolCytochrome P450 19A1enzyme
DB01406DanazolAndrogen receptortarget
DB01406DanazolProgesterone receptortarget
DB01406DanazolCytochrome P450 3A4enzyme
DB09123DienogestCytochrome P450 3A4enzyme
DB09123DienogestProgesterone receptortarget
DB09123DienogestAndrogen receptortarget
DB11979ElagolixGonadotropin-releasing hormone receptortarget
DB11979ElagolixCytochrome P450 3A Subfamilyenzyme
DB11979ElagolixCytochrome P450 2D6enzyme
DB11979ElagolixCytochrome P450 2C8enzyme
DB11979ElagolixP-glycoprotein 1transporter
DB11979ElagolixSolute carrier organic anion transporter family member 1B1transporter
DB00783EstradiolEstrogen receptor alphatarget
DB00783EstradiolNuclear receptor subfamily 1 group I member 2target
DB00783EstradiolSex hormone-binding globulincarrier
DB00783EstradiolEstrogen receptor betatarget
DB00783EstradiolCytochrome P450 1A2enzyme
DB00783EstradiolUDP-glucuronosyltransferase 1-1enzyme
DB00783EstradiolSerum albumincarrier
DB00783EstradiolFatty acid-binding protein, intestinalcarrier
DB00783EstradiolCytochrome P450 3A4enzyme
DB00783EstradiolCytochrome P450 3A5enzyme
DB00783EstradiolCytochrome P450 3A7enzyme
DB00783EstradiolSolute carrier family 22 member 2transporter
DB00783EstradiolSolute carrier family 22 member 3transporter
DB00783EstradiolMultidrug resistance-associated protein 7transporter
DB00783EstradiolSolute carrier family 22 member 11transporter
DB00783EstradiolATP-binding cassette sub-family G member 2transporter
DB00783EstradiolSolute carrier organic anion transporter family member 1B1transporter
DB00783EstradiolP-glycoprotein 1transporter
DB00783EstradiolCytochrome P450 1A1enzyme
DB00783EstradiolCytochrome P450 1B1enzyme
DB00783EstradiolCytochrome P450 2C19enzyme
DB00783EstradiolCytochrome P450 2C8enzyme
DB00783EstradiolCytochrome P450 2C9enzyme
DB00783EstradiolSolute carrier family 22 member 8transporter
DB00783EstradiolSolute carrier organic anion transporter family member 1B3transporter
DB00783EstradiolSolute carrier organic anion transporter family member 1C1transporter
DB00783EstradiolNeuronal acetylcholine receptor subunit alpha-4target
DB00783EstradiolG-protein coupled estrogen receptor 1target
DB00783EstradiolATP synthase subunit atarget
DB00783EstradiolBeclin-1target
DB00783EstradiolUDP-glucuronosyltransferase 2B15enzyme
DB00783EstradiolCatechol O-methyltransferaseenzyme
DB00783EstradiolUDP-glucuronosyltransferases (UGTs)enzyme
DB00783EstradiolCytochrome P450 19A1enzyme
DB00823Ethynodiol diacetateEstrogen receptor alphatarget
DB00823Ethynodiol diacetateProgesterone receptortarget
DB00823Ethynodiol diacetateCytochrome P450 3A4enzyme
DB00014GoserelinLutropin-choriogonadotropic hormone receptortarget
DB00014GoserelinGonadotropin-releasing hormone receptortarget
DB00007LeuprolideGonadotropin-releasing hormone receptortarget
DB00367LevonorgestrelProgesterone receptortarget
DB00367LevonorgestrelEstrogen receptor alphatarget
DB00367Levonorgestrel3-oxo-5-alpha-steroid 4-dehydrogenase 1target
DB00367LevonorgestrelCytochrome P450 3A4enzyme
DB00367LevonorgestrelAndrogen receptortarget
DB00367LevonorgestrelSex hormone-binding globulintarget
DB00367LevonorgestrelGlucocorticoid receptortarget
DB00367LevonorgestrelCytochrome P450 3A5enzyme
DB12474LynestrenolCytochrome P450 3A4enzyme
DB12474LynestrenolCytochrome P450 2C9enzyme
DB12474LynestrenolCytochrome P450 2C19enzyme
DB00603Medroxyprogesterone acetateProgesterone receptortarget
DB00603Medroxyprogesterone acetateEstrogen receptor alphatarget
DB00603Medroxyprogesterone acetateCytochrome P450 3A4enzyme
DB00603Medroxyprogesterone acetateCytochrome P450 2C8enzyme
DB00603Medroxyprogesterone acetate3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2enzyme
DB00603Medroxyprogesterone acetateCytochrome P450 2C9enzyme
DB00603Medroxyprogesterone acetateCytochrome P450 3A1enzyme
DB00603Medroxyprogesterone acetateSerum albumincarrier
DB00603Medroxyprogesterone acetateP-glycoprotein 1target
DB00603Medroxyprogesterone acetateGABA(A) Receptortarget
DB00603Medroxyprogesterone acetateP-glycoprotein 1transporter
DB01357MestranolEstrogen receptor alphatarget
DB01357MestranolCytochrome P450 2C9enzyme
DB01357MestranolCytochrome P450 3A4enzyme
DB01357MestranolCytochrome P450 2C8enzyme
DB00666NafarelinGonadotropin-releasing hormone receptortarget
DB00666NafarelinPutative gonadotropin-releasing hormone II receptortarget
DB00717NorethisteroneProgesterone receptortarget
DB00717NorethisteroneP-glycoprotein 1transporter
DB00717NorethisteroneCytochrome P450 2C19enzyme
DB00717NorethisteroneSerum albumincarrier
DB00717NorethisteroneSex hormone-binding globulincarrier
DB00717NorethisteroneAldo-keto reductase family 1 member C4enzyme
DB00717Norethisterone3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2enzyme
DB00717Norethisterone3-oxo-5-alpha-steroid 4-dehydrogenaseenzyme
DB00717Norethisterone3-oxo-5-beta-steroid 4-dehydrogenaseenzyme
DB00717NorethisteroneCytochrome P450 3A4enzyme
DB00717NorethisteroneCytochrome P450 1A2enzyme
DB00717NorethisteroneCytochrome P450 2A6enzyme
DB00717NorethisteroneGlucocorticoid receptortarget
DB00717NorethisteroneAndrogen receptortarget
DB09389NorgestrelProgesterone receptortarget
DB09389Norgestrel3-oxo-5-alpha-steroid 4-dehydrogenase 1target
DB09389NorgestrelAndrogen receptortarget
DB09389NorgestrelCytochrome P450 3A4enzyme
DB09389NorgestrelCytochrome P450 19A1enzyme
DB11853RelugolixSerum albumincarrier
DB11853RelugolixAlpha-1-acid glycoprotein 1carrier
DB11853RelugolixP-glycoprotein 1transporter
DB11853RelugolixATP-binding cassette sub-family G member 2transporter
DB11853RelugolixCytochrome P450 3A Subfamilyenzyme
DB11853RelugolixCytochrome P450 2C8enzyme
DB11853RelugolixCytochrome P450 2B6enzyme
DB11853RelugolixGonadotropin-releasing hormone receptortarget
DrugDrug NamePhaseStatusCount
DB00026Anakinra0Recruiting1
DB09123Dienogest0Completed1
DB11979Elagolix0Active Not Recruiting1
DB11979Elagolix0Recruiting1
DB00898Ethanol0Completed1
DB16024Indocyanine green0Completed2
DB00007Leuprolide0Active Not Recruiting1
DB01399Salsalate0Recruiting1
DB01217Anastrozole1Completed1
DB01076Atorvastatin1Completed1
DB00112Bevacizumab1Unknown Status1
DB00196Fluconazole1Completed1
DB01221Ketamine1Recruiting1
DB00367Levonorgestrel1Completed1
DB01110Miconazole1Completed1
DB00683Midazolam1Completed2
DB00218Moxifloxacin1Completed1
DB11853Relugolix1Completed1
DB01045Rifampicin1Completed1
DB01041Thalidomide1Terminated1
DB11971Vilaprisan1Completed1
DB08916Afatinib1 / 2Withdrawn1
DB06626Axitinib1 / 2Withdrawn1
DB00050Cetrorelix1 / 2Completed1
DB00097Choriogonadotropin alfa1 / 2Completed1
DB09126Chorionic Gonadotropin (Human)1 / 2Completed1
DB15690Fluoroestradiol F-181 / 2Enrolling by Invitation1
DB00644Gonadorelin1 / 2Completed1
DB06080Linifanib1 / 2Withdrawn1
DB00603Medroxyprogesterone acetate1 / 2Completed1
DB00032Menotropins1 / 2Completed1
DB00666Nafarelin1 / 2Completed1
DB06825Triptorelin1 / 2Completed1
DB01217Anastrozole2Completed1
DB00126Ascorbic acid2Completed1
DB06680Asoprisnil2Completed3
DB09059Atosiban2Recruiting1
DB16851Bentamapimod2Completed1
DB00248Cabergoline2Completed1
DB00248Cabergoline2Recruiting1
DB00050Cetrorelix2Completed1
DB00286Conjugated estrogens2Completed1
DB01406Danazol2Completed2
DB09123Dienogest2Completed1
DB09123Dienogest2Withdrawn1
DB11074Dimethicone2Recruiting1
DB05694Elagolix2Completed1
DB11979Elagolix2Completed3
DB11979Elagolix2Terminated1
DB12116Epigallocatechin gallate2Completed1
DB00783Estradiol2Recruiting1
DB06597Estradiol sulfamate2Completed1
DB00977Ethinylestradiol2Completed1
DB00099Filgrastim2Unknown Status1
DB11242Gelatin2Not Yet Recruiting1
DB00644Gonadorelin2Completed1
DB14307Green tea leaf2Completed1
DB00065Infliximab2Completed1
DB01006Letrozole2Active Not Recruiting1
DB00007Leuprolide2Completed7
DB00007Leuprolide2Recruiting1
DB00367Levonorgestrel2Completed1
DB00281Lidocaine2Completed1
DB00281Lidocaine2Recruiting1
DB17083Linzagolix2Completed1
DB00603Medroxyprogesterone acetate2Completed1
DB01065Melatonin2Completed1
DB00916Metronidazole2Withdrawn1
DB00717Norethisterone2Completed3
DB00717Norethisterone2Not Yet Recruiting1
DB00957Norgestimate2Completed1
DB00540Nortriptyline2Recruiting1
DB11058Petrolatum2Recruiting1
DB06832Prinaberel2Completed2
DB09097Quinagolide2Completed1
DB00481Raloxifene2Completed1
DB11853Relugolix2Completed2
DB00412Rosiglitazone2Terminated1
DB11135Selenium2Completed1
DB13978Selisistat2Withdrawn1
DB12335Tanezumab2Terminated1
DB05253Telapristone acetate2Completed1
DB05253Telapristone acetate2Terminated2
DB05253Telapristone acetate2Withdrawn1
DB08653Tryptamine2Completed1
DB11971Vilaprisan2Terminated1
DB00163Vitamin E2Completed1
DB01593Zinc2Completed1
DB09123Dienogest2 / 3Recruiting1
DB09123Dienogest2 / 3Suspended1
DB01395Drospirenone2 / 3Recruiting1
DB00977Ethinylestradiol2 / 3Recruiting1
DB00977Ethinylestradiol2 / 3Suspended1
DB00644Gonadorelin2 / 3Recruiting1
DB00367Levonorgestrel2 / 3Suspended1
DB14009Medical Cannabis2 / 3Recruiting1
DB00834Mifepristone2 / 3Completed1
DB01132Pioglitazone2 / 3Withdrawn1
DB00412Rosiglitazone2 / 3Withdrawn1
DB06825Triptorelin2 / 3Recruiting1
DB09061Cannabidiol3Recruiting1
DB04839Cyproterone acetate3Unknown Status1
DB01406Danazol3Recruiting1
DB06699Degarelix3Completed1
DB09123Dienogest3Completed4
DB09123Dienogest3Recruiting1
DB01395Drospirenone3Completed1
DB11979Elagolix3Completed5
DB11979Elagolix3Recruiting4
DB11979Elagolix3Terminated1
DB00783Estradiol3Completed2
DB00783Estradiol3Recruiting1
DB00783Estradiol3Terminated1
DB00783Estradiol3Unknown Status1
DB00644Gonadorelin3Recruiting1
DB00644Gonadorelin3Unknown Status2
DB01221Ketamine3Recruiting1
DB00007Leuprolide3Completed3
DB00007Leuprolide3Unknown Status1
DB17083Linzagolix3Active Not Recruiting1
DB17083Linzagolix3Completed1
DB17083Linzagolix3Terminated2
DB00704Naltrexone3Terminated1
DB00717Norethisterone3Completed3
DB00717Norethisterone3Recruiting2
DB00717Norethisterone3Terminated2
DB00717Norethisterone3Unknown Status1
DB00396Progesterone3Unknown Status1
DB11853Relugolix3Completed2
DB11853Relugolix3Recruiting1
DB06825Triptorelin3Completed1
DB06825Triptorelin3Unknown Status2
DB00945Acetylsalicylic acid4Recruiting1
DB01217Anastrozole4Completed1
DB01076Atorvastatin4Suspended1
DB06401Bazedoxifene4Recruiting1
DB06724Calcium carbonate4Not Yet Recruiting1
DB13528Chlormadinone4Unknown Status1
DB00169Cholecalciferol4Not Yet Recruiting1
DB00575Clonidine4Recruiting1
DB01406Danazol4Completed1
DB09123Dienogest4Recruiting1
DB09123Dienogest4Unknown Status1
DB00783Estradiol4Completed1
DB00783Estradiol4Recruiting1
DB00783Estradiol4Unknown Status1
DB00898Ethanol4Completed1
DB00977Ethinylestradiol4Completed2
DB00977Ethinylestradiol4Not Yet Recruiting1
DB00977Ethinylestradiol4Unknown Status1
DB00294Etonogestrel4Completed1
DB06730Gestodene4Completed1
DB00644Gonadorelin4Completed1
DB00644Gonadorelin4Not Yet Recruiting1
DB00644Gonadorelin4Recruiting1
DB00014Goserelin4Completed2
DB00014Goserelin4Recruiting1
DB00014Goserelin4Unknown Status1
DB00007Leuprolide4Completed2
DB00007Leuprolide4Not Yet Recruiting1
DB00367Levonorgestrel4Completed2
DB00367Levonorgestrel4Unknown Status1
DB00603Medroxyprogesterone acetate4Completed1
DB14123Menthol4Unknown Status1
DB00916Metronidazole4Recruiting1
DB00717Norethisterone4Completed1
DB02709Resveratrol4Completed1
DB00728Rocuronium4Completed1
DB00641Simvastatin4Recruiting1
DB09070Tibolone4Not Yet Recruiting1
DB06825Triptorelin4Completed2
DB08867Ulipristal4Unknown Status1
DB11094Vitamin D4Unknown Status1
DB01076AtorvastatinNot AvailableUnknown Status1
DB00882ClomifeneNot AvailableWithdrawn1
DB00304DesogestrelNot AvailableCompleted1
DB00304DesogestrelNot AvailableUnknown Status1
DB08809Dichloroacetic acidNot AvailableUnknown Status1
DB09123DienogestNot AvailableCompleted8
DB09123DienogestNot AvailableRecruiting1
DB09123DienogestNot AvailableUnknown Status1
DB01075DiphenhydramineNot AvailableCompleted1
DB00378DydrogesteroneNot AvailableCompleted3
DB00898EthanolNot AvailableUnknown Status1
DB00977EthinylestradiolNot AvailableUnknown Status2
DB00644GonadorelinNot AvailableCompleted5
DB00644GonadorelinNot AvailableRecruiting1
DB00644GonadorelinNot AvailableUnknown Status1
DB00014GoserelinNot AvailableCompleted1
DB00581LactuloseNot AvailableCompleted1
DB01006LetrozoleNot AvailableCompleted1
DB00007LeuprolideNot AvailableCompleted4
DB00281LidocaineNot AvailableCompleted1
DB00742MannitolNot AvailableCompleted1
DB00717NorethisteroneNot AvailableCompleted1
DB14043PalmidrolNot AvailableCompleted1
DB00175PravastatinNot AvailableNot Yet Recruiting1
DB00175PravastatinNot AvailableWithdrawn1
DB00296RopivacaineNot AvailableWithdrawn1
DB09070TiboloneNot AvailableNot Yet Recruiting1
DB06825TriptorelinNot AvailableRecruiting1
DB06825TriptorelinNot AvailableUnknown Status1