Showing BioInteractions for Formoterol (DB00983)

BioInteractor utilizes data on drug-target, -enzyme and -transporter associations to provide insight on drug-drug interactions. It allows you to identify, for instance, which drugs act similarly on the same target. Such drugs may have additive pharmacodynamic effects if given concomitantly. Conversely, two drugs may antagonize the beneficial effects of each other by having opposite actions on a specific drug target. BioInteractor uses ranked drug-enzyme association information to predict enzyme-mediated drug interactions that may be clinically relevant.
Interacting GroupInteracting Drugs
Formoterol is a Beta-2 adrenergic receptor agonist
1Beta-2 adrenergic receptor antagonistsAlprenolol, Arotinolol, Asenapine, Atenolol, Betaxolol, Bevantolol, Bisoprolol, Bupranolol, Carteolol, Carvedilol, Desipramine, Labetalol, Levobunolol, Metipranolol, Metoprolol, Nadolol, Nebivolol, Oxprenolol, Penbutolol, Propafenone, Propranolol, Sotalol, Timolol
2Beta-2 adrenergic receptor agonistsAlbuterol, Arbutamine, Arformoterol, Bambuterol, Bedoradrine, Celiprolol, Clenbuterol, Dipivefrin, Dobutamine, Doxofylline, Droxidopa, Ephedra sinica root, Ephedrine, Epinephrine, Etafedrine, Fenoterol, Indacaterol, Isoetharine, Isoprenaline, Levosalbutamol, Norepinephrine, Olodaterol, Orciprenaline, Phenylpropanolamine, Pirbuterol, Procaterol, Protokylol, Racepinephrine, Ritodrine, Salmeterol, Terbutaline, Vilanterol
3Beta-2 adrenergic receptor partial agonistsAcebutolol, Bopindolol, Penbutolol, Pindolol, Pseudoephedrine
4Beta-2 adrenergic receptor bindersCabergoline
5Beta-2 adrenergic receptor ligandsAripiprazole
Interacting GroupInteracting Drugs
Formoterol is a Beta-1 adrenergic receptor agonist
1Beta-1 adrenergic receptor antagonistsAlprenolol, Arotinolol, Asenapine, Atenolol, Betaxolol, Bevantolol, Bisoprolol, Bupranolol, Carvedilol, Celiprolol, Dronedarone, Esmolol, Labetalol, Levobetaxolol, Levobunolol, Metipranolol, Metoprolol, Nadolol, Nebivolol, Oxprenolol, Penbutolol, Practolol, Propafenone, Propranolol, Ranolazine, Sotalol, Terbutaline, Timolol
2Beta-1 adrenergic receptor agonistsAlbuterol, Arbutamine, Clenbuterol, DL-Methylephedrine, Dobutamine, Droxidopa, Ephedra sinica root, Ephedrine, Epinephrine, Fenoterol, Isoetharine, Isoprenaline, Norepinephrine, Phenylpropanolamine, Pirbuterol, Pseudoephedrine, Racepinephrine
3Beta-1 adrenergic receptor partial agonistsAcebutolol, Bopindolol, Carteolol, Penbutolol, Pindolol, Pseudoephedrine, Xamoterol
4Beta-1 adrenergic receptor bindersCabergoline, Loxapine
5Beta-1 adrenergic receptor ligandsAripiprazole, Vortioxetine
6Beta-1 adrenergic receptor inverse agonistsSalmeterol
7Beta-1 adrenergic receptor inhibitorsLamotrigine
Interacting GroupInteracting Drugs
Formoterol is a Beta-3 adrenergic receptor agonist
1Beta-3 adrenergic receptor agonistsArbutamine, Celiprolol, Clenbuterol, Droxidopa, Ephedra sinica root, Fenoterol, Isoprenaline, Mirabegron, Nebivolol, Norepinephrine, Pindolol, Racepinephrine, Solabegron, Terbutaline, Vibegron
2Beta-3 adrenergic receptor antagonistsAlprenolol, Bupranolol, Propranolol
3Beta-3 adrenergic receptor inverse agonistsSalmeterol
Interacting GroupInteracting Drugs
Formoterol is a Cytochrome P450 2D6 substrate
1Cytochrome P450 2D6 substrates4-Methoxyamphetamine, 5-methoxy-N,N-dimethyltryptamine, Acebutolol, Acetaminophen, Almotriptan, Alogliptin, Alprenolol, Aminophenazone, Amitriptyline, Amoxapine, Amphetamine, Amprenavir, Anisodamine, Antipyrine, Aprindine, Arformoterol, Aripiprazole, Aripiprazole lauroxil, Arotinolol, Asenapine, Astemizole, Asunaprevir, Atenolol, Atomoxetine, Azelastine, Azimilide, Befunolol, Benzyl alcohol, Bepridil, Betaxolol, Bevantolol, Bicifadine, Bopindolol, Bortezomib, Brexpiprazole, Bucindolol, Bufuralol, Bupivacaine, Bupranolol, Buprenorphine, Buspirone, Butyrfentanyl, Caffeine, Cannabidiol, Cariprazine, Carteolol, Carvedilol, Celecoxib, Celiprolol, Cevimeline, Chloroquine, Chlorpheniramine, Chlorpromazine, Chlorzoxazone, Ciclesonide, Cilostazol, Cinnarizine, Citalopram, Clevidipine, Clomipramine, Clonidine, Cloranolol, Clozapine, Codeine, Cyclobenzaprine, Dacomitinib, Dapagliflozin, Dapoxetine, Darifenacin, Dasabuvir, Debrisoquine, Delavirdine, Desipramine, Deutetrabenazine, Dexchlorpheniramine, Dexchlorpheniramine maleate, Dexfenfluramine, Dextroamphetamine, Dextromethorphan, Dextropropoxyphene, Dihydrocodeine, Diltiazem, Diphenhydramine, Dolasetron, Domperidone, Donepezil, Dosulepin, Doxazosin, Doxepin, Dronedarone, Duloxetine, Elagolix, Eletriptan, Eliglustat, Enasidenib, Encainide, Enclomiphene, Encorafenib, Epanolol, Epinastine, Erlotinib, Esatenolol, Escitalopram, Esmirtazapine, Esmolol, Ethylmorphine, Fenfluramine, Fesoterodine, Flecainide, Flunarizine, Fluoxetine, Fluvastatin, Fluvoxamine, Fusidic acid, Galantamine, Gefitinib, Haloperidol, Hydrocodone, Hydroxychloroquine, Ibrutinib, Idarubicin, Iloperidone, Imatinib, Imipramine, Indenolol, Ipecac, Istradefylline, Ixazomib, Labetalol, Landiolol, Letermovir, Levobetaxolol, Levobunolol, Levomilnacipran, Lidocaine, Lisdexamfetamine, Lofexidine, Loperamide, Lopinavir, Loratadine, Lorcaserin, Lorpiprazole, Lysergic acid diethylamide, Maprotiline, Meclizine, Meperidine, Mephenytoin, Mepindolol, Mequitazine, Mesoridazine, Metamfetamine, Methadone, Methotrimeprazine, Methoxyflurane, Methylene blue, Metipranolol, Metoclopramide, Metoprolol, Mexiletine, Mianserin, Midodrine, Midomafetamine, Minaprine, Mirabegron, Mirtazapine, Moclobemide, Nabiximols, Nateglinide, Nebivolol, Nefazodone, Netupitant, Nevirapine, Nicergoline, Nicotine, Nortriptyline, Olanzapine, Oliceridine, Ondansetron, Opium, Osilodrostat, Oxamniquine, Oxprenolol, Oxycodone, Oxymorphone, Paliperidone, Palonosetron, Paroxetine, Penbutolol, Pentamidine, Perhexiline, Perospirone, Perphenazine, Phenacetin, Phenformin, Phenytoin, Pindolol, Piperazine, Pipotiazine, Pirfenidone, Pitolisant, Ponatinib, Practolol, Pralsetinib, Procainamide, Prochlorperazine, Progesterone, Promazine, Promethazine, Propacetamol, Propafenone, Propranolol, Quetiapine, Quinine, Ranolazine, Remdesivir, Remoxipride, Repinotan, Revefenacin, Ripretinib, Risperidone, Ritonavir, Rotigotine, Rucaparib, Rupatadine, Selegiline, Sertindole, Sertraline, Sildenafil, Simvastatin, Solifenacin, Sotalol, Sparteine, Tafenoquine, Talinolol, Tamoxifen, Tamsulosin, Tapentadol, Tegaserod, Terfenadine, Tertatolol, Tesmilifene, Tetrabenazine, Theophylline, Thioridazine, Ticlopidine, Timolol, Tiotropium, Tipranavir, Tolterodine, Trabectedin, Tramadol, Trazodone, Triclabendazole, Trimipramine, Umeclidinium, Umifenovir, Upadacitinib, Valbenazine, Venlafaxine, Vernakalant, Vilazodone, Vortioxetine, Yohimbine, Zolpidem, Zuclopenthixol
2Cytochrome P450 2D6 inhibitors1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine, Abemaciclib, Abiraterone, Acebutolol, Amiodarone, Amlodipine, Amodiaquine, Amoxapine, Artenimol, Asenapine, Asunaprevir, Atorvastatin, Azelastine, Bepridil, Berotralstat, Bicalutamide, Biperiden, Black cohosh, Buprenorphine, Bupropion, Cannabidiol, Celecoxib, Cerivastatin, Chloroquine, Chlorpheniramine, Chlorpromazine, Cimetidine, Cinacalcet, Cisapride, Citalopram, Clascoterone, Clemastine, Clinafloxacin, Clobazam, Clofazimine, Clomipramine, Clotrimazole, Clozapine, Cobicistat, Cocaine, Curcumin, Curcumin sulfate, Cyclosporine, Dacomitinib, Darifenacin, Darunavir, Delavirdine, Deramciclane, Desipramine, Desvenlafaxine, Dexchlorpheniramine, Dexchlorpheniramine maleate, Dexfenfluramine, Dexmedetomidine, Dextropropoxyphene, Diacerein, Dimethyl sulfoxide, Diphenhydramine, Dosulepin, Doxepin, Doxorubicin, Dronedarone, Duloxetine, Efavirenz, Elexacaftor, Eliglustat, Enasidenib, Entacapone, Epinastine, Escitalopram, Ethambutol, Etoricoxib, Everolimus, Fedratinib, Felodipine, Fenfluramine, Flecainide, Fluoxetine, Fluphenazine, Fluvoxamine, Fusidic acid, Gefitinib, Glycerol phenylbutyrate, Halofantrine, Haloperidol, Hydroxychloroquine, Hydroxyurea, Hydroxyzine, Imatinib, Imipramine, Indinavir, Indisulam, Iproniazid, Isavuconazole, Isoniazid, Ketoconazole, Labetalol, Lansoprazole, Lasmiditan, Lenvatinib, Lercanidipine, Lidocaine, Lisdexamfetamine, Lomustine, Loratadine, Lorcaserin, Lumefantrine, Manidipine, Medical Cannabis, Melperone, Menadione, Mepyramine, Methadone, Methimazole, Methotrimeprazine, Methylene blue, Metoclopramide, Metoprolol, Mibefradil, Miconazole, Midostaurin, Mifepristone, Mirabegron, Mizolastine, Moclobemide, Nabiximols, Naloxegol, Nefazodone, Nelfinavir, Nevirapine, Niacin, Nicardipine, Nicotinamide, Nifedipine, Nilotinib, Nortriptyline, Olanzapine, Omeprazole, Oritavancin, Orphenadrine, Osilodrostat, Ospemifene, Oxamniquine, Oxprenolol, Oxybutynin, Oxymetholone, Panobinostat, Paroxetine, Pazopanib, Peginterferon alfa-2b, Perhexiline, Perphenazine, Phenelzine, Phenylbutyric acid, Pimozide, Pindolol, Pipotiazine, Pitolisant, Primaquine, Proguanil, Promethazine, Propafenone, Propranolol, Quinidine, Quinine, Rabeprazole, Ranitidine, Ranolazine, Reboxetine, Rhein, Rilpivirine, Risperidone, Ritanserin, Ritonavir, Rolapitant, Rosiglitazone, Rotigotine, Rucaparib, Safinamide, Saquinavir, Selegiline, Sertraline, Sorafenib, Sparteine, St. John's Wort, Stiripentol, Sulconazole, Sulfanilamide, Sulfaphenazole, Tamoxifen, Tegaserod, Temsirolimus, Terbinafine, Terfenadine, Thioridazine, Thiothixene, Ticlopidine, Tipranavir, Tirbanibulin, Tranylcypromine, Trazodone, Triclabendazole, Tripelennamine, Trospium, Ubrogepant, Vemurafenib, Venlafaxine, Verapamil, Vernakalant, Vinblastine, Vinorelbine, Zafirlukast
3Cytochrome P450 2D6 inducersModafinil, Oritavancin
Interacting GroupInteracting Drugs
Formoterol is a Cytochrome P450 2C19 substrate
1Cytochrome P450 2C19 substrates(R)-warfarin, (S)-Warfarin, Acenocoumarol, Adinazolam, Albendazole, Almotriptan, Ambrisentan, Aminophenazone, Amiodarone, Amitriptyline, Antipyrine, Apixaban, Aprepitant, Arformoterol, Artemether, Asunaprevir, Atomoxetine, Axitinib, Azelastine, Barbital, Binimetinib, Bioallethrin, Bortezomib, Brivaracetam, Bromazepam, Bupivacaine, Cannabidiol, Capravirine, Carisoprodol, Cenobamate, Chlorpropamide, Cilostazol, Cisapride, Citalopram, Clobazam, Clomethiazole, Clomipramine, Clopidogrel, Clotiazepam, Clozapine, Cyclophosphamide, Dapsone, Dexibuprofen, Dexlansoprazole, Dexrabeprazole, Dextromethorphan, Diazepam, Diclofenac, Diltiazem, Diphenhydramine, Doxazosin, Doxepin, Eletriptan, Enasidenib, Encorafenib, Enfuvirtide, Escitalopram, Esketamine, Esomeprazole, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Etizolam, Etravirine, Fedratinib, Fenfluramine, Flunitrazepam, Fluoxetine, Fosphenytoin, Gliclazide, Glyburide, Guanfacine, Haloperidol, Hexobarbital, Hydrocodone, Ibuprofen, Ifosfamide, Imatinib, Imipramine, Indomethacin, Ixazomib, Ketobemidone, Labetalol, Lacosamide, Lansoprazole, Lapatinib, Levomilnacipran, Lofexidine, Lonafarnib, Loratadine, Lorcaserin, Lorlatinib, Lovastatin, Lumiracoxib, Lynestrenol, Macitentan, Medical Cannabis, Melatonin, Meperidine, Mephenytoin, Methadone, Methsuximide, Methylene blue, Methylphenobarbital, Moclobemide, Nabiximols, Nebivolol, Nelfinavir, Nicotine, Nilutamide, Norethisterone, Nortriptyline, Oliceridine, Omeprazole, Ospemifene, Oxiconazole, Oxymetazoline, Pantoprazole, Paroxetine, Pentamidine, Pentobarbital, Perphenazine, Phenacetin, Phenobarbital, Phenytoin, Piperaquine, Pipotiazine, Pirfenidone, Prasugrel, Praziquantel, Primidone, Progesterone, Proguanil, Promazine, Propofol, Propranolol, Quazepam, Quetiapine, Quinine, Rabeprazole, Ramelteon, Rilpivirine, Romidepsin, Rupatadine, Selegiline, Selumetinib, Seratrodast, Sertraline, Sildenafil, Simvastatin, St. John's Wort, Stiripentol, Tamoxifen, Tapentadol, Teniposide, Terbinafine, Testosterone, Testosterone cypionate, Testosterone enanthate, Testosterone undecanoate, Thalidomide, Thiopental, Thioridazine, Ticlopidine, Timolol, Tipranavir, Tofacitinib, Tolbutamide, Tolterodine, Trabectedin, Triclabendazole, Trimethadione, Trimipramine, Valproic acid, Verapamil, Vilazodone, Voriconazole, Vortioxetine, Voxelotor, Warfarin, Zolpidem, Zonisamide
2Cytochrome P450 2C19 inhibitorsAbiraterone, Alpelisib, Amiodarone, Amitriptyline, Amprenavir, Aprepitant, Armodafinil, Artenimol, Atorvastatin, Avasimibe, Azelastine, Benzbromarone, Bicalutamide, Bortezomib, Buprenorphine, Carbamazepine, Casimersen, Cenobamate, Chloramphenicol, Cimetidine, Cisapride, Citalopram, Clascoterone, Clevidipine, Clinafloxacin, Clozapine, Curcumin sulfate, Cyclosporine, Dabrafenib, Delavirdine, Dexlansoprazole, Diazepam, Dimethyl sulfoxide, Dosulepin, Dovitinib, Duloxetine, Elexacaftor, Enasidenib, Eslicarbazepine, Eslicarbazepine acetate, Esomeprazole, Ethambutol, Ethanol, Ethinylestradiol, Etoricoxib, Etravirine, Felbamate, Fenofibrate, Fluconazole, Fluoxetine, Fluvastatin, Fluvoxamine, Gefitinib, Gemfibrozil, Gestodene, Idelalisib, Imipramine, Indomethacin, Isavuconazole, Isoniazid, Ketoconazole, Lansoprazole, Lenvatinib, Letrozole, Lobeglitazone, Lonafarnib, Lopinavir, Loratadine, Losartan, Luliconazole, Lynestrenol, Manidipine, Memantine, Menadione, Mephenytoin, Methimazole, Methsuximide, Methylene blue, Miconazole, Midostaurin, Moclobemide, Modafinil, Naloxegol, Nicardipine, Nilutamide, Nilvadipine, Olanzapine, Omeprazole, Oritavancin, Osilodrostat, Oxcarbazepine, Pantoprazole, Phenelzine, Piperaquine, Progesterone, Quinine, Rabeprazole, Rifamycin, Rilpivirine, Rucaparib, Safinamide, Seproxetine, Sertraline, Sildenafil, Sitaxentan, Somapacitan, Somatotropin, Sorafenib, Stiripentol, Sulfanilamide, Telmisartan, Thalidomide, Ticlopidine, Tioconazole, Tipranavir, Tirbanibulin, Topiramate, Topiroxostat, Tranylcypromine, Triclabendazole, Troglitazone, Ubrogepant, Valproic acid, Vismodegib, Voriconazole, Warfarin, Zafirlukast, Zonisamide, Zucapsaicin
3Cytochrome P450 2C19 inducersAcetylsalicylic acid, Aminoglutethimide, Apalutamide, Artemether, Barbital, Betamethasone, Budesonide, Carbamazepine, Dabrafenib, Dexamethasone, Dexamethasone acetate, Efavirenz, Enzalutamide, Hydrocortisone, Hydroxyprogesterone caproate, Letermovir, Lumacaftor, Methylprednisolone, Midostaurin, Nelfinavir, Norethisterone, Opicapone, Phenobarbital, Phenytoin, Prednisolone phosphate, Prednisone, Primidone, Rifabutin, Rifampicin, Rifamycin, Rifapentine, Rifaximin, Ritonavir, Secobarbital, St. John's Wort
Interacting GroupInteracting Drugs
Formoterol is a Cytochrome P450 2C9 substrate
1Cytochrome P450 2C9 inhibitorsAbemaciclib, Abiraterone, Acetyl sulfisoxazole, Agomelatine, Amiodarone, Amodiaquine, Anastrozole, Aprepitant, Armodafinil, Atazanavir, Atorvastatin, Atovaquone, Avasimibe, Azelastine, Belinostat, Benzbromarone, Bicalutamide, Black cohosh, Bortezomib, Candesartan, Capecitabine, Casimersen, Ceritinib, Cerivastatin, Cimetidine, Cisapride, Cisplatin, Clascoterone, Clevidipine, Clinafloxacin, Clopidogrel, Clotrimazole, Crisaborole, Curcumin, Curcumin sulfate, Cyclizine, Delavirdine, Dexloxiglumide, Diacerein, Diethylstilbestrol, Doconexent, Dosulepin, Efavirenz, Elexacaftor, Enasidenib, Epinephrine, Estrone sulfate, Ethambutol, Ethanol, Etoricoxib, Etravirine, Felbamate, Felodipine, Fenofibrate, Flecainide, Floxuridine, Fluconazole, Fluorouracil, Fluoxetine, Fluvastatin, Fluvoxamine, Gefitinib, Gemfibrozil, Genistein, Ginkgo biloba, Glyburide, Imatinib, Iproniazid, Isavuconazole, Isoniazid, Ketoconazole, Ketoprofen, Lansoprazole, Leflunomide, Lenvatinib, Levofloxacin, Lifitegrast, Lobeglitazone, Lopinavir, Lumacaftor, Manidipine, Medical Cannabis, Medroxyprogesterone acetate, Mefenamic acid, Menadione, Methimazole, Methylene blue, Metronidazole, Miconazole, Midostaurin, Mifepristone, Modafinil, Nabilone, Nicardipine, Nifedipine, Nilotinib, Noscapine, Olanzapine, Opicapone, Oritavancin, Oxandrolone, Paroxetine, Pexidartinib, Phenylbutazone, Phenytoin, Pralsetinib, Pranlukast, Probenecid, Progesterone, Promethazine, Quinidine, Rabeprazole, Regorafenib, Rhein, Rifamycin, Rilpivirine, Rucaparib, Seproxetine, Sertraline, Sildenafil, Simvastatin, Sitaxentan, Sorafenib, Stiripentol, Sulconazole, Sulfadiazine, Sulfadimethoxine, Sulfamethizole, Sulfamethoxazole, Sulfamoxole, Sulfaphenazole, Sulfapyridine, Sulfinpyrazone, Sulfisoxazole, Suprofen, Tamoxifen, Teniposide, Ticagrelor, Ticlopidine, Tienilic acid, Tirbanibulin, Tolcapone, Topiroxostat, Torasemide, Tranylcypromine, Troglitazone, Ubrogepant, Valdecoxib, Valproic acid, Vemurafenib, Verapamil, Vismodegib, Voriconazole, Zafirlukast, Zucapsaicin
2Cytochrome P450 2C9 substrates(R)-warfarin, (S)-Warfarin, Aceclofenac, Acenocoumarol, Acetohexamide, Acetylsalicylic acid, Alosetron, Alprazolam, Aminophenazone, Amitriptyline, Amprenavir, Antipyrine, Apixaban, Arachidonic Acid, Arformoterol, Artemether, Asunaprevir, Atazanavir, Avanafil, Avapritinib, Azelastine, Bioallethrin, Bortezomib, Bosentan, Brivaracetam, Buprenorphine, Bupropion, Cabozantinib, Caffeine, Candesartan, Candesartan cilexetil, Cannabidiol, Capecitabine, Capravirine, Carbutamide, Carvedilol, Celecoxib, Chlorpropamide, Cinnarizine, Clopidogrel, Clozapine, Coumarin, Cyclophosphamide, Dacomitinib, Dapagliflozin, Dapsone, Desogestrel, Dexibuprofen, Dexloxiglumide, Dextromethorphan, Diazepam, Diclofenac, Dicoumarol, Diphenhydramine, Doconexent, Dolasetron, Donepezil, Dorzolamide, Doxazosin, Doxepin, Dronabinol, Duloxetine, Eletriptan, Enasidenib, Enzalutamide, Erdafitinib, Esketamine, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Estrone, Estrone sulfate, Ethinylestradiol, Etodolac, Etoricoxib, Etravirine, Febuxostat, Fenfluramine, Fluindione, Flunarizine, Flunitrazepam, Fluoxetine, Flurbiprofen, Fluvastatin, Fosphenytoin, Glibornuride, Gliclazide, Glimepiride, Glipizide, Gliquidone, Glisoxepide, Glyburide, Haloperidol, Halothane, Hexobarbital, Hydromorphone, Ibuprofen, Idarubicin, Ifosfamide, Imatinib, Indisulam, Indomethacin, Irbesartan, Istradefylline, Ixazomib, Ketamine, Ketobemidone, Ketoprofen, Ketorolac, Lacosamide, Leflunomide, Lesinurad, Licofelone, Lidocaine, Lonafarnib, Loratadine, Lornoxicam, Losartan, Lumiracoxib, Lynestrenol, Medical Cannabis, Mefenamic acid, Melatonin, Meloxicam, Mephenytoin, Mestranol, Metahexamide, Methadone, Methoxyflurane, Moclobemide, Montelukast, Nabiximols, Nabumetone, Naproxen, Nateglinide, Netupitant, Niclosamide, Nicotine, Norgestimate, Oliceridine, Olodaterol, Omeprazole, Ondansetron, Ospemifene, Paramethadione, Parecoxib, Perphenazine, Phenacetin, Phenobarbital, Phenprocoumon, Phenylbutazone, Phenytoin, Piperaquine, Pirfenidone, Piroxicam, Pitavastatin, Prasugrel, Primidone, Progesterone, Proguanil, Promazine, Propacetamol, Propofol, Quazepam, Quinidine, Quinine, Ramelteon, Rimegepant, Rofecoxib, Rosiglitazone, Rosuvastatin, Rupatadine, Ruxolitinib, Salicylic acid, Selegiline, Selumetinib, Seratrodast, Sertraline, Sildenafil, Siponimod, Sitaxentan, Sulfamethoxazole, Suprofen, Tamoxifen, Tapentadol, Temazepam, Tenoxicam, Terbinafine, Testosterone, Testosterone cypionate, Testosterone enanthate, Testosterone undecanoate, Thalidomide, Thiamylal, Tolazamide, Tolbutamide, Tolterodine, Torasemide, Trabectedin, Tranilast, Treprostinil, Tretinoin, Triclabendazole, Trifarotene, Trimethadione, Trimethoprim, Trimipramine, Troglitazone, Umbralisib, Umifenovir, Valdecoxib, Valproic acid, Valsartan, Verapamil, Vicriviroc, Vismodegib, Voriconazole, Vortioxetine, Voxelotor, Warfarin, Ximelagatran, Zafirlukast, Zaltoprofen, Zidovudine, Zileuton, Zolpidem, Zopiclone
3Cytochrome P450 2C9 inducersAlpelisib, Apalutamide, Aprepitant, Avatrombopag, Betamethasone, Bosentan, Budesonide, Carbamazepine, Dabrafenib, Dapsone, Delafloxacin, Enzalutamide, Fosaprepitant, Fosphenytoin, Hydrocortisone, Isavuconazole, Ivosidenib, Lansoprazole, Letermovir, Lopinavir, Lumacaftor, Methylprednisolone, Midostaurin, Modafinil, Nelfinavir, Nevirapine, Nifedipine, Peginterferon alfa-2b, Phenobarbital, Phenytoin, Pralsetinib, Prednisolone phosphate, Prednisone, Primidone, Rifabutin, Rifampicin, Rifamycin, Rifapentine, Ritonavir, Secobarbital, Vigabatrin, Warfarin
4Cytochrome P450 2C9 inactivatorsSuprofen
Interacting GroupInteracting Drugs
Formoterol is a Cytochrome P450 2A6 substrate
1Cytochrome P450 2A6 substratesAcetaminophen, Antipyrine, Apremilast, Arformoterol, Artesunate, Asunaprevir, Azelastine, Cenobamate, Chlorzoxazone, Cinnarizine, Cisapride, Clomethiazole, Clozapine, Cyclophosphamide, Dapagliflozin, Flunarizine, Flunitrazepam, Fluorouracil, Flurazepam, Halothane, Ifosfamide, Letrozole, Lidocaine, Lonafarnib, Lorcaserin, Methoxyflurane, Metronidazole, Montelukast, Nevirapine, Nicotine, Nifedipine, Norethisterone, Phenacetin, Phenytoin, Plitidepsin, Selegiline, Sevoflurane, Tamoxifen, Tegafur, Tegafur-uracil, Tretinoin, Valproic acid, Vortioxetine, Zidovudine
2Cytochrome P450 2A6 inhibitorsAmiodarone, Amphetamine, Azelastine, Clotrimazole, Ethambutol, Fenofibrate, Fomepizole, Isoniazid, Ketoconazole, Letrozole, Memantine, Menadione, Methimazole, Methoxsalen, Metyrapone, Miconazole, Nicotine, Nilvadipine, Pilocarpine, Rosiglitazone, Selegiline, Seratrodast, Tranylcypromine, Triclabendazole
3Cytochrome P450 2A6 inducersBetamethasone, Budesonide, Dexamethasone, Dexamethasone acetate, Eletriptan, Hydrocortisone, Methylprednisolone, Pentobarbital, Phenobarbital, Prednisolone phosphate, Prednisone, Progesterone, Rifampicin, Valproic acid
Interacting GroupInteracting Drugs
Formoterol is a UDP-glucuronosyltransferase 1A1 substrate
1UDP-glucuronosyltransferase 1A1 substratesBazedoxifene
2UDP-glucuronosyltransferase 1A1 inhibitorsOsilodrostat
Interacting GroupInteracting Drugs
Formoterol is a UDP-glucuronosyltransferase 1-8 substrate
1UDP-glucuronosyltransferase 1-8 substratesBazedoxifene, Diflunisal, Empagliflozin, Morphine, Mycophenolate mofetil, Nalmefene, Naproxen, Nintedanib, Propofol, Raloxifene, Troglitazone, Valproic acid
2UDP-glucuronosyltransferase 1-8 inhibitorsIsavuconazole
Interacting GroupInteracting Drugs
Formoterol is a UDP-glucuronosyltransferase 1-9 substrate
1UDP-glucuronosyltransferase 1-9 substratesAcetaminophen, Ambrisentan, Artenimol, Artesunate, Ataluren, Cabotegravir, Canagliflozin, Dabigatran etexilate, Dapagliflozin, Dexibuprofen, Diclofenac, Dolutegravir, Empagliflozin, Enasidenib, Entacapone, Ertugliflozin, Ethinylestradiol, Etodolac, Ezogabine, Febuxostat, Fenofibrate, Flurbiprofen, Fostamatinib, Gavestinel, Gemfibrozil, Glasdegib, Haloperidol, Ibuprofen, Indomethacin, Irinotecan, Ketobemidone, Labetalol, Lumiracoxib, Mycophenolate mofetil, Mycophenolic acid, Naproxen, Nateglinide, Oxazepam, Oxymetazoline, Phenytoin, Propacetamol, Propofol, Regorafenib, Seratrodast, Sorafenib, Tapentadol, Topiroxostat, Troglitazone, Umifenovir, Vadimezan, Valdecoxib, Valproic acid, Vericiguat, Zileuton
2UDP-glucuronosyltransferase 1-9 inhibitorsDeferasirox, Diflunisal, Eltrombopag, Fosphenytoin, Isavuconazole, Mefenamic acid, Methylene blue, Morniflumate, Niflumic acid, Phenytoin, Regorafenib, Rifampicin, Sorafenib, Umifenovir
Interacting GroupInteracting Drugs
Formoterol is a UDP-glucuronosyltransferase 2B7 substrate
1UDP-glucuronosyltransferase 2B7 substratesAcemetacin, Ambrisentan, Anastrozole, Artenimol, Artesunate, Bempedoic acid, Carbamazepine, Carvedilol, Cenobamate, Codeine, Dabigatran etexilate, Dapagliflozin, Dexibuprofen, Dextromethorphan, Diclofenac, Empagliflozin, Enasidenib, Epirubicin, Ertugliflozin, Ethinylestradiol, Etodolac, Ezetimibe, Febuxostat, Flurbiprofen, Fluvastatin, Gemfibrozil, Hydromorphone, Ibuprofen, Indomethacin, Ketorolac, Labetalol, Letrozole, Losartan, Lovastatin, Loxoprofen, Mitiglinide, Morphine, Mycophenolate mofetil, Mycophenolic acid, Nalmefene, Naproxen, Osilodrostat, Oxazepam, Pitavastatin, Silodosin, Simvastatin, Suprofen, Tamoxifen, Tapentadol, Troglitazone, Vadimezan, Valproic acid, Zaltoprofen, Zidovudine
2UDP-glucuronosyltransferase 2B7 inhibitorsChenodeoxycholic acid, Dovitinib, Flunitrazepam, Indomethacin, Ketoconazole, Mefenamic acid, Umifenovir
3UDP-glucuronosyltransferase 2B7 inducersPhenobarbital
Interacting GroupInteracting Drugs
Formoterol is a UDP-glucuronosyltransferase 2B15 substrate
1UDP-glucuronosyltransferase 2B15 substratesAcetaminophen, Dabigatran etexilate, Delafloxacin, Dextromethorphan, Enasidenib, Ezetimibe, Lorazepam, Morphine, Oxazepam, Propacetamol, Troglitazone, Valproic acid
2UDP-glucuronosyltransferase 2B15 inducersEstradiol
Interacting GroupInteracting Drugs
Formoterol is a Solute carrier family 22 member 1 substrate
1Solute carrier family 22 member 1 substratesAcetylcholine, Acyclovir, Agmatine, Amantadine, Buformin, Choline, Choline salicylate, Cimetidine, Codeine, Dexchlorpheniramine maleate, Dopamine, Epinephrine, Ganciclovir, Guanfacine, Imatinib, Lamivudine, Lamotrigine, Metformin, Nafamostat, Nintedanib, Norepinephrine, Pancuronium, Phenformin, Pramipexole, Prazosin, Quinine, Ranitidine, Rocuronium, Salmeterol, Spermidine, Spermine, Sulpiride, Thiamine, Tubocurarine
2Solute carrier family 22 member 1 inhibitorsAcyclovir, Amantadine, Chlorpheniramine, Choline, Choline salicylate, Cimetidine, Clopidogrel, Codeine, Dacomitinib, Desipramine, Dexchlorpheniramine maleate, Disopyramide, Doxazosin, Dronedarone, Efavirenz, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Ganciclovir, Gilteritinib, Guanfacine, Guanidine, Indinavir, Lasmiditan, Levofloxacin, Linagliptin, Lurbinectedin, Nelfinavir, Nevirapine, Nicotine, Nintedanib, Osilodrostat, Palbociclib, Phenoxybenzamine, Pitolisant, Prazosin, Probenecid, Procainamide, Progesterone, Quinidine, Quinine, Ranitidine, Reserpine, Rucaparib, Salmeterol, Saquinavir, Tirbanibulin, Verapamil
Interacting GroupInteracting Drugs
Formoterol is a Solute carrier family 22 member 1 inhibitor
1Solute carrier family 22 member 1 substratesAcetylcholine, Acyclovir, Agmatine, Amantadine, Buformin, Choline, Choline salicylate, Cimetidine, Codeine, Dexchlorpheniramine maleate, Dopamine, Epinephrine, Ganciclovir, Guanfacine, Imatinib, Lamivudine, Lamotrigine, Metformin, Nafamostat, Nintedanib, Norepinephrine, Pancuronium, Phenformin, Pramipexole, Prazosin, Quinine, Ranitidine, Rocuronium, Salmeterol, Spermidine, Spermine, Sulpiride, Thiamine, Tubocurarine
2Solute carrier family 22 member 1 inhibitorsAcyclovir, Amantadine, Chlorpheniramine, Choline, Choline salicylate, Cimetidine, Clopidogrel, Codeine, Dacomitinib, Desipramine, Dexchlorpheniramine maleate, Disopyramide, Doxazosin, Dronedarone, Efavirenz, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Ganciclovir, Gilteritinib, Guanfacine, Guanidine, Indinavir, Lasmiditan, Levofloxacin, Linagliptin, Lurbinectedin, Nelfinavir, Nevirapine, Nicotine, Nintedanib, Osilodrostat, Palbociclib, Phenoxybenzamine, Pitolisant, Prazosin, Probenecid, Procainamide, Progesterone, Quinidine, Quinine, Ranitidine, Reserpine, Rucaparib, Salmeterol, Saquinavir, Tirbanibulin, Verapamil
Interacting GroupInteracting Drugs
Formoterol is a Solute carrier family 22 member 4 substrate
1Solute carrier family 22 member 4 inhibitorsAmiloride, Aminohippuric acid, Arginine, Benzylpenicillin, Choline, Choline salicylate, Cimetidine, Clonidine, Desipramine, Guanidine, Imipramine, Levocarnitine, Levofloxacin, Lysine, Nicotine, Ofloxacin, Procainamide, Putrescine, Quinidine, Quinine, Spermidine, Spermine, Verapamil
2Solute carrier family 22 member 4 substratesCytarabine, Ipratropium, Levocarnitine, Testosterone cypionate, Testosterone enanthate, Testosterone undecanoate, Tiotropium
Interacting GroupInteracting Drugs
Formoterol is a Solute carrier family 22 member 5 substrate
1Solute carrier family 22 member 5 inhibitorsAcetylcholine, Aldosterone, Aminohippuric acid, Ampicillin, Arginine, Azidocillin, Benzylpenicillin, Cefadroxil, Cefalotin, Cefdinir, Cefepime, Cefixime, Cefradine, Ceftazidime, Cephalexin, Cephaloglycin, Choline, Choline salicylate, Cimetidine, Clonidine, Creatine, Cyclacillin, Dactinomycin, Desipramine, Diphenhydramine, Dopamine, Furosemide, Grepafloxacin, Guanidine, Histamine, Levamlodipine, Lidocaine, Lomefloxacin, Metamfetamine, Methacholine, Niacin, Nicotine, Norepinephrine, Norfloxacin, Ofloxacin, Probenecid, Procainamide, Quinidine, Quinine, Sparfloxacin, Thiamine, Valproic acid, Verapamil
2Solute carrier family 22 member 5 substratesAmphetamine, Ipratropium, Levocarnitine, Terbutaline, Tiotropium
Interacting GroupInteracting Drugs
Formoterol is a Solute carrier family 22 member 3 inhibitor
1Solute carrier family 22 member 3 inhibitorsCholine, Choline salicylate, Cimetidine, Clonidine, Desipramine, Dopamine, Estradiol, Estradiol acetate, Estradiol benzoate, Estradiol cypionate, Estradiol dienanthate, Estradiol valerate, Guanidine, Histamine, Imipramine, Irinotecan, Linagliptin, Melphalan, Metamfetamine, Nicotine, Norepinephrine, Phenoxybenzamine, Prazosin, Procainamide, Progesterone, Salmeterol, Vincristine
2Solute carrier family 22 member 3 substratesAdefovir dipivoxil, Agmatine, Amphetamine, Cimetidine, Guanidine, Lamivudine, Metformin, Norepinephrine, Oxaliplatin, Sulpiride, Testosterone cypionate, Testosterone enanthate