Showing BioInteractions for Cefazolin (DB01327)
BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting Group | Interacting Drugs | |
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Cefazolin is a Serum paraoxonase/arylesterase 1 inhibitor | ||
1 | Serum paraoxonase/arylesterase 1 inhibitors | Edetate calcium disodium anhydrous, Edetate disodium anhydrous |
2 | Serum paraoxonase/arylesterase 1 substrates | Drospirenone, Loteprednol etabonate |
3 | Serum paraoxonase/arylesterase 1 inducers | Zinc chloride, Zinc sulfate, unspecified form |
Interacting Group | Interacting Drugs | |
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Cefazolin is a Penicillin-binding protein 1A inhibitor | ||
1 | Penicillin-binding protein 1A inhibitors | Cefacetrile, Cefmetazole, Cefonicid, Cefoperazone, Cefoxitin, Cefpiramide, Cefradine, Ceftazidime, Ceftibuten, Ceftizoxime, Doripenem, Ertapenem, Imipenem, Latamoxef |
2 | Penicillin-binding protein 1A antagonists | Doripenem |
Interacting Group | Interacting Drugs | |
---|---|---|
Cefazolin is a Penicillin-binding protein 1B inhibitor | ||
1 | Penicillin-binding protein 1B inhibitors | Cefacetrile, Cefmetazole, Cefonicid, Cefoperazone, Cefoxitin, Cefpiramide, Cefroxadine, Ceftazidime, Ceftibuten, Ceftizoxime, Doripenem, Ertapenem, Imipenem, Latamoxef |
2 | Penicillin-binding protein 1B antagonists | Cephaloglycin, Doripenem |
Interacting Group | Interacting Drugs | |
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Cefazolin is a Penicillin-binding protein 2 inhibitor | ||
1 | Penicillin-binding protein 2 inhibitors | Amdinocillin, Cefepime, Cefonicid, Cefoperazone, Ceftazidime, Ceftibuten, Ceftolozane, Doripenem, Ertapenem, Imipenem, Mezlocillin |
2 | Penicillin-binding protein 2 antagonists | Doripenem |
Interacting Group | Interacting Drugs | |
---|---|---|
Cefazolin is a Penicillin-binding protein 1C inhibitor | ||
1 | Penicillin-binding protein 1C inhibitors | Ceftolozane |
Interacting Group | Interacting Drugs | |
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Cefazolin is a Peptidoglycan synthase FtsI inhibitor | ||
1 | Peptidoglycan synthase FtsI inhibitors | Cefepime, Cefmenoxime, Cefmetazole, Cefonicid, Cefoperazone, Cefoxitin, Cefpiramide, Cefpodoxime, Ceftazidime, Ceftibuten, Ertapenem |
Interacting Group | Interacting Drugs | |
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Cefazolin is a Interleukin-15 inhibitor |
Interacting Group | Interacting Drugs | |
---|---|---|
Cefazolin is a Interleukin-2 inhibitor | ||
1 | Interleukin-2 inhibitors | Pseudoephedrine |
Interacting Group | Interacting Drugs | |
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Cefazolin is a Thiopurine S-methyltransferase substrate | ||
1 | Thiopurine S-methyltransferase substrates | Azathioprine, Mercaptopurine |
2 | Thiopurine S-methyltransferase inhibitors | Bendroflumethiazide, Olsalazine, Trichlormethiazide |
Interacting Group | Interacting Drugs | |
---|---|---|
Cefazolin is a Solute carrier family 22 member 11 inhibitor | ||
1 | Solute carrier family 22 member 11 inhibitors | Aminohippuric acid, Aspartame, Benzylpenicillin, Bumetanide, Caprylic acid, Cefalotin, Cefamandole, Cefoperazone, Cefotaxime, Ceftriaxone, Cimetidine, Diclofenac, Dinoprostone, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Furosemide, Glutaric Acid, Ibuprofen, Indomethacin, Ketoprofen, Lesinurad, Novobiocin, Oxytetracycline, Phenylbutazone, Piroxicam, Probenecid, Salicylic acid, Tetracycline |
2 | Solute carrier family 22 member 11 substrates | Aminohippuric acid, Conjugated estrogens, Hydrochlorothiazide, Levocetirizine, Methotrexate, Oxytetracycline, Pravastatin, Relebactam |
Interacting Group | Interacting Drugs | |
---|---|---|
Cefazolin is a Multidrug resistance-associated protein 4 substrate | ||
1 | Multidrug resistance-associated protein 4 substrates | Adefovir dipivoxil, Alprostadil, Atorvastatin, Cyclic adenosine monophosphate, Dinoprostone, Fluciclovine (18F), Fluorouracil, Gadoxetic acid, Glutathione, Hydrochlorothiazide, Lamivudine, Mercaptopurine, Methotrexate, Nateglinide, Oseltamivir, Prasterone, Raloxifene, Rosuvastatin, Tenofovir, Tenofovir alafenamide, Tenofovir disoproxil, Zidovudine |
2 | Multidrug resistance-associated protein 4 inhibitors | Celecoxib, Cholic Acid, Conjugated estrogens, Cyclic adenosine monophosphate, Diclofenac, Dipyridamole, Flurbiprofen, Folic acid, Ibuprofen, Indomethacin, Ketoprofen, Methotrexate, Probenecid, Promethazine, Remdesivir, Rofecoxib, Rucaparib, Sildenafil, Sorafenib, Sulfinpyrazone, Sunitinib, Taurocholic acid, Tioguanine, Ursodeoxycholic acid, Verapamil |
3 | Multidrug resistance-associated protein 4 binders | Meloxicam |