Showing BioInteractions for Ephedrine (DB01364)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Ephedrine is a Alpha-1A adrenergic receptor agonist
1Alpha-1A adrenergic receptor agonists4-Methoxyamphetamine, Apraclonidine, Benzphetamine, Bromocriptine, Cirazoline, Clonidine, Dipivefrin, Droxidopa, Epinephrine, Ergometrine, Isometheptene, Lofexidine, Metaraminol, Methoxamine, Midodrine, Naphazoline, Norepinephrine, Pergolide, Phendimetrazine, Phenylephrine, Pseudoephedrine, Racepinephrine, Tetryzoline, Xylometazoline
2Alpha-1A adrenergic receptor antagonistsAcepromazine, Alfuzosin, Amitriptyline, Amoxapine, Aripiprazole, Aripiprazole lauroxil, Asenapine, Bevantolol, Bromocriptine, Carvedilol, Chlorpromazine, Clozapine, Dapiprazole, Doxazosin, Doxepin, Dronedarone, Droperidol, Flupentixol, Iloperidone, Imipramine, Indoramin, Methotrimeprazine, Nefazodone, Nicardipine, Nicergoline, Niguldipine, Nortriptyline, Olanzapine, Paliperidone, Phenoxybenzamine, Phentolamine, Pizotifen, Prazosin, Promazine, Propiomazine, Propiverine, Quinidine, Risperidone, Silodosin, Tamsulosin, Terazosin, Thioproperazine, Thioridazine, Tolazoline, Trazodone, Trifluoperazine, Trimipramine, Verapamil, Ziprasidone, Zuclopenthixol
3Alpha-1A adrenergic receptor partial agonistsErgotamine, Oxymetazoline, Xylometazoline
4Alpha-1A adrenergic receptor potentiatorsCarvedilol
5Alpha-1A adrenergic receptor inhibitorsAmitriptyline, Fenoldopam, Lamotrigine
6Alpha-1A adrenergic receptor bindersCabergoline, Loxapine
Interacting GroupInteracting Drugs
Ephedrine is a Sodium-dependent noradrenaline transporter inverse agonist
1Sodium-dependent noradrenaline transporter inhibitorsAmitriptyline, Amoxapine, Atomoxetine, Benzatropine, Bupropion, Chlorpheniramine, Clomipramine, Cocaine, Cyclobenzaprine, Desipramine, Desvenlafaxine, Dexmethylphenidate, Dextromethorphan, Diethylpropion, Dopamine, Dosulepin, Doxepin, Duloxetine, Escitalopram, Etoperidone, Ginkgo biloba, Imipramine, Ketamine, Levomilnacipran, Maprotiline, Mazindol, Meperidine, Methylphenidate, Mianserin, Milnacipran, Nefazodone, Netarsudil, Nortriptyline, Orphenadrine, Paroxetine, Phenmetrazine, Phentermine, Procaine, Protriptyline, Pseudoephedrine, Rauwolfia serpentina root, Reboxetine, Sertraline, Sibutramine, Tapentadol, Tramadol, Trimipramine, Venlafaxine, Viloxazine
2Sodium-dependent noradrenaline transporter partial agonistsGuanadrel
3Sodium-dependent noradrenaline transporter inducersDebrisoquine, Guanethidine
4Sodium-dependent noradrenaline transporter negative modulatorsDextroamphetamine, Ephedra sinica root, Metamfetamine, Midomafetamine, MMDA, Phendimetrazine
5Sodium-dependent noradrenaline transporter substratesDroxidopa, Iobenguane, Iobenguane sulfate I-123, Norepinephrine, Nortriptyline
6Sodium-dependent noradrenaline transporter bindersLoxapine
7Sodium-dependent noradrenaline transporter stimulatorsAmphetamine
8Sodium-dependent noradrenaline transporter blockersVortioxetine
9Sodium-dependent noradrenaline transporter antagonistsZotepine
Interacting GroupInteracting Drugs
Ephedrine is a Beta-1 adrenergic receptor agonist
1Beta-1 adrenergic receptor antagonistsAlprenolol, Arotinolol, Asenapine, Atenolol, Betaxolol, Bevantolol, Bisoprolol, Bupranolol, Carvedilol, Celiprolol, Dronedarone, Esmolol, Labetalol, Levobetaxolol, Levobunolol, Metipranolol, Metoprolol, Nadolol, Nebivolol, Oxprenolol, Penbutolol, Practolol, Propafenone, Propranolol, Ranolazine, Sotalol, Terbutaline, Timolol
2Beta-1 adrenergic receptor agonistsAlbuterol, Arbutamine, Clenbuterol, DL-Methylephedrine, Dobutamine, Droxidopa, Ephedra sinica root, Epinephrine, Fenoterol, Formoterol, Isoetharine, Isoprenaline, Norepinephrine, Phenylpropanolamine, Pirbuterol, Pseudoephedrine, Racepinephrine
3Beta-1 adrenergic receptor partial agonistsAcebutolol, Bopindolol, Carteolol, Penbutolol, Pindolol, Pseudoephedrine, Xamoterol
4Beta-1 adrenergic receptor bindersCabergoline, Loxapine
5Beta-1 adrenergic receptor ligandsAripiprazole, Vortioxetine
6Beta-1 adrenergic receptor inverse agonistsSalmeterol
7Beta-1 adrenergic receptor inhibitorsLamotrigine
Interacting GroupInteracting Drugs
Ephedrine is a Beta-2 adrenergic receptor agonist
1Beta-2 adrenergic receptor antagonistsAlprenolol, Arotinolol, Asenapine, Atenolol, Betaxolol, Bevantolol, Bisoprolol, Bupranolol, Carteolol, Carvedilol, Desipramine, Labetalol, Levobunolol, Metipranolol, Metoprolol, Nadolol, Nebivolol, Oxprenolol, Penbutolol, Propafenone, Propranolol, Sotalol, Timolol
2Beta-2 adrenergic receptor agonistsAlbuterol, Arbutamine, Arformoterol, Bambuterol, Bedoradrine, Celiprolol, Clenbuterol, Dipivefrin, Dobutamine, Doxofylline, Droxidopa, Ephedra sinica root, Epinephrine, Etafedrine, Fenoterol, Formoterol, Indacaterol, Isoetharine, Isoprenaline, Levosalbutamol, Norepinephrine, Olodaterol, Orciprenaline, Phenylpropanolamine, Pirbuterol, Procaterol, Protokylol, Racepinephrine, Ritodrine, Salmeterol, Terbutaline, Vilanterol
3Beta-2 adrenergic receptor partial agonistsAcebutolol, Bopindolol, Penbutolol, Pindolol, Pseudoephedrine
4Beta-2 adrenergic receptor bindersCabergoline
5Beta-2 adrenergic receptor ligandsAripiprazole
Interacting GroupInteracting Drugs
Ephedrine is a Cholinesterase substrate
1Cholinesterase inhibitorsAmbenonium, Aprotinin, Bambuterol, Betaine, Capsaicin, Chlorpromazine, Cinchocaine, Cisplatin, Decamethonium, Demecarium, Diethylcarbamazine, Echothiophate, Edrophonium, Galantamine, Hexafluronium, Isoflurophate, Ketamine, Malathion, Mechlorethamine, Mefloquine, Methylphosphinic Acid, Neostigmine, Nizatidine, Pancuronium, Pegvisomant, Perindopril, Phenserine, Pipecuronium, Procainamide, Procaine, Profenamine, Ramipril, Regramostim, Rivastigmine, Sulpiride, Tacrine, Terbutaline, Thiotepa, Tretamine, Triflupromazine
2Cholinesterase substratesAclidinium, Bambuterol, Benzonatate, Butamben, Butyrylthiocholine, Chloroprocaine, Clevidipine, Cocaine, Cyclopentolate, Dipivefrin, Doxacurium, Irinotecan, Mirabegron, Moxisylyte, Oxybuprocaine, Procaine, Propacetamol, Sar9, Met (O2)11-Substance P, Succinylcholine, Trimethaphan, Tubocurarine
3Cholinesterase ligandsButyric Acid, Ethyl dihydrogen phosphate, Phosphorylisopropane
4Cholinesterase antagonistsPyridostigmine
5Cholinesterase activatorsPralidoxime
6Cholinesterase inducersChlorphenesin, Donepezil, Pentagastrin, Triamcinolone
Interacting GroupInteracting Drugs
Ephedrine is a Acetylcholinesterase inhibitor
1Acetylcholinesterase inhibitorsAmbenonium, Decamethonium, Demecarium, Dipivefrin, Donepezil, Edrophonium, Galantamine, Gallamine triethiodide, Huperzine A, Isoflurophate, Itopride, Mefloquine, Methantheline, Minaprine, Neostigmine, Physostigmine, Pyridostigmine, Ranitidine, Rivastigmine, Tacrine, Tubocurarine, Tyrothricin
2Acetylcholinesterase antagonistsDimetacrine, Pyridostigmine
3Acetylcholinesterase activatorsPralidoxime
4Acetylcholinesterase substratesCarbamoylcholine