Atherosclerosis

Also known as: Atherosclerotic Disease / Atherosclerotic heart disease of native coronary artery / Atherosclerosis (morphologic abnormality) / Atheromatosis / Atherosclerotic cardiovascular disease / Arteriosclerotic vascular disease (disorder) / Arteriosclerosis / Arteriosclerosis (morphologic abnormality) / Vascular sclerosis (morphologic abnormality) / Senile endarteritis (disorder) / Senile arteritis (disorder) / Arteriovascular degeneration (disorder) / Atheromatous degeneration (morphologic abnormality) / Atheroma of artery (disorder) / Atheroma (morphologic abnormality) / Atheroma / Arteriolosclerosis / Arteriolosclerosis (morphologic abnormality) / Vascular degeneration (disorder)

DrugDrug NameDrug Description
DB01432CholestyramineA bile acid sequestrant used as an adjunct in the reduction of elevated serum cholesterol in patients with primary hypercholesterolemia, and for the relief of pruritus associated with partial biliary obstruction.
DB01095FluvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
DB00627NiacinA B vitamin used to treat hypertriglyceridemia and pellagra.
DB13327PicotamideA platelet aggregation inhibitor indicated in the treatment of myocardial infarction, thrombosis, cerebrovascular disorders, pulmonary emboli, and atherosclerosis.
DB01098RosuvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
DrugDrug NameTargetType
DB01432CholestyramineBile acidstarget
DB01095Fluvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
DB01095FluvastatinCytochrome P450 2C9enzyme
DB01095FluvastatinCytochrome P450 3A4enzyme
DB01095FluvastatinCytochrome P450 2C8enzyme
DB01095FluvastatinCytochrome P450 2D6enzyme
DB01095FluvastatinCytochrome P450 2C19enzyme
DB01095FluvastatinCytochrome P450 1A1enzyme
DB01095FluvastatinSolute carrier organic anion transporter family member 1B1transporter
DB01095FluvastatinSolute carrier organic anion transporter family member 1B3transporter
DB01095FluvastatinSolute carrier organic anion transporter family member 2B1transporter
DB01095FluvastatinSolute carrier family 15 member 1transporter
DB01095FluvastatinCytochrome P450 3A5enzyme
DB01095FluvastatinUDP-glucuronosyltransferase 1-1enzyme
DB01095FluvastatinUDP-glucuronosyltransferase 1-3enzyme
DB01095FluvastatinUDP-glucuronosyltransferase 2B7enzyme
DB01095FluvastatinCanalicular multispecific organic anion transporter 1transporter
DB01095FluvastatinCytochrome P450 2B6enzyme
DB01095FluvastatinHistone deacetylase 2target
DB00627NiacinHydroxycarboxylic acid receptor 2target
DB00627NiacinNicotinamide N-methyltransferasetarget
DB00627NiacinNicotinate-nucleotide pyrophosphorylase [carboxylating]target
DB00627NiacinHydroxycarboxylic acid receptor 3target
DB00627NiacinSolute carrier family 22 member 5transporter
DB00627NiacinSolute carrier organic anion transporter family member 2B1transporter
DB00627NiacinMonocarboxylate transporter 1transporter
DB00627NiacinCytochrome P450 2D6enzyme
DB00627NiacinSodium-coupled monocarboxylate transporter 1transporter
DB00627NiacinMonocarboxylate transporter 4transporter
DB00627NiacinThyroxine-binding globulincarrier
DB00627NiacinCytochrome P450 3A4enzyme
DB00627NiacinCytochrome P450 2E1enzyme
DB01098Rosuvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
DB01098RosuvastatinCytochrome P450 2C9enzyme
DB01098RosuvastatinMultidrug resistance-associated protein 4transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1A2transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1B3transporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 2B1transporter
DB01098RosuvastatinCystine/glutamate transportertransporter
DB01098RosuvastatinSolute carrier organic anion transporter family member 1B1transporter
DB01098RosuvastatinBile salt export pumptransporter
DB01098RosuvastatinATP-binding cassette sub-family G member 2transporter
DB01098RosuvastatinSerum albumincarrier
DB01098RosuvastatinCanalicular multispecific organic anion transporter 1transporter
DB01098RosuvastatinSolute carrier family 22 member 8transporter
DB01098RosuvastatinSodium/bile acid cotransportertransporter
DB01098RosuvastatinIntegrin alpha-Ltarget
DrugDrug NamePhaseStatusCount
DB11827Ertugliflozin0Active Not Recruiting1
DB00973Ezetimibe0Unknown Status1
DB01067Glipizide0Active Not Recruiting1
DB00635Prednisone0Completed1
DB01098Rosuvastatin0Completed2
DB00641Simvastatin0Unknown Status1
DB00945Acetylsalicylic acid1Completed1
DB09302Alirocumab1Completed1
DB00758Clopidogrel1Completed1
DB01394Colchicine1Recruiting1
DB06311Darapladib1Completed13
DB00343Diltiazem1Completed1
DB00973Ezetimibe1Completed1
DB06705Gadofosveset trisodium1Completed1
DB16024Indocyanine green1Completed1
DB12270Losmapimod1Completed2
DB14833MEDI60121Completed1
DB00683Midazolam1Completed1
DB05119Rilapladib1Completed3
DB01098Rosuvastatin1Completed2
DB09153Sodium chloride1Terminated1
DB12000Apabetalone1 / 2Completed1
DB00125Arginine1 / 2Unknown Status1
DB00959Methylprednisolone1 / 2Unknown Status1
DB14644Methylprednisolone hemisuccinate1 / 2Unknown Status1
DB00860Prednisolone1 / 2Unknown Status1
DB14631Prednisolone phosphate1 / 2Unknown Status1
DB00945Acetylsalicylic acid2Active Not Recruiting1
DB00945Acetylsalicylic acid2Completed1
DB12000Apabetalone2Completed1
DB00126Ascorbic acid2Terminated1
DB01076Atorvastatin2Recruiting1
DB12758Atreleuton2Completed1
DB06401Bazedoxifene2Recruiting1
DB11936Bempedoic acid2Recruiting1
DB06168Canakinumab2Completed1
DB00608Chloroquine2Completed1
DB00169Cholecalciferol2Completed1
DB00758Clopidogrel2Active Not Recruiting1
DB00758Clopidogrel2Completed2
DB01394Colchicine2Not Yet Recruiting1
DB00286Conjugated estrogens2Recruiting1
DB06311Darapladib2Completed4
DB00783Estradiol2Completed3
DB12469Fasudil2Completed1
DB01611Hydroxychloroquine2Completed1
DB16956L-Acetylleucine2Completed2
DB12270Losmapimod2Completed1
DB00227Lovastatin2Completed1
DB14833MEDI60122Completed1
DB15381Menaquinone2Unknown Status1
DB14936Menaquinone 62Unknown Status1
DB09112Nitrous acid2Unknown Status1
DB16653Orticumab2Completed1
DB12971Pactimibe2Completed1
DB00806Pentoxifylline2Completed2
DB12520Plozalizumab2Completed1
DB06209Prasugrel2Active Not Recruiting1
DB00396Progesterone2Completed1
DB00178Ramipril2Completed1
DB05119Rilapladib2Completed1
DB06372Rilonacept2Completed1
DB01098Rosuvastatin2Completed1
DB00203Sildenafil2Terminated1
DB01261Sitagliptin2Completed1
DB09153Sodium chloride2Unknown Status1
DB08816Ticagrelor2Active Not Recruiting1
DB00177Valsartan2Completed1
DB00163Vitamin E2Terminated1
DB09030Vorapaxar2Completed1
DB00945Acetylsalicylic acid2 / 3Unknown Status1
DB09026Aliskiren2 / 3Terminated1
DB00115Cyanocobalamin2 / 3Completed1
DB14476DL-alpha-Tocopherol2 / 3Completed1
DB00783Estradiol2 / 3Completed1
DB15058Flutemetamol2 / 3Unknown Status1
DB00158Folic acid2 / 3Completed1
DB00227Lovastatin2 / 3Completed1
DB00563Methotrexate2 / 3Recruiting1
DB01229Paclitaxel2 / 3Unknown Status1
DB00635Prednisone2 / 3Completed1
DB00165Pyridoxine2 / 3Completed1
DB01399Salsalate2 / 3Completed2
DB00197Troglitazone2 / 3Completed1
DB00284Acarbose3Completed1
DB00945Acetylsalicylic acid3Recruiting1
DB00945Acetylsalicylic acid3Terminated1
DB00945Acetylsalicylic acid3Unknown Status1
DB09302Alirocumab3Unknown Status1
DB00381Amlodipine3Completed2
DB11842Angiotensin II3Completed2
DB01076Atorvastatin3Completed7
DB01076Atorvastatin3Recruiting1
DB11936Bempedoic acid3Completed1
DB00542Benazepril3Completed1
DB06168Canakinumab3Completed1
DB00796Candesartan cilexetil3Completed2
DB06441Cangrelor3Completed1
DB06441Cangrelor3Terminated1
DB01136Carvedilol3Completed1
DB00310Chlorthalidone3Completed1
DB01166Cilostazol3Unknown Status1
DB00758Clopidogrel3Completed1
DB00758Clopidogrel3Terminated1
DB00758Clopidogrel3Unknown Status1
DB01394Colchicine3Recruiting2
DB00375Colestipol3Completed1
DB06311Darapladib3Completed1
DB00343Diltiazem3Completed1
DB00973Ezetimibe3Completed8
DB00973Ezetimibe3Terminated1
DB01023Felodipine3Completed1
DB01039Fenofibrate3Completed1
DB01095Fluvastatin3Completed1
DB00695Furosemide3Completed1
DB00222Glimepiride3Completed1
DB01067Glipizide3Completed1
DB01275Hydralazine3Completed1
DB00999Hydrochlorothiazide3Completed1
DB01306Insulin aspart3Completed1
DB01307Insulin detemir3Completed1
DB00047Insulin glargine3Completed1
DB00030Insulin human3Completed1
DB01249Iodixanol3Completed1
DB00722Lisinopril3Completed1
DB00331Metformin3Completed1
DB00264Metoprolol3Completed1
DB05528Mipomersen3Completed1
DB00688Mycophenolate mofetil3Terminated1
DB00627Niacin3Completed2
DB00627Niacin3Terminated1
DB00275Olmesartan3Completed1
DB01229Paclitaxel3Completed1
DB01132Pioglitazone3Completed1
DB00175Pravastatin3Completed1
DB00635Prednisone3Terminated1
DB00178Ramipril3Completed2
DB00912Repaglinide3Completed1
DB00206Reserpine3Completed1
DB00412Rosiglitazone3Completed3
DB01098Rosuvastatin3Completed7
DB00641Simvastatin3Completed5
DB00641Simvastatin3Terminated2
DB00877Sirolimus3Terminated1
DB11104Sulfur hexafluoride3Completed1
DB00864Tacrolimus3Terminated1
DB01162Terazosin3Completed1
DB08816Ticagrelor3Recruiting1
DB00302Tranexamic acid3Completed1
DB00384Triamterene3Completed1
DB00177Valsartan3Completed1
DB09030Vorapaxar3Completed2
DB05692Vorapaxar3Terminated1
DB09030Vorapaxar3Terminated1
DB00682Warfarin3Terminated1
DB06151Acetylcysteine4Unknown Status1
DB00945Acetylsalicylic acid4Completed7
DB00945Acetylsalicylic acid4Recruiting1
DB00945Acetylsalicylic acid4Suspended1
DB00945Acetylsalicylic acid4Terminated1
DB00945Acetylsalicylic acid4Unknown Status1
DB09302Alirocumab4Unknown Status1
DB00381Amlodipine4Terminated1
DB00335Atenolol4Completed2
DB01076Atorvastatin4Completed6
DB01076Atorvastatin4Recruiting1
DB01076Atorvastatin4Terminated3
DB01076Atorvastatin4Unknown Status3
DB01076Atorvastatin4Withdrawn1
DB13100Biguanide4Completed1
DB00201Caffeine4Completed1
DB01166Cilostazol4Completed1
DB00758Clopidogrel4Completed3
DB00758Clopidogrel4Suspended1
DB00758Clopidogrel4Unknown Status1
DB00758Clopidogrel4Withdrawn1
DB01394Colchicine4Recruiting1
DB00930Colesevelam4Completed1
DB00115Cyanocobalamin4Unknown Status1
DB14726Dabigatran4Terminated1
DB00514Dextromethorphan4Completed1
DB00975Dipyridamole4Completed2
DB00584Enalapril4Unknown Status1
DB00016Erythropoietin4Terminated1
DB00783Estradiol4Recruiting1
DB09303Evolocumab4Recruiting1
DB09303Evolocumab4Terminated1
DB01276Exenatide4Completed1
DB00973Ezetimibe4Completed7
DB00973Ezetimibe4Recruiting1
DB00973Ezetimibe4Terminated4
DB13873Fenofibric acid4Recruiting1
DB09279Fimasartan4Recruiting1
DB09398Fluoride ion F-184Completed1
DB01095Fluvastatin4Unknown Status1
DB00158Folic acid4Unknown Status1
DB01241Gemfibrozil4Withdrawn1
DB01611Hydroxychloroquine4Unknown Status1
DB08887Icosapent ethyl4Terminated1
DB01306Insulin aspart4Completed2
DB01307Insulin detemir4Completed1
DB00030Insulin human4Completed1
DB11629Laropiprant4Terminated1
DB00451Levothyroxine4Completed2
DB00722Lisinopril4Completed1
DB00678Losartan4Terminated1
DB04835Maraviroc4Completed1
DB00331Metformin4Completed3
DB00331Metformin4Recruiting1
DB00264Metoprolol4Completed1
DB09282Molsidomine4Completed1
DB00688Mycophenolate mofetil4Completed1
DB00688Mycophenolate mofetil4Unknown Status1
DB04861Nebivolol4Completed1
DB00627Niacin4Completed2
DB00627Niacin4Terminated2
DB00627Niacin4Unknown Status1
DB09539Omega-3-acid ethyl esters4Completed1
DB00946Phenprocoumon4Terminated1
DB01132Pioglitazone4Terminated1
DB08860Pitavastatin4Completed1
DB00571Propranolol4Completed1
DB00165Pyridoxine4Unknown Status1
DB00178Ramipril4Completed1
DB06155Rimonabant4Unknown Status1
DB06228Rivaroxaban4Completed1
DB01098Rosuvastatin4Completed6
DB01098Rosuvastatin4Terminated3
DB01098Rosuvastatin4Unknown Status1
DB11767Sarilumab4Unknown Status1
DB13928Semaglutide4Recruiting1
DB00641Simvastatin4Completed5
DB00641Simvastatin4Terminated1
DB00641Simvastatin4Unknown Status2
DB01261Sitagliptin4Completed2
DB00421Spironolactone4Completed1
DB00624Testosterone4Completed1
DB08816Ticagrelor4Completed1
DB08816Ticagrelor4Suspended1
DB08816Ticagrelor4Withdrawn1
DB15171Tirzepatide4Recruiting1
DB00162Vitamin A4Unknown Status2
DB00682Warfarin4Completed1
DB00054AbciximabNot AvailableCompleted1
DB15111Acetic acid C-11Not AvailableRecruiting1
DB03128AcetylcholineNot AvailableUnknown Status1
DB00945Acetylsalicylic acidNot AvailableCompleted3
DB00945Acetylsalicylic acidNot AvailableWithdrawn1
DB00051AdalimumabNot AvailableCompleted1
DB00640AdenosineNot AvailableUnknown Status1
DB09302AlirocumabNot AvailableActive Not Recruiting1
DB09026AliskirenNot AvailableUnknown Status1
DB11842Angiotensin IINot AvailableUnknown Status1
DB01076AtorvastatinNot AvailableActive Not Recruiting1
DB01076AtorvastatinNot AvailableCompleted4
DB01076AtorvastatinNot AvailableUnknown Status1
DB01076AtorvastatinNot AvailableWithdrawn1
DB00169CholecalciferolNot AvailableCompleted1
DB00758ClopidogrelNot AvailableCompleted1
DB01394ColchicineNot AvailableRecruiting1
DB00975DipyridamoleNot AvailableCompleted1
DB00584EnalaprilNot AvailableUnknown Status1
DB00005EtanerceptNot AvailableCompleted1
DB00973EzetimibeNot AvailableActive Not Recruiting1
DB00973EzetimibeNot AvailableWithdrawn1
DB01039FenofibrateNot AvailableCompleted1
DB00813FentanylNot AvailableWithdrawn1
DB13961Fish oilNot AvailableCompleted1
DB01095FluvastatinNot AvailableCompleted1
DB00158Folic acidNot AvailableCompleted1
DB00222GlimepirideNot AvailableCompleted1
DB01109HeparinNot AvailableWithdrawn1
DB14901InclisiranNot AvailableRecruiting1
DB00065InfliximabNot AvailableCompleted1
DB00678LosartanNot AvailableUnknown Status2
DB00563MethotrexateNot AvailableCompleted1
DB00683MidazolamNot AvailableWithdrawn1
DB00627NiacinNot AvailableCompleted3
DB00627NiacinNot AvailableTerminated1
DB00627NiacinNot AvailableUnknown Status1
DB01229PaclitaxelNot AvailableCompleted1
DB01132PioglitazoneNot AvailableCompleted2
DB14317PomegranateNot AvailableUnknown Status1
DB14500PotassiumNot AvailableRecruiting1
DB06228RivaroxabanNot AvailableCompleted1
DB00412RosiglitazoneNot AvailableCompleted1
DB01098RosuvastatinNot AvailableActive Not Recruiting1
DB01098RosuvastatinNot AvailableCompleted2
DB01098RosuvastatinNot AvailableWithdrawn1
DB12163SarpogrelateNot AvailableUnknown Status1
DB13928SemaglutideNot AvailableRecruiting1
DB00658SevelamerNot AvailableTerminated1
DB00641SimvastatinNot AvailableActive Not Recruiting1
DB00641SimvastatinNot AvailableCompleted4
DB00641SimvastatinNot AvailableWithdrawn1
DB11104Sulfur hexafluorideNot AvailableCompleted1
DB05679UstekinumabNot AvailableCompleted1
DB00177ValsartanNot AvailableCompleted1
DB11094Vitamin DNot AvailableCompleted1
DB00163Vitamin ENot AvailableCompleted1
DB14003alpha-Tocopherol acetateNot AvailableCompleted1