Showing BioInteractions for Metformin (DB00331)
BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting Group | Interacting Drugs | |
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Metformin is a 5'-AMP-activated protein kinase subunit beta-1 inducer | ||
1 | 5'-AMP-activated protein kinase subunit beta-1 activators | Adenosine phosphate |
Interacting Group | Interacting Drugs | |
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Metformin is a 5'-AMP-activated protein kinase subunit beta-1 activator | ||
1 | 5'-AMP-activated protein kinase subunit beta-1 activators | Adenosine phosphate |
Interacting Group | Interacting Drugs | |
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Metformin is a Electron transfer flavoprotein-ubiquinone oxidoreductase, mitochondrial inhibitor |
Interacting Group | Interacting Drugs | |
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Metformin is a Glycerol-3-phosphate dehydrogenase [NAD(+)], cytoplasmic inhibitor |
Interacting Group | Interacting Drugs | |
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Metformin is a Multidrug and toxin extrusion protein 1 substrate | ||
1 | Multidrug and toxin extrusion protein 1 substrates | Acyclovir, Cefradine, Cephalexin, Cimetidine, Ciprofloxacin, Emtricitabine, Estrone sulfate, Flecainide, Ganciclovir, Guanidine, Levofloxacin, N-methylnicotinamide, Nadolol, Procainamide, Relebactam, Sulpiride, Tetraethylammonium, Tipiracil, Topotecan, Trimethoprim |
2 | Multidrug and toxin extrusion protein 1 inhibitors | Abemaciclib, Apalutamide, Bictegravir, Brigatinib, Capmatinib, Cimetidine, Ciprofloxacin, Famotidine, Fedratinib, Flecainide, Gilteritinib, Glasdegib, Guanfacine, Istradefylline, Lasmiditan, Levofloxacin, Lofexidine, Methylene blue, Osilodrostat, Pemigatinib, Pexidartinib, Plazomicin, Pralsetinib, Pyrimethamine, Ranolazine, Remdesivir, Rifamycin, Rimegepant, Ripretinib, Risdiplam, Rucaparib, Selpercatinib, Tafenoquine, Tazemetostat, Tirbanibulin, Topotecan, Trilaciclib, Trimethoprim, Tucatinib, Verapamil |
Interacting Group | Interacting Drugs | |
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Metformin is a Equilibrative nucleoside transporter 4 substrate | ||
1 | Equilibrative nucleoside transporter 4 substrates | Adenosine |
Interacting Group | Interacting Drugs | |
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Metformin is a Solute carrier family 22 member 3 substrate | ||
1 | Solute carrier family 22 member 3 inhibitors | Choline, Choline salicylate, Cimetidine, Clonidine, Desipramine, Dopamine, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Formoterol, Guanidine, Histamine, Imipramine, Irinotecan, Linagliptin, Melphalan, Metamfetamine, Nicotine, Norepinephrine, Phenoxybenzamine, Prazosin, Procainamide, Progesterone, Salmeterol, Vincristine |
2 | Solute carrier family 22 member 3 substrates | Adefovir dipivoxil, Agmatine, Amphetamine, Cimetidine, Guanidine, Lamivudine, Norepinephrine, Oxaliplatin, Sulpiride, Testosterone cypionate, Testosterone enanthate |
Interacting Group | Interacting Drugs | |
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Metformin is a Multidrug and toxin extrusion protein 2 substrate | ||
1 | Multidrug and toxin extrusion protein 2 substrates | Acyclovir, Baricitinib, Cimetidine, Estrone sulfate, Ganciclovir, N-methylnicotinamide, Nadolol, Procainamide, Relebactam, Sulpiride, Topotecan, Trastuzumab deruxtecan, Trimethoprim |
2 | Multidrug and toxin extrusion protein 2 inhibitors | Abemaciclib, Apalutamide, Baricitinib, Brigatinib, Capmatinib, Cimetidine, Ciprofloxacin, Copanlisib, Fedratinib, Glasdegib, Istradefylline, Lasmiditan, Levofloxacin, Methylene blue, Pexidartinib, Plazomicin, Pralsetinib, Pyrimethamine, Ranolazine, Risdiplam, Rucaparib, Tafenoquine, Tazemetostat, Tirbanibulin, Trilaciclib, Trimethoprim, Tucatinib, Verapamil |