Showing BioInteractions for Relebactam (DB12377)
BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting Group | Interacting Drugs | |
---|---|---|
Relebactam is a Beta-lactamase TEM inhibitor | ||
1 | Beta-lactamase TEM inhibitors | Avibactam, Vaborbactam |
2 | Beta-lactamase TEM substrates | Benzylpenicillin, Imipenem |
Interacting Group | Interacting Drugs | |
---|---|---|
Relebactam is a Beta-lactamase SHV-1 inhibitor | ||
1 | Beta-lactamase SHV-1 inhibitors | Avibactam, Tazobactam |
2 | Beta-lactamase SHV-1 substrates | Imipenem |
Interacting Group | Interacting Drugs | |
---|---|---|
Relebactam is a Beta-lactamase CTX-M inhibitor | ||
1 | Beta-lactamase CTX-M inhibitors | Avibactam, Vaborbactam |
2 | Beta-lactamase CTX-M substrates | Imipenem |
Interacting Group | Interacting Drugs | |
---|---|---|
Relebactam is a Beta-lactamase (KPC-2) inhibitor | ||
1 | Beta-lactamase (KPC-2) inhibitors | Vaborbactam |
2 | Beta-lactamase (KPC-2) substrates | Imipenem |
Interacting Group | Interacting Drugs | |
---|---|---|
Relebactam is a Beta-lactamase inhibitor | ||
1 | Beta-lactamase inhibitors | Avibactam, Vaborbactam |
Interacting Group | Interacting Drugs | |
---|---|---|
Relebactam is a Solute carrier family 22 member 11 substrate | ||
1 | Solute carrier family 22 member 11 inhibitors | Aminohippuric acid, Aspartame, Benzylpenicillin, Bumetanide, Caprylic acid, Cefalotin, Cefamandole, Cefazolin, Cefoperazone, Cefotaxime, Ceftriaxone, Cimetidine, Diclofenac, Dinoprostone, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Furosemide, Glutaric Acid, Ibuprofen, Indomethacin, Ketoprofen, Lesinurad, Novobiocin, Oxytetracycline, Phenylbutazone, Piroxicam, Probenecid, Salicylic acid, Tetracycline |
2 | Solute carrier family 22 member 11 substrates | Aminohippuric acid, Conjugated estrogens, Hydrochlorothiazide, Levocetirizine, Methotrexate, Oxytetracycline, Pravastatin |
Interacting Group | Interacting Drugs | |
---|---|---|
Relebactam is a Multidrug and toxin extrusion protein 1 substrate | ||
1 | Multidrug and toxin extrusion protein 1 substrates | Acyclovir, Cefradine, Cephalexin, Cimetidine, Ciprofloxacin, Emtricitabine, Estrone sulfate, Flecainide, Ganciclovir, Guanidine, Levofloxacin, Metformin, N-methylnicotinamide, Nadolol, Procainamide, Tetraethylammonium, Tipiracil, Topotecan, Trimethoprim |
2 | Multidrug and toxin extrusion protein 1 inhibitors | Abemaciclib, Apalutamide, Bictegravir, Brigatinib, Capmatinib, Cimetidine, Ciprofloxacin, Famotidine, Fedratinib, Flecainide, Gilteritinib, Glasdegib, Guanfacine, Istradefylline, Lasmiditan, Levofloxacin, Lofexidine, Methylene blue, Osilodrostat, Pemigatinib, Pexidartinib, Plazomicin, Pralsetinib, Pyrimethamine, Ranolazine, Remdesivir, Rifamycin, Rimegepant, Ripretinib, Risdiplam, Rucaparib, Selpercatinib, Tafenoquine, Tazemetostat, Tirbanibulin, Topotecan, Trimethoprim, Tucatinib, Verapamil |
Interacting Group | Interacting Drugs | |
---|---|---|
Relebactam is a Multidrug and toxin extrusion protein 2 substrate | ||
1 | Multidrug and toxin extrusion protein 2 substrates | Acyclovir, Baricitinib, Cimetidine, Estrone sulfate, Ganciclovir, Metformin, N-methylnicotinamide, Nadolol, Procainamide, Topotecan, Trastuzumab deruxtecan, Trimethoprim |
2 | Multidrug and toxin extrusion protein 2 inhibitors | Abemaciclib, Apalutamide, Baricitinib, Brigatinib, Capmatinib, Cimetidine, Ciprofloxacin, Copanlisib, Fedratinib, Glasdegib, Istradefylline, Lasmiditan, Levofloxacin, Methylene blue, Pexidartinib, Plazomicin, Pralsetinib, Pyrimethamine, Ranolazine, Risdiplam, Rucaparib, Tafenoquine, Tazemetostat, Tirbanibulin, Trimethoprim, Tucatinib, Verapamil |