Showing BioInteractions for Fostamatinib (DB12010)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Fostamatinib is a Adenosine receptor A3 antagonist
1Adenosine receptor A3 antagonistsAminophylline, Caffeine
2Adenosine receptor A3 agonistsAdenosine
3Adenosine receptor A3 inhibitorsEnprofylline
Interacting GroupInteracting Drugs
Fostamatinib is a vesicular monoamine transporter 2 (VMAT2) inhibitor
1vesicular monoamine transporter 2 (VMAT2) antagonistsValbenazine
2vesicular monoamine transporter 2 (VMAT2) inhibitorsRauwolfia serpentina root
Interacting GroupInteracting Drugs
Fostamatinib is a Fatty-acid amide hydrolase 1 inhibitor
1Fatty-acid amide hydrolase 1 inhibitorsCannabidiol, Medical Cannabis, Nabiximols, Thiopental
2Fatty-acid amide hydrolase 1 substratesAcetaminophen, Propofol
3Fatty-acid amide hydrolase 1 inducersNabiximols
Interacting GroupInteracting Drugs
Fostamatinib is a Equilibrative nucleoside transporter 1 inhibitor
1Equilibrative nucleoside transporter 1 inhibitorsCannabidiol, Medical Cannabis, Nabiximols, Troglitazone
2Equilibrative nucleoside transporter 1 substratesCytarabine, Fludarabine, Fluorouracil, Gemcitabine, Mercaptopurine, Ribavirin, Tegafur-uracil, Trifluridine
3Equilibrative nucleoside transporter 1 inducersPemetrexed
Interacting GroupInteracting Drugs
Fostamatinib is a UDP-glucuronosyltransferase 1-1 inhibitor
1UDP-glucuronosyltransferase 1-1 substratesAbacavir, Acetaminophen, Alvocidib, Atorvastatin, Axitinib, Bictegravir, Binimetinib, Carvedilol, Cerivastatin, Deferasirox, Delafloxacin, Dexibuprofen, Dolutegravir, Eltrombopag, Enasidenib, Eslicarbazepine, Eslicarbazepine acetate, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Ethinylestradiol, Etoposide, Ezetimibe, Ezogabine, Flurbiprofen, Fluvastatin, Fulvestrant, Furosemide, Fusidic acid, Gavestinel, Gemfibrozil, Glipizide, Indacaterol, Indomethacin, Irinotecan, Ketoprofen, Labetalol, Letermovir, Levothyroxine, Liothyronine, Losartan, Lovastatin, Metronidazole, Migalastat, Minoxidil, Morphine, Muraglitazar, Mycophenolate mofetil, Mycophenolic acid, Naloxone, Naltrexone, Nintedanib, Norgestimate, Phenytoin, Propacetamol, Propofol, Raloxifene, Raltegravir, Sacituzumab govitecan, Selumetinib, Simvastatin, Suprofen, Tecovirimat, Tiagabine, Tramadol, Troglitazone, Valproic acid, Zidovudine, Zonisamide
2UDP-glucuronosyltransferase 1-1 inhibitorsAdenine, Atazanavir, Dacomitinib, Deferasirox, Eltrombopag, Enasidenib, Erlotinib, Ertugliflozin, Flunitrazepam, Flurbiprofen, Gemfibrozil, Glecaprevir, Indinavir, Indomethacin, Ketoconazole, Nilotinib, Paritaprevir, Pazopanib, Pexidartinib, Pibrentasvir, Probenecid, Propofol, Regorafenib, Rucaparib, Silibinin, Sodium aurothiomalate, Sorafenib, Ubrogepant, Valproic acid
3UDP-glucuronosyltransferase 1-1 inducersCarbamazepine, Desogestrel, Efavirenz, Ethinylestradiol, Nelfinavir, Phenobarbital, Phenytoin, Rifampicin, Testosterone propionate, Tipranavir, Zidovudine
Interacting GroupInteracting Drugs
Fostamatinib is a cGMP-specific 3',5'-cyclic phosphodiesterase inhibitor
1cGMP-specific 3',5'-cyclic phosphodiesterase inhibitorsAvanafil, Dipyridamole, Sildenafil, Tadalafil, Theophylline, Udenafil, Vardenafil
2cGMP-specific 3',5'-cyclic phosphodiesterase substratesMolsidomine
Interacting GroupInteracting Drugs
Fostamatinib is a Arachidonate 5-lipoxygenase inhibitor
1Arachidonate 5-lipoxygenase inhibitorsAminosalicylic acid, Balsalazide, Cannabidiol, Diacerein, Diethylcarbamazine, Hyperforin, Masoprocol, Meclofenamic acid, Medical Cannabis, Mesalazine, Minocycline, Morniflumate, Nabiximols, Rhein, Sulfasalazine, Zileuton
2Arachidonate 5-lipoxygenase substratesOmega-3 fatty acids, Omega-6 fatty acids
3Arachidonate 5-lipoxygenase antagonistsMorniflumate
4Arachidonate 5-lipoxygenase potentiatorsDiclofenac
Interacting GroupInteracting Drugs
Fostamatinib is a Cathepsin S inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Cathepsin L1 inhibitor
1Cathepsin L1 substratesTrastuzumab deruxtecan
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Fostamatinib is a Tyrosine-protein kinase ABL1 inhibitor
1Tyrosine-protein kinase ABL1 inhibitorsATP, Bosutinib, Brigatinib, Imatinib, Nilotinib, Ponatinib, Regorafenib
2Tyrosine-protein kinase ABL1 antagonistsRadotinib
3Tyrosine-protein kinase ABL1 substratesMagnesium gluconate
4Tyrosine-protein kinase ABL1 inducersMagnesium gluconate
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Fostamatinib is a Calcium-dependent protein kinase 1 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase PknB inhibitor
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Fostamatinib is a Ribosomal protein S6 kinase alpha-6 inhibitor
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Fostamatinib is a Non-receptor tyrosine-protein kinase TYK2 inhibitor
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Fostamatinib is a Atypical kinase COQ8A, mitochondrial inhibitor
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Fostamatinib is a Tyrosine-protein kinase JAK1 inhibitor
1Tyrosine-protein kinase JAK1 inhibitorsBaricitinib, Fedratinib, Filgotinib, Pralsetinib, Ruxolitinib, Tofacitinib, Upadacitinib
Interacting GroupInteracting Drugs
Fostamatinib is a Hepatocyte growth factor receptor inhibitor
1Hepatocyte growth factor receptor antagonistsCabozantinib
2Hepatocyte growth factor receptor inhibitorsAMG-208, Brigatinib, Capmatinib, Crizotinib
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Fostamatinib is a Serine/threonine-protein kinase NIM1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase MST4 inhibitor
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Fostamatinib is a cAMP-dependent protein kinase catalytic subunit alpha inhibitor
1cAMP-dependent protein kinase catalytic subunit alpha inhibitorsEllagic acid
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Fostamatinib is a Serine/threonine-protein kinase 24 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase 3 inhibitor
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Fostamatinib is a Tyrosine-protein kinase Tec inhibitor
1Tyrosine-protein kinase Tec inhibitorsZanubrutinib
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Fostamatinib is a Tyrosine-protein kinase SYK inhibitor
1Tyrosine-protein kinase SYK inhibitorsEllagic acid
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Fostamatinib is a Serine/threonine-protein kinase 33 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase 35 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase 36 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase 38 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase 38-like inhibitor
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Fostamatinib is a STE20/SPS1-related proline-alanine-rich protein kinase inhibitor
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Fostamatinib is a Serine/threonine-protein kinase TAO1 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase TAO2 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase TAO3 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase TBK1 inhibitor
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Fostamatinib is a Angiopoietin-1 receptor inhibitor
1Angiopoietin-1 receptor inhibitorsPonatinib, Regorafenib, Ripretinib, Vandetanib
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Fostamatinib is a Dual specificity testis-specific protein kinase 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a TGF-beta receptor type-1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a TGF-beta receptor type-2 inhibitor
1TGF-beta receptor type-2 agonistsForeskin fibroblast (neonatal), Foreskin keratinocyte (neonatal)
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Fostamatinib is a Tyrosine-protein kinase receptor Tie-1 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase tousled-like 1 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase tousled-like 2 inhibitor
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Fostamatinib is a TRAF2 and NCK-interacting protein kinase inhibitor
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Fostamatinib is a Non-receptor tyrosine-protein kinase TNK1 inhibitor
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Fostamatinib is a Activated CDC42 kinase 1 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase TNNI3K inhibitor
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Fostamatinib is a Testis-specific serine/threonine-protein kinase 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Dual specificity protein kinase TTK inhibitor
1Dual specificity protein kinase TTK inhibitorsBOS172722
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Fostamatinib is a Tyrosine-protein kinase TXK inhibitor
1Tyrosine-protein kinase TXK inhibitorsZanubrutinib
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Fostamatinib is a Tyrosine-protein kinase receptor TYRO3 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase ULK1 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase ULK2 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase ULK3 inhibitor
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Fostamatinib is a Wee1-like protein kinase inhibitor
1Wee1-like protein kinase inhibitorsAdavosertib
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Fostamatinib is a Tyrosine-protein kinase Yes inhibitor
1Tyrosine-protein kinase Yes inhibitorsDasatinib
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Fostamatinib is a Mitogen-activated protein kinase kinase kinase 19 inhibitor
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Fostamatinib is a Mitogen-activated protein kinase kinase kinase MLT inhibitor
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Fostamatinib is a Tyrosine-protein kinase ZAP-70 inhibitor
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Fostamatinib is a AP2-associated protein kinase 1 inhibitor
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Fostamatinib is a Tyrosine-protein kinase ABL2 inhibitor
1Tyrosine-protein kinase ABL2 inhibitorsATP
Interacting GroupInteracting Drugs
Fostamatinib is a Activin receptor type-1 inhibitor
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Fostamatinib is a Activin receptor type-1B inhibitor
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Fostamatinib is a Atypical kinase COQ8B, mitochondrial inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a ALK tyrosine kinase receptor inhibitor
1ALK tyrosine kinase receptor inhibitorsAlectinib, Brigatinib, Crizotinib, Gilteritinib, Lorlatinib
2ALK tyrosine kinase receptor antagonistsCeritinib
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Fostamatinib is a Ankyrin repeat and protein kinase domain-containing protein 1 inhibitor
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Fostamatinib is a Aurora kinase A inhibitor
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Fostamatinib is a Aurora kinase B inhibitor
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Fostamatinib is a Aurora kinase C inhibitor
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Fostamatinib is a Tyrosine-protein kinase receptor UFO inhibitor
1Tyrosine-protein kinase receptor UFO inhibitorsGilteritinib
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Fostamatinib is a Tyrosine-protein kinase Blk inhibitor
1Tyrosine-protein kinase Blk inhibitorsZanubrutinib
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Fostamatinib is a BMP-2-inducible protein kinase inhibitor
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Fostamatinib is a Bone morphogenetic protein receptor type-1B inhibitor
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Fostamatinib is a Bone morphogenetic protein receptor type-2 inhibitor
1Bone morphogenetic protein receptor type-2 ligandsDibotermin alfa
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Fostamatinib is a Cytoplasmic tyrosine-protein kinase BMX inhibitor
1Cytoplasmic tyrosine-protein kinase BMX inhibitorsZanubrutinib
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Fostamatinib is a Serine/threonine-protein kinase B-raf inhibitor
1Serine/threonine-protein kinase B-raf inhibitorsDabrafenib, Encorafenib, Regorafenib, Ripretinib, Sorafenib, Vemurafenib
2Serine/threonine-protein kinase B-raf antagonistsDabrafenib
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase BTK inhibitor
1Tyrosine-protein kinase BTK inhibitorsAbivertinib, Acalabrutinib, Ibrutinib, Zanubrutinib
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Fostamatinib is a Calcium/calmodulin-dependent protein kinase type 1 inhibitor
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Fostamatinib is a Calcium/calmodulin-dependent protein kinase type 1D inhibitor
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Fostamatinib is a Calcium/calmodulin-dependent protein kinase type 1G inhibitor
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Fostamatinib is a Calcium/calmodulin-dependent protein kinase type II subunit alpha inhibitor
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Fostamatinib is a Calcium/calmodulin-dependent protein kinase type II subunit beta inhibitor
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Fostamatinib is a Calcium/calmodulin-dependent protein kinase type II subunit delta inhibitor
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Fostamatinib is a Calcium/calmodulin-dependent protein kinase type II subunit gamma inhibitor
1Calcium/calmodulin-dependent protein kinase type II subunit gamma inhibitorsBosutinib
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Fostamatinib is a Calcium/calmodulin-dependent protein kinase kinase 1 inhibitor
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Fostamatinib is a Calcium/calmodulin-dependent protein kinase kinase 2 inhibitor
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Fostamatinib is a Peripheral plasma membrane protein CASK inhibitor
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Fostamatinib is a Kappa-casein inhibitor
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Fostamatinib is a Cyclin-dependent kinase 1 inhibitor
1Cyclin-dependent kinase 1 inhibitorsAlsterpaullone
2Cyclin-dependent kinase 1 bindersIndirubin-3'-monoxime, Olomoucine, SU9516
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Fostamatinib is a Serine/threonine-protein kinase MRCK gamma inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Cyclin-dependent kinase 4 inhibitor
1Cyclin-dependent kinase 4 inhibitorsAbemaciclib, Palbociclib, Ribociclib
2Cyclin-dependent kinase 4 antagonistsRibociclib
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Fostamatinib is a Cyclin-dependent kinase-like 1 inhibitor
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Fostamatinib is a Cyclin-dependent kinase-like 2 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase Chk1 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase Chk2 inhibitor
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Fostamatinib is a Citron Rho-interacting kinase inhibitor
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Fostamatinib is a Dual specificity protein kinase CLK1 inhibitor
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Fostamatinib is a Dual specificity protein kinase CLK2 inhibitor
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Fostamatinib is a Dual specificity protein kinase CLK3 inhibitor
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Fostamatinib is a Dual specificity protein kinase CLK4 inhibitor
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Fostamatinib is a Macrophage colony-stimulating factor 1 receptor inhibitor
1Macrophage colony-stimulating factor 1 receptor inhibitorsPexidartinib, Sunitinib
2Macrophage colony-stimulating factor 1 receptor antagonistsImatinib
3Macrophage colony-stimulating factor 1 receptor substratesErdafitinib
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase CSK inhibitor
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Fostamatinib is a Casein kinase I isoform alpha inhibitor
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Fostamatinib is a Casein kinase II subunit alpha inhibitor
1Casein kinase II subunit alpha inhibitorsEllagic acid
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Fostamatinib is a Casein kinase II subunit alpha' inhibitor
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Fostamatinib is a Death-associated protein kinase 1 inhibitor
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Fostamatinib is a Death-associated protein kinase 2 inhibitor
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Fostamatinib is a Death-associated protein kinase 3 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase DCLK1 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase DCLK2 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase DCLK3 inhibitor
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Fostamatinib is a Epithelial discoidin domain-containing receptor 1 inhibitor
1Epithelial discoidin domain-containing receptor 1 antagonistsImatinib
2Epithelial discoidin domain-containing receptor 1 inhibitorsPralsetinib
Interacting GroupInteracting Drugs
Fostamatinib is a Discoidin domain-containing receptor 2 inhibitor
1Discoidin domain-containing receptor 2 inhibitorsRegorafenib
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Fostamatinib is a Dual specificity tyrosine-phosphorylation-regulated kinase 1A inhibitor
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Fostamatinib is a Dual specificity tyrosine-phosphorylation-regulated kinase 1B inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Epidermal growth factor receptor inhibitor
1Epidermal growth factor receptor antagonistsCetuximab, Erlotinib, Gefitinib, Icotinib, Lapatinib, Lidocaine, Necitumumab, Zalutumumab
2Epidermal growth factor receptor suppressorsPanitumumab
3Epidermal growth factor receptor inhibitorsAbivertinib, Afatinib, Brigatinib, Dacomitinib, Neratinib, Olmutinib, Osimertinib, Vandetanib, Zanubrutinib
4Epidermal growth factor receptor agonistsForeskin keratinocyte (neonatal)
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Fostamatinib is a Eukaryotic translation initiation factor 2-alpha kinase 1 inhibitor
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Fostamatinib is a Interferon-induced, double-stranded RNA-activated protein kinase inhibitor
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Fostamatinib is a eIF-2-alpha kinase GCN2 inhibitor
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Fostamatinib is a Ephrin type-A receptor 1 inhibitor
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Fostamatinib is a Ephrin type-A receptor 2 inhibitor
1Ephrin type-A receptor 2 antagonistsDasatinib
2Ephrin type-A receptor 2 inhibitorsRegorafenib
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Fostamatinib is a Ephrin type-A receptor 3 inhibitor
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Fostamatinib is a Ephrin type-A receptor 4 inhibitor
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Fostamatinib is a Ephrin type-A receptor 5 inhibitor
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Fostamatinib is a Ephrin type-A receptor 6 inhibitor
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Fostamatinib is a Ephrin type-A receptor 7 inhibitor
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Fostamatinib is a Ephrin type-A receptor 8 inhibitor
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Fostamatinib is a Ephrin type-B receptor 1 inhibitor
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Fostamatinib is a Ephrin type-B receptor 2 inhibitor
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Fostamatinib is a Ephrin type-B receptor 4 inhibitor
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Fostamatinib is a Ephrin type-B receptor 6 inhibitor
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Fostamatinib is a Receptor tyrosine-protein kinase erbB-2 inhibitor
1Receptor tyrosine-protein kinase erbB-2 antagonistsLapatinib, Margetuximab
2Receptor tyrosine-protein kinase erbB-2 inhibitorsAfatinib, Brigatinib, Pertuzumab, Tucatinib, Zanubrutinib
Interacting GroupInteracting Drugs
Fostamatinib is a Receptor tyrosine-protein kinase erbB-4 inhibitor
1Receptor tyrosine-protein kinase erbB-4 inhibitorsAfatinib, Brigatinib, Zanubrutinib
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Fostamatinib is a Serine/threonine-protein kinase/endoribonuclease IRE1 inhibitor
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Fostamatinib is a Tyrosine-protein kinase Fer inhibitor
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Fostamatinib is a Tyrosine-protein kinase Fes/Fps inhibitor
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Fostamatinib is a Fibroblast growth factor receptor 1 inhibitor
1Fibroblast growth factor receptor 1 agonistsPalifermin
2Fibroblast growth factor receptor 1 inhibitorsErdafitinib, Lenvatinib, Nintedanib, Pemigatinib, Ponatinib, Pralsetinib, Regorafenib, Selpercatinib, Sorafenib
Interacting GroupInteracting Drugs
Fostamatinib is a Fibroblast growth factor receptor 2 inhibitor
1Fibroblast growth factor receptor 2 agonistsForeskin fibroblast (neonatal), Foreskin keratinocyte (neonatal), Palifermin
2Fibroblast growth factor receptor 2 bindersPalifermin
3Fibroblast growth factor receptor 2 antagonistsThalidomide
4Fibroblast growth factor receptor 2 inhibitorsErdafitinib, Lenvatinib, Nintedanib, Pemigatinib, Ponatinib, Pralsetinib, Regorafenib, Selpercatinib
5Fibroblast growth factor receptor 2 ligandsSucrosofate
Interacting GroupInteracting Drugs
Fostamatinib is a Fibroblast growth factor receptor 3 inhibitor
1Fibroblast growth factor receptor 3 inhibitorsErdafitinib, Lenvatinib, Nintedanib, Pazopanib, Pemigatinib, Ponatinib, Selpercatinib
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase Fgr inhibitor
1Tyrosine-protein kinase Fgr inhibitorsZanubrutinib
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Fostamatinib is a Vascular endothelial growth factor receptor 1 inhibitor
1Vascular endothelial growth factor receptor 1 inhibitorsAxitinib, Lenvatinib, Nintedanib, Pazopanib, Regorafenib, Selpercatinib, Sorafenib, Sunitinib
2Vascular endothelial growth factor receptor 1 agonistsForeskin fibroblast (neonatal), Polaprezinc
Interacting GroupInteracting Drugs
Fostamatinib is a Receptor-type tyrosine-protein kinase FLT3 inhibitor
1Receptor-type tyrosine-protein kinase FLT3 antagonistsMidostaurin, Sorafenib
2Receptor-type tyrosine-protein kinase FLT3 inhibitorsBrigatinib, Fedratinib, Gilteritinib, Midostaurin, Nintedanib, Pexidartinib, Ponatinib, Pralsetinib, Sunitinib
Interacting GroupInteracting Drugs
Fostamatinib is a Vascular endothelial growth factor receptor 3 inhibitor
1Vascular endothelial growth factor receptor 3 antagonistsSorafenib
2Vascular endothelial growth factor receptor 3 inhibitorsAxitinib, Lenvatinib, Nintedanib, Regorafenib, Selpercatinib, Sunitinib
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase mTOR inhibitor
1Serine/threonine-protein kinase mTOR ligandsRimiducid
2Serine/threonine-protein kinase mTOR inhibitorsEverolimus, Sirolimus, Temsirolimus
3Serine/threonine-protein kinase mTOR potentiatorsPimecrolimus
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase FRK inhibitor
1Tyrosine-protein kinase FRK inhibitorsRegorafenib, Zanubrutinib
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Fostamatinib is a Tyrosine-protein kinase Fyn inhibitor
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Fostamatinib is a Cyclin-G-associated kinase inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Glycogen synthase kinase-3 alpha inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Glycogen synthase kinase-3 beta inhibitor
1Glycogen synthase kinase-3 beta inhibitorsLithium cation
2Glycogen synthase kinase-3 beta antagonistsTideglusib
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase HCK inhibitor
1Tyrosine-protein kinase HCK inhibitorsBosutinib
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Fostamatinib is a Homeodomain-interacting protein kinase 2 inhibitor
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Fostamatinib is a Homeodomain-interacting protein kinase 3 inhibitor
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Fostamatinib is a Serine/threonine-protein kinase ICK inhibitor
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Fostamatinib is a Inhibitor of nuclear factor kappa-B kinase subunit beta inhibitor
1Inhibitor of nuclear factor kappa-B kinase subunit beta inhibitorsAcetylcysteine, Auranofin, Mesalazine, Sulfasalazine
2Inhibitor of nuclear factor kappa-B kinase subunit beta inducersArsenic trioxide
Interacting GroupInteracting Drugs
Fostamatinib is a Inhibitor of nuclear factor kappa-B kinase subunit epsilon inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Insulin receptor inhibitor
1Insulin receptor agonistsInsulin aspart, Insulin detemir, Insulin glargine, Insulin glulisine, Insulin human, Insulin lispro
2Insulin receptor bindersInsulin pork
3Insulin receptor ligandsInsulin degludec
4Insulin receptor activatorsChromic chloride
5Insulin receptor bindingsBrigatinib
Interacting GroupInteracting Drugs
Fostamatinib is a Insulin receptor-related protein inhibitor
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Fostamatinib is a Interleukin-1 receptor-associated kinase 1 inhibitor
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Fostamatinib is a Interleukin-1 receptor-associated kinase 3 inhibitor
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Fostamatinib is a Interleukin-1 receptor-associated kinase 4 inhibitor
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Fostamatinib is a Tyrosine-protein kinase ITK/TSK inhibitor
1Tyrosine-protein kinase ITK/TSK inhibitorsPazopanib, Zanubrutinib
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase JAK2 inhibitor
1Tyrosine-protein kinase JAK2 inhibitorsBaricitinib, Entrectinib, Fedratinib, Pralsetinib, Ruxolitinib, Tofacitinib, Zanubrutinib
2Tyrosine-protein kinase JAK2 antagonistsTofacitinib
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase JAK3 inhibitor
1Tyrosine-protein kinase JAK3 inhibitorsBaricitinib, Tofacitinib, Zanubrutinib
Interacting GroupInteracting Drugs
Fostamatinib is a Vascular endothelial growth factor receptor 2 inhibitor
1Vascular endothelial growth factor receptor 2 antagonistsCabozantinib, Midostaurin, Ramucirumab, Sorafenib
2Vascular endothelial growth factor receptor 2 inhibitorsAxitinib, Lenvatinib, Midostaurin, Nintedanib, Pazopanib, Ponatinib, Pralsetinib, Regorafenib, Ripretinib, Sunitinib
3Vascular endothelial growth factor receptor 2 substratesErdafitinib
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase SIK3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mast/stem cell growth factor receptor Kit inhibitor
1Mast/stem cell growth factor receptor Kit antagonistsDasatinib, Imatinib, Midostaurin, Nilotinib, Sorafenib
2Mast/stem cell growth factor receptor Kit inhibitorsAvapritinib, Lenvatinib, Midostaurin, Pazopanib, Pexidartinib, Ponatinib, Regorafenib, Ripretinib, Sunitinib
3Mast/stem cell growth factor receptor Kit agonistsAncestim
4Mast/stem cell growth factor receptor Kit substratesErdafitinib
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase LATS1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase Lck inhibitor
1Tyrosine-protein kinase Lck inhibitorsNintedanib, Ponatinib, Zanubrutinib
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Fostamatinib is a LIM domain kinase 1 inhibitor
1LIM domain kinase 1 antagonistsDabrafenib
2LIM domain kinase 1 inhibitorsDabrafenib
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Fostamatinib is a LIM domain kinase 2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Leucine-rich repeat serine/threonine-protein kinase 2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Leukocyte tyrosine kinase receptor inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase Lyn inhibitor
1Tyrosine-protein kinase Lyn inhibitorsNintedanib, Ponatinib
Interacting GroupInteracting Drugs
Fostamatinib is a Dual specificity mitogen-activated protein kinase kinase 2 inhibitor
1Dual specificity mitogen-activated protein kinase kinase 2 inhibitorsBinimetinib, Bosutinib, Selumetinib, Trametinib
2Dual specificity mitogen-activated protein kinase kinase 2 antagonistsTrametinib
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Fostamatinib is a Dual specificity mitogen-activated protein kinase kinase 3 inhibitor
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Fostamatinib is a Dual specificity mitogen-activated protein kinase kinase 5 inhibitor
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Fostamatinib is a Dual specificity mitogen-activated protein kinase kinase 6 inhibitor
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Fostamatinib is a Mitogen-activated protein kinase kinase kinase 1 inhibitor
1Mitogen-activated protein kinase kinase kinase 1 inhibitorsBinimetinib
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Fostamatinib is a Mitogen-activated protein kinase kinase kinase 10 inhibitor
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Fostamatinib is a Mitogen-activated protein kinase kinase kinase 11 inhibitor
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Fostamatinib is a Mitogen-activated protein kinase kinase kinase 12 inhibitor
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Fostamatinib is a Mitogen-activated protein kinase kinase kinase 13 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase 15 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase 2 inhibitor
1Mitogen-activated protein kinase kinase kinase 2 inhibitorsBosutinib
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase 3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase 4 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase 6 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase 9 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase kinase 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase kinase 2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase kinase 3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase kinase 4 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase kinase kinase kinase 5 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase 10 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase 13 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase 14 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase 15 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase 4 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase 7 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Mitogen-activated protein kinase 9 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a MAP kinase-activated protein kinase 5 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase MARK1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase MARK2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a MAP/microtubule affinity-regulating kinase 3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a MAP/microtubule affinity-regulating kinase 4 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a CLIP-associating protein 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Microtubule-associated serine/threonine-protein kinase 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Megakaryocyte-associated tyrosine-protein kinase inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Maternal embryonic leucine zipper kinase inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase Mer inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Misshapen-like kinase 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a MAP kinase-interacting serine/threonine-protein kinase 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a MAP kinase-interacting serine/threonine-protein kinase 2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Macrophage-stimulating protein receptor inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Muscle, skeletal receptor tyrosine-protein kinase inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Myosin light chain kinase, smooth muscle inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Myosin light chain kinase 2, skeletal/cardiac muscle inhibitor
1Myosin light chain kinase 2, skeletal/cardiac muscle inhibitorsPrenylamine
Interacting GroupInteracting Drugs
Fostamatinib is a Myosin light chain kinase 3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Myosin light chain kinase family member 4 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Myosin-IIIa inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase Nek1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase Nek11 inhibitor
1Serine/threonine-protein kinase Nek11 antagonistsDabrafenib
2Serine/threonine-protein kinase Nek11 inhibitorsDabrafenib
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase Nek2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase Nek3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase Nek4 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase Nek5 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase Nek9 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a High affinity nerve growth factor receptor inhibitor
1High affinity nerve growth factor receptor antagonistsImatinib
2High affinity nerve growth factor receptor agonistsAmitriptyline
3High affinity nerve growth factor receptor activatorsAmitriptyline
4High affinity nerve growth factor receptor inhibitorsEntrectinib, Larotrectinib, Pralsetinib, Regorafenib
5High affinity nerve growth factor receptor stimulatorsCenegermin
Interacting GroupInteracting Drugs
Fostamatinib is a BDNF/NT-3 growth factors receptor inhibitor
1BDNF/NT-3 growth factors receptor agonistsAmitriptyline
2BDNF/NT-3 growth factors receptor inhibitorsEntrectinib, Larotrectinib
Interacting GroupInteracting Drugs
Fostamatinib is a NT-3 growth factor receptor inhibitor
1NT-3 growth factor receptor inhibitorsEntrectinib, Larotrectinib, Pralsetinib
Interacting GroupInteracting Drugs
Fostamatinib is a NUAK family SNF1-like kinase 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a NUAK family SNF1-like kinase 2 inhibitor
1NUAK family SNF1-like kinase 2 activatorsBempedoic acid
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase OSR1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PAK 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PAK 2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PAK 3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PAK 4 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PAK 6 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PAK 5 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Cyclin-dependent kinase 16 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Cyclin-dependent kinase 17 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Platelet-derived growth factor receptor alpha inhibitor
1Platelet-derived growth factor receptor alpha inhibitorsLenvatinib, Midostaurin, Nintedanib, Pazopanib, Ponatinib, Regorafenib, Ripretinib, Sunitinib
2Platelet-derived growth factor receptor alpha antagonistsImatinib, Midostaurin, Olaratumab
3Platelet-derived growth factor receptor alpha agonistsForeskin keratinocyte (neonatal)
4Platelet-derived growth factor receptor alpha substratesErdafitinib
Interacting GroupInteracting Drugs
Fostamatinib is a Platelet-derived growth factor receptor beta inhibitor
1Platelet-derived growth factor receptor beta antagonistsDasatinib, Imatinib, Midostaurin, Sorafenib, Trapidil
2Platelet-derived growth factor receptor beta inhibitorsMidostaurin, Nintedanib, Pazopanib, Pexidartinib, Pralsetinib, Regorafenib, Ripretinib, Sunitinib
3Platelet-derived growth factor receptor beta agonistsForeskin fibroblast (neonatal), Polaprezinc
4Platelet-derived growth factor receptor beta substratesErdafitinib
Interacting GroupInteracting Drugs
Fostamatinib is a 3-phosphoinositide-dependent protein kinase 1 inhibitor
13-phosphoinositide-dependent protein kinase 1 inhibitorsCelecoxib
Interacting GroupInteracting Drugs
Fostamatinib is a Cyclin-dependent kinase 15 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Phosphatidylinositol 4-kinase beta inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform inhibitor
1Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform inhibitorsCaffeine, Copanlisib, Duvelisib, Idelalisib, TG100-115
Interacting GroupInteracting Drugs
Fostamatinib is a Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform inhibitor
1Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform inhibitorsDuvelisib, TG100-115
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase pim-1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase pim-3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Phosphatidylinositol 5-phosphate 4-kinase type-2 beta inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase N1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase N2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PLK1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PLK2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PLK3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PLK4 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a 5'-AMP-activated protein kinase catalytic subunit alpha-1 inhibitor
15'-AMP-activated protein kinase catalytic subunit alpha-1 activatorsAdenosine phosphate, Phenformin
Interacting GroupInteracting Drugs
Fostamatinib is a 5'-AMP-activated protein kinase inhibitor
15'-AMP-activated protein kinase activatorsAcetylsalicylic acid, Adenosine phosphate
25'-AMP-activated protein kinase inducersTopiramate
Interacting GroupInteracting Drugs
Fostamatinib is a cAMP-dependent protein kinase catalytic subunit beta inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Protein kinase C delta type inhibitor
1Protein kinase C delta type ligandsIngenol mebutate
Interacting GroupInteracting Drugs
Fostamatinib is a Protein kinase C epsilon type inhibitor
1Protein kinase C epsilon type activatorsBryostatin 1
Interacting GroupInteracting Drugs
Fostamatinib is a Protein kinase C gamma type (PRKCG) inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Protein kinase C iota type inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Protein kinase C theta type inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase D1 inhibitor
1Serine/threonine-protein kinase D1 activatorsBryostatin 1
Interacting GroupInteracting Drugs
Fostamatinib is a cGMP-dependent protein kinase 2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase PRP4 homolog inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Focal adhesion kinase 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Protein-tyrosine kinase 2-beta inhibitor
1Protein-tyrosine kinase 2-beta antagonistsLeflunomide
2Protein-tyrosine kinase 2-beta inhibitorsBaricitinib
Interacting GroupInteracting Drugs
Fostamatinib is a Protein-tyrosine kinase 6 inhibitor
1Protein-tyrosine kinase 6 inhibitorsVandetanib, Zanubrutinib
Interacting GroupInteracting Drugs
Fostamatinib is a RAF proto-oncogene serine/threonine-protein kinase inhibitor
1RAF proto-oncogene serine/threonine-protein kinase inhibitorsDabrafenib, Regorafenib, Sorafenib
2RAF proto-oncogene serine/threonine-protein kinase antagonistsDabrafenib
3RAF proto-oncogene serine/threonine-protein kinase agonistsCholecystokinin
Interacting GroupInteracting Drugs
Fostamatinib is a Proto-oncogene tyrosine-protein kinase receptor Ret inhibitor
1Proto-oncogene tyrosine-protein kinase receptor Ret antagonistsCabozantinib
2Proto-oncogene tyrosine-protein kinase receptor Ret inhibitorsLenvatinib, Ponatinib, Pralsetinib, Regorafenib, Selpercatinib, Sorafenib
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase RIO1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase RIO2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase RIO3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Receptor-interacting serine/threonine-protein kinase 1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Receptor-interacting serine/threonine-protein kinase 2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Receptor-interacting serine/threonine-protein kinase 4 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Rho-associated protein kinase 2 inhibitor
1Rho-associated protein kinase 2 inhibitorsNetarsudil, Ripasudil
Interacting GroupInteracting Drugs
Fostamatinib is a Proto-oncogene tyrosine-protein kinase ROS inhibitor
1Proto-oncogene tyrosine-protein kinase ROS inhibitorsEntrectinib
Interacting GroupInteracting Drugs
Fostamatinib is a Ribosomal protein S6 kinase alpha-1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Ribosomal protein S6 kinase alpha-3 inhibitor
1Ribosomal protein S6 kinase alpha-3 inhibitorsAcetylsalicylic acid
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase SBK1 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Uncharacterized serine/threonine-protein kinase SBK3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase Sgk3 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase SIK1 inhibitor
1Serine/threonine-protein kinase SIK1 antagonistsDabrafenib
2Serine/threonine-protein kinase SIK1 inhibitorsDabrafenib
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase SIK2 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a STE20-like serine/threonine-protein kinase inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a SNF-related serine/threonine-protein kinase inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Proto-oncogene tyrosine-protein kinase Src inhibitor
1Proto-oncogene tyrosine-protein kinase Src inhibitorsBosutinib, Nintedanib, Ponatinib, Tirbanibulin
Interacting GroupInteracting Drugs
Fostamatinib is a Tyrosine-protein kinase Srms inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase 10 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase 16 inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase 17A inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase 17B inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Serine/threonine-protein kinase 32A inhibitor
Interacting GroupInteracting Drugs
Fostamatinib is a Cytochrome P450 3A4 substrate
1Cytochrome P450 3A4 substrates(R)-warfarin, (S)-Warfarin, 1,2-Benzodiazepine, 3,5-diiodothyropropionic acid, 5-androstenedione, 6-O-benzylguanine, 9-aminocamptothecin, Abemaciclib, Abiraterone, Acalabrutinib, Acenocoumarol, Acetaminophen, Adinazolam, Agmatine, Albendazole, Alclometasone, Aldosterone, Alfentanil, Alfuzosin, Aliskiren, Almotriptan, Alogliptin, Alosetron, Alpelisib, alpha-Tocopherol acetate, Alprazolam, Ambrisentan, Ambroxol, Amcinonide, Aminophenazone, Aminophylline, Amiodarone, Amitriptyline, Amlodipine, Amprenavir, Anastrozole, Androstenedione, Antipyrine, Apalutamide, Apixaban, Apremilast, Aprepitant, Aranidipine, Argatroban, Aripiprazole, Aripiprazole lauroxil, Artemether, Asenapine, Astemizole, Asunaprevir, Atazanavir, Atorvastatin, Atovaquone, Avanafil, Avapritinib, Axitinib, Azelastine, Azelnidipine, Azimilide, Azithromycin, Balaglitazone, Baloxavir marboxil, Banoxantrone, Baricitinib, Barnidipine, Beclomethasone dipropionate, Bedaquiline, Belinostat, Bencyclane, Benidipine, Benzphetamine, Bepridil, Betamethasone, Betamethasone phosphate, Bexarotene, Bezafibrate, Bicalutamide, Bictegravir, Bimatoprost, Bioallethrin, Bisoprolol, Blonanserin, Boceprevir, Bortezomib, Bosentan, Bosutinib, Brentuximab vedotin, Brexpiprazole, Brigatinib, Brinzolamide, Brivaracetam, Bromocriptine, Brotizolam, Budesonide, Bupivacaine, Buprenorphine, Buspirone, Busulfan, Butyrfentanyl, Cabazitaxel, Cabergoline, Cabozantinib, Caffeine, Calanolide A, Calcitriol, Canagliflozin, Cannabidiol, Capmatinib, Capravirine, Carbamazepine, Carboxyamidotriazole, Cariprazine, Caroverine, Carvedilol, Celecoxib, Cenobamate, Ceritinib, Cerivastatin, Cethromycin, Cevimeline, Chenodeoxycholic acid, Chlormadinone, Chloroquine, Chlorpheniramine, Chlorzoxazone, Cholecalciferol, Ciclesonide, Ciglitazone, Cilnidipine, Cilostazol, Cinacalcet, Cinnarizine, Cisapride, Citalopram, Clarithromycin, Clevidipine, Clindamycin, Clobazam, Clobetasol, Clobetasol propionate, Clobetasone, Clofibrate, Clomethiazole, Clomipramine, Clonazepam, Clonidine, Clopidogrel, Clorazepic acid, Clotiazepam, Clotrimazole, Clozapine, Cobicistat, Cobimetinib, Cocaine, Codeine, Colchicine, Conivaptan, Conjugated estrogens, Copanlisib, Corticosterone, Corticotropin, Cortisone acetate, Crizotinib, Cyclandelate, Cyclobenzaprine, Cyclophosphamide, Cyclosporine, Cyproterone acetate, Cytarabine, Dabrafenib, Daclatasvir, Dacomitinib, Dapagliflozin, Dapoxetine, Dapsone, Darifenacin, Darodipine, Darolutamide, Darunavir, Dasabuvir, Dasatinib, Daunorubicin, Deflazacort, Delamanid, Delavirdine, Demegestone, Desogestrel, Desonide, Desoxycorticosterone acetate, Desoxycorticosterone pivalate, Desvenlafaxine, Deutetrabenazine, Dexamethasone, Dexamethasone acetate, Dexamethasone isonicotinate, Dexchlorpheniramine maleate, Dexlansoprazole, Dexloxiglumide, Dexniguldipine, Dextromethorphan, Dextropropoxyphene, Dexverapamil, Diazepam, Diclofenac, Dienogest, Diethylstilbestrol, Difluocortolone, Difluprednate, Digitoxin, Dihydro-alpha-ergocryptine, Dihydrocodeine, Dihydroergocornine, Dihydroergocristine, Dihydroergocryptine, Dihydroergotamine, Diltiazem, Diphenadione, Disopyramide, Disulfiram, Docetaxel, Dofetilide, Dolasetron, Domperidone, Donepezil, Doravirine, Dotarizine, Doxazosin, Doxepin, Doxorubicin, Doxycycline, Dronabinol, Dronedarone, Drospirenone, Duvelisib, Dydrogesterone, Ebastine, Efavirenz, Efonidipine, Elbasvir, Eletriptan, Elexacaftor, Eliglustat, Elvitegravir, Emopamil, Enasidenib, Encorafenib, Enfortumab vedotin, Entrectinib, Enzalutamide, Eperisone, Epinastine, Eplerenone, Equilenin, Equilin, Eravacycline, Erdafitinib, Ergoloid mesylate, Ergometrine, Ergotamine, Erlotinib, Erythromycin, Escitalopram, Esketamine, Esomeprazole, Estazolam, Esterified estrogens, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Estramustine, Estrone, Estrone sulfate, Eszopiclone, Ethanol, Ethinylestradiol, Ethosuximide, Ethyl biscoumacetate, Ethylmorphine, Ethynodiol diacetate, Etizolam, Etonogestrel, Etoposide, Etoricoxib, Etravirine, Etynodiol, Everolimus, Exemestane, Fedratinib, Felbamate, Felodipine, Fendiline, Fenfluramine, Fentanyl, Fesoterodine, Finasteride, Fish oil, Flibanserin, Flucloxacillin, Fludrocortisone, Flumethasone, Flunarizine, Flunisolide, Flunitrazepam, Fluocinolone acetonide, Fluocinonide, Fluocortolone, Fluorometholone, Fluoxetine, Fluprednidene, Fluprednisolone, Fluprednisolone acetate, Flurandrenolide, Flurazepam, Fluspirilene, Flutamide, Fluticasone, Fluticasone furoate, Fluticasone propionate, Fluvastatin, Fluvoxamine, Fosamprenavir, Fosaprepitant, Fosnetupitant, Fosphenytoin, Fostemsavir, Fulvestrant, Fusidic acid, Galantamine, Gallopamil, Gefitinib, Gemfibrozil, Gestodene, Gestrinone, Gilteritinib, Glasdegib, Glyburide, Granisetron, Grazoprevir, Grepafloxacin, Guanfacine, Halcinonide, Halofantrine, Haloperidol, Halothane, HE3286, Hydrocodone, Hydrocortisone, Hydrocortisone aceponate, Hydrocortisone acetate, Hydrocortisone butyrate, Hydrocortisone cypionate, Hydrocortisone phosphate, Hydrocortisone probutate, Hydrocortisone succinate, Hydrocortisone valerate, Hydroxychloroquine, Hydroxyprogesterone, Hydroxyprogesterone caproate, Hydroxyzine, Ibrutinib, Ibuprofen, Icotinib, Idelalisib, Ifosfamide, Iloperidone, Imatinib, Imidafenacin, Imipramine, Imiquimod, Indacaterol, Indalpine, Indapamide, Indinavir, Ipecac, Irinotecan, Isavuconazole, Isavuconazonium, Isotretinoin, Isradipine, Istradefylline, Itraconazole, Ivabradine, Ivacaftor, Ivermectin, Ivosidenib, Ixabepilone, Ixazomib, Ketamine, Ketazolam, Ketobemidone, Ketoconazole, Lacidipine, Lacosamide, Lansoprazole, Lapatinib, Laquinimod, Larotrectinib, Lefamulin, Lemborexant, Lenvatinib, Lercanidipine, Letrozole, Levacetylmethadol, Levamlodipine, Levobupivacaine, Levocetirizine, Levomenthol, Levomilnacipran, Levonorgestrel, Lidocaine, Lidoflazine, Linagliptin, Liotrix, Lisuride, Lobeglitazone, Lomerizine, Lomitapide, Lonafarnib, Loperamide, Lopinavir, Loratadine, Lorazepam, Lorcaserin, Lorpiprazole, Losartan, Loteprednol etabonate, Lovastatin, Lumefantrine, Lurasidone, Lurbinectedin, Lynestrenol, Lysergic acid diethylamide, Macimorelin, Macitentan, Manidipine, Maraviroc, Medrogestone, Medroxyprogesterone acetate, Medrysone, Mefloquine, Megestrol acetate, Melengestrol, Meloxicam, Meperidine, Meprednisone, Mestranol, Methadone, Methaqualone, Methotrexate, Methoxyflurane, Methylergometrine, Methylprednisolone, Methylprednisone, Methyltestosterone, Methysergide, Metoclopramide, Metoprolol, Mexazolam, Mexiletine, Mianserin, Mibefradil, Midazolam, Midecamycin, Midostaurin, Mifepristone, Milnacipran, Mirabegron, Mirtazapine, Modafinil, Mometasone, Mometasone furoate, Montelukast, Morphine, Mycophenolate mofetil, Nabiximols, Naftopidil, Naloxegol, Nateglinide, Nebivolol, Nefazodone, Nelfinavir, Neratinib, Netoglitazone, Netupitant, Nevirapine, Nicardipine, Nicotine, Nifedipine, Niguldipine, Nilotinib, Niludipine, Nilvadipine, Nimesulide, Nimodipine, Nintedanib, Nisoldipine, Nitrazepam, Nitrendipine, Nomegestrol, Nomegestrol acetate, Norelgestromin, Norethindrone enanthate, Norethisterone, Norethynodrel, Norgestimate, Norgestrel, Nortriptyline, Nylidrin, Odanacatib, Olaparib, Oliceridine, Olopatadine, Omeprazole, Ondansetron, Opium, Orphenadrine, Osilodrostat, Osimertinib, Ospemifene, Otilonium, Oxybutynin, Oxycodone, Oxymorphone, Ozanimod, Paclitaxel, Palbociclib, Paliperidone, Palonosetron, Panobinostat, Pantoprazole, Paramethadione, Paramethasone, Parecoxib, Paricalcitol, Paritaprevir, Paroxetine, Pazopanib, Pemigatinib, Penfluridol, Perampanel, Perhexiline, Perospirone, Perphenazine, Pexidartinib, Phenacetin, Phenprocoumon, Phentermine, Phenytoin, Pimecrolimus, Pimozide, Pinacidil, Pinaverium, Pioglitazone, Piperaquine, Pipotiazine, Pitolisant, Plitidepsin, Polatuzumab vedotin, Pomalidomide, Ponatinib, Posaconazole, Pralsetinib, Pranlukast, Prasugrel, Prazepam, Praziquantel, Prednicarbate, Prednisolone, Prednisolone acetate, Prednisolone phosphate, Prednisone, Prednylidene, Pregnenolone, Prenylamine, Pretomanid, Primaquine, Progesterone, Promazine, Promegestone, Propacetamol, Propafenone, Propiverine, Propranolol, Prucalopride, Quazepam, Quetiapine, Quinacrine, Quingestanol, Quinidine, Quinine, Rabeprazole, Ramelteon, Ranolazine, Reboxetine, Regorafenib, Remdesivir, Repaglinide, Retapamulin, Ribociclib, Rifabutin, Rifalazil, Rifapentine, Rifaximin, Rilpivirine, Rimegepant, Rimexolone, Rimonabant, Riociguat, Ripretinib, Risdiplam, Risperidone, Ritonavir, Rivaroxaban, Rivoglitazone, Rofecoxib, Roflumilast, Rolapitant, Romidepsin, Ropivacaine, Rosiglitazone, Rotigotine, Roxithromycin, Rucaparib, Rufinamide, Rupatadine, Ruxolitinib, Safinamide, Salmeterol, Saquinavir, Saxagliptin, Segesterone acetate, Selegiline, Seletracetam, Selexipag, Selinexor, Selpercatinib, Selumetinib, Seratrodast, Sertindole, Sertraline, Sevoflurane, Sibutramine, Sildenafil, Silodosin, Simeprevir, Simvastatin, Siponimod, Sirolimus, Sitagliptin, SN-38, Solifenacin, Sonidegib, Sorafenib, St. John's Wort, Sufentanil, Sulfadiazine, Sulfamethoxazole, Sulfinpyrazone, Sunitinib, Suvorexant, Synthetic Conjugated Estrogens, A, Synthetic Conjugated Estrogens, B, Tacrolimus, Tadalafil, Tamoxifen, Tamsulosin, Tasimelteon, Tasosartan, Taurochenodeoxycholic acid, Tazemetostat, Telaprevir, Telithromycin, Temazepam, Temsirolimus, Tenapanor, Teniposide, Tenofovir, Tenofovir alafenamide, Terbinafine, Terfenadine, Terguride, Terodiline, Tesmilifene, Testosterone, Testosterone cypionate, Testosterone enanthate, Testosterone propionate, Testosterone undecanoate, Tetracycline, Tetrahydropalmatine, Tetrandrine, Tezacaftor, Theophylline, Thiamylal, Thiotepa, Tiagabine, Tianeptine, Ticagrelor, Tinidazole, Tiotropium, Tipranavir, Tirbanibulin, Tocofersolan, Tocopherol, Tofacitinib, Tolfenamic acid, Tolterodine, Tolvaptan, Toremifene, Trabectedin, Tramadol, Tranilast, Trastuzumab deruxtecan, Trastuzumab emtansine, Trazodone, Tretinoin, Triamcinolone, Triazolam, Triclabendazole, Trifarotene, Trimebutine, Trimethadione, Trimethoprim, Troleandomycin, Ubrogepant, Udenafil, Ulipristal, Umifenovir, Upadacitinib, Valbenazine, Valdecoxib, Vandetanib, Vanoxerine, Vardenafil, Velpatasvir, Vemurafenib, Venetoclax, Venlafaxine, Verapamil, Vibegron, Vicriviroc, Vilanterol, Vilazodone, Vinblastine, Vincristine, Vindesine, Vinflunine, Vinorelbine, Vinpocetine, Vismodegib, Vitamin D, Vitamin E, Vorapaxar, Voriconazole, Vortioxetine, Voxelotor, Voxilaprevir, Warfarin, WIN 55212-2, Yohimbine, Zafirlukast, Zaleplon, Zanubrutinib, Zidovudine, Zileuton, Ziprasidone, Zolpidem, Zomepirac, Zonisamide, Zopiclone, Zotepine, Zuclopenthixol
2Cytochrome P450 3A4 inducersAcetaminophen, Amcinonide, Aminoglutethimide, Amprenavir, Apalutamide, Aprepitant, Aprobarbital, Armodafinil, Artemether, Asunaprevir, Avasimibe, Azatadine, Barbital, Beclomethasone dipropionate, Betamethasone, Betamethasone phosphate, Bexarotene, Bosentan, Budesonide, Calcitriol, Carbamazepine, Cefradine, Cenobamate, Cerivastatin, Chlorphenesin, Chlorpromazine, Clevidipine, Clobazam, Clobetasol, Clobetasol propionate, Clocortolone acetate, Clofibrate, Cloprednol, Clotrimazole, Clozapine, Corticotropin, Cortisone, Cortisone acetate, Cortivazol, Cyclophosphamide, Dabrafenib, Deferasirox, Deflazacort, Delafloxacin, Desonide, Dexamethasone, Dexamethasone acetate, Dexamethasone isonicotinate, Dicloxacillin, Difluocortolone, Echinacea, Efavirenz, Enasidenib, Enzalutamide, Esketamine, Eslicarbazepine, Eslicarbazepine acetate, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Ethanol, Etoposide, Etravirine, Felbamate, Flucloxacillin, Flunisolide, Fluocinolone acetonide, Fluocinonide, Fluocortolone, Fluorometholone, Fluprednidene, Fluprednidene acetate, Fluticasone, Fluticasone furoate, Formestane, Fosaprepitant, Fosphenytoin, Genistein, Glycerol phenylbutyrate, Griseofulvin, Halometasone, Hydrocortamate, Hydrocortisone, Hydrocortisone aceponate, Hydrocortisone acetate, Hydrocortisone butyrate, Hydrocortisone probutate, Hydrocortisone succinate, Hydrocortisone valerate, Idelalisib, Ifosfamide, Isavuconazole, Isavuconazonium, Ivermectin, Ivosidenib, Ketamine, Lansoprazole, Lenvatinib, Lesinurad, Lumacaftor, Lumefantrine, Medroxyprogesterone acetate, Medrysone, Melengestrol acetate, Meperidine, Meprednisone, Metamizole, Methadone, Methylprednisolone, Methylprednisolone hemisuccinate, Metyrapone, Midostaurin, Mifepristone, Mitotane, Modafinil, Mometasone, Mometasone furoate, Nafcillin, Nevirapine, Nifedipine, Norgestimate, Omeprazole, Oritavancin, Orlistat, Osimertinib, Oxcarbazepine, Oxiconazole, Paclitaxel, Paramethasone, Pegvisomant, Pentobarbital, Perampanel, Pexidartinib, Phenobarbital, Phenylbutazone, Phenytoin, Pioglitazone, Pitolisant, Pralsetinib, Prednicarbate, Prednisolone, Prednisolone acetate, Prednisolone hemisuccinate, Prednisolone phosphate, Prednisone, Prednisone acetate, Prednylidene, Primidone, Probenecid, Progesterone, Propacetamol, Quinine, Rifabutin, Rifampicin, Rifamycin, Rifapentine, Rifaximin, Rimexolone, Rofecoxib, Rufinamide, Sarilumab, Seratrodast, Siltuximab, St. John's Wort, Sulfinpyrazone, Tamoxifen, Terbinafine, Terfenadine, Tesmilifene, Testosterone, Testosterone cypionate, Testosterone enanthate, Testosterone undecanoate, Thiamylal, Tocilizumab, Topiramate, Topotecan, Trametinib, Triamcinolone, Troglitazone, Vemurafenib, Vinblastine, Vitamin E, Warfarin
3Cytochrome P450 3A4 inhibitors6-Deoxyerythronolide B, Abametapir, Abemaciclib, Abiraterone, Acalabrutinib, Acetazolamide, Aldesleukin, Amiodarone, Amphotericin B, Amprenavir, Anastrozole, Aprepitant, Arsenic trioxide, Astemizole, Atazanavir, AVE9633, Azelastine, Azithromycin, Barnidipine, Benidipine, Berotralstat, Bicalutamide, Bifonazole, Black cohosh, Boceprevir, Bosutinib, Brefeldin A, Brentuximab vedotin, Bromocriptine, Bryostatin 1, Buprenorphine, Cabergoline, Candicidin, Capsaicin, Carbomycin, Caspofungin, Cenobamate, Ceritinib, Cerivastatin, Cethromycin, Chloramphenicol, Chlorzoxazone, Cimetidine, Ciprofloxacin, Citalopram, Clarithromycin, Clascoterone, Clevidipine, Clindamycin, Clofazimine, Clotrimazole, Clozapine, Cobicistat, Colchicine, Coltuximab ravtansine, Conivaptan, Crizotinib, Curcumin, Curcumin sulfate, Cyclosporine, Cyproterone acetate, Dalfopristin, Danazol, Danoprevir, Dapoxetine, Darunavir, Dasatinib, Daunorubicin, Delavirdine, Desipramine, Desvenlafaxine, Dexamethasone, Dexamethasone acetate, Dexamethasone isonicotinate, Dextropropoxyphene, Diazepam, Diclofenac, Diethylstilbestrol, Dihydroergotamine, Diltiazem, Dimethyl sulfoxide, Dirithromycin, Ditiocarb, Docetaxel, Doramectin, Dovitinib, Doxorubicin, Doxycycline, Dronedarone, Econazole, Edetate calcium disodium anhydrous, Edetate disodium anhydrous, Efavirenz, Efonidipine, Elbasvir, Elexacaftor, Elvitegravir, Enasidenib, Epinephrine, Epofolate, Epothilone D, Eprinomectin, Ergotamine, Erlotinib, Erythromycin, Ethanol, Etoposide, Etoricoxib, Ezetimibe, Felodipine, Fidaxomicin, Fluconazole, Fluoxetine, Flurithromycin, Fluticasone, Fluticasone furoate, Fluticasone propionate, Fluvastatin, Fluvoxamine, Fosamprenavir, Fosaprepitant, Fosnetupitant, Fusidic acid, Gefitinib, Ginkgo biloba, Glecaprevir, Glyburide, GPI-1485, Haloperidol, Hydralazine, Idelalisib, Ifosfamide, Imatinib, Indalpine, Indinavir, Indisulam, Irbesartan, Isavuconazole, Isavuconazonium, Isradipine, Itraconazole, Ivacaftor, Ixabepilone, Ketazolam, Ketoconazole, Kitasamycin, KOS-1584, Lanreotide, Lansoprazole, Lapatinib, Lenvatinib, Lercanidipine, Lestaurtinib, Letermovir, Levosalbutamol, Linagliptin, Lomustine, Lonafarnib, Loperamide, Lopinavir, Loratadine, Lorvotuzumab mertansine, Losartan, Lovastatin, Luliconazole, Manidipine, Medical Cannabis, Mefloquine, Mepartricin, Mequitazine, Methadone, Methimazole, Methylene blue, Methylergometrine, Metronidazole, Metyrapone, Mibefradil, Miconazole, Midazolam, Midecamycin, Midostaurin, Mifepristone, Milnacipran, Miocamycin, Mirtazapine, Mirvetuximab soravtansine, Mitemcinal, Mitoxantrone, Naloxone, Natamycin, Nefazodone, Nelfinavir, Netupitant, Niacin, Nicardipine, Nicotinamide, Nifedipine, Nilotinib, Nilvadipine, Nitric Oxide, Norfloxacin, Noscapine, Octreotide, Olanzapine, Olaparib, Oleandomycin, Omeprazole, Oritavancin, Orphenadrine, Osilodrostat, Osimertinib, Oxcarbazepine, Oxetacaine, Oxybutynin, Oxymetholone, Palbociclib, Paramethasone, Paroxetine, Pasireotide, Patupilone, Pazopanib, Peppermint oil, Pergolide, Pexidartinib, Phenelzine, Pilocarpine, Pimecrolimus, Pimozide, Piperaquine, Piperine, Posaconazole, Pralsetinib, Primaquine, Quinidine, Quinine, Quinupristin, Rabeprazole, Raloxifene, Ranitidine, Ranolazine, Reboxetine, Regorafenib, Remacemide, Remdesivir, Resveratrol, Ribociclib, Ridaforolimus, Rifamycin, Rilpivirine, Rimegepant, Ritonavir, Rokitamycin, Roxithromycin, Rucaparib, Rutin, Sagopilone, Salbutamol, Saquinavir, Saracatinib, Sarilumab, Selamectin, Seproxetine, Simeprevir, Sitaxentan, SN-38, Solithromycin, Somatostatin, Sorafenib, Stiripentol, Sulfanilamide, Sunitinib, Tamoxifen, Telaprevir, Telithromycin, Teniposide, Terfenadine, Tesmilifene, Testosterone cypionate, Testosterone enanthate, Testosterone undecanoate, Tetracycline, Ticagrelor, Tildipirosin, Tilmicosin, Tioconazole, Tipranavir, Tirbanibulin, Tofisopam, Topiroxostat, Topotecan, Toremifene, Trastuzumab emtansine, Triclabendazole, Troleandomycin, Tylosin, Tylvalosin, Valproic acid, Vapreotide, Venetoclax, Verapamil, Vinblastine, Voriconazole, WIN 55212-2, Zafirlukast, Zimelidine
Interacting GroupInteracting Drugs
Fostamatinib is a Cytochrome P450 3A4 inhibitor
1Cytochrome P450 3A4 substrates(R)-warfarin, (S)-Warfarin, 1,2-Benzodiazepine, 3,5-diiodothyropropionic acid, 5-androstenedione, 6-O-benzylguanine, 9-aminocamptothecin, Abemaciclib, Abiraterone, Acalabrutinib, Acenocoumarol, Acetaminophen, Adinazolam, Agmatine, Albendazole, Alclometasone, Aldosterone, Alfentanil, Alfuzosin, Aliskiren, Almotriptan, Alogliptin, Alosetron, Alpelisib, alpha-Tocopherol acetate, Alprazolam, Ambrisentan, Ambroxol, Amcinonide, Aminophenazone, Aminophylline, Amiodarone, Amitriptyline, Amlodipine, Amprenavir, Anastrozole, Androstenedione, Antipyrine, Apalutamide, Apixaban, Apremilast, Aprepitant, Aranidipine, Argatroban, Aripiprazole, Aripiprazole lauroxil, Artemether, Asenapine, Astemizole, Asunaprevir, Atazanavir, Atorvastatin, Atovaquone, Avanafil, Avapritinib, Axitinib, Azelastine, Azelnidipine, Azimilide, Azithromycin, Balaglitazone, Baloxavir marboxil, Banoxantrone, Baricitinib, Barnidipine, Beclomethasone dipropionate, Bedaquiline, Belinostat, Bencyclane, Benidipine, Benzphetamine, Bepridil, Betamethasone, Betamethasone phosphate, Bexarotene, Bezafibrate, Bicalutamide, Bictegravir, Bimatoprost, Bioallethrin, Bisoprolol, Blonanserin, Boceprevir, Bortezomib, Bosentan, Bosutinib, Brentuximab vedotin, Brexpiprazole, Brigatinib, Brinzolamide, Brivaracetam, Bromocriptine, Brotizolam, Budesonide, Bupivacaine, Buprenorphine, Buspirone, Busulfan, Butyrfentanyl, Cabazitaxel, Cabergoline, Cabozantinib, Caffeine, Calanolide A, Calcitriol, Canagliflozin, Cannabidiol, Capmatinib, Capravirine, Carbamazepine, Carboxyamidotriazole, Cariprazine, Caroverine, Carvedilol, Celecoxib, Cenobamate, Ceritinib, Cerivastatin, Cethromycin, Cevimeline, Chenodeoxycholic acid, Chlormadinone, Chloroquine, Chlorpheniramine, Chlorzoxazone, Cholecalciferol, Ciclesonide, Ciglitazone, Cilnidipine, Cilostazol, Cinacalcet, Cinnarizine, Cisapride, Citalopram, Clarithromycin, Clevidipine, Clindamycin, Clobazam, Clobetasol, Clobetasol propionate, Clobetasone, Clofibrate, Clomethiazole, Clomipramine, Clonazepam, Clonidine, Clopidogrel, Clorazepic acid, Clotiazepam, Clotrimazole, Clozapine, Cobicistat, Cobimetinib, Cocaine, Codeine, Colchicine, Conivaptan, Conjugated estrogens, Copanlisib, Corticosterone, Corticotropin, Cortisone acetate, Crizotinib, Cyclandelate, Cyclobenzaprine, Cyclophosphamide, Cyclosporine, Cyproterone acetate, Cytarabine, Dabrafenib, Daclatasvir, Dacomitinib, Dapagliflozin, Dapoxetine, Dapsone, Darifenacin, Darodipine, Darolutamide, Darunavir, Dasabuvir, Dasatinib, Daunorubicin, Deflazacort, Delamanid, Delavirdine, Demegestone, Desogestrel, Desonide, Desoxycorticosterone acetate, Desoxycorticosterone pivalate, Desvenlafaxine, Deutetrabenazine, Dexamethasone, Dexamethasone acetate, Dexamethasone isonicotinate, Dexchlorpheniramine maleate, Dexlansoprazole, Dexloxiglumide, Dexniguldipine, Dextromethorphan, Dextropropoxyphene, Dexverapamil, Diazepam, Diclofenac, Dienogest, Diethylstilbestrol, Difluocortolone, Difluprednate, Digitoxin, Dihydro-alpha-ergocryptine, Dihydrocodeine, Dihydroergocornine, Dihydroergocristine, Dihydroergocryptine, Dihydroergotamine, Diltiazem, Diphenadione, Disopyramide, Disulfiram, Docetaxel, Dofetilide, Dolasetron, Domperidone, Donepezil, Doravirine, Dotarizine, Doxazosin, Doxepin, Doxorubicin, Doxycycline, Dronabinol, Dronedarone, Drospirenone, Duvelisib, Dydrogesterone, Ebastine, Efavirenz, Efonidipine, Elbasvir, Eletriptan, Elexacaftor, Eliglustat, Elvitegravir, Emopamil, Enasidenib, Encorafenib, Enfortumab vedotin, Entrectinib, Enzalutamide, Eperisone, Epinastine, Eplerenone, Equilenin, Equilin, Eravacycline, Erdafitinib, Ergoloid mesylate, Ergometrine, Ergotamine, Erlotinib, Erythromycin, Escitalopram, Esketamine, Esomeprazole, Estazolam, Esterified estrogens, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Estramustine, Estrone, Estrone sulfate, Eszopiclone, Ethanol, Ethinylestradiol, Ethosuximide, Ethyl biscoumacetate, Ethylmorphine, Ethynodiol diacetate, Etizolam, Etonogestrel, Etoposide, Etoricoxib, Etravirine, Etynodiol, Everolimus, Exemestane, Fedratinib, Felbamate, Felodipine, Fendiline, Fenfluramine, Fentanyl, Fesoterodine, Finasteride, Fish oil, Flibanserin, Flucloxacillin, Fludrocortisone, Flumethasone, Flunarizine, Flunisolide, Flunitrazepam, Fluocinolone acetonide, Fluocinonide, Fluocortolone, Fluorometholone, Fluoxetine, Fluprednidene, Fluprednisolone, Fluprednisolone acetate, Flurandrenolide, Flurazepam, Fluspirilene, Flutamide, Fluticasone, Fluticasone furoate, Fluticasone propionate, Fluvastatin, Fluvoxamine, Fosamprenavir, Fosaprepitant, Fosnetupitant, Fosphenytoin, Fostemsavir, Fulvestrant, Fusidic acid, Galantamine, Gallopamil, Gefitinib, Gemfibrozil, Gestodene, Gestrinone, Gilteritinib, Glasdegib, Glyburide, Granisetron, Grazoprevir, Grepafloxacin, Guanfacine, Halcinonide, Halofantrine, Haloperidol, Halothane, HE3286, Hydrocodone, Hydrocortisone, Hydrocortisone aceponate, Hydrocortisone acetate, Hydrocortisone butyrate, Hydrocortisone cypionate, Hydrocortisone phosphate, Hydrocortisone probutate, Hydrocortisone succinate, Hydrocortisone valerate, Hydroxychloroquine, Hydroxyprogesterone, Hydroxyprogesterone caproate, Hydroxyzine, Ibrutinib, Ibuprofen, Icotinib, Idelalisib, Ifosfamide, Iloperidone, Imatinib, Imidafenacin, Imipramine, Imiquimod, Indacaterol, Indalpine, Indapamide, Indinavir, Ipecac, Irinotecan, Isavuconazole, Isavuconazonium, Isotretinoin, Isradipine, Istradefylline, Itraconazole, Ivabradine, Ivacaftor, Ivermectin, Ivosidenib, Ixabepilone, Ixazomib, Ketamine, Ketazolam, Ketobemidone, Ketoconazole, Lacidipine, Lacosamide, Lansoprazole, Lapatinib, Laquinimod, Larotrectinib, Lefamulin, Lemborexant, Lenvatinib, Lercanidipine, Letrozole, Levacetylmethadol, Levamlodipine, Levobupivacaine, Levocetirizine, Levomenthol, Levomilnacipran, Levonorgestrel, Lidocaine, Lidoflazine, Linagliptin, Liotrix, Lisuride, Lobeglitazone, Lomerizine, Lomitapide, Lonafarnib, Loperamide, Lopinavir, Loratadine, Lorazepam, Lorcaserin, Lorpiprazole, Losartan, Loteprednol etabonate, Lovastatin, Lumefantrine, Lurasidone, Lurbinectedin, Lynestrenol, Lysergic acid diethylamide, Macimorelin, Macitentan, Manidipine, Maraviroc, Medrogestone, Medroxyprogesterone acetate, Medrysone, Mefloquine, Megestrol acetate, Melengestrol, Meloxicam, Meperidine, Meprednisone, Mestranol, Methadone, Methaqualone, Methotrexate, Methoxyflurane, Methylergometrine, Methylprednisolone, Methylprednisone, Methyltestosterone, Methysergide, Metoclopramide, Metoprolol, Mexazolam, Mexiletine, Mianserin, Mibefradil, Midazolam, Midecamycin, Midostaurin, Mifepristone, Milnacipran, Mirabegron, Mirtazapine, Modafinil, Mometasone, Mometasone furoate, Montelukast, Morphine, Mycophenolate mofetil, Nabiximols, Naftopidil, Naloxegol, Nateglinide, Nebivolol, Nefazodone, Nelfinavir, Neratinib, Netoglitazone, Netupitant, Nevirapine, Nicardipine, Nicotine, Nifedipine, Niguldipine, Nilotinib, Niludipine, Nilvadipine, Nimesulide, Nimodipine, Nintedanib, Nisoldipine, Nitrazepam, Nitrendipine, Nomegestrol, Nomegestrol acetate, Norelgestromin, Norethindrone enanthate, Norethisterone, Norethynodrel, Norgestimate, Norgestrel, Nortriptyline, Nylidrin, Odanacatib, Olaparib, Oliceridine, Olopatadine, Omeprazole, Ondansetron, Opium, Orphenadrine, Osilodrostat, Osimertinib, Ospemifene, Otilonium, Oxybutynin, Oxycodone, Oxymorphone, Ozanimod, Paclitaxel, Palbociclib, Paliperidone, Palonosetron, Panobinostat, Pantoprazole, Paramethadione, Paramethasone, Parecoxib, Paricalcitol, Paritaprevir, Paroxetine, Pazopanib, Pemigatinib, Penfluridol, Perampanel, Perhexiline, Perospirone, Perphenazine, Pexidartinib, Phenacetin, Phenprocoumon, Phentermine, Phenytoin, Pimecrolimus, Pimozide, Pinacidil, Pinaverium, Pioglitazone, Piperaquine, Pipotiazine, Pitolisant, Plitidepsin, Polatuzumab vedotin, Pomalidomide, Ponatinib, Posaconazole, Pralsetinib, Pranlukast, Prasugrel, Prazepam, Praziquantel, Prednicarbate, Prednisolone, Prednisolone acetate, Prednisolone phosphate, Prednisone, Prednylidene, Pregnenolone, Prenylamine, Pretomanid, Primaquine, Progesterone, Promazine, Promegestone, Propacetamol, Propafenone, Propiverine, Propranolol, Prucalopride, Quazepam, Quetiapine, Quinacrine, Quingestanol, Quinidine, Quinine, Rabeprazole, Ramelteon, Ranolazine, Reboxetine, Regorafenib, Remdesivir, Repaglinide, Retapamulin, Ribociclib, Rifabutin, Rifalazil, Rifapentine, Rifaximin, Rilpivirine, Rimegepant, Rimexolone, Rimonabant, Riociguat, Ripretinib, Risdiplam, Risperidone, Ritonavir, Rivaroxaban, Rivoglitazone, Rofecoxib, Roflumilast, Rolapitant, Romidepsin, Ropivacaine, Rosiglitazone, Rotigotine, Roxithromycin, Rucaparib, Rufinamide, Rupatadine, Ruxolitinib, Safinamide, Salmeterol, Saquinavir, Saxagliptin, Segesterone acetate, Selegiline, Seletracetam, Selexipag, Selinexor, Selpercatinib, Selumetinib, Seratrodast, Sertindole, Sertraline, Sevoflurane, Sibutramine, Sildenafil, Silodosin, Simeprevir, Simvastatin, Siponimod, Sirolimus, Sitagliptin, SN-38, Solifenacin, Sonidegib, Sorafenib, St. John's Wort, Sufentanil, Sulfadiazine, Sulfamethoxazole, Sulfinpyrazone, Sunitinib, Suvorexant, Synthetic Conjugated Estrogens, A, Synthetic Conjugated Estrogens, B, Tacrolimus, Tadalafil, Tamoxifen, Tamsulosin, Tasimelteon, Tasosartan, Taurochenodeoxycholic acid, Tazemetostat, Telaprevir, Telithromycin, Temazepam, Temsirolimus, Tenapanor, Teniposide, Tenofovir, Tenofovir alafenamide, Terbinafine, Terfenadine, Terguride, Terodiline, Tesmilifene, Testosterone, Testosterone cypionate, Testosterone enanthate, Testosterone propionate, Testosterone undecanoate, Tetracycline, Tetrahydropalmatine, Tetrandrine, Tezacaftor, Theophylline, Thiamylal, Thiotepa, Tiagabine, Tianeptine, Ticagrelor, Tinidazole, Tiotropium, Tipranavir, Tirbanibulin, Tocofersolan, Tocopherol, Tofacitinib, Tolfenamic acid, Tolterodine, Tolvaptan, Toremifene, Trabectedin, Tramadol, Tranilast, Trastuzumab deruxtecan, Trastuzumab emtansine, Trazodone, Tretinoin, Triamcinolone, Triazolam, Triclabendazole, Trifarotene, Trimebutine, Trimethadione, Trimethoprim, Troleandomycin, Ubrogepant, Udenafil, Ulipristal, Umifenovir, Upadacitinib, Valbenazine, Valdecoxib, Vandetanib, Vanoxerine, Vardenafil, Velpatasvir, Vemurafenib, Venetoclax, Venlafaxine, Verapamil, Vibegron, Vicriviroc, Vilanterol, Vilazodone, Vinblastine, Vincristine, Vindesine, Vinflunine, Vinorelbine, Vinpocetine, Vismodegib, Vitamin D, Vitamin E, Vorapaxar, Voriconazole, Vortioxetine, Voxelotor, Voxilaprevir, Warfarin, WIN 55212-2, Yohimbine, Zafirlukast, Zaleplon, Zanubrutinib, Zidovudine, Zileuton, Ziprasidone, Zolpidem, Zomepirac, Zonisamide, Zopiclone, Zotepine, Zuclopenthixol
2Cytochrome P450 3A4 inducersAcetaminophen, Amcinonide, Aminoglutethimide, Amprenavir, Apalutamide, Aprepitant, Aprobarbital, Armodafinil, Artemether, Asunaprevir, Avasimibe, Azatadine, Barbital, Beclomethasone dipropionate, Betamethasone, Betamethasone phosphate, Bexarotene, Bosentan, Budesonide, Calcitriol, Carbamazepine, Cefradine, Cenobamate, Cerivastatin, Chlorphenesin, Chlorpromazine, Clevidipine, Clobazam, Clobetasol, Clobetasol propionate, Clocortolone acetate, Clofibrate, Cloprednol, Clotrimazole, Clozapine, Corticotropin, Cortisone, Cortisone acetate, Cortivazol, Cyclophosphamide, Dabrafenib, Deferasirox, Deflazacort, Delafloxacin, Desonide, Dexamethasone, Dexamethasone acetate, Dexamethasone isonicotinate, Dicloxacillin, Difluocortolone, Echinacea, Efavirenz, Enasidenib, Enzalutamide, Esketamine, Eslicarbazepine, Eslicarbazepine acetate, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Ethanol, Etoposide, Etravirine, Felbamate, Flucloxacillin, Flunisolide, Fluocinolone acetonide, Fluocinonide, Fluocortolone, Fluorometholone, Fluprednidene, Fluprednidene acetate, Fluticasone, Fluticasone furoate, Formestane, Fosaprepitant, Fosphenytoin, Genistein, Glycerol phenylbutyrate, Griseofulvin, Halometasone, Hydrocortamate, Hydrocortisone, Hydrocortisone aceponate, Hydrocortisone acetate, Hydrocortisone butyrate, Hydrocortisone probutate, Hydrocortisone succinate, Hydrocortisone valerate, Idelalisib, Ifosfamide, Isavuconazole, Isavuconazonium, Ivermectin, Ivosidenib, Ketamine, Lansoprazole, Lenvatinib, Lesinurad, Lumacaftor, Lumefantrine, Medroxyprogesterone acetate, Medrysone, Melengestrol acetate, Meperidine, Meprednisone, Metamizole, Methadone, Methylprednisolone, Methylprednisolone hemisuccinate, Metyrapone, Midostaurin, Mifepristone, Mitotane, Modafinil, Mometasone, Mometasone furoate, Nafcillin, Nevirapine, Nifedipine, Norgestimate, Omeprazole, Oritavancin, Orlistat, Osimertinib, Oxcarbazepine, Oxiconazole, Paclitaxel, Paramethasone, Pegvisomant, Pentobarbital, Perampanel, Pexidartinib, Phenobarbital, Phenylbutazone, Phenytoin, Pioglitazone, Pitolisant, Pralsetinib, Prednicarbate, Prednisolone, Prednisolone acetate, Prednisolone hemisuccinate, Prednisolone phosphate, Prednisone, Prednisone acetate, Prednylidene, Primidone, Probenecid, Progesterone, Propacetamol, Quinine, Rifabutin, Rifampicin, Rifamycin, Rifapentine, Rifaximin, Rimexolone, Rofecoxib, Rufinamide, Sarilumab, Seratrodast, Siltuximab, St. John's Wort, Sulfinpyrazone, Tamoxifen, Terbinafine, Terfenadine, Tesmilifene, Testosterone, Testosterone cypionate, Testosterone enanthate, Testosterone undecanoate, Thiamylal, Tocilizumab, Topiramate, Topotecan, Trametinib, Triamcinolone, Troglitazone, Vemurafenib, Vinblastine, Vitamin E, Warfarin
3Cytochrome P450 3A4 inhibitors6-Deoxyerythronolide B, Abametapir, Abemaciclib, Abiraterone, Acalabrutinib, Acetazolamide, Aldesleukin, Amiodarone, Amphotericin B, Amprenavir, Anastrozole, Aprepitant, Arsenic trioxide, Astemizole, Atazanavir, AVE9633, Azelastine, Azithromycin, Barnidipine, Benidipine, Berotralstat, Bicalutamide, Bifonazole, Black cohosh, Boceprevir, Bosutinib, Brefeldin A, Brentuximab vedotin, Bromocriptine, Bryostatin 1, Buprenorphine, Cabergoline, Candicidin, Capsaicin, Carbomycin, Caspofungin, Cenobamate, Ceritinib, Cerivastatin, Cethromycin, Chloramphenicol, Chlorzoxazone, Cimetidine, Ciprofloxacin, Citalopram, Clarithromycin, Clascoterone, Clevidipine, Clindamycin, Clofazimine, Clotrimazole, Clozapine, Cobicistat, Colchicine, Coltuximab ravtansine, Conivaptan, Crizotinib, Curcumin, Curcumin sulfate, Cyclosporine, Cyproterone acetate, Dalfopristin, Danazol, Danoprevir, Dapoxetine, Darunavir, Dasatinib, Daunorubicin, Delavirdine, Desipramine, Desvenlafaxine, Dexamethasone, Dexamethasone acetate, Dexamethasone isonicotinate, Dextropropoxyphene, Diazepam, Diclofenac, Diethylstilbestrol, Dihydroergotamine, Diltiazem, Dimethyl sulfoxide, Dirithromycin, Ditiocarb, Docetaxel, Doramectin, Dovitinib, Doxorubicin, Doxycycline, Dronedarone, Econazole, Edetate calcium disodium anhydrous, Edetate disodium anhydrous, Efavirenz, Efonidipine, Elbasvir, Elexacaftor, Elvitegravir, Enasidenib, Epinephrine, Epofolate, Epothilone D, Eprinomectin, Ergotamine, Erlotinib, Erythromycin, Ethanol, Etoposide, Etoricoxib, Ezetimibe, Felodipine, Fidaxomicin, Fluconazole, Fluoxetine, Flurithromycin, Fluticasone, Fluticasone furoate, Fluticasone propionate, Fluvastatin, Fluvoxamine, Fosamprenavir, Fosaprepitant, Fosnetupitant, Fusidic acid, Gefitinib, Ginkgo biloba, Glecaprevir, Glyburide, GPI-1485, Haloperidol, Hydralazine, Idelalisib, Ifosfamide, Imatinib, Indalpine, Indinavir, Indisulam, Irbesartan, Isavuconazole, Isavuconazonium, Isradipine, Itraconazole, Ivacaftor, Ixabepilone, Ketazolam, Ketoconazole, Kitasamycin, KOS-1584, Lanreotide, Lansoprazole, Lapatinib, Lenvatinib, Lercanidipine, Lestaurtinib, Letermovir, Levosalbutamol, Linagliptin, Lomustine, Lonafarnib, Loperamide, Lopinavir, Loratadine, Lorvotuzumab mertansine, Losartan, Lovastatin, Luliconazole, Manidipine, Medical Cannabis, Mefloquine, Mepartricin, Mequitazine, Methadone, Methimazole, Methylene blue, Methylergometrine, Metronidazole, Metyrapone, Mibefradil, Miconazole, Midazolam, Midecamycin, Midostaurin, Mifepristone, Milnacipran, Miocamycin, Mirtazapine, Mirvetuximab soravtansine, Mitemcinal, Mitoxantrone, Naloxone, Natamycin, Nefazodone, Nelfinavir, Netupitant, Niacin, Nicardipine, Nicotinamide, Nifedipine, Nilotinib, Nilvadipine, Nitric Oxide, Norfloxacin, Noscapine, Octreotide, Olanzapine, Olaparib, Oleandomycin, Omeprazole, Oritavancin, Orphenadrine, Osilodrostat, Osimertinib, Oxcarbazepine, Oxetacaine, Oxybutynin, Oxymetholone, Palbociclib, Paramethasone, Paroxetine, Pasireotide, Patupilone, Pazopanib, Peppermint oil, Pergolide, Pexidartinib, Phenelzine, Pilocarpine, Pimecrolimus, Pimozide, Piperaquine, Piperine, Posaconazole, Pralsetinib, Primaquine, Quinidine, Quinine, Quinupristin, Rabeprazole, Raloxifene, Ranitidine, Ranolazine, Reboxetine, Regorafenib, Remacemide, Remdesivir, Resveratrol, Ribociclib, Ridaforolimus, Rifamycin, Rilpivirine, Rimegepant, Ritonavir, Rokitamycin, Roxithromycin, Rucaparib, Rutin, Sagopilone, Salbutamol, Saquinavir, Saracatinib, Sarilumab, Selamectin, Seproxetine, Simeprevir, Sitaxentan, SN-38, Solithromycin, Somatostatin, Sorafenib, Stiripentol, Sulfanilamide, Sunitinib, Tamoxifen, Telaprevir, Telithromycin, Teniposide, Terfenadine, Tesmilifene, Testosterone cypionate, Testosterone enanthate, Testosterone undecanoate, Tetracycline, Ticagrelor, Tildipirosin, Tilmicosin, Tioconazole, Tipranavir, Tirbanibulin, Tofisopam, Topiroxostat, Topotecan, Toremifene, Trastuzumab emtansine, Triclabendazole, Troleandomycin, Tylosin, Tylvalosin, Valproic acid, Vapreotide, Venetoclax, Verapamil, Vinblastine, Voriconazole, WIN 55212-2, Zafirlukast, Zimelidine
Interacting GroupInteracting Drugs
Fostamatinib is a UDP-glucuronosyltransferase 1-9 substrate
1UDP-glucuronosyltransferase 1-9 substratesAcetaminophen, Ambrisentan, Artenimol, Artesunate, Ataluren, Canagliflozin, Dabigatran etexilate, Dapagliflozin, Dexibuprofen, Diclofenac, Dolutegravir, Empagliflozin, Enasidenib, Entacapone, Ertugliflozin, Ethinylestradiol, Etodolac, Ezogabine, Fenofibrate, Flurbiprofen, Formoterol, Gavestinel, Gemfibrozil, Glasdegib, Haloperidol, Ibuprofen, Indomethacin, Irinotecan, Ketobemidone, Labetalol, Lumiracoxib, Mycophenolate mofetil, Mycophenolic acid, Naproxen, Nateglinide, Oxazepam, Phenytoin, Propacetamol, Propofol, Regorafenib, Seratrodast, Sorafenib, Tapentadol, Topiroxostat, Troglitazone, Umifenovir, Vadimezan, Valdecoxib, Valproic acid, Zileuton
2UDP-glucuronosyltransferase 1-9 inhibitorsDeferasirox, Diflunisal, Eltrombopag, Fosphenytoin, Isavuconazole, Mefenamic acid, Methylene blue, Morniflumate, Niflumic acid, Phenytoin, Regorafenib, Rifampicin, Sorafenib, Umifenovir
Interacting GroupInteracting Drugs
Fostamatinib is a ATP-binding cassette sub-family G member 2 inhibitor
1ATP-binding cassette sub-family G member 2 substratesAbemaciclib, Afatinib, Allopurinol, Alpelisib, Alvocidib, Apixaban, Artesunate, Baricitinib, Berotralstat, Brigatinib, Camptothecin, Carboplatin, Celecoxib, Cerivastatin, Cisplatin, Cladribine, Clofarabine, Conjugated estrogens, Copanlisib, Dabrafenib, Dacomitinib, Dactinomycin, Darolutamide, Dasatinib, Daunorubicin, Delafloxacin, Docetaxel, Dolutegravir, Donepezil, Doxorubicin, Duvelisib, Empagliflozin, Enasidenib, Ertugliflozin, Etoposide, Ezetimibe, Fimasartan, Fluorouracil, Folic acid, Fostemsavir, Gefitinib, Glasdegib, Glecaprevir, Glyburide, Idelalisib, Imatinib, Irinotecan, Ivermectin, Lamivudine, Larotrectinib, Leflunomide, Lenvatinib, Lusutrombopag, Methotrexate, Mitoxantrone, Mycophenolate mofetil, Nifurtimox, Nilotinib, Nitrofurantoin, Ombitasvir, Osimertinib, Oxaliplatin, Ozanimod, Palbociclib, Pantoprazole, Pazopanib, Pemigatinib, Pibrentasvir, Pitavastatin, Ponatinib, Pralatrexate, Pralsetinib, Prasterone, Pravastatin, Prazosin, Raloxifene, Revefenacin, Riluzole, Rimegepant, Riociguat, Ripretinib, Risdiplam, Rivaroxaban, Rosuvastatin, Rucaparib, Selpercatinib, Selumetinib, Simeprevir, Sofosbuvir, Sorafenib, Sulfasalazine, Sumatriptan, Talazoparib, Tamoxifen, Tazemetostat, Tegaserod, Teniposide, Tenofovir alafenamide, Teriflunomide, Testosterone, Testosterone cypionate, Testosterone enanthate, Testosterone undecanoate, Tezacaftor, Topotecan, Trastuzumab deruxtecan, Tucatinib, Ubrogepant, Upadacitinib, Velpatasvir, Vemurafenib, Vincristine, Voxilaprevir, Zidovudine
2ATP-binding cassette sub-family G member 2 inhibitorsAbemaciclib, Afatinib, Alectinib, Avatrombopag, Baricitinib, Beclomethasone dipropionate, Brigatinib, Buprenorphine, Cabazitaxel, Caffeine, Cannabidiol, Capmatinib, Clofazimine, Cobicistat, Cyclosporine, Dabrafenib, Daclatasvir, Dacomitinib, Daidzin, Darolutamide, Dasabuvir, Dasatinib, Dexamethasone, Dexamethasone acetate, Diethylstilbestrol, Dovitinib, Dronabinol, Elacridar, Eltrombopag, Enasidenib, Erlotinib, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Estrone, Fedratinib, Fostemsavir, Fusidic acid, Gefitinib, Genistein, Gilteritinib, Glasdegib, Glecaprevir, Hesperetin, Imatinib, Isavuconazole, Istradefylline, Lansoprazole, Lasmiditan, Letermovir, Lonafarnib, Medical Cannabis, Nabiximols, Naringenin, Nelfinavir, Nilotinib, Novobiocin, Olaparib, Omeprazole, Palbociclib, Pantoprazole, Paritaprevir, Pibrentasvir, Ponatinib, Pralsetinib, Progesterone, Quercetin, Rabeprazole, Regorafenib, Relugolix, Rilpivirine, Ripretinib, Ritonavir, Rolapitant, Rucaparib, Safinamide, Saquinavir, Selpercatinib, Simeprevir, Sorafenib, Sulfasalazine, Sunitinib, Tafamidis, Taurocholic acid, Telmisartan, Teriflunomide, Topiroxostat, Upadacitinib, Vandetanib, Velpatasvir, Vemurafenib, Venetoclax, Vismodegib, Voxilaprevir
3ATP-binding cassette sub-family G member 2 inducersApalutamide, Cholesterol, Dovitinib, Progesterone, Venlafaxine
4ATP-binding cassette sub-family G member 2 antagonistsZafirlukast
5ATP-binding cassette sub-family G member 2 weak inhibitorsCobimetinib
6ATP-binding cassette sub-family G member 2 transportersLedipasvir
7ATP-binding cassette sub-family G member 2 modulatorsAvapritinib
Interacting GroupInteracting Drugs
Fostamatinib is a ATP-binding cassette sub-family B member 5 substrate
1ATP-binding cassette sub-family B member 5 substratesAmrubicin, Baloxavir marboxil, Bilastine, Brentuximab vedotin, Brigatinib, Dasabuvir, Delafloxacin, Naldemedine, Vinflunine
2ATP-binding cassette sub-family B member 5 inhibitorsBilastine, Brigatinib, Dofequidar, Lofexidine
3ATP-binding cassette sub-family B member 5 inducersDoxycycline