Showing BioInteractions for Pizotifen (DB06153)
BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting Group | Interacting Drugs | |
---|---|---|
Pizotifen is a 5-hydroxytryptamine receptor 2B antagonist | ||
1 | 5-hydroxytryptamine receptor 2B antagonists | Amoxapine, Asenapine, Cariprazine, Clomipramine, Cyclobenzaprine, Doxepin, Lisuride, Methysergide, Minaprine, PRX-08066, Tegaserod, Triflupromazine, Yohimbine |
2 | 5-hydroxytryptamine receptor 2B agonists | Apomorphine, Bromocriptine, Cabergoline, Dihydroergotamine, Fenfluramine, Lysergic acid diethylamide, Midomafetamine, Paroxetine, Pergolide, Zolmitriptan |
3 | 5-hydroxytryptamine receptor 2B binders | Mianserin |
4 | 5-hydroxytryptamine receptor 2B inverse agonists | Aripiprazole |
Interacting Group | Interacting Drugs | |
---|---|---|
Pizotifen is a 5-hydroxytryptamine receptor 1B antagonist | ||
1 | 5-hydroxytryptamine receptor 1B agonists | Almotriptan, Apomorphine, Bromocriptine, Cabergoline, Dihydroergotamine, Eletriptan, Ergotamine, Frovatriptan, Lisuride, Naratriptan, Oxymetazoline, Pergolide, Rizatriptan, Sumatriptan, Zolmitriptan |
2 | 5-hydroxytryptamine receptor 1B antagonists | Amoxapine, Aripiprazole, Asenapine, Clozapine, Penbutolol, Ziprasidone |
3 | 5-hydroxytryptamine receptor 1B ligands | Aripiprazole, Quetiapine |
4 | 5-hydroxytryptamine receptor 1B partial agonists | Vortioxetine, Yohimbine |
5 | 5-hydroxytryptamine receptor 1B binders | Amitriptyline, Loxapine, Methysergide |
Interacting Group | Interacting Drugs | |
---|---|---|
Pizotifen is a 5-hydroxytryptamine receptor 1D antagonist | ||
1 | 5-hydroxytryptamine receptor 1D agonists | Almotriptan, Apomorphine, Bromocriptine, Cabergoline, Dihydroergotamine, Eletriptan, Ergotamine, Fenfluramine, Frovatriptan, Lisuride, Lofexidine, Naratriptan, Oxymetazoline, Pergolide, Rizatriptan, Sumatriptan, Zolmitriptan |
2 | 5-hydroxytryptamine receptor 1D antagonists | Aripiprazole, Clozapine, Paliperidone, Risperidone, Ziprasidone |
3 | 5-hydroxytryptamine receptor 1D ligands | Aripiprazole, Quetiapine |
4 | 5-hydroxytryptamine receptor 1D partial agonists | Yohimbine |
5 | 5-hydroxytryptamine receptor 1D binders | Amitriptyline, Loxapine, Trimipramine |
Interacting Group | Interacting Drugs | |
---|---|---|
Pizotifen is a Alpha-1B adrenergic receptor antagonist | ||
1 | Alpha-1B adrenergic receptor antagonists | Acepromazine, Alfuzosin, Amitriptyline, Aripiprazole, Aripiprazole lauroxil, Brexpiprazole, Bromocriptine, Carvedilol, Chlorpromazine, Clozapine, Dapiprazole, Dextroamphetamine, Doxepin, Dronedarone, Imipramine, Methotrimeprazine, Nicardipine, Nortriptyline, Olanzapine, Paliperidone, Periciazine, Phenoxybenzamine, Phentolamine, Prazosin, Quinidine, Risperidone, Silodosin, Tamsulosin, Terazosin, Thioproperazine, Thioridazine, Trimipramine, Verapamil, Ziprasidone |
2 | Alpha-1B adrenergic receptor partial agonists | Cirazoline, Ergotamine, Modafinil |
3 | Alpha-1B adrenergic receptor agonists | Bromocriptine, Clonidine, Droxidopa, Epinephrine, Methoxamine, Midodrine, Norepinephrine, Oxymetazoline, Pergolide, Phendimetrazine, Phenylephrine, Racepinephrine, Xylometazoline |
4 | Alpha-1B adrenergic receptor binders | Cabergoline, Loxapine |
5 | Alpha-1B adrenergic receptor inhibitors | Fenoldopam |
Interacting Group | Interacting Drugs | |
---|---|---|
Pizotifen is a Alpha-1D adrenergic receptor antagonist | ||
1 | Alpha-1D adrenergic receptor antagonists | Alfuzosin, Amitriptyline, Carvedilol, Dapiprazole, Doxazosin, Doxepin, Dronedarone, Epinephrine, Imipramine, Methotrimeprazine, Nicardipine, Nortriptyline, Phenoxybenzamine, Phentolamine, Prazosin, Quinidine, Racepinephrine, Silodosin, Tamsulosin, Terazosin, Verapamil |
2 | Alpha-1D adrenergic receptor agonists | Bromocriptine, Clonidine, Droxidopa, Midodrine, Norepinephrine, Oxymetazoline, Pergolide, Phenylephrine, Xylometazoline |
3 | Alpha-1D adrenergic receptor partial agonists | Cirazoline, Ergotamine |
4 | Alpha-1D adrenergic receptor inhibitors | Fenoldopam |
5 | Alpha-1D adrenergic receptor binders | Cabergoline, Methoxamine |
Interacting Group | Interacting Drugs | |
---|---|---|
Pizotifen is a Alpha-2B adrenergic receptor antagonist | ||
1 | Alpha-2B adrenergic receptor antagonists | Aripiprazole, Asenapine, Cabergoline, Carvedilol, Celiprolol, Clozapine, Dronedarone, Fenoldopam, Methotrimeprazine, Mianserin, Paliperidone, Phenoxybenzamine, Quetiapine, Risperidone, Rotigotine, Yohimbine, Ziprasidone |
2 | Alpha-2B adrenergic receptor agonists | Apomorphine, Apraclonidine, Brimonidine, Bromocriptine, Clonidine, Droxidopa, Ephedra sinica root, Epinephrine, Etomidate, Metamfetamine, Norepinephrine, Oxymetazoline, Racepinephrine, Xylometazoline |
3 | Alpha-2B adrenergic receptor ligands | Aripiprazole |
4 | Alpha-2B adrenergic receptor binders | Guanabenz, Guanfacine, Loxapine, Prazosin, Tolazoline |
Interacting Group | Interacting Drugs | |
---|---|---|
Pizotifen is a Alpha-2C adrenergic receptor antagonist | ||
1 | Alpha-2C adrenergic receptor antagonists | Aripiprazole, Asenapine, Brexpiprazole, Cabergoline, Carvedilol, Celiprolol, Clozapine, Dronedarone, Fenoldopam, Iloperidone, Lurasidone, Methotrimeprazine, Mianserin, Phenoxybenzamine, Quetiapine, Risperidone, Yohimbine, Ziprasidone |
2 | Alpha-2C adrenergic receptor agonists | Agmatine, Apomorphine, Brimonidine, Bromocriptine, Clonidine, Droxidopa, Ephedra sinica root, Metamfetamine, Norepinephrine, Oxymetazoline, Paliperidone, Racepinephrine, Xylometazoline |
3 | Alpha-2C adrenergic receptor binders | Loxapine, Tolazoline |
Interacting Group | Interacting Drugs | |
---|---|---|
Pizotifen is a UDP-glucuronosyltransferase 2B10 substrate | ||
1 | UDP-glucuronosyltransferase 2B10 substrates | Amitriptyline, Cyclobenzaprine, Ketotifen, Osilodrostat |
2 | UDP-glucuronosyltransferase 2B10 inhibitors | Amitriptyline |